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4YHP
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Crystal structure of 309M3-B Fab in complex with H3K9me3 peptide
分子名称: Fab Heavy Chain, Fab Light Chain, H3K9me3 peptide
著者Hattori, T, Dementieva, I.S, Montano, S.P, Koide, S.
登録日2015-02-27
公開日2016-02-10
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.53 Å)
主引用文献Antigen clasping by two antigen-binding sites of an exceptionally specific antibody for histone methylation.
Proc.Natl.Acad.Sci.USA, 113, 2016
8ONE
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Crystal Structure of full-length Human Lysyl Hydroxylase LH3 - Asp190Ser mutant - Cocrystal with Fe2+, Mn2+, UDP-Glucose
分子名称: 2-OXOGLUTARIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Mattoteia, D, De Marco, M, Pinnola, A, Faravelli, S, Scietti, L, Forneris, F.
登録日2023-04-02
公開日2023-07-19
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Identification of Regulatory Molecular "Hot Spots" for LH/PLOD Collagen Glycosyltransferase Activity.
Int J Mol Sci, 24, 2023
1M9I
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Crystal Structure Of Phosphorylation-Mimicking Mutant T356D Of Annexin VI
分子名称: Annexin VI, CALCIUM ION
著者Freye-Minks, C, Kretsinger, R.H, Creutz, C.E.
登録日2002-07-29
公開日2002-08-07
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.65 Å)
主引用文献Structural and Dynamic Changes in Human Annexin VI Induced by a Phosphorylation-Mimicking Mutation, T356D
Biochemistry, 42, 2003
4YIG
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vaccinia virus D4/A20(1-50) in complex with dsDNA containing an abasic site and free uracyl
分子名称: DNA (5'-D(*AP*AP*GP*AP*TP*AP*AP*CP*AP*G)-3'), DNA (5'-D(*CP*TP*GP*TP*(ORP)P*AP*TP*CP*TP*T)-3'), DNA polymerase processivity factor component A20, ...
著者tarbouriech, N, burmeister, W.P, iseni, F.
登録日2015-03-02
公開日2015-06-10
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Crystal Structure of the Vaccinia Virus Uracil-DNA Glycosylase in Complex with DNA.
J.Biol.Chem., 290, 2015
1ML5
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Structure of the E. coli ribosomal termination complex with release factor 2
分子名称: 30S 16S RIBOSOMAL RNA, 30S RIBOSOMAL PROTEIN S10, 30S RIBOSOMAL PROTEIN S11, ...
著者Klaholz, B.P, Pape, T, Zavialov, A.V, Myasnikov, A.G, Orlova, E.V, Vestergaard, B, Ehrenberg, M, van Heel, M.
登録日2002-08-30
公開日2003-01-14
最終更新日2024-02-14
実験手法ELECTRON MICROSCOPY (14 Å)
主引用文献Structure of the Escherichia coli ribosomal termination complex with release factor 2
Nature, 421, 2003
4YIV
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Crystal structure of engineered TgAMA1 lacking the DII loop
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Apical membrane antigen AMA1, CADMIUM ION, ...
著者Parker, M.L, Boulanger, M.J.
登録日2015-03-02
公開日2015-05-20
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.93 Å)
主引用文献An Extended Surface Loop on Toxoplasma gondii Apical Membrane Antigen 1 (AMA1) Governs Ligand Binding Selectivity.
Plos One, 10, 2015
1M9R
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human endothelial nitric oxide synthase with 3-Bromo-7-Nitroindazole bound
分子名称: 3-BROMO-7-NITROINDAZOLE, PROTOPORPHYRIN IX CONTAINING FE, ZINC ION, ...
著者Rosenfeld, R.J, Garcin, E.D, Panda, K, Andersson, G, Aberg, A, Wallace, A.V, Stuehr, D.J, Tainer, J.A, Getzoff, E.D.
登録日2002-07-29
公開日2002-08-14
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.56 Å)
主引用文献Conformational Changes in Nitric Oxide Synthases Induced by Chlorzoxazone and Nitroindazoles: Crystallographic and Computational Analyses of Inhibitor Potency
Biochemistry, 41, 2002
4YJ3
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Crystal structure of tubulin bound to compound 2
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 6-(4-ethoxyphenyl)-3-(2-methoxyphenyl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine, CALCIUM ION, ...
著者McNamara, D.E, Torres, J.Z, Yeates, T.O.
登録日2015-03-03
公開日2015-05-27
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (3.75 Å)
主引用文献Structures of potent anticancer compounds bound to tubulin.
Protein Sci., 24, 2015
1MA6
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BU of 1ma6 by Molmil
TPY4 Tachyplesin I tyrosine mutant in the presence of dodecylphosphocholine micelles (300 mM)
分子名称: Tachyplesin I
著者Laederach, A, Andreotti, A.H, Fulton, D.B.
登録日2002-07-31
公開日2002-10-16
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Solution and micelle-bound structures of tachyplesin I and its active linear derivatives
Biochemistry, 41, 2002
4YKK
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Mnemiopsis leidyi ML032222a iGluR LBD D-serine complex
分子名称: D-SERINE, GLYCINE, MAGNESIUM ION, ...
著者Alberstein, R.G, Mayer, M.L.
登録日2015-03-04
公開日2015-10-21
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.38 Å)
主引用文献Glycine activated ion channel subunits encoded by ctenophore glutamate receptor genes.
Proc.Natl.Acad.Sci.USA, 112, 2015
1MB4
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Crystal structure of aspartate semialdehyde dehydrogenase from vibrio cholerae with NADP and S-methyl-l-cysteine sulfoxide
分子名称: Aspartate-Semialdehyde Dehydrogenase, CYSTEINE, NADPH DIHYDRO-NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE
著者Blanco, J, Moore, R.A, Kabaleeswaran, V, Viola, R.E.
登録日2002-08-02
公開日2003-01-07
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.84 Å)
主引用文献A structural Basis for the Mechanism of Aspartate-beta-semialdehyde Dehydrogenase from Vibrio Cholerae
Protein Sci., 12, 2003
4YL7
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BU of 4yl7 by Molmil
Crystal structure of the indole prenyltransferase MpnD from Marinactinospora thermotolerans
分子名称: Aromatic prenyltransferase
著者Mori, T, Morita, H, Abe, I.
登録日2015-03-05
公開日2016-03-16
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.601 Å)
主引用文献Manipulation of prenylation reactions by structure-based engineering of bacterial indolactam prenyltransferases.
Nat Commun, 7, 2016
1MNM
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YEAST MATALPHA2/MCM1/DNA TERNARY TRANSCRIPTION COMPLEX CRYSTAL STRUCTURE
分子名称: DNA (STE6 OPERATOR DNA), PROTEIN (MAT ALPHA-2 TRANSCRIPTIONAL REPRESSOR), PROTEIN (MCM1 TRANSCRIPTIONAL REGULATOR)
著者Tan, S, Richmond, T.J.
登録日1997-11-03
公開日1998-03-18
最終更新日2023-08-02
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Crystal structure of the yeast MATalpha2/MCM1/DNA ternary complex.
Nature, 391, 1998
1MBU
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BU of 1mbu by Molmil
Crystal Structure Analysis of ClpSN heterodimer
分子名称: ATP-Dependent clp Protease ATP-Binding Subunit clp A, BIS-(2-HYDROXYETHYL)AMINO-TRIS(HYDROXYMETHYL)METHANE YTTRIUM, CHLORIDE ION, ...
著者Guo, F, Esser, L, Singh, S.K, Maurizi, M.R, Xia, D.
登録日2002-08-03
公開日2002-12-11
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal Structure of the Heterodimeric Complex of the Adaptor, ClpS, with the N-domain of the AAA+ Chaperone, ClpA
J.Biol.Chem., 277, 2002
4YLL
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BU of 4yll by Molmil
Crystal structure of DYRK1AA in complex with 10-Bromo-substituted 11H-indolo[3,2-c]quinolone-6-carboxylic acid inhibitor 5t
分子名称: 1,2-ETHANEDIOL, 10-bromo-2-iodo-11H-indolo[3,2-c]quinoline-6-carboxylic acid, Dual specificity tyrosine-phosphorylation-regulated kinase 1A, ...
著者Chaikuad, A, Falke, H, Krojer, T, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Kunick, C, Knapp, S, Structural Genomics Consortium (SGC)
登録日2015-03-05
公開日2015-03-25
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献10-Iodo-11H-indolo[3,2-c]quinoline-6-carboxylic Acids Are Selective Inhibitors of DYRK1A.
J.Med.Chem., 58, 2015
4YM0
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BU of 4ym0 by Molmil
Crystal structure of the human galectin-4 C-terminal carbohydrate recognition domain in complex with lacto-N-tetraose (LNT)
分子名称: GLYCEROL, Galectin-4, beta-D-galactopyranose-(1-3)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Bum-Erdene, K, Blanchard, H.
登録日2015-03-06
公開日2015-07-01
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structural characterization of human galectin-4 C-terminal domain: elucidating the molecular basis for recognition of glycosphingolipids, sulfated saccharides and blood group antigens.
Febs J., 282, 2015
1MGN
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BU of 1mgn by Molmil
HIS64(E7)-> TYR APOMYOGLOBIN AS A REAGENT FOR MEASURING RATES OF HEMIN DISSOCIATION
分子名称: METMYOGLOBIN, PROTOPORPHYRIN IX CONTAINING FE, SULFATE ION
著者Hargrove, M.S, Quillin, M.L, Phillips Jr, G.N.
登録日1993-10-29
公開日1994-01-31
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献His64(E7)-->Tyr apomyoglobin as a reagent for measuring rates of hemin dissociation.
J.Biol.Chem., 269, 1994
4YM9
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Crystal structure of Porcine Pancreatic Elastase (PPE) in complex with the novel inhibitor JM102
分子名称: 2-ethyl-2-(hydroxymethyl)-N-(6-methylpyridin-3-yl)butanamide, ACETATE ION, Chymotrypsin-like elastase family member 1, ...
著者Hofbauer, S, Brito, J.A, Mulchande, J, Nogly, P, Pessanha, M, Moreira, R, Archer, M.
登録日2015-03-06
公開日2016-06-29
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Clickable 4-Oxo-beta-lactam-Based Selective Probing for Human Neutrophil Elastase Related Proteomes.
ChemMedChem, 11, 2016
1MC8
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Crystal Structure of Flap Endonuclease-1 R42E mutant from Pyrococcus horikoshii
分子名称: Flap Endonuclease-1
著者Matsui, E, Musti, K.V, Abe, J, Yamazaki, K, Matsui, I, Harata, K.
登録日2002-08-06
公開日2002-10-16
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Molecular Structure and Novel DNA Binding Sites Located in Loops of Flap Endonuclease-1 from Pyrococcus horikoshii
J.BIOL.CHEM., 277, 2002
4YMI
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Crystal structure of probable nicotinate-nucleotide adenylyltransferase from Mycobacterium abcessus in complex with NADP
分子名称: ADENINE, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, Probable nicotinate-nucleotide adenylyltransferase
著者Seattle Structural Genomics Center for Infectious Disease (SSGCID)
登録日2015-03-06
公開日2016-03-09
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Crystal structure of probable nicotinate-nucleotide adenylyltransferase from Mycobacterium abcessus in complex with NADP
to be published
1MJZ
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STRUCTURE OF INORGANIC PYROPHOSPHATASE MUTANT D97N
分子名称: INORGANIC PYROPHOSPHATASE
著者Oganesyan, V, Harutyunyan, E.H, Avaeva, S.M, Huber, R.
登録日1997-02-08
公開日1997-12-03
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Three-dimensional structures of mutant forms of E. coli inorganic pyrophosphatase with Asp-->Asn single substitution in positions 42, 65, 70, and 97.
Biochemistry Mosc., 63, 1998
4YMS
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Crystal structure of an amino acid ABC transporter
分子名称: ABC-type amino acid transport system, permease component, ABC-type polar amino acid transport system, ...
著者Ge, J, Yu, J, Yang, M.
登録日2015-03-07
公開日2015-04-22
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structural basis for substrate specificity of an amino acid ABC transporter
Proc.Natl.Acad.Sci.USA, 112, 2015
1MCL
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PRINCIPLES AND PITFALLS in DESIGNING SITE DIRECTED PEPTIDE LIGANDS
分子名称: IMMUNOGLOBULIN LAMBDA DIMER MCG (LIGHT CHAIN), N-ACETYL-D-HIS-L-PRO-OH
著者Edmundson, A.B, Harris, D.L, Fan, Z.-C, Guddat, L.W.
登録日1993-02-25
公開日1994-01-31
最終更新日2017-11-29
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Principles and pitfalls in designing site-directed peptide ligands.
Proteins, 16, 1993
4YN5
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Catalytic domain of Bacillus sp. JAMB-750 GH26 Endo-beta-1,4-mannanase
分子名称: CACODYLATE ION, Mannan endo-1,4-beta-mannosidase
著者Shimane, Y, Ohta, Y, Usami, R, Hatada, Y.
登録日2015-03-09
公開日2016-03-09
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Crystal structure of Bacillus sp. JAMB-750 GH26 Endo-beta-1,4-mannanase
To Be Published
1MI2
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SOLUTION STRUCTURE OF MURINE MACROPHAGE INFLAMMATORY PROTEIN-2, NMR, 20 STRUCTURES
分子名称: MACROPHAGE INFLAMMATORY PROTEIN-2
著者Shao, W, Jerva, L.F, West, J, Lolis, E, Schweitzer, B.I.
登録日1997-10-24
公開日1998-04-29
最終更新日2022-02-23
実験手法SOLUTION NMR
主引用文献Solution structure of murine macrophage inflammatory protein-2.
Biochemistry, 37, 1998

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