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7TNN
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Complex GGNN of AMPA-subtype iGluR GluA2 in complex with auxiliary subunit gamma2 (Stargazin) at low glutamate concentration (20 uM) in the presence of cyclothiazide (100 uM)
分子名称: CYCLOTHIAZIDE, GLUTAMIC ACID, Isoform Flip of Glutamate receptor 2,Voltage-dependent calcium channel gamma-3 subunit chimera
著者Yelshanskaya, M.V, Sobolevsky, A.I.
登録日2022-01-21
公開日2022-04-20
最終更新日2022-05-18
実験手法ELECTRON MICROSCOPY (3.91 Å)
主引用文献Opening of glutamate receptor channel to subconductance levels.
Nature, 605, 2022
7TNL
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Complex GNGN1 of AMPA-subtype iGluR GluA2 in complex with auxiliary subunit gamma2 (Stargazin) at low glutamate concentration (20 uM) in the presence of cyclothiazide (100 uM)
分子名称: CYCLOTHIAZIDE, GLUTAMIC ACID, Isoform Flip of Glutamate receptor 2,Voltage-dependent calcium channel gamma-3 subunit chimera
著者Yelshanskaya, M.V, Sobolevsky, A.I.
登録日2022-01-21
公開日2022-04-20
最終更新日2022-05-18
実験手法ELECTRON MICROSCOPY (3.59 Å)
主引用文献Opening of glutamate receptor channel to subconductance levels.
Nature, 605, 2022
7TNJ
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Complex NNNN of AMPA-subtype iGluR GluA2 in complex with auxiliary subunit gamma2 (Stargazin) at low glutamate concentration (20 uM) in the presence of cyclothiazide (100 uM)
分子名称: CYCLOTHIAZIDE, Isoform Flip of Glutamate receptor 2,Voltage-dependent calcium channel gamma-3 subunit chimera
著者Yelshanskaya, M.V, Sobolevsky, A.I.
登録日2022-01-21
公開日2022-04-20
最終更新日2022-05-18
実験手法ELECTRON MICROSCOPY (4.02 Å)
主引用文献Opening of glutamate receptor channel to subconductance levels.
Nature, 605, 2022
7TNP
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Complex GGGG of AMPA-subtype iGluR GluA2 in complex with auxiliary subunit gamma2 (Stargazin) at low glutamate concentration (20 uM) in the presence of cyclothiazide (100 uM)
分子名称: CYCLOTHIAZIDE, GLUTAMIC ACID, Isoform Flip of Glutamate receptor 2,Voltage-dependent calcium channel gamma-3 subunit chimera
著者Yelshanskaya, M.V, Sobolevsky, A.I.
登録日2022-01-21
公開日2022-04-20
最終更新日2022-05-18
実験手法ELECTRON MICROSCOPY (3.96 Å)
主引用文献Opening of glutamate receptor channel to subconductance levels.
Nature, 605, 2022
5CJ7
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Human DNA polymerase lambda L431A mutant- MgdTTP binary and complex with 6 paired DNA
分子名称: DNA (5'-D(*CP*AP*GP*TP*AP*C)-3'), DNA (5'-D(P*GP*TP*AP*CP*TP*G)-3'), DNA polymerase lambda, ...
著者Liu, M.S, Tsai, M.D.
登録日2015-07-14
公開日2016-02-24
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.901 Å)
主引用文献Structural Mechanism for the Fidelity Modulation of DNA Polymerase lambda
J.Am.Chem.Soc., 138, 2016
3CSG
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BU of 3csg by Molmil
Crystal Structure of Monobody YS1(MBP-74)/Maltose Binding Protein Fusion Complex
分子名称: Maltose-binding protein Monobody YS1 Fusion
著者Gilbreth, R.N, Koide, S.
登録日2008-04-09
公開日2008-07-22
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.798 Å)
主引用文献A Dominant Conformational Role for Amino Acid Diversity in Minimalist Protein-Protein Interfaces
J.Mol.Biol., 381, 2008
1E3W
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BU of 1e3w by Molmil
Rat brain 3-hydroxyacyl-CoA dehydrogenase binary complex with NADH and 3-keto butyrate
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, ACETOACETIC ACID, NICOTINAMIDE-ADENINE-DINUCLEOTIDE, ...
著者Powell, A.J, Read, J.A, Brady, R.L.
登録日2000-06-26
公開日2001-05-25
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Recognition of Structurally Diverse Substrates by Type II 3-Hydroxyacyl-Coa Dehydrogenase (Hadh II) Amyloid-Beta Binding Alcohol Dehydrogenase (Abad)
J.Mol.Biol., 303, 2000
1E3S
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Rat brain 3-hydroxyacyl-CoA dehydrogenase binary complex with NADH
分子名称: NICOTINAMIDE-ADENINE-DINUCLEOTIDE, SHORT CHAIN 3-HYDROXYACYL-COA DEHYDROGENASE
著者Powell, A.J, Read, J.A, Banfield, M.J, Brady, R.L.
登録日2000-06-22
公開日2001-05-25
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Recognition of Structurally Diverse Substrates by Type II 3-Hydroxyacyl-Coa Dehydrogenase (Hadh II) Amyloid-Beta Binding Alcohol Dehydrogenase (Abad)
J.Mol.Biol., 303, 2000
1QZY
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BU of 1qzy by Molmil
Human Methionine Aminopeptidase in complex with bengamide inhibitor LAF153 and cobalt
分子名称: (E)-(2R,3R,4S,5R)-3,4,5-TRIHYDROXY-2-METHOXY-8,8-DIMETHYL-NON-6-ENOIC ACID ((3S,6R)-6-HYDROXY-2-OXO-AZEPAN-3-YL)-AMIDE, COBALT (II) ION, Methionine aminopeptidase 2, ...
著者Eck, M.J, Song, H.K, Morollo, A.
登録日2003-09-18
公開日2003-11-25
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Proteomics-based target identification: bengamides as a new class of methionine aminopeptidase inhibitors.
J.Biol.Chem., 278, 2003
3D1K
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BU of 3d1k by Molmil
R/T intermediate quaternary structure of an antarctic fish hemoglobin in an alpha(CO)-beta(pentacoordinate) state
分子名称: ACETYL GROUP, CARBON MONOXIDE, Hemoglobin subunit alpha-1, ...
著者Vitagliano, L, Vergara, A, Bonomi, G, Merlino, A, Mazzarella, L.
登録日2008-05-06
公開日2008-08-05
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.25 Å)
主引用文献Spectroscopic and crystallographic characterization of a tetrameric hemoglobin oxidation reveals structural features of the functional intermediate relaxed/tense state.
J.Am.Chem.Soc., 130, 2008
8CTA
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BU of 8cta by Molmil
Minimal 2:2 Ternary Complex between BI-224436 bound HIV-1 Integrase Catalytic Core Domain Dimer and Carboxy Terminal Domains
分子名称: (2S)-tert-butoxy[4-(2,3-dihydropyrano[4,3,2-de]quinolin-7-yl)-2-methylquinolin-3-yl]acetic acid, 1,2-ETHANEDIOL, Integrase
著者Gupta, K, Van Duyne, G.D, Eilers, G, Bushman, F.D.
登録日2022-05-13
公開日2023-02-22
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.93 Å)
主引用文献Structure of a HIV-1 IN-Allosteric inhibitor complex at 2.93 angstrom resolution: Routes to inhibitor optimization.
Plos Pathog., 19, 2023
1QJZ
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BU of 1qjz by Molmil
Three Dimensional Structure of Physalis Mottle Virus : Implications for the Viral Assembly
分子名称: COAT PROTEIN
著者Krishna, S.S, Hiremath, C.N, Munshi, S.K, Prahadeeswaran, D, Sastri, M, Savithri, H.S, Murthy, M.R.N.
登録日1999-07-07
公開日1999-07-08
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (3.8 Å)
主引用文献Three Dimensional Structure of Physalis Movirus: Implications for the Viral Assembly
J.Mol.Biol., 289, 1999
1CSH
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BU of 1csh by Molmil
A very short hydrogen bond provides only moderate stabilization of an enzyme: inhibitor complex of citrate synthase
分子名称: AMIDOCARBOXYMETHYLDETHIA COENZYME *A, CITRATE SYNTHASE, OXALOACETATE ION
著者Usher, K.C, Remington, S.J.
登録日1994-03-07
公開日1994-04-30
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献A very short hydrogen bond provides only moderate stabilization of an enzyme-inhibitor complex of citrate synthase.
Biochemistry, 33, 1994
2SHK
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BU of 2shk by Molmil
THE THREE-DIMENSIONAL STRUCTURE OF SHIKIMATE KINASE FROM ERWINIA CHRYSANTHEMI COMPLEXED WITH ADP
分子名称: ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, SHIKIMATE KINASE
著者Krell, T, Coggins, J.R, Lapthorn, A.J.
登録日1997-10-27
公開日1998-11-18
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Crystallization and preliminary X-ray crystallographic analysis of shikimate kinase from Erwinia chrysanthemi.
Acta Crystallogr.,Sect.D, 53, 1997
1H4T
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BU of 1h4t by Molmil
Prolyl-tRNA synthetase from Thermus thermophilus complexed with L-proline
分子名称: PROLINE, PROLYL-TRNA SYNTHETASE, ZINC ION
著者Yaremchuk, A, Tukalo, M, Cusack, S.
登録日2001-05-14
公開日2001-06-18
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献A Succession of Substrate Induced Conformational Changes Ensures the Amino Acid Specificity of Thermus Thermophilus Prolyl-tRNA Synthetase: Comparison with Histidyl-tRNA Synthetase
J.Mol.Biol., 309, 2001
4C13
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BU of 4c13 by Molmil
x-ray crystal structure of Staphylococcus aureus MurE with UDP-MurNAc- Ala-Glu-Lys
分子名称: CHLORIDE ION, MAGNESIUM ION, PHOSPHATE ION, ...
著者Ruane, K.M, Roper, D.I, Fulop, V, Barreteau, H, Boniface, A, Dementin, S, Blanot, D, Mengin-Lecreulx, D, Gobec, S, Dessen, A, Dowson, C.G, Lloyd, A.J.
登録日2013-08-09
公開日2013-10-02
最終更新日2021-03-17
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Discovery of a first-in-class CDK2 selective degrader for AML differentiation therapy.
Nat.Chem.Biol., 2021
3CSB
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BU of 3csb by Molmil
Crystal Structure of Monobody YSX1/Maltose Binding Protein Fusion Complex
分子名称: 1,2-ETHANEDIOL, DI(HYDROXYETHYL)ETHER, MANGANESE (II) ION, ...
著者Gilbreth, R.N, Koide, S.
登録日2008-04-09
公開日2008-07-22
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.999 Å)
主引用文献A Dominant Conformational Role for Amino Acid Diversity in Minimalist Protein-Protein Interfaces
J.Mol.Biol., 381, 2008
1HC7
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BU of 1hc7 by Molmil
Prolyl-tRNA synthetase from Thermus thermophilus
分子名称: PROLYL-TRNA SYNTHETASE, ZINC ION
著者Yaremchuk, A, Tukalo, M, Cusack, S.
登録日2001-04-26
公開日2001-06-18
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.43 Å)
主引用文献A Succession of Substrate Induced Conformational Changes Ensures the Amino Acid Specificity of Thermus Thermophilus Prolyl-tRNA Synthetase: Comparison with Histidyl-tRNA Synthetase
J.Mol.Biol., 309, 2001
1JQN
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BU of 1jqn by Molmil
Crystal structure of E.coli phosphoenolpyruvate carboxylase in complex with Mn2+ and DCDP
分子名称: 3,3-DICHLORO-2-PHOSPHONOMETHYL-ACRYLIC ACID, ASPARTIC ACID, MANGANESE (II) ION, ...
著者Matsumura, H, Kai, Y.
登録日2001-08-07
公開日2003-01-14
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Crystal structures of C4 form maize and quaternary complex of E. coli phosphoenolpyruvate carboxylases.
Structure, 10, 2002
1H4S
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BU of 1h4s by Molmil
Prolyl-tRNA synthetase from Thermus thermophilus complexed with tRNApro(CGG) and a prolyl-adenylate analogue
分子名称: '5'-O-(N-(L-PROLYL)-SULFAMOYL)ADENOSINE, PROLYL-TRNA SYNTHETASE, SULFATE ION, ...
著者Yaremchuk, A, Tukalo, M, Cusack, S.
登録日2001-05-14
公開日2001-06-18
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.85 Å)
主引用文献A Succession of Substrate Induced Conformational Changes Ensures the Amino Acid Specificity of Thermus Thermophilus Prolyl-tRNA Synthetase: Comparison with Histidyl-tRNA Synthetase
J.Mol.Biol., 309, 2001
8DSO
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BU of 8dso by Molmil
Structure of cIAP1, BTK and BCCov
分子名称: (4S)-4-[2-(2-{4-[(2E)-4-{(3R)-3-[4-amino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}-4-oxobut-2-en-1-yl]piperazin-1-yl}ethoxy)acetamido]-1-{(2S)-2-cyclohexyl-2-[(N-methyl-L-alanyl)amino]acetyl}-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]-L-prolinamide bound form, Baculoviral IAP repeat-containing protein 2, Tyrosine-protein kinase BTK, ...
著者Schiemer, J.S, Calabrese, M.F.
登録日2022-07-22
公開日2023-03-08
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (2.334 Å)
主引用文献A covalent BTK ternary complex compatible with targeted protein degradation.
Nat Commun, 14, 2023
7U8P
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Structure of porcine kidney V-ATPase with SidK, Rotary State 1
分子名称: ADENOSINE-5'-DIPHOSPHATE, ATPase H(+)-transporting lysosomal accessory protein 2, ATPase H+ transporting accessory protein 1, ...
著者Tan, Y.Z, Keon, K.A.
登録日2022-03-09
公開日2022-07-06
最終更新日2024-02-14
実験手法ELECTRON MICROSCOPY (3.7 Å)
主引用文献CryoEM of endogenous mammalian V-ATPase interacting with the TLDc protein mEAK-7.
Life Sci Alliance, 5, 2022
7U8R
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BU of 7u8r by Molmil
Structure of porcine kidney V-ATPase with SidK, Rotary State 3
分子名称: ADENOSINE-5'-DIPHOSPHATE, ATPase H(+)-transporting lysosomal accessory protein 2, ATPase H+ transporting accessory protein 1, ...
著者Tan, Y.Z, Keon, K.A.
登録日2022-03-09
公開日2022-07-06
最終更新日2024-02-14
実験手法ELECTRON MICROSCOPY (3.8 Å)
主引用文献CryoEM of endogenous mammalian V-ATPase interacting with the TLDc protein mEAK-7.
Life Sci Alliance, 5, 2022
3DRC
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BU of 3drc by Molmil
INVESTIGATION OF THE FUNCTIONAL ROLE OF TRYPTOPHAN-22 IN ESCHERICHIA COLI DIHYDROFOLATE REDUCTASE BY SITE-DIRECTED MUTAGENESIS
分子名称: CALCIUM ION, CHLORIDE ION, DIHYDROFOLATE REDUCTASE, ...
著者Oatley, S.J, Kraut, J.
登録日1992-09-22
公開日1994-01-31
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Investigation of the functional role of tryptophan-22 in Escherichia coli dihydrofolate reductase by site-directed mutagenesis.
Biochemistry, 30, 1991
7U8Q
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Structure of porcine kidney V-ATPase with SidK, Rotary State 2
分子名称: ADENOSINE-5'-DIPHOSPHATE, ATPase H(+)-transporting lysosomal accessory protein 2, ATPase H+ transporting accessory protein 1, ...
著者Tan, Y.Z, Keon, K.A.
登録日2022-03-09
公開日2022-07-06
最終更新日2024-02-14
実験手法ELECTRON MICROSCOPY (4.1 Å)
主引用文献CryoEM of endogenous mammalian V-ATPase interacting with the TLDc protein mEAK-7.
Life Sci Alliance, 5, 2022

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