Loading
PDBj
メニューPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

6QCI
DownloadVisualize
BU of 6qci by Molmil
Structure of XIAP-BIR1 V86E mutant
分子名称: DI(HYDROXYETHYL)ETHER, E3 ubiquitin-protein ligase XIAP, SODIUM ION, ...
著者Sorrentino, L, Cossu, F, Milani, M, Mastrangelo, E.
登録日2018-12-28
公開日2019-05-01
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structure-Activity Relationship of NF023 Derivatives Binding to XIAP-BIR1.
Chemistryopen, 8, 2019
3FUQ
DownloadVisualize
BU of 3fuq by Molmil
Glycosylated SV2 and Gangliosides as Dual Receptors for Botulinum Neurotoxin Serotype F
分子名称: BoNT/F (Neurotoxin type F)
著者Fu, Z, Chen, C, Barbieri, J.T, Kim, J.-J.P, Baldwin, M.R.
登録日2009-01-14
公開日2009-06-16
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Glycosylated SV2 and gangliosides as dual receptors for botulinum neurotoxin serotype F
Biochemistry, 48, 2009
6QE9
DownloadVisualize
BU of 6qe9 by Molmil
The X-ray structure of the adduct formed in the reaction between bovine pancreatic ribonuclease and complex I, a pentacoordinate Pt(II) compound containing 2,9-dimethyl-1,10-phenanthroline, dimethylfumarate, methyl and iodine as ligands
分子名称: Ribonuclease pancreatic, SULFATE ION, pentacoordinate Pt(II) compound
著者Merlino, A, Ferraro, G.
登録日2019-01-07
公開日2019-02-27
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.03 Å)
主引用文献Reaction with Proteins of a Five-Coordinate Platinum(II) Compound.
Int J Mol Sci, 20, 2019
6Q2Y
DownloadVisualize
BU of 6q2y by Molmil
Crystal structure of NDM-1 beta-lactamase in complex with broad spectrum boronic inhibitor cpd3
分子名称: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, CALCIUM ION, Metallo-beta-lactamase type 2, ...
著者Maso, L, Quotadamo, A, Bellio, P, Montanari, M, Venturelli, A, Celenza, G, Costi, M.P, Tondi, D, Cendron, L.
登録日2018-12-03
公開日2019-04-24
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1 Å)
主引用文献X-ray Crystallography Deciphers the Activity of Broad-Spectrum Boronic Acid beta-Lactamase Inhibitors.
Acs Med.Chem.Lett., 10, 2019
6RYV
DownloadVisualize
BU of 6ryv by Molmil
Copper oxidase from Colletotrichum graminicola
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, COPPER (II) ION, Kelch domain-containing protein, ...
著者Offen, W.A, Henrissat, B, Davies, G.J.
登録日2019-06-12
公開日2019-11-13
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Discovery of a Fungal Copper Radical Oxidase with High Catalytic Efficiency toward 5-Hydroxymethylfurfural and Benzyl Alcohols for Bioprocessing
Acs Catalysis, 2020
3JXI
DownloadVisualize
BU of 3jxi by Molmil
Crystal structure of the chicken TRPV4 ankyrin repeat domain
分子名称: Vanilloid receptor-related osmotically activated channel protein
著者Phelps, C.B, Wang, R.R, Gaudet, R.
登録日2009-09-19
公開日2009-12-22
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Mutations in TRPV4 cause Charcot-Marie-Tooth disease type 2C.
Nat.Genet., 42, 2010
6WC5
DownloadVisualize
BU of 6wc5 by Molmil
Crystal Structure of a Ternary MEF2B/NKX2-5/myocardin enhancer DNA Complex
分子名称: Homeobox protein Nkx-2.5, Myocardin enhancer DNA, Myocyte-specific enhancer factor 2B
著者Chen, L, Lei, X.
登録日2020-03-29
公開日2020-07-22
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Crystal Structures of Ternary Complexes of MEF2 and NKX2-5 Bound to DNA Reveal a Disease Related Protein-Protein Interaction Interface.
J.Mol.Biol., 432, 2020
6RZA
DownloadVisualize
BU of 6rza by Molmil
Cryo-EM structure of the human inner arm dynein DNAH7 microtubule binding domain bound to microtubules
分子名称: Cytoplasmic dynein 1 heavy chain 1,Dynein heavy chain 7, axonemal,Cytoplasmic dynein 1 heavy chain 1, GUANOSINE-5'-DIPHOSPHATE, ...
著者Lacey, S.E, He, S, Scheres, S.H.W, Carter, A.P.
登録日2019-06-13
公開日2019-07-10
最終更新日2024-05-22
実験手法ELECTRON MICROSCOPY (4.5 Å)
主引用文献Cryo-EM of dynein microtubule-binding domains shows how an axonemal dynein distorts the microtubule.
Elife, 8, 2019
6S04
DownloadVisualize
BU of 6s04 by Molmil
Crystal structure of an inverting family GH156 exosialidase from uncultured bacterium pG7 in complex with N-glycolylneuraminic acid
分子名称: ACETATE ION, GLYCEROL, N-glycolyl-beta-neuraminic acid, ...
著者Bule, P, Blagova, E, Chuzel, L, Taron, C.H, Davies, G.J.
登録日2019-06-13
公開日2019-11-06
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Inverting family GH156 sialidases define an unusual catalytic motif for glycosidase action.
Nat Commun, 10, 2019
6QG0
DownloadVisualize
BU of 6qg0 by Molmil
Structure of eIF2B-eIF2 (phosphorylated at Ser51) complex (model 1)
分子名称: Eukaryotic translation initiation factor 2 subunit alpha, Eukaryotic translation initiation factor 2 subunit beta, Eukaryotic translation initiation factor 2 subunit gamma, ...
著者Llacer, J.L, Gordiyenko, Y, Ramakrishnan, V.
登録日2019-01-10
公開日2019-06-26
最終更新日2019-12-18
実験手法ELECTRON MICROSCOPY (4.2 Å)
主引用文献Structural basis for the inhibition of translation through eIF2 alpha phosphorylation.
Nat Commun, 10, 2019
3JZQ
DownloadVisualize
BU of 3jzq by Molmil
Human MDMX liganded with a 12mer peptide inhibitor (pDIQ)
分子名称: Protein Mdm4, SULFATE ION, pDIQ peptide (12mer)
著者Schonbrunn, E, Phan, J.
登録日2009-09-24
公開日2009-11-10
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structure-based design of high affinity peptides inhibiting the interaction of p53 with MDM2 and MDMX.
J.Biol.Chem., 285, 2010
6Q45
DownloadVisualize
BU of 6q45 by Molmil
F1-ATPase from Fusobacterium nucleatum
分子名称: ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, ATP synthase epsilon chain, ...
著者Petri, J, Nakatani, Y, Montgomery, M.G, Ferguson, S.A, Aragao, D, Leslie, A.G.W, Heikal, A, Walker, J.E, Cook, G.M.
登録日2018-12-05
公開日2019-07-10
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (3.6 Å)
主引用文献Structure of F1-ATPase from the obligate anaerobe Fusobacterium nucleatum.
Open Biology, 9, 2019
6RGY
DownloadVisualize
BU of 6rgy by Molmil
Revisiting pH-gated conformational switch. Complex HK853-RR468 pH 7.5
分子名称: ADENOSINE-5'-DIPHOSPHATE, CITRIC ACID, MAGNESIUM ION, ...
著者Mideros-Mora, C, Casino, P, Marina, A.
登録日2019-04-18
公開日2020-02-19
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Revisiting the pH-gated conformational switch on the activities of HisKA-family histidine kinases.
Nat Commun, 11, 2020
6RI2
DownloadVisualize
BU of 6ri2 by Molmil
Single crystal serial study of the inhibition of laccases from Steccherinum murashkinskyi by chloride anions at sub-atomic resolution. Twentieth structure of the series with 4065 KGy dose.
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CHLORIDE ION, COPPER (II) ION, ...
著者Polyakov, K.M, Gavryushov, S, Fedorova, T.V, Glazunova, O.A, Popov, A.N.
登録日2019-04-23
公開日2019-05-01
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.09 Å)
主引用文献The subatomic resolution study of laccase inhibition by chloride and fluoride anions using single-crystal serial crystallography: insights into the enzymatic reaction mechanism.
Acta Crystallogr D Struct Biol, 75, 2019
6QKT
DownloadVisualize
BU of 6qkt by Molmil
Crystal Structure of the Fluoroacetate Dehalogenase RPA1163 - Tyr219Phe - Fluoroacetate soaked 24hr - Glycolate bound
分子名称: Fluoroacetate dehalogenase, GLYCOLIC ACID
著者Mehrabi, P, Kim, T.H, Prosser, R.S, Pai, E.F.
登録日2019-01-30
公開日2019-06-26
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.512 Å)
主引用文献Substrate-Based Allosteric Regulation of a Homodimeric Enzyme.
J.Am.Chem.Soc., 141, 2019
6S6Z
DownloadVisualize
BU of 6s6z by Molmil
Structure of beta-Galactosidase from Thermotoga maritima
分子名称: Beta-galactosidase, MAGNESIUM ION
著者Miguez-Amil, S, Jimenez-Ortega, E, Ramirez Escudero, M, Sanz-Aparicio, J, Fernandez-Leiro, R.
登録日2019-07-04
公開日2020-03-18
最終更新日2024-05-22
実験手法ELECTRON MICROSCOPY (2 Å)
主引用文献The cryo-EM Structure ofThermotoga maritimabeta-Galactosidase: Quaternary Structure Guides Protein Engineering.
Acs Chem.Biol., 15, 2020
6WIS
DownloadVisualize
BU of 6wis by Molmil
Copper resistance protein copG- Form 1
分子名称: ACETATE ION, COPPER (II) ION, DUF411 domain-containing protein, ...
著者Hausrath, A.C, Ly, A, McEvoy, M.M.
登録日2020-04-10
公開日2020-06-24
最終更新日2020-08-19
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献The bacterial copper resistance protein CopG contains a cysteine-bridged tetranuclear copper cluster.
J.Biol.Chem., 295, 2020
6Q50
DownloadVisualize
BU of 6q50 by Molmil
Structure of MPT-4, a mannose phosphorylase from Leishmania mexicana, in complex with phosphate ion
分子名称: 1,2-ETHANEDIOL, MPT-4, PHOSPHATE ION, ...
著者Sobala, L.F, Males, A, Bastidas, L.M, Ward, T, Sernee, M.F, Ralton, J.E, Nero, T.L, Cobbold, S, Kloehn, J, Viera-Lara, M, Stanton, L, Hanssen, E, Parker, M.W, Williams, S.J, McConville, M.J, Davies, G.J.
登録日2018-12-06
公開日2019-09-25
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献A Family of Dual-Activity Glycosyltransferase-Phosphorylases Mediates Mannogen Turnover and Virulence in Leishmania Parasites.
Cell Host Microbe, 26, 2019
3K42
DownloadVisualize
BU of 3k42 by Molmil
Crystal structure of sCD-MPR mutant E19Q/K137M pH 7.0
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Cation-dependent mannose-6-phosphate receptor, SN-GLYCEROL-1-PHOSPHATE, ...
著者Olson, L.J, Sun, G, Bohnsack, R.N, Peterson, F.C, Dahms, N.M, Kim, J.J.P.
登録日2009-10-05
公開日2009-11-24
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Intermonomer interactions are essential for lysosomal enzyme binding by the cation-dependent mannose 6-phosphate receptor.
Biochemistry, 49, 2010
6Q6C
DownloadVisualize
BU of 6q6c by Molmil
Pore-modulating toxins exploit inherent slow inactivation to block K+ channels
分子名称: 1,2-ETHANEDIOL, Kunitz-type conkunitzin-S1, NITRATE ION, ...
著者Karbat, I, Gueta, H, Fine, S, Szanto, T, Hamer-Rogotner, S, Dym, O, Frolow, F, Gordon, D, Panyi, G, Gurevitz, M, Reuveny, E.
登録日2018-12-10
公開日2019-08-21
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献Pore-modulating toxins exploit inherent slow inactivation to block K+channels.
Proc.Natl.Acad.Sci.USA, 116, 2019
6WGY
DownloadVisualize
BU of 6wgy by Molmil
Crystal structure of a Putative citrate synthase 2 from Mycobacterium bovis in complex with citrate
分子名称: CITRIC ACID, IODIDE ION, Putative citrate synthase 2
著者Seattle Structural Genomics Center for Infectious Disease (SSGCID)
登録日2020-04-06
公開日2020-04-22
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal structure of a Putative citrate synthase 2 from Mycobacterium bovis in complex with citrate
to be published
6RYX
DownloadVisualize
BU of 6ryx by Molmil
Copper oxidase from Colletotrichum graminicola
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, COPPER (II) ION, DI(HYDROXYETHYL)ETHER, ...
著者Offen, W.A, Henrissat, B, Davies, G.J.
登録日2019-06-12
公開日2019-11-13
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.65 Å)
主引用文献Discovery of a Fungal Copper Radical Oxidase with High Catalytic Efficiency toward 5-Hydroxymethylfurfural and Benzyl Alcohols for Bioprocessing
Acs Catalysis, 2020
3K77
DownloadVisualize
BU of 3k77 by Molmil
X-ray crystal structure of XRCC1
分子名称: DNA repair protein XRCC1
著者Cuneo, M.J, London, R.E.
登録日2009-10-12
公開日2010-04-28
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.597 Å)
主引用文献Oxidation state of the XRCC1 N-terminal domain regulates DNA polymerase beta binding affinity.
Proc.Natl.Acad.Sci.USA, 107, 2010
6WDV
DownloadVisualize
BU of 6wdv by Molmil
Crystal Structure of Danio rerio Histone Deacetylase 10 in Complex with Dimethylaminomethylindole Phenylhydroxamate Inhibitor
分子名称: 4-({3-[(dimethylamino)methyl]-1H-indol-1-yl}methyl)-N-hydroxybenzamide, PHOSPHATE ION, POTASSIUM ION, ...
著者Herbst-Gervasoni, C.J, Christianson, D.W.
登録日2020-04-01
公開日2020-07-22
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structural Basis for the Selective Inhibition of HDAC10, the Cytosolic Polyamine Deacetylase.
Acs Chem.Biol., 15, 2020
6QIH
DownloadVisualize
BU of 6qih by Molmil
Pancreatic Bovine Trypsin with a boronic acid inhibitor
分子名称: CALCIUM ION, Cationic trypsin, DI(HYDROXYETHYL)ETHER, ...
著者Santos-Silva, T, Correia, H.D.
登録日2019-01-18
公開日2020-02-05
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.42 Å)
主引用文献Pancreatic Bovine Trypsin with a boronic acid inhibitor
To Be Published

224004

件を2024-08-21に公開中

PDB statisticsPDBj update infoContact PDBjnumon