5BS0
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![BU of 5bs0 by Molmil](/molmil-images/mine/5bs0) | MAGE-A3 Reactive TCR in complex with Titin Epitope in HLA-A1 | 分子名称: | Beta-2-microglobulin, GLYCEROL, HLA class I histocompatibility antigen, ... | 著者 | Raman, M.C.C, Rizkallah, P.J, Simmons, R, Donellan, Z, Dukes, J, Bossi, G, LeProvost, G, Mahon, T, Hickman, E, Lomax, M, Oates, J, Hassan, N, Vuidepot, A, Sami, M, Cole, D.K, Jakobsen, B.K. | 登録日 | 2015-06-01 | 公開日 | 2016-03-02 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Direct molecular mimicry enables off-target cardiovascular toxicity by an enhanced affinity TCR designed for cancer immunotherapy. Sci Rep, 6, 2016
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1T2I
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4V1S
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![BU of 4v1s by Molmil](/molmil-images/mine/4v1s) | Structure of the GH76 alpha-mannanase BT2949 from Bacteroides thetaiotaomicron | 分子名称: | ALPHA-1,6-MANNANASE, GLYCEROL | 著者 | Thompson, A.J, Cuskin, F, Spears, R.J, Dabin, J, Turkenburg, J.P, Gilbert, H.J, Davies, G.J. | 登録日 | 2014-10-02 | 公開日 | 2015-02-11 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Structure of the Gh76 Alpha-Mannanase Homolog, Bt2949, from the Gut Symbiont Bacteroides Thetaiotaomicron Acta Crystallogr.,Sect.D, 71, 2015
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4WAJ
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1SZ2
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![BU of 1sz2 by Molmil](/molmil-images/mine/1sz2) | Crystal structure of E. coli glucokinase in complex with glucose | 分子名称: | Glucokinase, beta-D-glucopyranose | 著者 | Lunin, V.V, Li, Y, Schrag, J.D, Iannuzzi, P, Matte, A, Cygler, M. | 登録日 | 2004-04-02 | 公開日 | 2004-11-16 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Crystal structures of Escherichia coli ATP-dependent glucokinase and its complex with glucose J.Bacteriol., 186, 2004
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4WAK
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6D43
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4WAM
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4WLA
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1UA2
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![BU of 1ua2 by Molmil](/molmil-images/mine/1ua2) | Crystal Structure of Human CDK7 | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, Cell division protein kinase 7 | 著者 | Lolli, G, Lowe, E.D, Brown, N.R, Johnson, L.N. | 登録日 | 2004-08-11 | 公開日 | 2004-12-07 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (3.02 Å) | 主引用文献 | The Crystal Structure of Human CDK7 and Its Protein Recognition Properties Structure, 12, 2004
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6WE2
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![BU of 6we2 by Molmil](/molmil-images/mine/6we2) | Human PARP14 (ARTD8), catalytic fragment in complex with RBN012759 | 分子名称: | 1,2-ETHANEDIOL, 7-(cyclopropylmethoxy)-5-fluoro-2-{[(trans-4-hydroxycyclohexyl)sulfanyl]methyl}quinazolin-4(3H)-one, Isoform 1 of Protein mono-ADP-ribosyltransferase PARP14 | 著者 | Swinger, K.K, Schenkel, L.B, Kuntz, K.W. | 登録日 | 2020-04-01 | 公開日 | 2021-03-24 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.66 Å) | 主引用文献 | A potent and selective PARP14 inhibitor decreases protumor macrophage gene expression and elicits inflammatory responses in tumor explants. Cell Chem Biol, 28, 2021
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6UDC
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![BU of 6udc by Molmil](/molmil-images/mine/6udc) | Spectroscopic and structural characterization of a genetically encoded direct sensor for protein-ligand interactions | 分子名称: | BIOTIN, Streptavidin | 著者 | Mills, J.H, Gleason, P.R, Simmons, C.R, Henderson, J.N, Kartchner, B.K. | 登録日 | 2019-09-19 | 公開日 | 2020-09-23 | 最終更新日 | 2021-10-13 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structural Origins of Altered Spectroscopic Properties upon Ligand Binding in Proteins Containing a Fluorescent Noncanonical Amino Acid. Biochemistry, 60, 2021
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4WL9
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6UC3
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![BU of 6uc3 by Molmil](/molmil-images/mine/6uc3) | Spectroscopic and structural characterization of a genetically encoded direct sensor for protein-ligand interactions | 分子名称: | BIOTIN, Streptavidin | 著者 | Mills, J.H, Gleason, P.R, Simmons, C.R, Henderson, J.N, Kartchner, B.K. | 登録日 | 2019-09-13 | 公開日 | 2020-09-16 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.84 Å) | 主引用文献 | Structural Origins of Altered Spectroscopic Properties upon Ligand Binding in Proteins Containing a Fluorescent Noncanonical Amino Acid. Biochemistry, 60, 2021
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6UD1
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![BU of 6ud1 by Molmil](/molmil-images/mine/6ud1) | Spectroscopic and structural characterization of a genetically encoded direct sensor for protein-ligand interactions | 分子名称: | CHLORIDE ION, Streptavidin | 著者 | Mills, J.H, Gleason, P.R, Simmons, C.R, Henderson, J.N, Kartchner, B.K. | 登録日 | 2019-09-18 | 公開日 | 2021-02-10 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Structural Origins of Altered Spectroscopic Properties upon Ligand Binding in Proteins Containing a Fluorescent Noncanonical Amino Acid. Biochemistry, 60, 2021
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7KL8
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![BU of 7kl8 by Molmil](/molmil-images/mine/7kl8) | Structure of F420 binding protein Rv1558 from Mycobacterium tuberculosis with F420 bound | 分子名称: | COENZYME F420, COENZYME F420-3, Deazaflavin-dependent nitroreductase, ... | 著者 | Lee, B.M, Tan, L.L, Jackson, C.J. | 登録日 | 2020-10-29 | 公開日 | 2021-03-24 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.469 Å) | 主引用文献 | Potency boost of a Mycobacterium tuberculosis dihydrofolate reductase inhibitor by multienzyme F 420 H 2 -dependent reduction. Proc.Natl.Acad.Sci.USA, 118, 2021
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2Z98
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2Z9C
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5LU6
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![BU of 5lu6 by Molmil](/molmil-images/mine/5lu6) | Heptose isomerase mutant - H64Q | 分子名称: | 1,2-ETHANEDIOL, D-ALTRO-HEPT-2-ULOSE 7-PHOSPHATE, GLYCEROL, ... | 著者 | Vivoli, M, Harmer, N.J, Pang, J. | 登録日 | 2016-09-08 | 公開日 | 2017-12-06 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.67 Å) | 主引用文献 | A half-site multimeric enzyme achieves its cooperativity without conformational changes. Sci Rep, 7, 2017
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2YDE
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![BU of 2yde by Molmil](/molmil-images/mine/2yde) | FACTOR INHIBITING HIF-1 ALPHA IN COMPLEX WITH S-2-HYDROXYGLUTARATE | 分子名称: | (2S)-2-HYDROXYPENTANEDIOIC ACID, FE (III) ION, GLYCEROL, ... | 著者 | Chowdhury, R, Clifton, I.J, Schofield, C.J. | 登録日 | 2011-03-18 | 公開日 | 2011-03-30 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.28 Å) | 主引用文献 | The oncometabolite 2-hydroxyglutarate inhibits histone lysine demethylases. EMBO Rep., 12, 2011
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2YBP
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![BU of 2ybp by Molmil](/molmil-images/mine/2ybp) | JMJD2A COMPLEXED WITH R-2-HYDROXYGLUTARATE AND HISTONE H3K36me3 PEPTIDE (30-41) | 分子名称: | (2R)-2-hydroxypentanedioic acid, GLYCEROL, HISTONE H3.1T, ... | 著者 | Chowdhury, R, McDonough, M.A, Schofield, C.J. | 登録日 | 2011-03-09 | 公開日 | 2011-03-30 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.02 Å) | 主引用文献 | The oncometabolite 2-hydroxyglutarate inhibits histone lysine demethylases. EMBO Rep., 12, 2011
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4ABI
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![BU of 4abi by Molmil](/molmil-images/mine/4abi) | Co-complex structure of bovine trypsin with a modified Bowman-Birk inhibitor (PtA)SFTI-1(1,14), that was 1,4-disubstituted with a 1,2,3- trizol to mimic a trans amide bond | 分子名称: | CALCIUM ION, CATIONIC TRYPSIN, DIMETHYLFORMAMIDE, ... | 著者 | Schmelz, S, Empting, M, Tischler, M, Nasu, D, Heinz, D, Kolmar, H. | 登録日 | 2011-12-08 | 公開日 | 2012-03-07 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Braces for the Peptide Backbone: Insights Into Structure-Activity Relation-Ships of Protease Inhibitor Mimics with Locked Amide Conformations Angew.Chem.Int.Ed.Engl., 51, 2012
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7L05
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![BU of 7l05 by Molmil](/molmil-images/mine/7l05) | Complex of novel maytansinoid M24 bound to T2R-TTL (two tubulin alpha/beta heterodimers, RB3 stathmin-like domain, and tubulin tyrosine ligase) | 分子名称: | (1S,2R,3S,5S,6S,16E,18E,20R,21S)-11-chloro-21-hydroxy-12,20-dimethoxy-2,5,9,16-tetramethyl-8,23-dioxo-4,24-dioxa-9,22-diazatetracyclo[19.3.1.1~10,14~.0~3,5~]hexacosa-10(26),11,13,16,18-pentaen-6-yl (2S)-2-{methyl[3-(methylamino)propanoyl]amino}propanoate (non-preferred name), 1,2-ETHANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, ... | 著者 | Franklin, M.C. | 登録日 | 2020-12-11 | 公開日 | 2021-12-22 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.21 Å) | 主引用文献 | A Biparatopic Antibody-Drug Conjugate to Treat MET-Expressing Cancers, Including Those that Are Unresponsive to MET Pathway Blockade. Mol.Cancer Ther., 20, 2021
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2Z9D
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2YC0
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![BU of 2yc0 by Molmil](/molmil-images/mine/2yc0) | FACTOR INHIBITING HIF-1 ALPHA IN COMPLEX WITH R-2-HYDROXYGLUTARATE | 分子名称: | (2R)-2-hydroxypentanedioic acid, FE (II) ION, GLYCEROL, ... | 著者 | Chowdhury, R, Clifton, I.J, Schofield, C.J. | 登録日 | 2011-03-10 | 公開日 | 2011-03-30 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.15 Å) | 主引用文献 | The oncometabolite 2-hydroxyglutarate inhibits histone lysine demethylases. EMBO Rep., 12, 2011
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