8SKN
Crystal structure of compound 3-bound human Dynamin-1-like protein GTPase-BSE fusion
Summary for 8SKN
Entry DOI | 10.2210/pdb8skn/pdb |
Descriptor | Dynamin-1-like protein GTPase-BSE fusion, N-[4-(azetidin-1-yl)-2-(4-methylphenyl)quinolin-6-yl]-2-methylpropanamide, 1,2-ETHANEDIOL, ... (4 entities in total) |
Functional Keywords | inhibitor, hydrolase-inhibitor complex, hydrolase/inhibitor |
Biological source | Homo sapiens (human) More |
Total number of polymer chains | 2 |
Total formula weight | 86161.53 |
Authors | |
Primary citation | Furuya, T.,Lin, J.,Afanaseva, A.,Molz, L.,Lagu, B.,Ma, B. Discovery of Potent Allosteric DRP1 Inhibitors by Disrupting Protein-Protein Interaction with MiD49. Acs Med.Chem.Lett., 14:1095-1099, 2023 Cited by PubMed: 37583827DOI: 10.1021/acsmedchemlett.3c00223 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.41 Å) |
Structure validation
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