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8U1D
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BU of 8u1d by Molmil
Cryo-EM structure of vaccine-elicited CD4 binding site antibody DH1285 bound to HIV-1 CH505TFchim.6R.SOSIP.664v4.1 Env Local Refinement
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, DH1285 Heavy Chain, DH1285 Light Chain, ...
著者Thakur, B, Stalls, V.D, Acharya, P.
登録日2023-08-31
公開日2024-01-03
最終更新日2025-06-04
実験手法ELECTRON MICROSCOPY (4.25 Å)
主引用文献Vaccine induction of CD4-mimicking HIV-1 broadly neutralizing antibody precursors in macaques.
Cell, 187, 2024
6QV6
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BU of 6qv6 by Molmil
CryoEM structure of the human ClC-1 chloride channel, membrane domain
分子名称: Chloride channel protein 1
著者Wang, K.T, Gourdon, P.E, Zhou, Z.H.
登録日2019-03-01
公開日2019-05-08
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (3.63 Å)
主引用文献Structure of the human ClC-1 chloride channel.
Plos Biol., 17, 2019
6QVB
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BU of 6qvb by Molmil
CryoEM structure of the human ClC-1 chloride channel, CBS state 3
分子名称: Chloride channel protein 1
著者Wang, K.T, Gourdon, P.E, Zhou, Z.H.
登録日2019-03-01
公開日2019-05-08
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (4.34 Å)
主引用文献Structure of the human ClC-1 chloride channel.
Plos Biol., 17, 2019
8YVR
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BU of 8yvr by Molmil
Crystal structure of GH65 alpha-1,2-glucosidase from Flavobacterium johnsoniae in complex with 1-deoxynojirimycin
分子名称: 1,2-ETHANEDIOL, 1-DEOXYNOJIRIMYCIN, Candidate alpha glycoside phosphorylase Glycoside hydrolase family 65
著者Nakamura, S, Miyazaki, T.
登録日2024-03-29
公開日2025-03-19
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structural insights into the inhibition mechanism of glucosidase inhibitors toward kojibiose hydrolase belonging to glycoside hydrolase family 65.
Biosci.Biotechnol.Biochem., 89, 2024
7RI1
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BU of 7ri1 by Molmil
Crystal structure of anti-HIV llama VHH antibody J3 in complex with HIV-1 C1086 gp120
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Glycoprotein 120, Lamma VHH antibody J3, ...
著者Zhou, T, Kwong, P.D.
登録日2021-07-19
公開日2022-03-30
最終更新日2024-10-30
実験手法X-RAY DIFFRACTION (2.55 Å)
主引用文献Structural basis for llama nanobody recognition and neutralization of HIV-1 at the CD4-binding site.
Structure, 30, 2022
6QVU
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BU of 6qvu by Molmil
CryoEM structure of the human ClC-1 chloride channel, low pH
分子名称: Chloride channel protein 1
著者Wang, K.T, Gourdon, P.E, Zhou, Z.H.
登録日2019-03-05
公開日2019-05-08
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (4.2 Å)
主引用文献Structure of the human ClC-1 chloride channel.
Plos Biol., 17, 2019
8D3Z
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BU of 8d3z by Molmil
Crystal structure of GalS1 in complex with Manganese from Populus trichocarpas
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Galactan synthase, ...
著者Pereira, J.H, Prabhakar, P.K, Urbanowicz, B.R, Adams, P.D.
登録日2022-06-01
公開日2023-03-15
最終更新日2024-10-30
実験手法X-RAY DIFFRACTION (2.56 Å)
主引用文献Structural and biochemical insight into a modular beta-1,4-galactan synthase in plants.
Nat.Plants, 9, 2023
8HRV
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BU of 8hrv by Molmil
dutpase of helicobacter pylori 26695
分子名称: 1,2-ETHANEDIOL, 2'-DEOXYURIDINE 5'-ALPHA,BETA-IMIDO-TRIPHOSPHATE, Deoxyuridine 5'-triphosphate nucleotidohydrolase, ...
著者Kumari, K, Gourinath, S.
登録日2022-12-16
公開日2024-01-17
最終更新日2025-03-26
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural analysis of dUTPase from Helicobacter pylori reveals unusual activity for dATP.
Int.J.Biol.Macromol., 282, 2024
8SAL
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BU of 8sal by Molmil
CryoEM structure of VRC01-CH848.0358.80
分子名称: CH0848.3.D0358.80.06CHIM.DS.6R.SOSIP gp120, CH0848.3.D0358.80.06CHIM.DS.6R.SOSIP gp41, VCR01 variable heavy chain, ...
著者Henderson, R, Zhou, Y, Stalls, V, Bartesaghi, B, Acharya, P.
登録日2023-04-01
公開日2023-04-19
最終更新日2025-05-21
実験手法ELECTRON MICROSCOPY (4.9 Å)
主引用文献Structural basis for breadth development in the HIV-1 V3-glycan targeting DH270 antibody clonal lineage.
Nat Commun, 14, 2023
8SAT
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BU of 8sat by Molmil
CryoEM structure of VRC01-CH848.10.17
分子名称: CH848.10.17 gp120, CH848.10.17 gp41, VRC01-variable heavy chain, ...
著者Henderson, R, Zhou, Y, Stalls, V, Bartesaghi, B, Acharya, P.
登録日2023-04-02
公開日2023-04-19
最終更新日2025-05-28
実験手法ELECTRON MICROSCOPY (4.5 Å)
主引用文献Structural basis for breadth development in the HIV-1 V3-glycan targeting DH270 antibody clonal lineage.
Nat Commun, 14, 2023
8UA2
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BU of 8ua2 by Molmil
Crystal Structure of infected cell protein 0 (ICP0) from herpes simplex virus 1 (proteolyzed fragment)
分子名称: IODIDE ION, RL2
著者Lovell, S, Kashipathy, M, Battaile, K.P, Cooper, A, Davido, D.
登録日2023-09-20
公開日2024-02-28
最終更新日2024-06-19
実験手法X-RAY DIFFRACTION (2.65 Å)
主引用文献HSV-1 ICP0 dimer domain adopts a novel beta-barrel fold.
Proteins, 92, 2024
8DJ1
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BU of 8dj1 by Molmil
Crystal structure of NavAb V126T as a basis for the human Nav1.7 Inherited Erythromelalgia S241T mutation
分子名称: 1,2-DIMYRISTOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 3-[(3-CHOLAMIDOPROPYL)DIMETHYLAMMONIO]-1-PROPANESULFONATE, Ion transport protein
著者Wisedchaisri, G, Gamal El-Din, T.M, Zheng, N, Catterall, W.A.
登録日2022-06-29
公開日2023-04-12
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Structural basis for severe pain caused by mutations in the S4-S5 linkers of voltage-gated sodium channel Na V 1.7.
Proc.Natl.Acad.Sci.USA, 120, 2023
8TY6
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BU of 8ty6 by Molmil
Disulfide-stabilized HIV-1 CA hexamer in complex with PQBP1 Nt
分子名称: Capsid protein p24
著者Piacentini, J, Pornillos, O, Ganser-Pornillos, B.K.
登録日2023-08-24
公開日2024-03-06
最終更新日2024-11-06
実験手法ELECTRON MICROSCOPY (3.3 Å)
主引用文献Molecular Determinants of PQBP1 Binding to the HIV-1 Capsid Lattice.
J.Mol.Biol., 436, 2024
6GPK
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BU of 6gpk by Molmil
Crystal structure of human GDP-D-mannose 4,6-dehydratase (E157Q) in complex with GDP-Man
分子名称: 1,2-ETHANEDIOL, GDP-mannose 4,6 dehydratase, GLYCEROL, ...
著者Pfeiffer, M, Krojer, T, Johansson, C, von Delft, F, Bountra, C, Arrowsmith, C.H, Edwards, A, Nidetzky, B, Oppermann, U, Structural Genomics Consortium (SGC)
登録日2018-06-06
公開日2018-07-18
最終更新日2024-05-15
実験手法X-RAY DIFFRACTION (1.47 Å)
主引用文献A Parsimonious Mechanism of Sugar Dehydration by Human GDP-Mannose-4,6-dehydratase.
Acs Catalysis, 9, 2019
6QVC
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BU of 6qvc by Molmil
CryoEM structure of the human ClC-1 chloride channel, CBS state 1
分子名称: Chloride channel protein 1
著者Wang, K.T, Gourdon, P.E, Zhou, Z.H.
登録日2019-03-01
公開日2019-05-08
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (4 Å)
主引用文献Structure of the human ClC-1 chloride channel.
Plos Biol., 17, 2019
8SKN
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BU of 8skn by Molmil
Crystal structure of compound 3-bound human Dynamin-1-like protein GTPase-BSE fusion
分子名称: 1,2-ETHANEDIOL, Dynamin-1-like protein GTPase-BSE fusion, N-[4-(azetidin-1-yl)-2-(4-methylphenyl)quinolin-6-yl]-2-methylpropanamide
著者Ma, B.
登録日2023-04-20
公開日2023-08-30
実験手法X-RAY DIFFRACTION (2.41 Å)
主引用文献Discovery of Potent Allosteric DRP1 Inhibitors by Disrupting Protein-Protein Interaction with MiD49.
Acs Med.Chem.Lett., 14, 2023
6YB4
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BU of 6yb4 by Molmil
Crystal structure of human ATAD2 bromodomain in complex with N-(4-bromo-3-(3-methylpyrrolidin-1-yl)sulfonyl)phenyl)-2-(-4-cyclopropyl-4-methyl-2,5-dioxoimidazolidin-1-yl)acetamide
分子名称: 1,2-ETHANEDIOL, ATPase family AAA domain-containing protein 2, SULFATE ION, ...
著者Chung, C.
登録日2020-03-15
公開日2020-05-06
最終更新日2024-05-15
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Optimization of Potent ATAD2 and CECR2 Bromodomain Inhibitors with an Atypical Binding Mode.
J.Med.Chem., 63, 2020
8ZD8
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BU of 8zd8 by Molmil
NMR structure of the (CGG-dsDNA:ND=) 1:1 complex
分子名称: DNA (5'-D(*CP*AP*TP*TP*CP*GP*GP*TP*TP*AP*G)-3'), DNA (5'-D(*CP*TP*AP*AP*CP*GP*GP*AP*AP*TP*G)-3'), ~{N}-(7-methyl-1,8-naphthyridin-2-yl)-3-[[3-[(7-methyl-1,8-naphthyridin-2-yl)amino]-3-oxidanylidene-propyl]amino]propanamide
著者Sakurabayashi, S, Furuita, K, Yamada, T, Nomura, M, Nakatani, K, Kojima, C.
登録日2024-05-01
公開日2025-04-30
実験手法SOLUTION NMR
主引用文献NMR structure of the (CGG-dsDNA:ND=) 1:1 complex
To Be Published
7R97
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BU of 7r97 by Molmil
Crystal structure of postcleavge complex of Escherichia coli RNase III
分子名称: 1,2-ETHANEDIOL, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CHLORIDE ION, ...
著者Dharavath, S, Shaw, G.X, Ji, X.
登録日2021-06-28
公開日2022-07-20
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.804 Å)
主引用文献Structural basis for Dicer-like function of an engineered RNase III variant and insights into the reaction trajectory of two-Mg 2+ -ion catalysis.
Rna Biol., 19, 2022
6HY3
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BU of 6hy3 by Molmil
Three-dimensional structure of AgaC from Zobellia galactanivorans
分子名称: 1,2-ETHANEDIOL, Beta-agarase C, GLYCEROL, ...
著者Naretto, A, Fanuel, M, Ropartz, D, Rogniaux, H, Larocque, R, Czjzek, M, Tellier, C, Michel, G.
登録日2018-10-19
公開日2019-03-13
最終更新日2024-11-06
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献The agar-specific hydrolaseZgAgaC from the marine bacteriumZobellia galactanivoransdefines a new GH16 protein subfamily.
J.Biol.Chem., 294, 2019
5XXD
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BU of 5xxd by Molmil
Crystal structure of SmyD3 in complex with covalent inhibitor 1
分子名称: S-ADENOSYLMETHIONINE, Smyd3 methyltransferase, ZINC ION, ...
著者Baburajendran, N, Anna E, J.
登録日2017-07-03
公開日2018-08-29
最終更新日2024-11-13
実験手法X-RAY DIFFRACTION (2.314 Å)
主引用文献Crystal structure of SmyD3 in complex with covalent inhibitor 1
To Be Published
7RJ2
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BU of 7rj2 by Molmil
Co-crystal structure of lenacapavir bound to Q67H/N74D mutant of disulfide stabilized HIV-1 CA hexamer
分子名称: CHLORIDE ION, Capsid protein p24, IODIDE ION, ...
著者Bester, S.M, Kvaratskhelia, M.
登録日2021-07-20
公開日2022-07-27
最終更新日2024-12-25
実験手法X-RAY DIFFRACTION (2.32 Å)
主引用文献Structural and Mechanistic Bases of Viral Resistance to HIV-1 Capsid Inhibitor Lenacapavir.
Mbio, 13, 2022
7RHM
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BU of 7rhm by Molmil
Structure of Q67H/N74D mutant of disulfide stabilized HIV-1 CA hexamer
分子名称: CAPSID PROTEIN P24, CHLORIDE ION, IODIDE ION
著者Bester, S.M, Kvaratskhelia, M.
登録日2021-07-17
公開日2022-07-27
最終更新日2024-10-23
実験手法X-RAY DIFFRACTION (2.16 Å)
主引用文献Structural and Mechanistic Bases of Viral Resistance to HIV-1 Capsid Inhibitor Lenacapavir.
Mbio, 13, 2022
6ZK6
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BU of 6zk6 by Molmil
Protein Phosphatase 1 (PP1) T320E mutant
分子名称: FE (III) ION, MANGANESE (II) ION, PHOSPHATE ION, ...
著者Salvi, F, Barabas, O, Koehn, M.
登録日2020-06-29
公開日2020-11-18
最終更新日2024-11-06
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Towards Dissecting the Mechanism of Protein Phosphatase-1 Inhibition by Its C-Terminal Phosphorylation.
Chembiochem, 22, 2021
6Z4V
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BU of 6z4v by Molmil
Crystal structure of the neurotensin receptor 1 (NTSR1-H4bmx) in complex with NTS8-13
分子名称: ARG-PRO-TYR-ILE-LEU, Neurotensin receptor type 1,Neurotensin receptor type 1,DARPin
著者Deluigi, M, Klipp, A, Hilge, M, Merklinger, L, Klenk, C, Plueckthun, A.
登録日2020-05-25
公開日2021-02-10
最終更新日2024-11-13
実験手法X-RAY DIFFRACTION (2.595 Å)
主引用文献Complexes of the neurotensin receptor 1 with small-molecule ligands reveal structural determinants of full, partial, and inverse agonism.
Sci Adv, 7, 2021

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