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6FCK
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CHK1 KINASE IN COMPLEX WITH COMPOUND 13
分子名称: 2-phenyl-4-[[(3~{S})-piperidin-3-yl]amino]-1~{H}-indole-7-carboxamide, SULFATE ION, Serine/threonine-protein kinase Chk1
著者Read, J.A, Breed, J.
登録日2017-12-20
公開日2018-01-17
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Adventures in Scaffold Morphing: Discovery of Fused Ring Heterocyclic Checkpoint Kinase 1 (CHK1) Inhibitors.
J. Med. Chem., 61, 2018
6FC8
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CHK1 KINASE IN COMPLEX WITH COMPOUND 13
分子名称: 2-(3-fluorophenyl)-4-[[(3~{S})-piperidin-3-yl]amino]thieno[3,2-c]pyridine-7-carboxamide, SULFATE ION, Serine/threonine-protein kinase Chk1
著者Read, J.A, Breed, J.
登録日2017-12-20
公開日2018-01-17
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.61 Å)
主引用文献Adventures in Scaffold Morphing: Discovery of Fused Ring Heterocyclic Checkpoint Kinase 1 (CHK1) Inhibitors.
J. Med. Chem., 61, 2018
1W5S
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BU of 1w5s by Molmil
Structure of the Aeropyrum Pernix ORC2 protein (ADP form)
分子名称: ADENOSINE-5'-DIPHOSPHATE, ORIGIN RECOGNITION COMPLEX SUBUNIT 2 ORC2, SULFATE ION
著者Singleton, M.R, Morales, R, Grainge, I, Cook, N, Isupov, M.N, Wigley, D.B.
登録日2004-08-09
公開日2004-10-05
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Conformational Changes Induced by Nucleotide Binding in Cdc6/Orc from Aeropyrum Pernix
J.Mol.Biol., 343, 2004
1WCN
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BU of 1wcn by Molmil
NMR structure of the carboxyterminal domains of Escherichia coli NusA
分子名称: TRANSCRIPTION ELONGATION PROTEIN NUSA
著者Eisenmann, A, Schwarz, S, Schweimer, K, Roesch, P.
登録日2004-11-18
公開日2005-08-31
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献The E. Coli Nusa Carboxy-Terminal Domains are Structurally Similar and Show Specific Rnap- and Lambdan Interactions
Protein Sci., 14, 2005
6GY2
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BU of 6gy2 by Molmil
Crystal structure of human Plk1-PBD in complex with WSSSLATPPTLSSpTVLI phosphopeptide from BRCA2
分子名称: GLYCEROL, Phosphopeptide of BRCA2, Serine/threonine-protein kinase PLK1
著者Miron, S, Ropars, V, Zinn-Justin, S.
登録日2018-06-28
公開日2019-07-10
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (3.11 Å)
主引用文献Proper chromosome alignment depends on BRCA2 phosphorylation by PLK1.
Nat Commun, 11, 2020
1Z96
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BU of 1z96 by Molmil
Crystal structure of the Mud1 UBA domain
分子名称: UBA-domain protein mud1
著者Trempe, J.-F, Brown, N.R, Lowe, E.D, Noble, M.E.M, Gordon, C, Campbell, I.D, Johnson, L.N, Endicott, J.A.
登録日2005-03-31
公開日2005-10-04
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Mechanism of Lys48-linked polyubiquitin chain recognition by the Mud1 UBA domain
Embo J., 24, 2005
6H2V
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BU of 6h2v by Molmil
Crystal structure of human METTL5-TRMT112 complex, the 18S rRNA m6A1832 methyltransferase at 2.5A resolution
分子名称: 1,2-ETHANEDIOL, 2-(2-METHOXYETHOXY)ETHANOL, DI(HYDROXYETHYL)ETHER, ...
著者van Tran, N, Graille, M.
登録日2018-07-16
公開日2019-07-31
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.49 Å)
主引用文献The human 18S rRNA m6A methyltransferase METTL5 is stabilized by TRMT112.
Nucleic Acids Res., 47, 2019
8ADD
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BU of 8add by Molmil
Viral tegument-like DUBs
分子名称: ATP-dependent DNA helicase
著者Erven, I, Abraham, E.T, Hermanns, T, Hofmann, K, Baumann, U.
登録日2022-07-08
公開日2023-02-15
最終更新日2024-09-04
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献A widely distributed family of eukaryotic and bacterial deubiquitinases related to herpesviral large tegument proteins.
Nat Commun, 13, 2022
6EKA
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BU of 6eka by Molmil
Solid-state MAS NMR structure of the HELLF prion amyloid fibrils
分子名称: Podospora anserina S mat+ genomic DNA chromosome 3, supercontig 2
著者Martinez, D, Daskalov, A, Andreas, L, Bardiaux, B, Coustou, V, Stanek, J, Berbon, M, Noubhani, M, Kauffmann, B, Wall, J.S, Pintacuda, G, Saupe, S.J, Habenstein, B, Loquet, A.
登録日2017-09-25
公開日2018-10-10
最終更新日2024-06-19
実験手法SOLID-STATE NMR
主引用文献Structural and molecular basis of cross-seeding barriers in amyloids
Proc.Natl.Acad.Sci.USA, 118, 2021
2AEO
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BU of 2aeo by Molmil
Crystal structure of cisplatinated bovine Cu,Zn superoxide dismutase
分子名称: COPPER (II) ION, Cisplatin, Superoxide dismutase [Cu-Zn], ...
著者Calderone, V, Casini, A, Mangani, S, Messori, L, Orioli, P.L.
登録日2005-07-23
公開日2006-05-02
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structural investigation of cisplatin-protein interactions: selective platination of His19 in a cuprozinc superoxide dismutase.
Angew. Chem. Int. Ed. Engl., 45, 2006
1Y98
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BU of 1y98 by Molmil
Structure of the BRCT repeats of BRCA1 bound to a CtIP phosphopeptide.
分子名称: Breast cancer type 1 susceptibility protein, COBALT (II) ION, CtIP PHOSPHORYLATED PEPTIDE, ...
著者Varma, A.K, Brown, R.S, Birrane, G, Ladias, J.A.A.
登録日2004-12-14
公開日2005-08-30
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural Basis for Cell Cycle Checkpoint Control by the BRCA1-CtIP Complex.
Biochemistry, 44, 2005
3L2D
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BU of 3l2d by Molmil
Glycocyamine kinase, beta-beta homodimer from marine worm Namalycastis sp.
分子名称: Glycocyamine kinase beta chain
著者Lim, K, Pullalarevu, S, Herzberg, O.
登録日2009-12-15
公開日2010-03-02
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structural basis for the mechanism and substrate specificity of glycocyamine kinase, a phosphagen kinase family member.
Biochemistry, 49, 2010
3L2E
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Glycocyamine kinase, alpha-beta heterodimer from marine worm Namalycastis sp.
分子名称: Glycocyamine kinase alpha chain, Glycocyamine kinase beta chain
著者Lim, K, Pullalarevu, S, Herzberg, O.
登録日2009-12-15
公開日2010-03-02
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Structural basis for the mechanism and substrate specificity of glycocyamine kinase, a phosphagen kinase family member.
Biochemistry, 49, 2010
6I8M
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BU of 6i8m by Molmil
THE CATALYTIC FRAGMENT OF POLY(ADP-RIBOSE) POLYMERASE COMPLEXED WITH ISOINDOLINONE INHIBITOR
分子名称: (1~{S})-2-(1-cyclohexylpiperidin-4-yl)-1-methyl-3-oxidanylidene-1~{H}-isoindole-4-carboxamide, Poly [ADP-ribose] polymerase 1
著者Casale, E, Papeo, G, Montagnoli, A.
登録日2018-11-20
公開日2019-05-01
最終更新日2024-05-15
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Discovery of Stereospecific PARP-1 Inhibitor Isoindolinone NMS-P515.
Acs Med.Chem.Lett., 10, 2019
6J0D
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BU of 6j0d by Molmil
Crystal structure of OsSUF4
分子名称: ZINC ION, transcription factor
著者Wang, B, Luo, Q.
登録日2018-12-24
公開日2019-11-06
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献The transcription factor OsSUF4 interacts with SDG725 in promoting H3K36me3 establishment.
Nat Commun, 10, 2019
6J0W
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BU of 6j0w by Molmil
Crystal Structure of Yeast Rtt107 and Nse6
分子名称: Peptide from DNA repair protein KRE29, Regulator of Ty1 transposition protein 107
著者Wan, B, Wu, J, Lei, M.
登録日2018-12-27
公開日2019-08-14
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Molecular Basis for Control of Diverse Genome Stability Factors by the Multi-BRCT Scaffold Rtt107.
Mol.Cell, 75, 2019
5CNV
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BU of 5cnv by Molmil
Crystal structure of the dATP inhibited E. coli class Ia ribonucleotide reductase complex bound to GDP and TTP at 3.20 Angstroms resolution
分子名称: 2'-DEOXYADENOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ...
著者Chen, P.Y.-T, Zimanyi, C.M, Funk, M.A, Drennan, C.L.
登録日2015-07-18
公開日2016-01-20
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Molecular basis for allosteric specificity regulation in class Ia ribonucleotide reductase from Escherichia coli.
Elife, 5, 2016
2RS7
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BU of 2rs7 by Molmil
Solution structure of the second dsRBD from RNA helicase A
分子名称: ATP-dependent RNA helicase A
著者Nagata, T, Muto, Y, Tsuda, K, Inoue, M, Kigawa, T, Terada, T, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2011-11-29
公開日2012-03-14
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Solution structures of the double-stranded RNA-binding domains from RNA helicase A
Proteins, 80, 2012
2RS6
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BU of 2rs6 by Molmil
Solution structure of the N-terminal dsRBD from RNA helicase A
分子名称: ATP-dependent RNA helicase A
著者Nagata, T, Muto, Y, Tsuda, K, Inoue, M, Kigawa, T, Terada, T, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2011-11-29
公開日2012-03-14
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Solution structures of the double-stranded RNA-binding domains from RNA helicase A
Proteins, 80, 2012
5CNS
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BU of 5cns by Molmil
Crystal structure of the dATP inhibited E. coli class Ia ribonucleotide reductase complex bound to CDP and dATP at 2.97 Angstroms resolution
分子名称: 2'-DEOXYADENOSINE 5'-TRIPHOSPHATE, 2'-DEOXYADENOSINE-5'-DIPHOSPHATE, CYTIDINE-5'-DIPHOSPHATE, ...
著者Chen, P.Y.-T, Zimanyi, C.M, Funk, M.A, Drennan, C.L.
登録日2015-07-18
公開日2016-01-20
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.975 Å)
主引用文献Molecular basis for allosteric specificity regulation in class Ia ribonucleotide reductase from Escherichia coli.
Elife, 5, 2016
6H2U
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BU of 6h2u by Molmil
Crystal structure of human METTL5-TRMT112 complex, the 18S rRNA m6A1832 methyltransferase at 1.6A resolution
分子名称: 1,2-ETHANEDIOL, Methyltransferase-like protein 5, Multifunctional methyltransferase subunit TRM112-like protein, ...
著者van Tran, N, Graille, M.
登録日2018-07-16
公開日2019-07-31
最終更新日2019-09-18
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献The human 18S rRNA m6A methyltransferase METTL5 is stabilized by TRMT112.
Nucleic Acids Res., 47, 2019
5CNT
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BU of 5cnt by Molmil
Crystal structure of the dATP inhibited E. coli class Ia ribonucleotide reductase complex bound to UDP and dATP at 3.25 Angstroms resolution
分子名称: 2'-DEOXYADENOSINE 5'-TRIPHOSPHATE, MAGNESIUM ION, MU-OXO-DIIRON, ...
著者Chen, P.Y.-T, Zimanyi, C.M, Funk, M.A, Drennan, C.L.
登録日2015-07-18
公開日2016-01-20
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (3.25 Å)
主引用文献Molecular basis for allosteric specificity regulation in class Ia ribonucleotide reductase from Escherichia coli.
Elife, 5, 2016
5CNU
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BU of 5cnu by Molmil
Crystal structure of the dATP inhibited E. coli class Ia ribonucleotide reductase complex bound to ADP and dGTP at 3.40 Angstroms resolution
分子名称: 2'-DEOXYADENOSINE-5'-DIPHOSPHATE, 2'-DEOXYGUANOSINE-5'-TRIPHOSPHATE, ADENOSINE-5'-DIPHOSPHATE, ...
著者Chen, P.Y.-T, Zimanyi, C.M, Funk, M.A, Drennan, C.L.
登録日2015-07-18
公開日2016-01-20
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (3.4 Å)
主引用文献Molecular basis for allosteric specificity regulation in class Ia ribonucleotide reductase from Escherichia coli.
Elife, 5, 2016
6JCG
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BU of 6jcg by Molmil
Room temperature structure of HIV-1 Integrase catalytic core domain by serial femtosecond crystallography.
分子名称: CACODYLATE ION, Integrase
著者Park, J.H, Shi, Y, Han, J, Li, X, Kim, T.H, Yun, J.H.
登録日2019-01-28
公開日2019-07-17
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Non-Cryogenic Structure and Dynamics of HIV-1 Integrase Catalytic Core Domain by X-ray Free-Electron Lasers.
Int J Mol Sci, 20, 2019
6JCF
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Cryogenic structure of HIV-1 Integrase catalytic core domain by synchrotron
分子名称: CACODYLATE ION, Integrase
著者Park, J.H, Han, J, Kim, T.H, Yun, J.H, Lee, W.
登録日2019-01-28
公開日2019-07-17
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.153 Å)
主引用文献Non-Cryogenic Structure and Dynamics of HIV-1 Integrase Catalytic Core Domain by X-ray Free-Electron Lasers.
Int J Mol Sci, 20, 2019

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