6SVL
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1BYL
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5ME7
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![BU of 5me7 by Molmil](/molmil-images/mine/5me7) | Crystal Structure of eiF4E from C. melo | 分子名称: | Eukaryotic transcription initiation factor 4E, GLYCEROL | 著者 | Querol-Audi, J, Silva, C, Miras, M, Aranda-Regules, M, Verdaguer, N. | 登録日 | 2016-11-14 | 公開日 | 2017-08-23 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Structure of eIF4E in Complex with an eIF4G Peptide Supports a Universal Bipartite Binding Mode for Protein Translation. Plant Physiol., 174, 2017
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6SSH
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2HAP
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![BU of 2hap by Molmil](/molmil-images/mine/2hap) | STRUCTURE OF A HAP1-18/DNA COMPLEX REVEALS THAT PROTEIN/DNA INTERACTIONS CAN HAVE DIRECT ALLOSTERIC EFFECTS ON TRANSCRIPTIONAL ACTIVATION | 分子名称: | DNA (5'-D(*AP*CP*GP*CP*TP*AP*TP*TP*AP*TP*CP*GP*CP*TP*AP*TP*TP*AP*GP*T)-3'), DNA (5'-D(*AP*CP*TP*AP*AP*TP*AP*GP*CP*GP*AP*TP*AP*AP*TP*AP*GP*CP*GP*T)-3'), PROTEIN (HEME ACTIVATOR PROTEIN), ... | 著者 | King, D.A, Zhang, L, Guarente, L, Marmorstein, R. | 登録日 | 1998-09-17 | 公開日 | 1999-11-10 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Structure of HAP1-18-DNA implicates direct allosteric effect of protein-DNA interactions on transcriptional activation. Nat.Struct.Biol., 6, 1999
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7K66
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![BU of 7k66 by Molmil](/molmil-images/mine/7k66) | Structure of Blood Coagulation Factor VIII in Complex with an Anti-C1 Domain Pathogenic Antibody Inhibitor | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2A9 heavy chain, ... | 著者 | Childers, K.C, Gish, J, Jarvis, L, Peters, S, Garrels, C, Smith, I.W, Spencer, H.T, Spiegel, P.C. | 登録日 | 2020-09-18 | 公開日 | 2020-10-14 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (3.92 Å) | 主引用文献 | Structure of blood coagulation factor VIII in complex with an anti-C1 domain pathogenic antibody inhibitor. Blood, 137, 2021
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8FNB
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2HAC
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![BU of 2hac by Molmil](/molmil-images/mine/2hac) | Structure of Zeta-Zeta Transmembrane Dimer | 分子名称: | T-cell surface glycoprotein CD3 zeta chain | 著者 | Chou, J.J, Wucherpfennig, K.W, Schnell, J.R, Call, M.E. | 登録日 | 2006-06-12 | 公開日 | 2006-10-31 | 最終更新日 | 2021-10-20 | 実験手法 | SOLUTION NMR | 主引用文献 | The structure of the zetazeta transmembrane dimer reveals features essential for its assembly with the T cell receptor. Cell(Cambridge,Mass.), 127, 2006
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6NOU
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![BU of 6nou by Molmil](/molmil-images/mine/6nou) | An scFv derived from ixekizumab | 分子名称: | GLYCEROL, scFv derived from ixekizumab | 著者 | Durbin, J.D, Clawson, D.K, Lu, F, Tian, Y, Lu, J, Atwell, S. | 登録日 | 2019-01-16 | 公開日 | 2019-06-19 | 最終更新日 | 2019-08-14 | 実験手法 | X-RAY DIFFRACTION (1.914 Å) | 主引用文献 | Development of tibulizumab, a tetravalent bispecific antibody targeting BAFF and IL-17A for the treatment of autoimmune disease. Mabs, 11, 2019
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6SW6
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8FNA
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![BU of 8fna by Molmil](/molmil-images/mine/8fna) | Crystal structure of the C-terminal Fg domain of human TNR | 分子名称: | CALCIUM ION, GLYCEROL, Tenascin-R | 著者 | Bouyain, S. | 登録日 | 2022-12-27 | 公開日 | 2023-07-12 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Protein-protein interactions between tenascin-R and RPTP zeta /phosphacan are critical to maintain the architecture of perineuronal nets. J.Biol.Chem., 299, 2023
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6SD5
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![BU of 6sd5 by Molmil](/molmil-images/mine/6sd5) | Structure of the RBM2 inner ring of Salmonella flagella MS-ring protein FliF with 22-fold symmetry applied | 分子名称: | Flagellar M-ring protein | 著者 | Johnson, S, Fong, Y.H, Deme, J.C, Furlong, E.J, Kuhlen, L, Lea, S.M. | 登録日 | 2019-07-26 | 公開日 | 2020-03-18 | 最終更新日 | 2024-05-22 | 実験手法 | ELECTRON MICROSCOPY (3.1 Å) | 主引用文献 | Symmetry mismatch in the MS-ring of the bacterial flagellar rotor explains the structural coordination of secretion and rotation. Nat Microbiol, 5, 2020
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6O06
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![BU of 6o06 by Molmil](/molmil-images/mine/6o06) | Extracellular factors prime enterovirus particles for uncoating | 分子名称: | VP1, VP2, VP3 | 著者 | Domanska, A, Ruokolainen, V, Pelliccia, M, Laajala, M, Butcher, S.J, Marjomaki, V.S. | 登録日 | 2019-02-15 | 公開日 | 2019-06-12 | 最終更新日 | 2024-03-20 | 実験手法 | ELECTRON MICROSCOPY (3.6 Å) | 主引用文献 | Extracellular Albumin and Endosomal Ions Prime Enterovirus Particles for Uncoating That Can Be Prevented by Fatty Acid Saturation. J.Virol., 93, 2019
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6SVC
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![BU of 6svc by Molmil](/molmil-images/mine/6svc) | Protein allostery of the WW domain at atomic resolution: apo structure | 分子名称: | Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 | 著者 | Strotz, D, Orts, J, Friedmann, M, Guntert, P, Vogeli, B, Riek, R. | 登録日 | 2019-09-18 | 公開日 | 2020-09-30 | 最終更新日 | 2024-06-19 | 実験手法 | SOLUTION NMR | 主引用文献 | Protein Allostery at Atomic Resolution. Angew.Chem.Int.Ed.Engl., 59, 2020
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8SMV
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![BU of 8smv by Molmil](/molmil-images/mine/8smv) | GPR161 Gs heterotrimer | 分子名称: | CHOLESTEROL, G-protein coupled receptor 161, Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, ... | 著者 | Hoppe, N, Manglik, A, Harrison, S. | 登録日 | 2023-04-26 | 公開日 | 2024-02-21 | 最終更新日 | 2024-03-20 | 実験手法 | ELECTRON MICROSCOPY (2.74 Å) | 主引用文献 | GPR161 structure uncovers the redundant role of sterol-regulated ciliary cAMP signaling in the Hedgehog pathway. Biorxiv, 2023
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5KDF
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![BU of 5kdf by Molmil](/molmil-images/mine/5kdf) | Inorganic pyrophosphatase from Mycobacterium tuberculosis in complex with inhibitor 6 and inorganic pyrophosphate | 分子名称: | CALCIUM ION, Inorganic pyrophosphatase, PYROPHOSPHATE 2-, ... | 著者 | Pang, A.H, Garzan, A, Garneau-Tsodikova, S, Tsodikov, O.V. | 登録日 | 2016-06-08 | 公開日 | 2016-09-28 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.45 Å) | 主引用文献 | Discovery of Allosteric and Selective Inhibitors of Inorganic Pyrophosphatase from Mycobacterium tuberculosis. ACS Chem. Biol., 11, 2016
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6C26
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![BU of 6c26 by Molmil](/molmil-images/mine/6c26) | The Cryo-EM structure of a eukaryotic oligosaccharyl transferase complex | 分子名称: | (4R,7R)-4-hydroxy-N,N,N-trimethyl-4,9-dioxo-7-[(undecanoyloxy)methyl]-3,5,8-trioxa-4lambda~5~-phosphadocosan-1-aminium, 2-acetamido-2-deoxy-beta-D-glucopyranose, Dolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1, ... | 著者 | Bai, L, Li, H. | 登録日 | 2018-01-06 | 公開日 | 2018-01-31 | 最終更新日 | 2020-07-29 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | The atomic structure of a eukaryotic oligosaccharyltransferase complex. Nature, 555, 2018
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5MRA
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![BU of 5mra by Molmil](/molmil-images/mine/5mra) | human SCBD (sorcin calcium binding domain) in complex with doxorubicin | 分子名称: | DIMETHYL SULFOXIDE, DOXORUBICIN, MAGNESIUM ION, ... | 著者 | Ilari, A, Fiorillo, A, Colotti, G, Genovese, I. | 登録日 | 2016-12-22 | 公開日 | 2017-11-29 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (3.74 Å) | 主引用文献 | Binding of doxorubicin to Sorcin impairs cell death and increases drug resistance in cancer cells. Cell Death Dis, 8, 2017
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1BND
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![BU of 1bnd by Molmil](/molmil-images/mine/1bnd) | STRUCTURE OF THE BRAIN-DERIVED NEUROTROPHIC FACTOR(SLASH)NEUROTROPHIN 3 HETERODIMER | 分子名称: | BRAIN DERIVED NEUROTROPHIC FACTOR, ISOPROPYL ALCOHOL, NEUROTROPHIN 3 | 著者 | Robinson, R.C, Radziejewski, C, Stuart, D.I, Jones, E.Y. | 登録日 | 1994-12-12 | 公開日 | 1996-04-04 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structure of the brain-derived neurotrophic factor/neurotrophin 3 heterodimer. Biochemistry, 34, 1995
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5NBW
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1G2K
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![BU of 1g2k by Molmil](/molmil-images/mine/1g2k) | HIV-1 PROTEASE WITH CYCLIC SULFAMIDE INHIBITOR, AHA047 | 分子名称: | 3-(7-BENZYL-4,5-DIHYDROXY-1,1-DIOXO-3,6-BIS-PHENOXYMETHYL-1L6-[1,2,7]THIADIAZEPAN-2-YLMETHYL)-N-METHYL-BENZAMIDE, PROTEASE RETROPEPSIN | 著者 | Lindberg, J, Unge, T. | 登録日 | 2000-10-20 | 公開日 | 2001-06-01 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Synthesis and comparative molecular field analysis (CoMFA) of symmetric and nonsymmetric cyclic sulfamide HIV-1 protease inhibitors. J.Med.Chem., 44, 2001
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8FN8
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6SPK
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![BU of 6spk by Molmil](/molmil-images/mine/6spk) | A4V MUTANT OF HUMAN SOD1 WITH EBSELEN DERIVATIVE 6 | 分子名称: | 2-selanyl-~{N}-[3-[4-(trifluoromethyl)phenyl]phenyl]benzamide, CHLORIDE ION, DIMETHYL SULFOXIDE, ... | 著者 | Chantadul, V, Amporndanai, K, Wright, G, Shahid, M, Antonyuk, S, Hasnain, S. | 登録日 | 2019-09-01 | 公開日 | 2020-03-18 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.77 Å) | 主引用文献 | Ebselen as template for stabilization of A4V mutant dimer for motor neuron disease therapy. Commun Biol, 3, 2020
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5KGX
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![BU of 5kgx by Molmil](/molmil-images/mine/5kgx) | HIV1 catalytic core domain in complex with an inhibitor (2~{S})-2-[3-(3,4-dihydro-2~{H}-chromen-6-yl)-1-methyl-indol-2-yl]-2-[(2-methylpropan-2-yl)oxy]ethanoic acid | 分子名称: | (2S)-tert-butoxy[3-(3,4-dihydro-2H-1-benzopyran-6-yl)-1-methyl-1H-indol-2-yl]acetic acid, Integrase, SULFATE ION | 著者 | Feng, L, Kobe, M, Kvaratskhelia, M. | 登録日 | 2016-06-13 | 公開日 | 2016-10-19 | 最終更新日 | 2018-03-07 | 実験手法 | X-RAY DIFFRACTION (2.67 Å) | 主引用文献 | Indole-based allosteric inhibitors of HIV-1 integrase. Bioorg.Med.Chem.Lett., 26, 2016
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6C8W
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