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6HGM
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Crystal structure of Alpha1-antichymotrypsin variant NewBG-III-allo: an allosterically controlled new binding globulin with an unprecedentedly high ligand release efficacy
分子名称: 1,2-ETHANEDIOL, Alpha-1-antichymotrypsin, CALCIUM ION, ...
著者Schmidt, K, Muller, Y.A.
登録日2018-08-23
公開日2019-05-29
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.369 Å)
主引用文献NewBG: A surrogate corticosteroid-binding globulin with an unprecedentedly high ligand release efficacy.
J.Struct.Biol., 207, 2019
6HGL
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Crystal structure of Alpha1-antichymotrypsin variant NewBG-III: a new binding globulin in complex with testosterone
分子名称: Alpha-1-antichymotrypsin, TESTOSTERONE
著者Schmidt, K, Muller, Y.A.
登録日2018-08-23
公開日2019-05-29
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.92 Å)
主引用文献NewBG: A surrogate corticosteroid-binding globulin with an unprecedentedly high ligand release efficacy.
J.Struct.Biol., 207, 2019
6HGK
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Crystal structure of Alpha1-antichymotrypsin variant NewBG-III: a new binding globulin in complex with progesterone
分子名称: 1,2-ETHANEDIOL, Alpha-1-antichymotrypsin, PROGESTERONE
著者Schmidt, K, Muller, Y.A.
登録日2018-08-23
公開日2019-05-29
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.855 Å)
主引用文献NewBG: A surrogate corticosteroid-binding globulin with an unprecedentedly high ligand release efficacy.
J.Struct.Biol., 207, 2019
6HGJ
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BU of 6hgj by Molmil
Crystal structure of Alpha1-antichymotrypsin variant NewBG-III: a new binding globulin in complex with aldosterone
分子名称: 1,2-ETHANEDIOL, ALDOSTERONE, Alpha-1-antichymotrypsin
著者Schmidt, K, Muller, Y.A.
登録日2018-08-23
公開日2019-05-29
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.825 Å)
主引用文献NewBG: A surrogate corticosteroid-binding globulin with an unprecedentedly high ligand release efficacy.
J.Struct.Biol., 207, 2019
6HX4
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BU of 6hx4 by Molmil
Fab fragment of a native monomer-selective antibody in complex with alpha-1-antitrypsin
分子名称: Alpha-1-antitrypsin, Fab 1D9 heavy chain, Fab 1D9 light chain
著者Elliston, E.L.K, Miranda, E, Perez, J, Jagger, A.M, Lomas, D.A, Irving, J.A.
登録日2018-10-15
公開日2019-10-30
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.95 Å)
主引用文献Characterisation of a monoclonal antibody conformationally-selective for native alpha-1-antitrypsin
To Be Published
6HGE
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BU of 6hge by Molmil
Crystal structure of Alpha1-antichymotrypsin variant NewBG-I in the uncleaved S-conformation
分子名称: Alpha-1-antichymotrypsin
著者Gardill, B.R, Schmidt, K, Muller, Y.A.
登録日2018-08-23
公開日2019-05-29
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献NewBG: A surrogate corticosteroid-binding globulin with an unprecedentedly high ligand release efficacy.
J.Struct.Biol., 207, 2019
6HGI
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BU of 6hgi by Molmil
Crystal structure of Alpha1-antichymotrypsin variant NewBG-III: a new binding globulin in complex with corticosterone
分子名称: Alpha-1-antichymotrypsin, CORTICOSTERONE
著者Schmidt, K, Muller, Y.A.
登録日2018-08-23
公開日2019-05-29
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.517 Å)
主引用文献NewBG: A surrogate corticosteroid-binding globulin with an unprecedentedly high ligand release efficacy.
J.Struct.Biol., 207, 2019
6I7U
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Alpha-1-antitrypsin (Ala250Met) in the native conformation
分子名称: Alpha-1-antitrypsin
著者Aldobiyan, I, Lomas, D.A, Irving, J.A.
登録日2018-11-19
公開日2019-11-27
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献Structural determinants of instability in alpha-1-antitrypsin
To Be Published
6HGN
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Crystal structure of Alpha1-antichymotrypsin variant DBS-II-allo-L55V: an allosterically controlled doxorubicin-binding serpin with an unprecedentedly high ligand release efficacy
分子名称: 1,2-ETHANEDIOL, Alpha-1-antichymotrypsin
著者Schmidt, K, Muller, Y.A.
登録日2018-08-23
公開日2019-05-29
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.478 Å)
主引用文献NewBG: A surrogate corticosteroid-binding globulin with an unprecedentedly high ligand release efficacy.
J.Struct.Biol., 207, 2019
6IAY
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BU of 6iay by Molmil
Alpha-1-antitrypsin Queen's (Lys154Asn) variant
分子名称: Alpha-1-antitrypsin, GLYCINE
著者Aldobiyan, I, Lomas, D.A, Irving, J.A.
登録日2018-11-28
公開日2019-12-18
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structural determinants of instability in alpha-1-antitrypsin
To Be Published
6KGA
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BU of 6kga by Molmil
Structure of Ovalbumin from Emu (Dromaius novaehollandiae)
分子名称: Ovalbumin
著者Yasutake, Y, Maehashi, K, Matano, M, Takeuchi, J.
登録日2019-07-11
公開日2019-07-24
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献Structure of Emu (Dromaius novaehollandiae) ovalbumin revealed alpha-1-antitrypsin-like domain-swapped trimer.
To Be Published
1AS4
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BU of 1as4 by Molmil
CLEAVED ANTICHYMOTRYPSIN A349R
分子名称: ACETATE ION, ANTICHYMOTRYPSIN
著者Lukacs, C.M, Christianson, D.W.
登録日1997-08-12
公開日1998-02-25
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Engineering an anion-binding cavity in antichymotrypsin modulates the "spring-loaded" serpin-protease interaction.
Biochemistry, 37, 1998
1C5G
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BU of 1c5g by Molmil
PLASMINOGEN ACTIVATOR INHIBITOR-1
分子名称: PLASMINOGEN ACTIVATOR INHIBITOR-1
著者Goldsmith, E.J.
登録日1999-12-07
公開日1999-12-17
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Engineering of plasminogen activator inhibitor-1 to reduce the rate of latency transition.
Nat.Struct.Biol., 2, 1995
1C8O
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BU of 1c8o by Molmil
2.9 A STRUCTURE OF CLEAVED VIRAL SERPIN CRMA
分子名称: ICE INHIBITOR
著者Simonovic, M, Gettins, P.G.W, Volz, K.
登録日2000-06-01
公開日2000-09-06
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Crystal structure of viral serpin crmA provides insights into its mechanism of cysteine proteinase inhibition.
Protein Sci., 9, 2000
1B3K
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BU of 1b3k by Molmil
Plasminogen activator inhibitor-1
分子名称: PLASMINOGEN ACTIVATOR INHIBITOR-1
著者Sharp, A.M, Stein, P.E, Pannu, N.S, Read, R.J.
登録日1998-12-11
公開日1999-12-11
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.99 Å)
主引用文献The active conformation of plasminogen activator inhibitor 1, a target for drugs to control fibrinolysis and cell adhesion.
Structure Fold.Des., 7, 1999
1ATH
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BU of 1ath by Molmil
THE INTACT AND CLEAVED HUMAN ANTITHROMBIN III COMPLEX AS A MODEL FOR SERPIN-PROTEINASE INTERACTIONS
分子名称: ANTITHROMBIN III
著者Schreuder, H.A, Hol, W.G.J.
登録日1993-12-14
公開日1995-02-07
最終更新日2017-11-29
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献The intact and cleaved human antithrombin III complex as a model for serpin-proteinase interactions.
Nat.Struct.Biol., 1, 1994
1ATU
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BU of 1atu by Molmil
UNCLEAVED ALPHA-1-ANTITRYPSIN
分子名称: ALPHA-1-ANTITRYPSIN
著者Ryu, S.-E, Choi, H.-J.
登録日1997-05-11
公開日1997-08-20
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献The native strains in the hydrophobic core and flexible reactive loop of a serine protease inhibitor: crystal structure of an uncleaved alpha1-antitrypsin at 2.7 A.
Structure, 4, 1996
1D5S
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BU of 1d5s by Molmil
CRYSTAL STRUCTURE OF CLEAVED ANTITRYPSIN POLYMER
分子名称: P1-ARG ANTITRYPSIN
著者Dunstone, M.A, Dai, W, Whisstock, J.C, Rossjohn, J, Pike, R.N, Feil, S.C, Le Bonneic, B.F, Parker, M.W, Bottomley, S.P.
登録日1999-10-11
公開日2000-04-02
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Cleaved antitrypsin polymers at atomic resolution.
Protein Sci., 9, 2000
1ATT
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BU of 1att by Molmil
CRYSTAL STRUCTURE OF CLEAVED BOVINE ANTITHROMBIN III AT 3.2 ANGSTROMS RESOLUTION
分子名称: ANTITHROMBIN III
著者Mourey, L, Samama, J.P, Delarue, M, Moras, D.
登録日1993-03-29
公開日1994-07-31
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Crystal structure of cleaved bovine antithrombin III at 3.2 A resolution.
J.Mol.Biol., 232, 1993
1AZX
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BU of 1azx by Molmil
ANTITHROMBIN/PENTASACCHARIDE COMPLEX
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 3,4-di-O-methyl-2,6-di-O-sulfo-alpha-D-glucopyranose-(1-4)-2,3-di-O-methyl-beta-D-glucopyranuronic acid-(1-4)-2,3,6-tri-O-sulfo-alpha-D-glucopyranose-(1-4)-3-O-methyl-2-O-sulfo-alpha-L-idopyranuronic acid-(1-4)-methyl 2,3,6-tri-O-sulfo-alpha-D-glucopyranoside, ANTITHROMBIN
著者Jin, L, Abrahams, J.P, Skinner, R, Petitou, M, Pike, R.N, Carrell, R.W.
登録日1997-11-23
公開日1999-01-13
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献The anticoagulant activation of antithrombin by heparin.
Proc.Natl.Acad.Sci.USA, 94, 1997
1DB2
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CRYSTAL STRUCTURE OF NATIVE PLASMINOGEN ACTIVATOR INHIBITOR-1
分子名称: PLASMINOGEN ACTIVATOR INHIBITOR-1
著者Nar, H, Bauer, M, Stassen, J.M, Lang, D, Gils, A, Declerck, P.
登録日1999-11-02
公開日1999-11-10
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Plasminogen activator inhibitor 1. Structure of the native serpin, comparison to its other conformers and implications for serpin inactivation.
J.Mol.Biol., 297, 2000
1E03
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PLASMA ALPHA ANTITHROMBIN-III AND PENTASACCHARIDE
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 3,4-di-O-methyl-2,6-di-O-sulfo-alpha-D-glucopyranose-(1-4)-2,3-di-O-methyl-beta-D-glucopyranuronic acid-(1-4)-2,3,6-tri-O-sulfo-alpha-D-glucopyranose-(1-4)-3-O-methyl-2-O-sulfo-alpha-L-idopyranuronic acid-(1-4)-methyl 2,3,6-tri-O-sulfo-alpha-D-glucopyranoside, ...
著者McCoy, A.J, Jin, L, Abrahams, J.-P, Skinner, R, Carrell, R.W.
登録日2000-03-09
公開日2000-06-02
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Structure of Beta-Antithrombin and the Effect of Glycosylation on Antithrombin'S Heparin Affinity and Activity.
J.Mol.Biol., 326, 2003
1DZH
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BU of 1dzh by Molmil
P14-FLUORESCEIN-N135Q-S380C-ANTITHROMBIN-III
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ANTITHROMBIN-III, ...
著者Mccoy, A.J, Huntington, J.A, Carrell, R.W.
登録日2000-02-28
公開日2000-05-26
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (2.85 Å)
主引用文献The Conformational Activation of Antithrombin. A 2. 85-A Structure of a Fluorescein Derivative Reveals an Electrostatic Link between the Hinge and Heparin Binding Regions.
J.Biol.Chem., 275, 2000
1A7C
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HUMAN PLASMINOGEN ACTIVATOR INHIBITOR TYPE-1 IN COMPLEX WITH A PENTAPEPTIDE
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[beta-D-ribopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, PENTAPEPTIDE, ...
著者Xue, Y, Inghardt, T, Sjolin, L, Deinum, J.
登録日1998-03-12
公開日1999-03-23
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Interfering with the inhibitory mechanism of serpins: crystal structure of a complex formed between cleaved plasminogen activator inhibitor type 1 and a reactive-centre loop peptide
Structure, 6, 1998
1E05
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PLASMA ALPHA ANTITHROMBIN-III
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ANTITHROMBIN-III, ...
著者McCoy, A.J, Skinner, R, Abrahams, J.-P, Pei, X.Y, Carrell, R.W.
登録日2000-03-09
公開日2000-06-02
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (2.62 Å)
主引用文献Structure of Beta-Antithrombin and the Effect of Glycosylation on Antithrombin'S Heparin Affinity and Activity.
J.Mol.Biol., 326, 2003

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