1CQP
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![BU of 1cqp by Molmil](/molmil-images/mine/1cqp) | CRYSTAL STRUCTURE ANALYSIS OF THE COMPLEX LFA-1 (CD11A) I-DOMAIN / LOVASTATIN AT 2.6 A RESOLUTION | 分子名称: | ANTIGEN CD11A (P180), LOVASTATIN, MAGNESIUM ION | 著者 | Kallen, J, Welzenbach, K, Ramage, P, Geyl, D, Kriwacki, R, Legge, G, Cottens, S, Weitz-Schmidt, G, Hommel, U. | 登録日 | 1999-08-10 | 公開日 | 2000-08-07 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Structural basis for LFA-1 inhibition upon lovastatin binding to the CD11a I-domain. J.Mol.Biol., 292, 1999
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3NFF
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![BU of 3nff by Molmil](/molmil-images/mine/3nff) | Crystal structure of extended Dimerization module of RNA polymerase I subcomplex A49/A34.5 | 分子名称: | RNA polymerase I subunit A34.5, RNA polymerase I subunit A49 | 著者 | Geiger, S.R, Lorenzen, K, Schreieck, A, Hanecker, P, Kostrewa, D, Heck, A.J.R, Cramer, P. | 登録日 | 2010-06-10 | 公開日 | 2010-09-08 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (3.24 Å) | 主引用文献 | RNA Polymerase I Contains a TFIIF-Related DNA-Binding Subcomplex. Mol.Cell, 39, 2010
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3NFH
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![BU of 3nfh by Molmil](/molmil-images/mine/3nfh) | Crystal structure of tandem winged helix domain of RNA polymerase I subunit A49 (P4) | 分子名称: | DNA-directed RNA polymerase I subunit RPA49 | 著者 | Geiger, S.R, Lorenzen, K, Schreieck, A, Hanecker, P, Kostrewa, D, Heck, A.J.R, Cramer, P. | 登録日 | 2010-06-10 | 公開日 | 2010-09-08 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.17 Å) | 主引用文献 | RNA Polymerase I Contains a TFIIF-Related DNA-Binding Subcomplex. Mol.Cell, 39, 2010
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2KFT
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2KI0
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![BU of 2ki0 by Molmil](/molmil-images/mine/2ki0) | NMR Structure of a de novo designed beta alpha beta | 分子名称: | DS119 | 著者 | Liang, H, Chen, H, Fan, K, Wei, P, Guo, X, Jin, C, Zeng, C, Tang, C, Lai, L. | 登録日 | 2009-04-18 | 公開日 | 2009-10-20 | 最終更新日 | 2024-05-29 | 実験手法 | SOLUTION NMR | 主引用文献 | De novo design of a beta alpha beta motif. Angew.Chem.Int.Ed.Engl., 48, 2009
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2KIB
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![BU of 2kib by Molmil](/molmil-images/mine/2kib) | Protein Fibril | 分子名称: | NFGAIL segment from human islet amyloid polypeptide | 著者 | Nielsen, J.T, Bjerring, M, Jeppesen, M.D, Pedersen, R.O, Pedersen, J.M, Hein, K.L, Vosegaard, T, Skrydstrup, T, Otzen, D.E, Nielsen, N. | 登録日 | 2009-05-01 | 公開日 | 2009-09-08 | 最終更新日 | 2024-05-01 | 実験手法 | SOLID-STATE NMR | 主引用文献 | Unique identification of supramolecular structures in amyloid fibrils by solid-state NMR spectroscopy. Angew.Chem.Int.Ed.Engl., 48, 2009
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3NFI
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![BU of 3nfi by Molmil](/molmil-images/mine/3nfi) | Crystal structure of tandem winged helix domain of RNA polymerase I subunit A49 | 分子名称: | 2-{2-[2-(2-{2-[2-(2-ETHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHOXY]-ETHOXY}-ETHANOL, DNA-directed RNA polymerase I subunit RPA49 | 著者 | Geiger, S.R, Lorenzen, K, Schreieck, A, Hanecker, P, Kostrewa, D, Heck, A.J.R, Cramer, P. | 登録日 | 2010-06-10 | 公開日 | 2010-09-08 | 最終更新日 | 2015-03-25 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | RNA Polymerase I Contains a TFIIF-Related DNA-Binding Subcomplex. Mol.Cell, 39, 2010
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1OY2
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![BU of 1oy2 by Molmil](/molmil-images/mine/1oy2) | Coupling of Folding and Binding in the PTB Domain of the Signaling Protein Shc | 分子名称: | SHC transforming protein | 著者 | Farooq, A, Zeng, L, Yan, K.S, Ravichandran, K.S, Zhou, M.-M. | 登録日 | 2003-04-03 | 公開日 | 2004-04-06 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Coupling of Folding and Binding in the PTB Domain of the Signaling Protein Shc Structure, 11, 2003
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2IZS
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![BU of 2izs by Molmil](/molmil-images/mine/2izs) | Structure of casein kinase gamma 3 in complex with inhibitor | 分子名称: | CASEIN KINASE I ISOFORM GAMMA-3, CHLORIDE ION, MAGNESIUM ION, ... | 著者 | Bunkoczi, G, Salah, E, Rellos, P, Das, S, Fedorov, O, Savitsky, P, Debreczeni, J.E, Gileadi, O, Sundstrom, M, Edwards, A, Arrowsmith, C, Weigelt, J, von Delft, F, Knapp, S. | 登録日 | 2006-07-26 | 公開日 | 2006-08-01 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Inhibitor Binding by Casein Kinases To be Published
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2HA4
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![BU of 2ha4 by Molmil](/molmil-images/mine/2ha4) | Crystal structure of mutant S203A of mouse acetylcholinesterase complexed with acetylcholine | 分子名称: | ACETATE ION, ACETYLCHOLINE, Acetylcholinesterase, ... | 著者 | Bourne, Y, Radic, Z, Sulzenbacher, G, Kim, E, Taylor, P, Marchot, P. | 登録日 | 2006-06-12 | 公開日 | 2006-07-18 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.56 Å) | 主引用文献 | Substrate and product trafficking through the active center gorge of acetylcholinesterase analyzed by crystallography and equilibrium binding J.Biol.Chem., 281, 2006
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1N3J
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![BU of 1n3j by Molmil](/molmil-images/mine/1n3j) | Structure and Substrate of a Histone H3 Lysine Methyltransferase from Paramecium Bursaria Chlorella Virus 1 | 分子名称: | Histone H3 Lysine Methyltransferase | 著者 | Manzur, K.L, Farooq, A, Zeng, L, Plotnikova, O, Sachchidanand, Koch, A.W, Zhou, M.-M. | 登録日 | 2002-10-28 | 公開日 | 2003-01-28 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | A dimeric viral SET domain methyltransferase specific to Lys27 of histone H3. Nat.Struct.Biol., 10, 2003
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2HA8
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![BU of 2ha8 by Molmil](/molmil-images/mine/2ha8) | Methyltransferase Domain of Human TAR (HIV-1) RNA binding protein 1 | 分子名称: | S-ADENOSYL-L-HOMOCYSTEINE, TAR (HIV-1) RNA loop binding protein | 著者 | Min, J, Wu, H, Zeng, H, Loppnau, P, Battaile, K, Weigelt, J, Sundstrom, M, Arrowsmith, C.H, Edwards, A.M, Bochkarev, A, Plotnikov, A.N, Structural Genomics Consortium (SGC) | 登録日 | 2006-06-12 | 公開日 | 2006-07-11 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | The Crystal Structure of Methyltransferase Domain of Human TAR (HIV-1) RNA binding protein 1 in complex with S-adenosyl-L-homocystein. To be Published
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1N6B
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![BU of 1n6b by Molmil](/molmil-images/mine/1n6b) | Microsomal Cytochrome P450 2C5/3LVdH Complex with a dimethyl derivative of sulfaphenazole | 分子名称: | 4-METHYL-N-METHYL-N-(2-PHENYL-2H-PYRAZOL-3-YL)BENZENESULFONAMIDE, Cytochrome P450 2C5, PROTOPORPHYRIN IX CONTAINING FE, ... | 著者 | Wester, M.R, Johnson, E.F, Marques-Soares, C, Dansette, P.M, Mansuy, D, Stout, C.D. | 登録日 | 2002-11-09 | 公開日 | 2003-06-03 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structure of a Substrate Complex of Mammalian Cytochrome P450 2C5 at 2.3 A Resolution: Evidence
for Multiple Substrate Binding Modes Biochemistry, 42, 2003
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6HO6
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1N72
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![BU of 1n72 by Molmil](/molmil-images/mine/1n72) | Structure and Ligand of a Histone Acetyltransferase Bromodomain | 分子名称: | HISTONE ACETYLTRANSFERASE | 著者 | Dhalluin, C, Carlson, J.E, Zeng, L, He, C, Aggarwal, A.K, Zhou, M.-M. | 登録日 | 2002-11-12 | 公開日 | 2002-12-11 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Structure and Ligand of a Histone Acetyltransferase Bromodomain Nature, 399, 1999
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3NKV
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![BU of 3nkv by Molmil](/molmil-images/mine/3nkv) | Crystal structure of Rab1b covalently modified with AMP at Y77 | 分子名称: | ADENOSINE MONOPHOSPHATE, BARIUM ION, MAGNESIUM ION, ... | 著者 | Mueller, M.P, Peters, H, Blankenfeldt, W, Goody, R.S, Itzen, A. | 登録日 | 2010-06-21 | 公開日 | 2010-08-04 | 最終更新日 | 2017-08-23 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | The Legionella effector protein DrrA AMPylates the membrane traffic regulator Rab1b. Science, 329, 2010
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6HYI
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![BU of 6hyi by Molmil](/molmil-images/mine/6hyi) | Regulatory subunit of a cAMP-independent protein kinase A from Trypanosoma cruzi at 1.4 A resolution in complex with inosine | 分子名称: | INOSINE, Protein kinase A regulatory subunit | 著者 | Volpato Santos, Y, Lorentzen, E, Basquin, J, Boshart, M. | 登録日 | 2018-10-22 | 公開日 | 2019-11-13 | 最終更新日 | 2024-04-10 | 実験手法 | X-RAY DIFFRACTION (1.39944851 Å) | 主引用文献 | Purine nucleosides replace cAMP in allosteric regulation of PKA in trypanosomatid pathogens. Elife, 12, 2024
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6HYQ
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1PWU
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![BU of 1pwu by Molmil](/molmil-images/mine/1pwu) | Crystal Structure of Anthrax Lethal Factor complexed with (3-(N-hydroxycarboxamido)-2-isobutylpropanoyl-Trp-methylamide), a known small molecule inhibitor of matrix metalloproteases. | 分子名称: | 3-(N-HYDROXYCARBOXAMIDO)-2-ISOBUTYLPROPANOYL-TRP-METHYLAMIDE, Lethal factor, ZINC ION | 著者 | Wong, T.Y, Schwarzenbacher, R, Liddington, R.C. | 登録日 | 2003-07-02 | 公開日 | 2004-02-03 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | The structural basis for substrate and inhibitor selectivity of the anthrax lethal factor. Nat.Struct.Mol.Biol., 11, 2004
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2KNJ
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![BU of 2knj by Molmil](/molmil-images/mine/2knj) | NMR structure of microplusin a antimicrobial peptide from Rhipicephalus (Boophilus) microplus | 分子名称: | Microplusin preprotein | 著者 | Pires, J.R, Rezende, C.A, Silva, F.D, Daffre, S. | 登録日 | 2009-08-26 | 公開日 | 2009-10-13 | 最終更新日 | 2022-03-16 | 実験手法 | SOLUTION NMR | 主引用文献 | Structure and mode of action of microplusin, a copper II-chelating antimicrobial peptide from the cattle tick Rhipicephalus (Boophilus) microplus. J.Biol.Chem., 284, 2009
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1PLP
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![BU of 1plp by Molmil](/molmil-images/mine/1plp) | SOLUTION STRUCTURE OF THE CYTOPLASMIC DOMAIN OF PHOSPHOLAMBAN | 分子名称: | PHOSPHOLAMBAN | 著者 | Mortishire-Smith, R.J, Pitzenberger, S.M, Burke, C.J, Middaugh, C.R, Garsky, V.M, Johnson, R.G. | 登録日 | 1995-05-01 | 公開日 | 1995-07-31 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of the cytoplasmic domain of phopholamban: phosphorylation leads to a local perturbation in secondary structure. Biochemistry, 34, 1995
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1E4K
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![BU of 1e4k by Molmil](/molmil-images/mine/1e4k) | CRYSTAL STRUCTURE OF SOLUBLE HUMAN IGG1 FC FRAGMENT-FC-GAMMA RECEPTOR III COMPLEX | 分子名称: | FC FRAGMENT OF HUMAN IGG1, LOW AFFINITY IMMUNOGLOBULIN GAMMA FC RECEPTOR III, alpha-D-galactopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-6)-[2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-3)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Sondermann, P, Huber, R, Oosthuizen, V, Jacob, U. | 登録日 | 2000-07-07 | 公開日 | 2000-08-06 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | The 3.2A Crystal Structure of the Human Igg1 Fc Fragment-Fc-Gamma-Riii Complex Nature, 406, 2000
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2HA6
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![BU of 2ha6 by Molmil](/molmil-images/mine/2ha6) | Crystal structure of mutant S203A of mouse acetylcholinesterase complexed with succinylcholine | 分子名称: | 2,2'-[(1,4-DIOXOBUTANE-1,4-DIYL)BIS(OXY)]BIS(N,N,N-TRIMETHYLETHANAMINIUM), ACETIC ACID, Acetylcholinesterase, ... | 著者 | Bourne, Y, Radic, Z, Sulzenbacher, G, Kim, E, Taylor, P, Marchot, P. | 登録日 | 2006-06-12 | 公開日 | 2006-07-18 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Substrate and product trafficking through the active center gorge of acetylcholinesterase analyzed by crystallography and equilibrium binding J.Biol.Chem., 281, 2006
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2HA7
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![BU of 2ha7 by Molmil](/molmil-images/mine/2ha7) | Crystal structure of mutant S203A of mouse acetylcholinesterase complexed with butyrylthiocholine | 分子名称: | 2-(BUTYRYLSULFANYL)-N,N,N-TRIMETHYLETHANAMINIUM, 2-(TRIMETHYLAMMONIUM)ETHYL THIOL, Acetylcholinesterase, ... | 著者 | Bourne, Y, Radic, Z, Sulzenbacher, G, Kim, E, Taylor, P, Marchot, P. | 登録日 | 2006-06-12 | 公開日 | 2006-07-18 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.66 Å) | 主引用文献 | Substrate and product trafficking through the active center gorge of acetylcholinesterase analyzed by crystallography and equilibrium binding J.Biol.Chem., 281, 2006
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3OUF
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![BU of 3ouf by Molmil](/molmil-images/mine/3ouf) | Structure of a K+ selective NaK mutant | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, POTASSIUM ION, Potassium channel protein | 著者 | Derebe, M.G, Sauer, D.B, Zeng, W, Alam, A, Shi, N, Jiang, Y. | 登録日 | 2010-09-14 | 公開日 | 2011-01-12 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Tuning the ion selectivity of tetrameric cation channels by changing the number of ion binding sites. Proc.Natl.Acad.Sci.USA, 108, 2011
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