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7AA4
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BU of 7aa4 by Molmil
Structure of ClpC1-NTD bound to a CymA analogue
分子名称: Negative regulator of genetic competence ClpC/mecB, polymer Cyclomarin A analogue
著者Meinhart, A, Morreale, F.E, Kaiser, M, Clausen, T.
登録日2020-09-03
公開日2021-08-11
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.68 Å)
主引用文献BacPROTACs mediate targeted protein degradation in bacteria.
Cell, 185, 2022
3TV6
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BU of 3tv6 by Molmil
Human B-Raf Kinase Domain in Complex with a Methoxypyrazolopyridinyl Benzamide Inhibitor
分子名称: 2,6-difluoro-N-(3-methoxy-2H-pyrazolo[3,4-b]pyridin-5-yl)-3-[(propylsulfonyl)amino]benzamide, Serine/threonine-protein kinase B-raf
著者Voegtli, W.C, Sturgis, H.L, Wu, W.-I.
登録日2011-09-19
公開日2011-10-05
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献Pyrazolopyridine Inhibitors of B-Raf(V600E). Part 1: The Development of Selective, Orally Bioavailable, and Efficacious Inhibitors.
ACS Med Chem Lett, 2, 2011
1E0E
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BU of 1e0e by Molmil
N-terminal zinc-binding HHCC domain of HIV-2 integrase
分子名称: HUMAN IMMUNODEFICIENCY VIRUS TYPE 2 INTEGRASE, ZINC ION
著者Eijkelenboom, A.P.A.M, Van Den ent, F.M.I, Plasterk, R.H.A, Kaptein, R, Boelens, R.
登録日2000-03-25
公開日2001-03-19
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Refined Solution Structure of the Dimeric N-Terminal Hhcc Domain of HIV-2 Integrase
J.Biomol.NMR, 18, 2000
3FD7
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BU of 3fd7 by Molmil
Crystal structure of Onconase C87A/C104A-ONC
分子名称: 1,2-ETHANEDIOL, GLYCEROL, Protein P-30, ...
著者Neumann, P, Schulenburg, C, Arnold, U, Ulbrich-Hofmann, R, Stubbs, M.T.
登録日2008-11-25
公開日2009-12-08
最終更新日2024-11-06
実験手法X-RAY DIFFRACTION (1.531 Å)
主引用文献Impact of the C-terminal disulfide bond on the folding and stability of onconase.
Chembiochem, 11, 2010
9ATV
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BU of 9atv by Molmil
X-ray co-crystal structure of NCGC00685960 / NCATS-SM9335 in NNMT
分子名称: (8M)-8-{3-[(3S)-1-(2-cyclohexylethyl)piperidin-3-yl]-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl}quinolin-2(1H)-one, Nicotinamide N-methyltransferase
著者Olland, A, White, A, Suto, R.
登録日2024-02-27
公開日2025-03-05
実験手法X-RAY DIFFRACTION (2.413 Å)
主引用文献NNMT inhibition blocks cancer-associated fibroblast-mediated immunosuppressi on
To Be Published
9ARJ
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BU of 9arj by Molmil
CryoEM structure of BoNT-NTNH-OrfX2 complex from Clostridium botulinum E1, major class
分子名称: Botulinum neurotoxin, Peptidase M27, Toxin
著者Gao, L.
登録日2024-02-23
公開日2025-01-22
最終更新日2025-05-28
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Botulinum neurotoxins exploit host digestive proteases to boost their oral toxicity via activating OrfXs/P47.
Nat.Struct.Mol.Biol., 32, 2025
9ARK
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BU of 9ark by Molmil
CryoEM structure of BoNT-NTNH-OrfX2 complex from Clostridium botulinum E1, minor class
分子名称: Botulinum neurotoxin, Peptidase M27, Toxin
著者Gao, L.
登録日2024-02-23
公開日2025-01-22
最終更新日2025-05-28
実験手法ELECTRON MICROSCOPY (4.1 Å)
主引用文献Botulinum neurotoxins exploit host digestive proteases to boost their oral toxicity via activating OrfXs/P47.
Nat.Struct.Mol.Biol., 32, 2025
9ARL
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BU of 9arl by Molmil
CryoEM structure of BoNT-NTNH-OrfX2 complex from Clostridium botulinum strain A1-ST7B, major class
分子名称: Botulinum neurotoxin type A, NtnH, OrfX2
著者Gao, L.
登録日2024-02-23
公開日2025-01-22
最終更新日2025-05-28
実験手法ELECTRON MICROSCOPY (4 Å)
主引用文献Botulinum neurotoxins exploit host digestive proteases to boost their oral toxicity via activating OrfXs/P47.
Nat.Struct.Mol.Biol., 32, 2025
7Y43
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BU of 7y43 by Molmil
Crystal structure of the KAT6A WH domain and its bound double stranded DNA
分子名称: DNA (5'-D(*GP*GP*AP*GP*TP*GP*CP*GP*CP*AP*CP*TP*CP*C)-3'), Histone acetyltransferase KAT6A, MAGNESIUM ION
著者Wang, Z, Jia, Y.
登録日2022-06-13
公開日2023-01-18
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献The histone acetyltransferase KAT6A is recruited to unmethylated CpG islands via a DNA binding winged helix domain.
Nucleic Acids Res., 51, 2023
4EIG
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BU of 4eig by Molmil
CA1698 camel antibody fragment in complex with DHFR
分子名称: CA1698 camel antibody fragment, Dihydrofolate reductase
著者Oyen, D, Srinivasan, V.
登録日2012-04-05
公開日2013-04-24
最終更新日2024-11-06
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Mechanistic analysis of allosteric and non-allosteric effects arising from nanobody binding to two epitopes of the dihyrofolate reductase of Escherichia coli.
Biochim.Biophys.Acta, 1834, 2013
4EIZ
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BU of 4eiz by Molmil
Structure of Nb113 bound to apoDHFR
分子名称: Dihydrofolate reductase, Nb113 Camel antibody fragment
著者Oyen, D, Srinivasan, V.
登録日2012-04-06
公開日2013-04-24
最終更新日2024-11-20
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Mechanistic analysis of allosteric and non-allosteric effects arising from nanobody binding to two epitopes of the dihyrofolate reductase of Escherichia coli.
Biochim.Biophys.Acta, 1834, 2013
5O8D
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BU of 5o8d by Molmil
Mutant of class II CPD photolyase from Methanosarcina mazei - Y345F
分子名称: Deoxyribodipyrimidine photolyase, FLAVIN-ADENINE DINUCLEOTIDE, GLYCEROL, ...
著者Ignatz, E, Essen, L.-O.
登録日2017-06-13
公開日2017-09-13
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Nicotinamide Adenine Dinucleotides Arrest Photoreduction of Class II DNA Photolyases in FADH ̇ State.
Photochem. Photobiol., 94, 2018
4EJ1
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BU of 4ej1 by Molmil
Binding of Nb113 camelid antibody fragment with the binary DHFR:folate complex
分子名称: Dihydrofolate reductase, FOLIC ACID, Nb113 camelid antibody fragment, ...
著者Oyen, D, Srinivasan, V.
登録日2012-04-06
公開日2013-04-24
最終更新日2024-11-20
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Mechanistic analysis of allosteric and non-allosteric effects arising from nanobody binding to two epitopes of the dihyrofolate reductase of Escherichia coli.
Biochim.Biophys.Acta, 1834, 2013
1O58
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BU of 1o58 by Molmil
Crystal structure of O-acetylserine sulfhydrylase (TM0665) from Thermotoga maritima at 1.80 A resolution
分子名称: O-acetylserine sulfhydrylase, PHOSPHATE ION
著者Joint Center for Structural Genomics (JCSG)
登録日2003-08-20
公開日2003-09-02
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Crystal structure of O-acetylserine sulfhydrylase (TM0665) from Thermotoga maritima at 1.8 A resolution
Proteins, 56, 2004
4FGV
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BU of 4fgv by Molmil
Crystal structure of free CRM1 (crystal form 1)
分子名称: Chromosome region maintenance 1 (CRM1) or Exportin 1 (Xpo1)
著者Monecke, T, Neumann, P, Dickmanns, A, Ficner, R.
登録日2012-06-05
公開日2013-01-23
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.941 Å)
主引用文献Structural basis for cooperativity of CRM1 export complex formation.
Proc.Natl.Acad.Sci.USA, 110, 2013
1O2D
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BU of 1o2d by Molmil
Crystal structure of Alcohol dehydrogenase, iron-containing (TM0920) from Thermotoga maritima at 1.30 A resolution
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Alcohol dehydrogenase, iron-containing, ...
著者Joint Center for Structural Genomics (JCSG)
登録日2003-02-27
公開日2003-06-10
最終更新日2024-11-20
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献Crystal structure of an iron-containing 1,3-propanediol dehydrogenase (TM0920) from Thermotoga maritima at 1.3 A resolution
Proteins, 54, 2004
4FHB
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BU of 4fhb by Molmil
Enhancing DHFR catalysis by binding of an allosteric regulator nanobody (Nb179)
分子名称: Dihydrofolate reductase, FOLIC ACID, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ...
著者Oyen, D.
登録日2012-06-06
公開日2013-04-24
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Mechanistic analysis of allosteric and non-allosteric effects arising from nanobody binding to two epitopes of the dihyrofolate reductase of Escherichia coli.
Biochim.Biophys.Acta, 1834, 2013
5O9Z
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BU of 5o9z by Molmil
Cryo-EM structure of a pre-catalytic human spliceosome primed for activation (B complex)
分子名称: 116 kDa U5 small nuclear ribonucleoprotein component, Homo sapiens RNA, U6 small nuclear 1 (RNU6-1), ...
著者Bertram, K, Kastner, B.
登録日2017-06-20
公開日2017-08-16
最終更新日2025-07-09
実験手法ELECTRON MICROSCOPY (4.5 Å)
主引用文献Cryo-EM Structure of a Pre-catalytic Human Spliceosome Primed for Activation.
Cell, 170, 2017
5O86
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BU of 5o86 by Molmil
Mutant of claas II CPD photolyase from Methanosarcina mazei - W388F
分子名称: Deoxyribodipyrimidine photolyase, FLAVIN-ADENINE DINUCLEOTIDE, GLYCEROL, ...
著者Ignatz, E, Essen, L.-O.
登録日2017-06-12
公開日2017-09-13
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.687 Å)
主引用文献Nicotinamide Adenine Dinucleotides Arrest Photoreduction of Class II DNA Photolyases in FADH ̇ State.
Photochem. Photobiol., 94, 2018
2KB6
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BU of 2kb6 by Molmil
Solution structure of onconase C87A/C104A
分子名称: Protein P-30
著者Weininger, U, Schulenburg, C, Arnold, U, Ulbrich-Hofmann, R, Balbach, J.
登録日2008-11-21
公開日2009-11-24
最終更新日2024-10-30
実験手法SOLUTION NMR
主引用文献Impact of the C-terminal disulfide bond on the folding and stability of onconase.
Chembiochem, 11, 2010
2LFJ
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BU of 2lfj by Molmil
Solution structure of the monomeric derivative of BS-RNase
分子名称: Seminal ribonuclease
著者Spadaccini, R, Picone, D.
登録日2011-07-06
公開日2012-02-08
最終更新日2024-10-30
実験手法SOLUTION NMR
主引用文献NMR Studies on Structure and Dynamics of the Monomeric Derivative of BS-RNase: New Insights for 3D Domain Swapping.
Plos One, 7, 2012
7BL6
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BU of 7bl6 by Molmil
50S-ObgE-GMPPNP particle
分子名称: 23S ribosomal RNA, 50S ribosomal protein L13, 50S ribosomal protein L14, ...
著者Hilal, T, Nikolay, R, Schmidt, S, Spahn, C.M.T.
登録日2021-01-18
公開日2021-05-12
最終更新日2024-05-01
実験手法ELECTRON MICROSCOPY (4 Å)
主引用文献Snapshots of native pre-50S ribosomes reveal a biogenesis factor network and evolutionary specialization.
Mol.Cell, 81, 2021
7BL2
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BU of 7bl2 by Molmil
pre-50S-ObgE particle state 1
分子名称: 23S ribosomal RNA, 50S ribosomal protein L11, 50S ribosomal protein L13, ...
著者Hilal, T, Nikolay, R, Schmidt, S, Spahn, C.M.T.
登録日2021-01-18
公開日2021-05-12
最終更新日2024-05-01
実験手法ELECTRON MICROSCOPY (3.7 Å)
主引用文献Snapshots of native pre-50S ribosomes reveal a biogenesis factor network and evolutionary specialization.
Mol.Cell, 81, 2021
7BL3
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BU of 7bl3 by Molmil
pre-50S-ObgE particle state 2
分子名称: 23S ribosomal RNA, 50S ribosomal protein L11, 50S ribosomal protein L13, ...
著者Hilal, T, Nikolay, R, Spahn, C.M.T.
登録日2021-01-18
公開日2021-05-12
最終更新日2024-10-23
実験手法ELECTRON MICROSCOPY (3.5 Å)
主引用文献Snapshots of native pre-50S ribosomes reveal a biogenesis factor network and evolutionary specialization.
Mol.Cell, 81, 2021
7BL5
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BU of 7bl5 by Molmil
pre-50S-ObgE particle
分子名称: 23S ribosomal RNA, 50S ribosomal protein L10, 50S ribosomal protein L11, ...
著者Hilal, T, Nikolay, R, Spahn, C.M.T, Schmidt, S.
登録日2021-01-18
公開日2021-05-12
最終更新日2025-04-09
実験手法ELECTRON MICROSCOPY (3.3 Å)
主引用文献Snapshots of native pre-50S ribosomes reveal a biogenesis factor network and evolutionary specialization.
Mol.Cell, 81, 2021

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