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8YTR
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The structure of Cu(II)-CopC from Thioalkalivibrio paradoxus
分子名称: COPPER (II) ION, CopC domain-containing protein, DI(HYDROXYETHYL)ETHER
著者Kulikova, O.G, Solovieva, A.Y, Varfolomeeva, L.A, Dergousova, N.I, Nikolaeva, A.Y, Boyko, K.M, Tikhonova, T.V, Popov, V.O.
登録日2024-03-26
公開日2024-04-24
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献The structure of Cu(II)-CopC from Thioalkalivibrio paradoxus
To Be Published
8YTQ
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BU of 8ytq by Molmil
The structure of apoCopC from Thioalkalivibrio paradoxus
分子名称: ACETATE ION, COPPER (II) ION, CopC domain-containing protein, ...
著者Kulikova, O.G, Solovieva, A.Y, Varfolomeeva, L.A, Dergousova, N.I, Boyko, K.M, Tikhonova, T.V, Popov, V.O.
登録日2024-03-26
公開日2024-04-24
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献The structure of apoCopC from Thioalkalivibrio paradoxus
To Be Published
8YTP
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Single-chain Fv antibody of E11 complex with NP-glycine under reducing conditions
分子名称: 2-[2-(3-nitro-4-oxidanyl-phenyl)ethanoylamino]ethanoic acid, Single-chain Fv antibody of E11
著者Yoshida, M, Hanazono, Y, Numoto, N, Ito, N, Oda, M.
登録日2024-03-26
公開日2024-07-03
最終更新日2024-07-10
実験手法X-RAY DIFFRACTION (1.36 Å)
主引用文献Affinity-matured antibody with a disulfide bond in H-CDR3 loop.
Arch.Biochem.Biophys., 758, 2024
8YTO
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BU of 8yto by Molmil
Single-chain Fv antibody of E11 complex with NP-glycine
分子名称: 2-[2-(3-nitro-4-oxidanyl-phenyl)ethanoylamino]ethanoic acid, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, GLYCEROL, ...
著者Yoshida, M, Hanazono, Y, Numoto, N, Ito, N, Oda, M.
登録日2024-03-26
公開日2024-07-03
最終更新日2024-07-10
実験手法X-RAY DIFFRACTION (1.04 Å)
主引用文献Affinity-matured antibody with a disulfide bond in H-CDR3 loop.
Arch.Biochem.Biophys., 758, 2024
8YTN
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BU of 8ytn by Molmil
Single-chain Fv antibody of E11
分子名称: GLYCEROL, Single-chain Fv antibody of E11
著者Yoshida, M, Hanazono, Y, Numoto, N, Ito, N, Oda, M.
登録日2024-03-26
公開日2024-07-03
最終更新日2024-07-10
実験手法X-RAY DIFFRACTION (1.72 Å)
主引用文献Affinity-matured antibody with a disulfide bond in H-CDR3 loop.
Arch.Biochem.Biophys., 758, 2024
8YTI
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BU of 8yti by Molmil
Crystal Structure of Nucleosome-H1x Linker Histone Assembly (sticky-169a DNA fragment)
分子名称: CALCIUM ION, CHLORIDE ION, DNA (169-MER), ...
著者Adhireksan, Z, Qiuye, B, Padavattan, S, Davey, C.A.
登録日2024-03-26
公開日2024-04-03
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Linker Histones Associate Heterogeneously with Nucleosomes in the Condensed State
To Be Published
8YTE
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BU of 8yte by Molmil
Crystal Structure of TrkA D5 domain in complex with macrocyclic peptide
分子名称: 1,2-ETHANEDIOL, AMINOMETHYLAMIDE, High affinity nerve growth factor receptor, ...
著者Yamada, T, Mihara, K, Ueda, T, Yamauchi, D, Shimizu, M, Ando, A, Mayumi, K, Nakata, Z, Mikamiyama, H.
登録日2024-03-25
公開日2024-07-10
最終更新日2024-07-24
実験手法X-RAY DIFFRACTION (2.26 Å)
主引用文献Discovery and Hit to Lead Optimization of Macrocyclic Peptides as Novel Tropomyosin Receptor Kinase A Antagonists.
J.Med.Chem., 67, 2024
8YTD
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Crystal Structure of TrkA D5 domain in complex with two different macrocyclic peptides
分子名称: 1,2-ETHANEDIOL, High affinity nerve growth factor receptor, Macrocyclic Peptide
著者Yamada, T, Mihara, K, Ueda, T, Yamauchi, D, Shimizu, M, Ando, A, Mayumi, K, Nakata, Z, Mikamiyama, H.
登録日2024-03-25
公開日2024-07-10
最終更新日2024-07-24
実験手法X-RAY DIFFRACTION (2.34 Å)
主引用文献Discovery and Hit to Lead Optimization of Macrocyclic Peptides as Novel Tropomyosin Receptor Kinase A Antagonists.
J.Med.Chem., 67, 2024
8YT5
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BU of 8yt5 by Molmil
SP1746 treated with EDTA, in complex with ADP
分子名称: ADENOSINE-5'-DIPHOSPHATE, FE (III) ION, bis(5'-nucleosyl)-tetraphosphatase (symmetrical)
著者Jin, Y, Niu, L, Ke, J.
登録日2024-03-25
公開日2024-05-08
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structural and biochemical characterization of a nucleotide hydrolase from Streptococcus pneumonia.
Structure, 2024
8YT4
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Structure of Aquifex aeolicus Lumazine Synthase by Cryo-Electron Microscopy to 1.42 Angstrom Resolution
分子名称: 6,7-dimethyl-8-ribityllumazine synthase, PHOSPHATE ION
著者Savva, C.G, Sobhy, M.A, De Biasio, A, Hamdan, S.M.
登録日2024-03-24
公開日2024-04-10
最終更新日2024-07-24
実験手法ELECTRON MICROSCOPY (1.42 Å)
主引用文献Structure of Aquifex aeolicus lumazine synthase by cryo-electron microscopy to 1.42 angstrom resolution.
Iucrj, 2024
8YSX
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canine immunoproteasome 20S subunit in complex with compound 2
分子名称: Proteasome subunit alpha type, Proteasome subunit beta, Proteasome subunit beta type-8, ...
著者Kashima, A, Arai, Y.
登録日2024-03-24
公開日2024-07-31
実験手法ELECTRON MICROSCOPY (2.2 Å)
主引用文献Optimization of alpha-amido boronic acids via cryo-electron microscopy analysis: Discovery of a novel highly selective immunoproteasome subunit LMP7 ( beta 5i)/LMP2 ( beta 1i) dual inhibitor.
Bioorg.Med.Chem., 109, 2024
8YSA
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BU of 8ysa by Molmil
The co-crystal structure of SARS-CoV-2 Mpro in complex with compound H102
分子名称: 3C-like proteinase nsp5, BOC-TBG-PHE-ELL
著者Zheng, W.Y, Fu, L.F, Feng, Y, Han, P, Qi, J.X.
登録日2024-03-22
公開日2024-05-08
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Discovery, Biological Activity, and Structural Mechanism of a Potent Inhibitor of SARS-CoV-2 Main Protease
To Be Published
8YRV
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BU of 8yrv by Molmil
Crystal structure of D-amino acid transaminase from Haliscomenobacter hydrossis complexed with 3-aminooxypropionic acid
分子名称: 3-[(~{E})-[2-methyl-3-oxidanyl-5-(phosphonooxymethyl)pyridin-4-yl]methylideneamino]oxypropanoic acid, Aminotransferase class IV, MAGNESIUM ION
著者Matyuta, I.O, Bakunova, A.K, Nikolaeva, A.Y, Popov, V.O, Boyko, K.M.
登録日2024-03-21
公開日2024-04-17
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Crystal structure of D-amino acid transaminase from Haliscomenobacter hydrossis complexed with 3-aminooxypropionic acid
To Be Published
8YRU
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BU of 8yru by Molmil
Crystal structure of D-amino acid transaminase from Haliscomenobacter hydrossis (apo form) after 15 sec of soaking with phenylhydrazine
分子名称: ACETATE ION, Aminotransferase class IV, [6-methyl-5-oxidanyl-4-[(2-phenylhydrazinyl)methyl]pyridin-3-yl]methyl dihydrogen phosphate
著者Matyuta, I.O, Bakunova, A.K, Minyaev, M.E, Popov, V.O, Boyko, K.M.
登録日2024-03-21
公開日2024-04-17
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal structure of D-amino acid transaminase from Haliscomenobacter hydrossis (apo form) after 15 sec of soaking with phenylhydrazine
To Be Published
8YRT
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BU of 8yrt by Molmil
Crystal structure of D-amino acid transaminase from Haliscomenobacter hydrossis in the holo form obtained at pH 7.0
分子名称: Aminotransferase class IV, PYRIDOXAL-5'-PHOSPHATE
著者Matyuta, I.O, Bakunova, A.K, Minyaev, M.E, Popov, V.O, Boyko, K.M.
登録日2024-03-21
公開日2024-04-17
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal structure of D-amino acid transaminase from Haliscomenobacter hydrossis in the holo form obtained at pH 7.0
To Be Published
8YRP
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BU of 8yrp by Molmil
SARS-CoV-2 Delta Spike in complex with JM-1A
分子名称: JM-1A Heavy Chain, JM-1A Light Chain, Spike glycoprotein
著者Nguyen, V.H.T, Chen, X.
登録日2024-03-21
公開日2024-06-05
最終更新日2024-06-26
実験手法ELECTRON MICROSCOPY (3.64 Å)
主引用文献The presence of broadly neutralizing anti-SARS-CoV-2 RBD antibodies elicited by primary series and booster dose of COVID-19 vaccine.
Plos Pathog., 20, 2024
8YRO
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BU of 8yro by Molmil
SARS-CoV-2 Delta Spike in complex with JL-8C
分子名称: JL-8C Heavy Chain, JL-8C Light Chain, Spike glycoprotein
著者Nguyen, V.H.T, Chen, X.
登録日2024-03-21
公開日2024-06-05
最終更新日2024-06-26
実験手法ELECTRON MICROSCOPY (3.27 Å)
主引用文献The presence of broadly neutralizing anti-SARS-CoV-2 RBD antibodies elicited by primary series and booster dose of COVID-19 vaccine.
Plos Pathog., 20, 2024
8YRJ
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BU of 8yrj by Molmil
Mouse Fc epsilon RI
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, High affinity immunoglobulin epsilon receptor subunit alpha, High affinity immunoglobulin epsilon receptor subunit beta, ...
著者Zhang, Z, Yui, M, Ohto, U, Shimizu, T.
登録日2024-03-21
公開日2024-07-17
実験手法ELECTRON MICROSCOPY (3.87 Å)
主引用文献Mouse Fc epsilon RI
To Be Published
8YRH
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BU of 8yrh by Molmil
Complex of SARS-CoV-2 main protease and Rosmarinic acid
分子名称: (2R)-3-(3,4-dihydroxyphenyl)-2-{[(2E)-3-(3,4-dihydroxyphenyl)prop-2-enoyl]oxy}propanoic acid, 3C-like proteinase nsp5
著者Wang, Q.S, Li, Q.H.
登録日2024-03-21
公開日2024-07-03
実験手法X-RAY DIFFRACTION (1.841 Å)
主引用文献Structural basis of rosmarinic acid inhibitory mechanism on SARS-CoV-2 main protease.
Biochem.Biophys.Res.Commun., 724, 2024
8YRG
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BU of 8yrg by Molmil
CryoEM structure of fospropofol-bound MRGPRX4-Gq complex
分子名称: Gs-mini-Gq chimera, Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1, ...
著者Cao, C, Fay, J.F, Roth, B.L.
登録日2024-03-21
公開日2024-05-22
実験手法ELECTRON MICROSCOPY (3.14 Å)
主引用文献MRGPRX4 mediates phospho-drug-associated pruritus in a humanized mouse model.
Sci Transl Med, 16, 2024
8YRF
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BU of 8yrf by Molmil
Crystal structure of LmrR with V15 replaced by unnatural amino acid 4-amino-L-phenyl-cysteine
分子名称: 1,2-ETHANEDIOL, Transcriptional regulator, PadR-like family
著者Zhou, Z, Huang, W.
登録日2024-03-21
公開日2024-04-24
実験手法X-RAY DIFFRACTION (2.66 Å)
主引用文献Crystal structure of LmrR with V15 replaced by unnatural amino acid 4-amino-L-phenyl-cysteine
To Be Published
8YRC
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Chlorinated YabJ from Staphylococcus aureus
分子名称: CHLORIDE ION, OXYGEN ATOM, SODIUM ION, ...
著者Jeong, C, Kim, H.J.
登録日2024-03-21
公開日2024-04-24
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献YabJ from Staphylococcus aureus entraps chlorides within its pocket.
Biochem.Biophys.Res.Commun., 710, 2024
8YR7
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BU of 8yr7 by Molmil
Crystal structure of human dishevelled 2 (Dvl2) PDZ domain fused with WGEF internal peptide motif
分子名称: Segment polarity protein dishevelled homolog DVL-2,Rho guanine nucleotide exchange factor 19
著者Omble, A, Mahajan, S, Kulkarni, K.A.
登録日2024-03-20
公開日2024-05-29
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Dishevelled2 activates WGEF via its interaction with a unique internal peptide motif of the GEF.
Commun Biol, 7, 2024
8YR4
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BU of 8yr4 by Molmil
Cryo-EM structure of the human ABCB6 in complex with Cd(II):Phytochelatin 2
分子名称: ATP-binding cassette sub-family B member 6, CADMIUM ION, GAMMA-D-GLUTAMIC ACID, ...
著者Choi, S.H, Lee, S.S, Lee, H.Y, Kim, S, Kim, J.W, Jin, M.S.
登録日2024-03-20
公開日2024-06-19
実験手法ELECTRON MICROSCOPY (3.1 Å)
主引用文献Cryo-EM structure of cadmium-bound human ABCB6.
Commun Biol, 7, 2024
8YR3
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Cryo-EM structure of the human ABCB6 in complex with Cd(II):GSH
分子名称: ATP-binding cassette sub-family B member 6, CADMIUM ION, GLUTATHIONE
著者Choi, S.H, Lee, S.S, Lee, H.Y, Kim, S, Kim, J.W, Jin, M.S.
登録日2024-03-20
公開日2024-06-19
実験手法ELECTRON MICROSCOPY (3.2 Å)
主引用文献Cryo-EM structure of cadmium-bound human ABCB6.
Commun Biol, 7, 2024

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件を2024-08-14に公開中

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