3UY6
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![BU of 3uy6 by Molmil](/molmil-images/mine/3uy6) | |
3UPP
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![BU of 3upp by Molmil](/molmil-images/mine/3upp) | |
3UPO
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![BU of 3upo by Molmil](/molmil-images/mine/3upo) | |
3UPN
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![BU of 3upn by Molmil](/molmil-images/mine/3upn) | |
3UN7
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![BU of 3un7 by Molmil](/molmil-images/mine/3un7) | |
3UE3
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![BU of 3ue3 by Molmil](/molmil-images/mine/3ue3) | Crystal structure of Acinetobacter baumanni PBP3 | 分子名称: | Septum formation, penicillin binding protein 3, peptidoglycan synthetase | 著者 | Han, S. | 登録日 | 2011-10-28 | 公開日 | 2011-12-14 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Distinctive attributes of beta-lactam target proteins in Acinetobacter baumannii relevant to development of new antibiotics J.Am.Chem.Soc., 133, 2011
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3UE1
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![BU of 3ue1 by Molmil](/molmil-images/mine/3ue1) | Crystal strucuture of Acinetobacter baumanni PBP1A in complex with MC-1 | 分子名称: | (4S,7Z)-7-(2-amino-1,3-thiazol-4-yl)-1-[({4-[(2R)-2,3-dihydroxypropyl]-3-(4,5-dihydroxypyridin-2-yl)-5-oxo-4,5-dihydro- 1H-1,2,4-triazol-1-yl}sulfonyl)amino]-4-formyl-10,10-dimethyl-1,6-dioxo-9-oxa-2,5,8-triazaundec-7-en-11-oate, Penicillin-binding protein 1a | 著者 | Han, S. | 登録日 | 2011-10-28 | 公開日 | 2011-12-14 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (2.73 Å) | 主引用文献 | Distinctive attributes of beta-lactam target proteins in Acinetobacter baumannii relevant to development of new antibiotics J.Am.Chem.Soc., 133, 2011
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3UE0
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![BU of 3ue0 by Molmil](/molmil-images/mine/3ue0) | Crystal structure of Acinetobacter baumannii PBP1a in complex with Aztreonam | 分子名称: | 2-({[(1Z)-1-(2-amino-1,3-thiazol-4-yl)-2-oxo-2-{[(2S,3S)-1-oxo-3-(sulfoamino)butan-2-yl]amino}ethylidene]amino}oxy)-2-methylpropanoic acid, Penicillin-binding protein 1a | 著者 | Han, S. | 登録日 | 2011-10-28 | 公開日 | 2011-12-14 | 最終更新日 | 2013-06-26 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Distinctive attributes of beta-lactam target proteins in Acinetobacter baumannii relevant to development of new antibiotics J.Am.Chem.Soc., 133, 2011
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3UDX
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![BU of 3udx by Molmil](/molmil-images/mine/3udx) | Crystal structure of Acinetobacter baumannii PBP1a in complex with Imipenem | 分子名称: | (5R)-5-[(1S,2R)-1-formyl-2-hydroxypropyl]-3-[(2-{[(E)-iminomethyl]amino}ethyl)sulfanyl]-4,5-dihydro-1H-pyrrole-2-carboxylic acid, Penicillin-binding protein 1a | 著者 | Han, S. | 登録日 | 2011-10-28 | 公開日 | 2011-12-14 | 最終更新日 | 2013-06-26 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Distinctive attributes of beta-lactam target proteins in Acinetobacter baumannii relevant to development of new antibiotics J.Am.Chem.Soc., 133, 2011
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3UDI
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3UDF
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![BU of 3udf by Molmil](/molmil-images/mine/3udf) | Crystal structure of Apo PBP1a from Acinetobacter baumannii | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, Penicillin-binding protein 1a | 著者 | Han, S. | 登録日 | 2011-10-28 | 公開日 | 2011-12-14 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Distinctive attributes of beta-lactam target proteins in Acinetobacter baumannii relevant to development of new antibiotics J.Am.Chem.Soc., 133, 2011
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3QNC
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![BU of 3qnc by Molmil](/molmil-images/mine/3qnc) | Crystal Structure of a Rationally Designed OXA-10 Variant Showing Carbapenemase Activity, OXA-10loop48 | 分子名称: | 1,2-ETHANEDIOL, CARBON DIOXIDE, Oxacillinase, ... | 著者 | De Luca, F, Benvenuti, M, Carboni, F, Pozzi, C, Rossolini, G.M, Mangani, S, Docquier, J.D. | 登録日 | 2011-02-08 | 公開日 | 2011-11-02 | 最終更新日 | 2023-12-06 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Evolution to carbapenem-hydrolyzing activity in noncarbapenemase class D {beta}-lactamase OXA-10 by rational protein design. Proc.Natl.Acad.Sci.USA, 108, 2011
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3QNB
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![BU of 3qnb by Molmil](/molmil-images/mine/3qnb) | Crystal Structure of an Engineered OXA-10 Variant with Carbapenemase Activity, OXA-10loop24 | 分子名称: | 1,2-ETHANEDIOL, Oxacillinase, SULFATE ION | 著者 | De Luca, F, Benvenuti, M, Carboni, F, Pozzi, C, Rossolini, G.M, Mangani, S, Docquier, J.D. | 登録日 | 2011-02-08 | 公開日 | 2011-11-02 | 最終更新日 | 2023-12-06 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Evolution to carbapenem-hydrolyzing activity in noncarbapenemase class D {beta}-lactamase OXA-10 by rational protein design. Proc.Natl.Acad.Sci.USA, 108, 2011
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3Q82
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![BU of 3q82 by Molmil](/molmil-images/mine/3q82) | Meropenem acylated BlaR1 sensor domain from Staphylococcus aureus | 分子名称: | (4R,5S)-3-{[(3S,5S)-5-(dimethylcarbamoyl)pyrrolidin-3-yl]sulfanyl}-5-[(2S,3R)-3-hydroxy-1-oxobutan-2-yl]-4-methyl-4,5-dihydro-1H-pyrrole-2-carboxylic acid, Beta-lactamase regulatory protein BlaR1, GLYCEROL | 著者 | Borbulevych, O.Y, Mobashery, S, Baker, B.M. | 登録日 | 2011-01-05 | 公開日 | 2011-07-20 | 最終更新日 | 2013-01-09 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Lysine Nzeta-decarboxylation switch and activation of the beta-lactam sensor domain of BlaR1 protein of methicillin-resistant Staphylococcus aureus. J.Biol.Chem., 286, 2011
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3Q81
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![BU of 3q81 by Molmil](/molmil-images/mine/3q81) | Imipenem acylated BlaR1 sensor domain from Staphylococcus aureus | 分子名称: | (5R)-5-[(1S,2R)-1-formyl-2-hydroxypropyl]-3-[(2-{[(E)-iminomethyl]amino}ethyl)sulfanyl]-4,5-dihydro-1H-pyrrole-2-carboxylic acid, Beta-lactamase regulatory protein BlaR1, GLYCEROL | 著者 | Borbulevych, O.Y, Mobashery, S, Baker, B.M. | 登録日 | 2011-01-05 | 公開日 | 2011-07-20 | 最終更新日 | 2013-01-09 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Lysine Nzeta-decarboxylation switch and activation of the beta-lactam sensor domain of BlaR1 protein of methicillin-resistant Staphylococcus aureus. J.Biol.Chem., 286, 2011
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3Q7Z
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![BU of 3q7z by Molmil](/molmil-images/mine/3q7z) | CBAP-acylated BlaR1 sensor domain from Staphylococcus aureus | 分子名称: | (2R,4S)-2-[(1R)-1-{[(2'-carboxybiphenyl-2-yl)carbonyl]amino}-2-oxoethyl]-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid, Beta-lactamase regulatory protein BlaR1 | 著者 | Borbulevych, O.Y, Mobashery, S, Baker, B.M. | 登録日 | 2011-01-05 | 公開日 | 2011-07-06 | 最終更新日 | 2017-11-08 | 実験手法 | X-RAY DIFFRACTION (1.87 Å) | 主引用文献 | Lysine Nzeta-decarboxylation switch and activation of the beta-lactam sensor domain of BlaR1 protein of methicillin-resistant Staphylococcus aureus. J.Biol.Chem., 286, 2011
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3Q7V
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3PBT
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![BU of 3pbt by Molmil](/molmil-images/mine/3pbt) | Crystal structure of PBP3 complexed with MC-1 | 分子名称: | (4S,7Z)-7-(2-amino-1,3-thiazol-4-yl)-1-[({4-[(2R)-2,3-dihydroxypropyl]-3-(4,5-dihydroxypyridin-2-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl}sulfonyl)amino]-4-formyl-10,10-dimethyl-1,6-dioxo-9-oxa-2,5,8-triazaundec-7-en-11-oate, Penicillin-binding protein 3 | 著者 | Han, S, Evdokimov, A. | 登録日 | 2010-10-20 | 公開日 | 2010-12-22 | 最終更新日 | 2012-02-08 | 実験手法 | X-RAY DIFFRACTION (1.641 Å) | 主引用文献 | Structural basis for effectiveness of siderophore-conjugated monocarbams against clinically relevant strains of Pseudomonas aeruginosa. Proc.Natl.Acad.Sci.USA, 107, 2010
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3PBS
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![BU of 3pbs by Molmil](/molmil-images/mine/3pbs) | Crystal structure of PBP3 complexed with aztreonam | 分子名称: | 2-({[(1Z)-1-(2-amino-1,3-thiazol-4-yl)-2-oxo-2-{[(2S,3S)-1-oxo-3-(sulfoamino)butan-2-yl]amino}ethylidene]amino}oxy)-2-methylpropanoic acid, Penicillin-binding protein 3 | 著者 | Han, S. | 登録日 | 2010-10-20 | 公開日 | 2010-12-22 | 最終更新日 | 2011-08-31 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structural basis for effectiveness of siderophore-conjugated monocarbams against clinically relevant strains of Pseudomonas aeruginosa. Proc.Natl.Acad.Sci.USA, 107, 2010
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3PBR
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![BU of 3pbr by Molmil](/molmil-images/mine/3pbr) | Crystal structure of PBP3 complexed with meropenem | 分子名称: | (4R,5S)-3-{[(3S,5S)-5-(dimethylcarbamoyl)pyrrolidin-3-yl]sulfanyl}-5-[(2S,3R)-3-hydroxy-1-oxobutan-2-yl]-4-methyl-4,5-dihydro-1H-pyrrole-2-carboxylic acid, Penicillin-binding protein 3 | 著者 | Han, S. | 登録日 | 2010-10-20 | 公開日 | 2010-12-22 | 最終更新日 | 2012-05-16 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Structural basis for effectiveness of siderophore-conjugated monocarbams against clinically relevant strains of Pseudomonas aeruginosa. Proc.Natl.Acad.Sci.USA, 107, 2010
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3PBQ
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![BU of 3pbq by Molmil](/molmil-images/mine/3pbq) | Crystal structure of PBP3 complexed with imipenem | 分子名称: | (5R)-5-[(1S,2R)-1-formyl-2-hydroxypropyl]-3-[(2-{[(E)-iminomethyl]amino}ethyl)sulfanyl]-4,5-dihydro-1H-pyrrole-2-carboxylic acid, Penicillin-binding protein 3 | 著者 | Han, S. | 登録日 | 2010-10-20 | 公開日 | 2010-12-22 | 最終更新日 | 2011-08-24 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Structural basis for effectiveness of siderophore-conjugated monocarbams against clinically relevant strains of Pseudomonas aeruginosa. Proc.Natl.Acad.Sci.USA, 107, 2010
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3PBO
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![BU of 3pbo by Molmil](/molmil-images/mine/3pbo) | Crystal structure of PBP3 complexed with ceftazidime | 分子名称: | ACYLATED CEFTAZIDIME, Penicillin-binding protein 3 | 著者 | Han, S. | 登録日 | 2010-10-20 | 公開日 | 2010-12-22 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.74 Å) | 主引用文献 | Structural basis for effectiveness of siderophore-conjugated monocarbams against clinically relevant strains of Pseudomonas aeruginosa. Proc.Natl.Acad.Sci.USA, 107, 2010
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3PBN
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![BU of 3pbn by Molmil](/molmil-images/mine/3pbn) | Crystal Structure of Apo PBP3 from Pseudomonas aeruginosa | 分子名称: | Penicillin-binding protein 3 | 著者 | Han, S. | 登録日 | 2010-10-20 | 公開日 | 2010-12-22 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structural basis for effectiveness of siderophore-conjugated monocarbams against clinically relevant strains of Pseudomonas aeruginosa. Proc.Natl.Acad.Sci.USA, 107, 2010
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3PAG
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![BU of 3pag by Molmil](/molmil-images/mine/3pag) | Crystal structure of the V130D mutant of OXA-24/40 in complex with doripenem | 分子名称: | (4R,5S)-5-[(2S,3R)-3-hydroxy-1-oxobutan-2-yl]-4-methyl-3-({(3S,5S)-5-[(sulfamoylamino)methyl]pyrrolidin-3-yl}sulfanyl)-4,5-dihydro-1H-pyrrole-2-carboxylic acid, Beta-lactamase, SULFATE ION | 著者 | Powers, R.A, Leonard, D.A, Schneider, K.D. | 登録日 | 2010-10-19 | 公開日 | 2011-01-19 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Structures of the Class D Carbapenemase OXA-24 from Acinetobacter baumannii in Complex with Doripenem. J.Mol.Biol., 406, 2011
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3PAE
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![BU of 3pae by Molmil](/molmil-images/mine/3pae) | Crystal structure of the K84D mutant of OXA-24/40 in complex with doripenem | 分子名称: | (4R,5S)-5-[(2S,3R)-3-hydroxy-1-oxobutan-2-yl]-4-methyl-3-({(3S,5S)-5-[(sulfamoylamino)methyl]pyrrolidin-3-yl}sulfanyl)-4,5-dihydro-1H-pyrrole-2-carboxylic acid, Beta-lactamase, SULFATE ION | 著者 | Powers, R.A, Leonard, D.A, Schneider, K.D. | 登録日 | 2010-10-19 | 公開日 | 2011-01-19 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structures of the Class D Carbapenemase OXA-24 from Acinetobacter baumannii in Complex with Doripenem. J.Mol.Biol., 406, 2011
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