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8UQ2
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Structure of human RyR2-S2808D in the subprimed state
分子名称: ADENOSINE-5'-TRIPHOSPHATE, Peptidyl-prolyl cis-trans isomerase FKBP1B, Ryanodine receptor 2, ...
著者Miotto, M.C, Marks, A.R.
登録日2023-10-23
公開日2023-11-15
実験手法ELECTRON MICROSCOPY (2.98 Å)
主引用文献Structural basis for ryanodine receptor type 2 leak in heart failure and arrhythmogenic disorders
To Be Published
8U4D
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BU of 8u4d by Molmil
TRPV1 in nanodisc bound with PI-Br4, consensus structure
分子名称: (2S)-2-[(9,10-dibromooctadecanoyl)oxy]-3-{[(S)-hydroxy{[(1S,2R,3R,4S,5S,6R)-2,3,4,5,6-pentahydroxycyclohexyl]oxy}phosphoryl]oxy}propyl (9R,10S)-9,10-dibromooctadecanoate, SODIUM ION, Transient receptor potential cation channel subfamily V member 1
著者Arnold, W.R, Julius, D, Cheng, Y.
登録日2023-09-10
公開日2024-05-08
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (2.2 Å)
主引用文献Structural basis of TRPV1 modulation by endogenous bioactive lipids.
Nat.Struct.Mol.Biol., 2024
8U43
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TRPV1 in nanodisc bound with PIP2-Br4
分子名称: (2S)-2-[(9,10-dibromooctadecanoyl)oxy]-3-{[(S)-hydroxy{[(1R,2R,3S,4R,5R,6S)-2,3,6-trihydroxy-4,5-bis(phosphonooxy)cyclohexyl]oxy}phosphoryl]oxy}propyl (9R,10S)-9,10-dibromooctadecanoate, 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, SODIUM ION, ...
著者Arnold, W.R, Julius, D, Cheng, Y.
登録日2023-09-08
公開日2024-05-08
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (2.4 Å)
主引用文献Structural basis of TRPV1 modulation by endogenous bioactive lipids.
Nat.Struct.Mol.Biol., 2024
8U3L
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TRPV1 in nanodisc bound with empty vanilloid binding pocket at 25C
分子名称: 1,2-DIACYL-GLYCEROL-3-SN-PHOSPHATE, SODIUM ION, Transient receptor potential cation channel subfamily V member 1
著者Arnold, W.R, Julius, D, Cheng, Y.
登録日2023-09-07
公開日2024-05-08
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (3.7 Å)
主引用文献Structural basis of TRPV1 modulation by endogenous bioactive lipids.
Nat.Struct.Mol.Biol., 2024
8U3J
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TRPV1 in nanodisc bound with empty vanilloid binding pocket at 4C
分子名称: 1,2-DIACYL-GLYCEROL-3-SN-PHOSPHATE, SODIUM ION, Transient receptor potential cation channel subfamily V member 1
著者Arnold, W.R, Julius, D, Cheng, Y.
登録日2023-09-07
公開日2024-05-08
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (2.9 Å)
主引用文献Structural basis of TRPV1 modulation by endogenous bioactive lipids.
Nat.Struct.Mol.Biol., 2024
8U3C
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TRPV1 in nanodisc bound with PI-Br4 bound in Conformation 2 (monomer)
分子名称: (2S)-2-[(9,10-dibromooctadecanoyl)oxy]-3-{[(S)-hydroxy{[(1S,2R,3R,4S,5S,6R)-2,3,4,5,6-pentahydroxycyclohexyl]oxy}phosphoryl]oxy}propyl (9R,10S)-9,10-dibromooctadecanoate, 1,2-DIACYL-GLYCEROL-3-SN-PHOSPHATE, 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, ...
著者Arnold, W.R, Julius, D, Cheng, Y.
登録日2023-09-07
公開日2024-05-08
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (2.3 Å)
主引用文献Structural basis of TRPV1 modulation by endogenous bioactive lipids.
Nat.Struct.Mol.Biol., 2024
8U3A
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BU of 8u3a by Molmil
TRPV1 in nanodisc bound with PI-Br4 bound in Conformation 1 (monomer)
分子名称: (2S)-2-[(9,10-dibromooctadecanoyl)oxy]-3-{[(S)-hydroxy{[(1S,2R,3R,4S,5S,6R)-2,3,4,5,6-pentahydroxycyclohexyl]oxy}phosphoryl]oxy}propyl (9R,10S)-9,10-dibromooctadecanoate, 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, SODIUM ION, ...
著者Arnold, W.R, Julius, D, Cheng, Y.
登録日2023-09-07
公開日2024-05-08
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (2.3 Å)
主引用文献Structural basis of TRPV1 modulation by endogenous bioactive lipids.
Nat.Struct.Mol.Biol., 2024
8U30
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TRPV1 in nanodisc bound with diC8-PIP2 in the closed state
分子名称: SODIUM ION, Transient receptor potential cation channel subfamily V member 1, [(2R)-2-octanoyloxy-3-[oxidanyl-[(1R,2R,3S,4R,5R,6S)-2,3,6-tris(oxidanyl)-4,5-diphosphonooxy-cyclohexyl]oxy-phosphoryl]oxy-propyl] octanoate
著者Arnold, W.R, Julius, D, Cheng, Y.
登録日2023-09-06
公開日2024-05-08
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (3 Å)
主引用文献Structural basis of TRPV1 modulation by endogenous bioactive lipids.
Nat.Struct.Mol.Biol., 2024
8U2Z
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TRPV1 in nanodisc bound with diC8-PIP2 in the dilated state
分子名称: 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, CHOLESTEROL, SODIUM ION, ...
著者Arnold, W.R, Julius, D, Cheng, Y.
登録日2023-09-06
公開日2024-05-08
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (3.6 Å)
主引用文献Structural basis of TRPV1 modulation by endogenous bioactive lipids.
Nat.Struct.Mol.Biol., 2024
8TLA
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BU of 8tla by Molmil
Human Type 3 IP3 Receptor - Higher-Order Inhibited State - Symmetry Mate 1
分子名称: ADENOSINE-5'-TRIPHOSPHATE, CALCIUM ION, D-MYO-INOSITOL-1,4,5-TRIPHOSPHATE, ...
著者Paknejad, N, Sapuru, V, Hite, R.K.
登録日2023-07-26
公開日2023-11-08
実験手法ELECTRON MICROSCOPY (3.2 Å)
主引用文献Structural titration reveals Ca 2+ -dependent conformational landscape of the IP 3 receptor.
Nat Commun, 14, 2023
8TL9
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Human Type 3 IP3 Receptor - Resting State (+IP3/ATP)
分子名称: ADENOSINE-5'-TRIPHOSPHATE, CALCIUM ION, D-MYO-INOSITOL-1,4,5-TRIPHOSPHATE, ...
著者Paknejad, N, Sapuru, V, Hite, R.K.
登録日2023-07-26
公開日2023-11-08
実験手法ELECTRON MICROSCOPY (3.3 Å)
主引用文献Structural titration reveals Ca 2+ -dependent conformational landscape of the IP 3 receptor.
Nat Commun, 14, 2023
8TKI
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Human Type 3 IP3 Receptor - Labile Resting State 2 (+IP3/ATP)
分子名称: ADENOSINE-5'-TRIPHOSPHATE, D-MYO-INOSITOL-1,4,5-TRIPHOSPHATE, Inositol 1,4,5-trisphosphate receptor type 3, ...
著者Paknejad, N, Sapuru, V, Hite, R.K.
登録日2023-07-25
公開日2023-11-08
実験手法ELECTRON MICROSCOPY (3.6 Å)
主引用文献Structural titration reveals Ca 2+ -dependent conformational landscape of the IP 3 receptor.
Nat Commun, 14, 2023
8TKH
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BU of 8tkh by Molmil
Human Type 3 IP3 Receptor - Labile Resting State 1 (+IP3/ATP)
分子名称: ADENOSINE-5'-TRIPHOSPHATE, D-MYO-INOSITOL-1,4,5-TRIPHOSPHATE, Inositol 1,4,5-trisphosphate receptor type 3, ...
著者Paknejad, N, Sapuru, V, Hite, R.K.
登録日2023-07-25
公開日2023-11-08
実験手法ELECTRON MICROSCOPY (3.5 Å)
主引用文献Structural titration reveals Ca 2+ -dependent conformational landscape of the IP 3 receptor.
Nat Commun, 14, 2023
8TKG
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BU of 8tkg by Molmil
Human Type 3 IP3 Receptor - Resting State (+IP3/ATP)
分子名称: 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, ADENOSINE-5'-TRIPHOSPHATE, CALCIUM ION, ...
著者Paknejad, N, Sapuru, V, Hite, R.K.
登録日2023-07-25
公開日2023-11-08
実験手法ELECTRON MICROSCOPY (2.5 Å)
主引用文献Structural titration reveals Ca 2+ -dependent conformational landscape of the IP 3 receptor.
Nat Commun, 14, 2023
8TKF
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Human Type 3 IP3 Receptor - Activated State (+IP3/ATP/JD Ca2+)
分子名称: 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, ADENOSINE-5'-TRIPHOSPHATE, CALCIUM ION, ...
著者Paknejad, N, Sapuru, V, Hite, R.K.
登録日2023-07-25
公開日2023-11-08
実験手法ELECTRON MICROSCOPY (3.2 Å)
主引用文献Structural titration reveals Ca 2+ -dependent conformational landscape of the IP 3 receptor.
Nat Commun, 14, 2023
8TKE
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BU of 8tke by Molmil
Human Type 3 IP3 Receptor - Preactivated+Ca2+ State (+IP3/ATP/JD Ca2+)
分子名称: ADENOSINE-5'-TRIPHOSPHATE, CALCIUM ION, D-MYO-INOSITOL-1,4,5-TRIPHOSPHATE, ...
著者Paknejad, N, Sapuru, V, Hite, R.K.
登録日2023-07-25
公開日2023-11-08
実験手法ELECTRON MICROSCOPY (3.6 Å)
主引用文献Structural titration reveals Ca 2+ -dependent conformational landscape of the IP 3 receptor.
Nat Commun, 14, 2023
8TKD
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BU of 8tkd by Molmil
Human Type 3 IP3 Receptor - Preactivated State (+IP3/ATP)
分子名称: ADENOSINE-5'-TRIPHOSPHATE, D-MYO-INOSITOL-1,4,5-TRIPHOSPHATE, Inositol 1,4,5-trisphosphate receptor type 3, ...
著者Paknejad, N, Sapuru, V, Hite, R.K.
登録日2023-07-25
公開日2023-11-08
実験手法ELECTRON MICROSCOPY (3.7 Å)
主引用文献Structural titration reveals Ca 2+ -dependent conformational landscape of the IP 3 receptor.
Nat Commun, 14, 2023
8TK8
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BU of 8tk8 by Molmil
Human Type 3 IP3 Receptor - Resting State (+IP3/ATP)
分子名称: 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, ADENOSINE-5'-TRIPHOSPHATE, D-MYO-INOSITOL-1,4,5-TRIPHOSPHATE, ...
著者Paknejad, N, Sapuru, V, Hite, R.K.
登録日2023-07-25
公開日2023-11-08
実験手法ELECTRON MICROSCOPY (2.7 Å)
主引用文献Structural titration reveals Ca 2+ -dependent conformational landscape of the IP 3 receptor.
Nat Commun, 14, 2023
8THH
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BU of 8thh by Molmil
Cryo-EM structure of Nav1.7 with LTG
分子名称: (6M)-6-(2,3-dichlorophenyl)-1,2,4-triazine-3,5-diamine, 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 1-O-OCTADECYL-SN-GLYCERO-3-PHOSPHOCHOLINE, ...
著者Fan, X, Huang, J, Yan, N.
登録日2023-07-16
公開日2023-11-22
実験手法ELECTRON MICROSCOPY (2.7 Å)
主引用文献Dual-pocket inhibition of Na v channels by the antiepileptic drug lamotrigine.
Proc.Natl.Acad.Sci.USA, 120, 2023
8THG
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Cryo-EM structure of Nav1.7 with RLZ
分子名称: 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 1-O-OCTADECYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Fan, X, Huang, J, Yan, N.
登録日2023-07-16
公開日2023-11-22
実験手法ELECTRON MICROSCOPY (2.9 Å)
主引用文献Dual-pocket inhibition of Na v channels by the antiepileptic drug lamotrigine.
Proc.Natl.Acad.Sci.USA, 120, 2023
8TF4
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BU of 8tf4 by Molmil
Wildtype rabbit TRPV5 into nanodiscs in the presence of PI(4,5)P2 and econazole
分子名称: 1-PALMITOYL-2-LINOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 1-[(2S)-2-[(4-CHLOROBENZYL)OXY]-2-(2,4-DICHLOROPHENYL)ETHYL]-1H-IMIDAZOLE, ERGOSTEROL, ...
著者De Jesus-Perez, J.J, Fluck, E.C, Moiseenkova-Bell, V.Y.
登録日2023-07-07
公開日2024-01-10
最終更新日2024-02-14
実験手法ELECTRON MICROSCOPY (2.86 Å)
主引用文献Structural mechanism of TRPV5 inhibition by econazole.
Structure, 32, 2024
8TF3
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Wildtype rabbit TRPV5 into nanodiscs in complex with econazole
分子名称: 1-PALMITOYL-2-LINOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 1-[(2S)-2-[(4-CHLOROBENZYL)OXY]-2-(2,4-DICHLOROPHENYL)ETHYL]-1H-IMIDAZOLE, ERGOSTEROL, ...
著者De Jesus-Perez, J.J, Fluck, E.C, Moiseenkova-Bell, V.Y.
登録日2023-07-07
公開日2024-01-10
最終更新日2024-02-14
実験手法ELECTRON MICROSCOPY (2.94 Å)
主引用文献Structural mechanism of TRPV5 inhibition by econazole.
Structure, 32, 2024
8TF2
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Wildtype rabbit TRPV5 into nanodiscs in Apo state
分子名称: 1-PALMITOYL-2-LINOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, ERGOSTEROL, Transient receptor potential cation channel subfamily V member 5
著者De Jesus-Perez, J.J, Fluck, E.C, Moiseenkova-Bell, V.Y.
登録日2023-07-07
公開日2024-01-10
最終更新日2024-02-14
実験手法ELECTRON MICROSCOPY (2.57 Å)
主引用文献Structural mechanism of TRPV5 inhibition by econazole.
Structure, 32, 2024
8TEO
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Shaker in low K+ (4mM K+)
分子名称: (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, POTASSIUM ION, Potassium voltage-gated channel protein Shaker
著者Tan, X, Swartz, K.J.
登録日2023-07-06
公開日2023-12-20
実験手法ELECTRON MICROSCOPY (2.39 Å)
主引用文献Eukaryotic Kv channel Shaker inactivates through selectivity filter dilation rather than collapse.
Sci Adv, 9, 2023
8T6L
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Cryo-EM structure of rat cardiac sodium channel NaV1.5 with batrachotoxin analog BTX-B
分子名称: (1R)-1-[(5aR,7aR,9R,11aS,11bS,12R,13aR)-9,12-dihydroxy-2,11a-dimethyl-1,2,3,4,7a,8,9,10,11,11a,12,13-dodecahydro-7H-9,11b-epoxy-13a,5a-prop[1]enophenanthro[2,1-f][1,4]oxazepin-14-yl]ethyl benzoate, (3beta,14beta,17beta,25R)-3-[4-methoxy-3-(methoxymethyl)butoxy]spirost-5-en, 1-palmitoyl-2-oleoyl-sn-glycero-3-phosphocholine, ...
著者Tonggu, L, Wisedchaisri, G, Gamal El-Din, T.M, Zheng, N, Catterall, W.A.
登録日2023-06-16
公開日2024-03-06
最終更新日2024-03-27
実験手法ELECTRON MICROSCOPY (3.3 Å)
主引用文献Dual receptor-sites reveal the structural basis for hyperactivation of sodium channels by poison-dart toxin batrachotoxin.
Nat Commun, 15, 2024

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件を2024-06-12に公開中

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