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1ESE
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BU of 1ese by Molmil
THE MOLECULAR MECHANISM OF ENANTIORECOGNITION BY ESTERASES
分子名称: DIETHYL PHOSPHONATE, ESTERASE
著者Wei, Y, Schottel, J.L, Derewenda, U, Swenson, L, Patkar, S, Derewenda, Z.S.
登録日1994-10-07
公開日1995-10-15
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献A novel variant of the catalytic triad in the Streptomyces scabies esterase.
Nat.Struct.Biol., 2, 1995
1EBV
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OVINE PGHS-1 COMPLEXED WITH SALICYL HYDROXAMIC ACID
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ACETIC ACID SALICYLOYL-AMINO-ESTER, ...
著者Loll, P.J, Sharkey, C.T, O'Connor, S.J, Fitzgerald, D.J.
登録日2000-01-24
公開日2000-02-24
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献O-acetylsalicylhydroxamic acid, a novel acetylating inhibitor of prostaglandin H2 synthase: structural and functional characterization of enzyme-inhibitor interactions.
Mol.Pharmacol., 60, 2001
1EQ0
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SOLUTION STRUCTURE OF 6-HYDROXYMETHYL-7,8-DIHYDROPTERIN PYROPHOSPHOKINASE COMPLEXED WITH MGAMPPCP
分子名称: 6-HYDROXYMETHYL-7,8-DIHYDROPTERIN PYROPHOSPHOKINASE
著者Shi, G, Yan, H.
登録日2000-03-30
公開日2001-11-07
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Unusual conformational changes in 6-hydroxymethyl-7,8-dihydropterin pyrophosphokinase as revealed by X-ray crystallography and NMR.
J.Biol.Chem., 276, 2001
1HT5
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THE 2.75 ANGSTROM RESOLUTION MODEL OF OVINE COX-1 COMPLEXED WITH METHYL ESTER FLURBIPROFEN
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, FLURBIPROFEN METHYL ESTER, PROSTAGLANDIN H2 SYNTHASE-1, ...
著者Selinsky, B.S, Gupta, K, Sharkey, C.T, Loll, P.J.
登録日2000-12-28
公開日2001-04-11
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.75 Å)
主引用文献Structural analysis of NSAID binding by prostaglandin H2 synthase: time-dependent and time-independent inhibitors elicit identical enzyme conformations.
Biochemistry, 40, 2001
1BCT
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THREE-DIMENSIONAL STRUCTURE OF PROTEOLYTIC FRAGMENT 163-231 OF BACTERIOOPSIN DETERMINED FROM NUCLEAR MAGNETIC RESONANCE DATA IN SOLUTION
分子名称: BACTERIORHODOPSIN
著者Nolde, D.E, Barsukov, I.L, Lomize, A.L, Arseniev, A.S.
登録日1993-07-07
公開日1994-04-30
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Three-dimensional structure of proteolytic fragment 163-231 of bacterioopsin determined from nuclear magnetic resonance data in solution.
Eur.J.Biochem., 206, 1992
1B82
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PRISTINE RECOMB. LIGNIN PEROXIDASE H8
分子名称: CALCIUM ION, PROTEIN (LIGNIN PEROXIDASE), PROTOPORPHYRIN IX CONTAINING FE
著者Blodig, W, Doyle, W.A, Smith, A.T, Piontek, K.
登録日1999-02-04
公開日1999-02-16
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Crystal structures of pristine and oxidatively processed lignin peroxidase expressed in Escherichia coli and of the W171F variant that eliminates the redox active tryptophan 171. Implications for the reaction mechanism.
J.Mol.Biol., 305, 2001
1F6D
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THE STRUCTURE OF UDP-N-ACETYLGLUCOSAMINE 2-EPIMERASE FROM E. COLI.
分子名称: CHLORIDE ION, SODIUM ION, UDP-N-ACETYLGLUCOSAMINE 2-EPIMERASE, ...
著者Campbell, R.E, Mosimann, S.C, Tanner, M.E, Strynadka, N.C.J.
登録日2000-06-21
公開日2000-12-13
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献The structure of UDP-N-acetylglucosamine 2-epimerase reveals homology to phosphoglycosyl transferases.
Biochemistry, 39, 2000
1B8G
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1-AMINOCYCLOPROPANE-1-CARBOXYLATE SYNTHASE
分子名称: PROTEIN (1-AMINOCYCLOPROPANE-1-CARBOXYLATE SYNTHASE), PYRIDOXAL-5'-PHOSPHATE
著者Capitani, G, Hohenester, E, Feng, L, Storici, P, Kirsch, J.F, Jansonius, J.N.
登録日1999-01-31
公開日2000-01-26
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.37 Å)
主引用文献Structure of 1-aminocyclopropane-1-carboxylate synthase, a key enzyme in the biosynthesis of the plant hormone ethylene.
J.Mol.Biol., 294, 1999
1GJH
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HUMAN BCL-2, ISOFORM 2
分子名称: PROTEIN (APOPTOSIS REGULATOR BCL-2 WITH PUTATIVE FLEXIBLE LOOP REPLACED WITH A PORTION OF APOPTOSIS REGULATOR BCL-X PROTEIN)
著者Petros, A.M, Medek, A, Nettesheim, D.G, Kim, D.H, Yoon, H.S, Swift, K, Matayoshi, E.D, Oltersdorf, T, Fesik, S.W.
登録日2001-05-31
公開日2001-06-13
最終更新日2023-12-27
実験手法SOLUTION NMR
主引用文献Solution structure of the antiapoptotic protein bcl-2.
Proc.Natl.Acad.Sci.USA, 98, 2001
1FZ6
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METHANE MONOOXYGENASE HYDROXYLASE, FORM II SOAKED IN 1 M METHANOL
分子名称: CALCIUM ION, FE (III) ION, METHANE MONOOXYGENASE COMPONENT A, ...
著者Whittington, D.A, Sazinsky, M.H, Lippard, S.J.
登録日2000-10-03
公開日2001-04-27
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献X-ray crystal structure of alcohol products bound at the active site of soluble methane monooxygenase hydroxylase.
J.Am.Chem.Soc., 123, 2001
1B1Y
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SEVENFOLD MUTANT OF BARLEY BETA-AMYLASE
分子名称: PROTEIN (BETA-AMYLASE), alpha-D-glucopyranose-(1-4)-beta-D-glucopyranose, beta-D-glucopyranose
著者Mikami, B, Yoon, H.J, Yoshigi, N.
登録日1998-11-25
公開日1998-12-02
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献The crystal structure of the sevenfold mutant of barley beta-amylase with increased thermostability at 2.5 A resolution.
J.Mol.Biol., 285, 1999
1G3G
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NMR STRUCTURE OF THE FHA1 DOMAIN OF YEAST RAD53
分子名称: PROTEIN KINASE SPK1
著者Yuan, C, Liao, H, Su, M, Yongkiettrakul, S, Byeon, I.-J.L, Tsai, M.-D.
登録日2000-10-24
公開日2001-01-10
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Structure of the FHA1 domain of yeast Rad53 and identification of binding sites for both FHA1 and its target protein Rad9
J.Mol.Biol., 304, 2000
1GMJ
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The structure of bovine IF1, the regulatory subunit of mitochondrial F-ATPase
分子名称: ATPASE INHIBITOR
著者Cabezon, E, Runswick, M.J, Leslie, A.G.W, Walker, J.E.
登録日2001-09-14
公開日2002-01-01
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献The Structure of Bovine If(1), the Regulatory Subunit of Mitochondrial F-ATPase.
Embo J., 20, 2001
1CQZ
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BU of 1cqz by Molmil
CRYSTAL STRUCTURE OF MURINE SOLUBLE EPOXIDE HYDROLASE.
分子名称: EPOXIDE HYDROLASE
著者Argiriadi, M.A, Morisseau, C, Hammock, B.D, Christianson, D.W.
登録日1999-08-12
公開日1999-11-19
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Detoxification of environmental mutagens and carcinogens: structure, mechanism, and evolution of liver epoxide hydrolase.
Proc.Natl.Acad.Sci.USA, 96, 1999
1FOL
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REDUCED BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH L-ARG(H4B-FREE)
分子名称: ACETATE ION, ARGININE, CACODYLATE ION, ...
著者Raman, C.S, Li, H, Martasek, P, Masters, B.S, Poulos, T.L.
登録日2000-08-28
公開日2001-07-20
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Crystallographic studies on endothelial nitric oxide synthase complexed with nitric oxide and mechanism-based inhibitors
Biochemistry, 40, 2001
1FOI
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BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH 1400W(H4B-FREE)
分子名称: ACETATE ION, CACODYLATE ION, GLYCEROL, ...
著者Raman, C.S, Li, H, Martasek, P, Masters, B.S.S, Poulos, T.L.
登録日2000-08-28
公開日2001-07-20
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.93 Å)
主引用文献Crystallographic studies on endothelial nitric oxide synthase complexed with nitric oxide and mechanism-based inhibitors.
Biochemistry, 40, 2001
4QKB
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Crystal structure of seleno-methionine labelled human ALKBH7 in complex with alpha-ketoglutarate and Mn(II)
分子名称: 2-OXOGLUTARIC ACID, Alpha-ketoglutarate-dependent dioxygenase alkB homolog 7, mitochondrial, ...
著者Wang, G, He, Q, Chen, Z.
登録日2014-06-05
公開日2014-08-20
最終更新日2015-10-21
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献The atomic resolution structure of human AlkB homolog 7 (ALKBH7), a key protein for programmed necrosis and fat metabolism
J.Biol.Chem., 289, 2014
4QL6
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Structure of C. trachomatis CT441
分子名称: Carboxy-terminal processing protease
著者Kohlmann, F, Hilgenfeld, R, Hansen, G.
登録日2014-06-10
公開日2014-11-05
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.97 Å)
主引用文献Structural basis of the proteolytic and chaperone activity of Chlamydia trachomatis CT441
J.Bacteriol., 197, 2015
4QXC
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Crystal structure of histone demethylase KDM2A-H3K36ME2 with NOG
分子名称: Histone H3.2, Lysine-specific demethylase 2A, N-OXALYLGLYCINE, ...
著者Cheng, Z.J, Patel, D.J.
登録日2014-07-19
公開日2014-11-05
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献A molecular threading mechanism underlies Jumonji lysine demethylase KDM2A regulation of methylated H3K36.
Genes Dev., 28, 2014
4QXB
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crystal structure of histone demethylase KDM2A-H3K36ME3 with NOG
分子名称: Histone H3.2, Lysine-specific demethylase 2A, N-OXALYLGLYCINE, ...
著者Cheng, Z.J, Patel, D.J.
登録日2014-07-19
公開日2014-11-05
最終更新日2019-07-17
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献A molecular threading mechanism underlies Jumonji lysine demethylase KDM2A regulation of methylated H3K36.
Genes Dev., 28, 2014
4QWN
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Histone demethylase KDM2A-H3K36ME1-alpha-KG complex structure
分子名称: 2-OXOGLUTARIC ACID, Histone H3.2, Lysine-specific demethylase 2A, ...
著者Cheng, Z.J, Patel, D.J.
登録日2014-07-16
公開日2014-11-05
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献A molecular threading mechanism underlies Jumonji lysine demethylase KDM2A regulation of methylated H3K36.
Genes Dev., 28, 2014
4QX8
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Crystal structure of histone demethylase kdm2a-h3k36me3 complex with alpha-kg
分子名称: 2-OXOGLUTARIC ACID, Histone H3.2, Lysine-specific demethylase 2A, ...
著者Cheng, Z.J, Patel, D.J.
登録日2014-07-19
公開日2014-11-05
最終更新日2018-01-24
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献A molecular threading mechanism underlies Jumonji lysine demethylase KDM2A regulation of methylated H3K36.
Genes Dev., 28, 2014
4R8Z
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Crystal Structure of PA4781 HD-GYP domain from Pseudomonas aeruginosa at 2.2A resolution showing a bi-metallic Ni ion center
分子名称: CHLORIDE ION, Cyclic di-GMP phosphodiesterase, NICKEL (II) ION
著者Giardina, G, Cutruzzolaa, F, Rinaldo, S, Stelitano, V.
登録日2014-09-03
公開日2015-03-04
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structural basis of functional diversification of the HD-GYP domain revealed by the Pseudomonas aeruginosa PA4781 protein, which displays an unselective bimetallic binding site.
J.Bacteriol., 197, 2015
4QT0
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Crystal structure of human muscle L-lactate dehydrogenase in complex with inhibitor 1, 3-{[3-CARBAMOYL-7-(2,4-DIMETHOXYPYRIMIDIN-5-YL)QUINOLIN-4-YL]AMINO}BENZOIC ACID
分子名称: 3-{[3-carbamoyl-7-(2,4-dimethoxypyrimidin-5-yl)quinolin-4-yl]amino}benzoic acid, L-lactate dehydrogenase A chain
著者Kolappan, S, Craig, L.
登録日2014-07-06
公開日2014-12-03
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Structures of lactate dehydrogenase A (LDHA) in apo, ternary and inhibitor-bound forms.
Acta Crystallogr.,Sect.D, 71, 2015
4QXH
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Crystal structure of histone demethylase KDM2A-H3K36ME1 with NOG
分子名称: Histone H3.2, Lysine-specific demethylase 2A, N-OXALYLGLYCINE, ...
著者Cheng, Z.J, Patel, D.J.
登録日2014-07-20
公開日2014-11-05
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献A molecular threading mechanism underlies Jumonji lysine demethylase KDM2A regulation of methylated H3K36.
Genes Dev., 28, 2014

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