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5BSB
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BU of 5bsb by Molmil
Lipomyces starkeyi levoglucosan kinase bound to levoglucosan
分子名称: Levoglucosan, Levoglucosan kinase, SULFATE ION
著者Bacik, J.P.
登録日2015-06-01
公開日2015-09-16
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Producing Glucose 6-Phosphate from Cellulosic Biomass: STRUCTURAL INSIGHTS INTO LEVOGLUCOSAN BIOCONVERSION.
J.Biol.Chem., 290, 2015
2F62
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BU of 2f62 by Molmil
Crystal structure of Nucleoside 2-deoxyribosyltransferase from Trypanosoma brucei at 1.5 A resolution with (2-ETHYLPHENYL)METHANOL bound
分子名称: (2-ETHYLPHENYL)METHANOL, GLYCEROL, Nucleoside 2-deoxyribosyltransferase, ...
著者Bosch, J, Robien, M.A, Hol, W.G.J, Structural Genomics of Pathogenic Protozoa Consortium (SGPP)
登録日2005-11-28
公開日2005-12-06
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Using fragment cocktail crystallography to assist inhibitor design of Trypanosoma brucei nucleoside 2-deoxyribosyltransferase.
J.Med.Chem., 49, 2006
4M2S
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BU of 4m2s by Molmil
Corrected Structure of Mouse P-glycoprotein bound to QZ59-RRR
分子名称: (4R,11R,18R)-4,11,18-tri(propan-2-yl)-6,13,20-triselena-3,10,17,22,23,24-hexaazatetracyclo[17.2.1.1~5,8~.1~12,15~]tetracosa-1(21),5(24),7,12(23),14,19(22)-hexaene-2,9,16-trione, Multidrug resistance protein 1A
著者Li, J, Jaimes, K.F, Aller, S.G.
登録日2013-08-05
公開日2013-11-13
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (4.4 Å)
主引用文献Refined structures of mouse P-glycoprotein.
Protein Sci., 23, 2014
2FKE
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BU of 2fke by Molmil
FK-506-BINDING PROTEIN: THREE-DIMENSIONAL STRUCTURE OF THE COMPLEX WITH THE ANTAGONIST L-685,818
分子名称: 8-DEETHYL-8-[BUT-3-ENYL]-ASCOMYCIN, FK506 BINDING PROTEIN
著者Becker, J.W, Mckeever, B.M, Rotonda, J.
登録日1993-01-27
公開日1994-01-31
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.72 Å)
主引用文献FK-506-binding protein: three-dimensional structure of the complex with the antagonist L-685,818.
J.Biol.Chem., 268, 1993
3AVT
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BU of 3avt by Molmil
Structure of viral RNA polymerase complex 1
分子名称: 3'-DEOXY-GUANOSINE-5'-TRIPHOSPHATE, CALCIUM ION, Elongation factor Ts, ...
著者Takeshita, D, Tomita, K.
登録日2011-03-08
公開日2012-01-18
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.607 Å)
主引用文献Molecular basis for RNA polymerization by Q beta replicase
Nat.Struct.Mol.Biol., 19, 2012
2SPZ
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BU of 2spz by Molmil
STAPHYLOCOCCAL PROTEIN A, Z-DOMAIN, NMR, 10 STRUCTURES
分子名称: IMMUNOGLOBULIN G BINDING PROTEIN A
著者Montelione, G.T, Tashiro, M, Tejero, R, Lyons, B.A.
登録日1998-07-29
公開日1998-08-05
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献High-resolution solution NMR structure of the Z domain of staphylococcal protein A.
J.Mol.Biol., 272, 1997
5A33
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BU of 5a33 by Molmil
Electron cryo-microscopy of Cowpea Mosaic Virus (CPMV) empty virus like particle (eVLP)
分子名称: RNA2 POLYPROTEIN
著者Hesketh, E.L, Meshcheriakova, Y, Dent, K.C, Saxena, P, Thompson, R, Cockburn, J.J, Lomonossoff, G.P, Ranson, N.A.
登録日2015-05-27
公開日2015-12-23
最終更新日2024-05-08
実験手法ELECTRON MICROSCOPY (3.04 Å)
主引用文献Mechanisms of assembly and genome packaging in an RNA virus revealed by high-resolution cryo-EM.
Nat Commun, 6, 2015
3AVU
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BU of 3avu by Molmil
Structure of viral RNA polymerase complex 2
分子名称: CALCIUM ION, Elongation factor Ts, Elongation factor Tu, ...
著者Takeshita, D, Tomita, K.
登録日2011-03-08
公開日2012-01-18
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.907 Å)
主引用文献Molecular basis for RNA polymerization by Q beta replicase
Nat.Struct.Mol.Biol., 19, 2012
3AVW
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BU of 3avw by Molmil
Structure of viral RNA polymerase complex 4
分子名称: 3'-DEOXY-GUANOSINE-5'-TRIPHOSPHATE, CALCIUM ION, Elongation factor Ts, ...
著者Takeshita, D, Tomita, K.
登録日2011-03-08
公開日2012-01-18
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.602 Å)
主引用文献Molecular basis for RNA polymerization by Q beta replicase
Nat.Struct.Mol.Biol., 19, 2012
3AV4
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BU of 3av4 by Molmil
Crystal structure of mouse DNA methyltransferase 1
分子名称: DNA (cytosine-5)-methyltransferase 1, ZINC ION
著者Takeshita, K, Suetake, I, Yamashita, E, Suga, M, Narita, H, Nakagawa, A, Tajima, S.
登録日2011-02-22
公開日2011-05-04
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.75 Å)
主引用文献Structural insight into maintenance methylation by mouse DNA methyltransferase 1 (Dnmt1).
Proc.Natl.Acad.Sci.USA, 108, 2011
3BLD
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BU of 3bld by Molmil
tRNA guanine transglycosylase V233G mutant preQ1 complex structure
分子名称: 7-DEAZA-7-AMINOMETHYL-GUANINE, GLYCEROL, Queuine tRNA-ribosyltransferase, ...
著者Tidten, N, Heine, A, Reuter, K, Klebe, G.
登録日2007-12-11
公開日2008-12-16
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (1.19 Å)
主引用文献Investigation of Specificity Determinants in Bacterial tRNA-Guanine Transglycosylase Reveals Queuine, the Substrate of Its Eucaryotic Counterpart, as Inhibitor
Plos One, 8, 2013
2GP6
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BU of 2gp6 by Molmil
X-ray crystal structure of Mycobacterium tuberculosis beta-ketoacyl acyl carrier protein synthase II (mtKasB)
分子名称: 3-oxoacyl-[acyl-carrier-protein] synthase 2
著者Sridharan, S, Sacchettini, J, TB Structural Genomics Consortium (TBSGC)
登録日2006-04-17
公開日2006-07-18
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献X-Ray Crystal Structure of Mycobacterium tuberculosis beta-Ketoacyl Acyl Carrier Protein Synthase II (mtKasB).
J.Mol.Biol., 366, 2007
7L6C
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BU of 7l6c by Molmil
Crystal Structure of Enoyl-[acyl-carrier-protein] reductase InhA from Mycobacterium abscessus in complex with NAD
分子名称: 1,2-ETHANEDIOL, Enoyl-[acyl-carrier-protein] reductase [NADH], NICOTINAMIDE-ADENINE-DINUCLEOTIDE, ...
著者Seattle Structural Genomics Center for Infectious Disease (SSGCID)
登録日2020-12-23
公開日2021-01-13
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Efficacy and Mode of Action of a Direct Inhibitor of Mycobacterium abscessus InhA.
Acs Infect Dis., 8, 2022
2F47
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BU of 2f47 by Molmil
Xray crystal structure of T4 lysozyme mutant L20/R63A liganded to methylguanidinium
分子名称: 1-METHYLGUANIDINE, BETA-MERCAPTOETHANOL, CHLORIDE ION, ...
著者Yousef, M.S, Bischoff, N, Dyer, C.M, Baase, W.A, Matthews, B.W.
登録日2005-11-22
公開日2006-04-25
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Guanidinium derivatives bind preferentially and trigger long-distance conformational changes in an engineered T4 lysozyme.
Protein Sci., 15, 2006
2UV0
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BU of 2uv0 by Molmil
Structure of the P. aeruginosa LasR ligand-binding domain bound to its autoinducer
分子名称: N-3-OXO-DODECANOYL-L-HOMOSERINE LACTONE, TRANSCRIPTIONAL ACTIVATOR PROTEIN LASR
著者Bottomley, M.J, Muraglia, E, Bazzo, R, Carfi, A.
登録日2007-03-08
公開日2007-03-27
最終更新日2019-07-24
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Molecular Insights Into Quorum Sensing in the Human Pathogen Pseudomonas Aeruginosa from the Structure of the Virulence Regulator Lasr Bound to its Autoinducer.
J.Biol.Chem., 282, 2007
2GVV
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BU of 2gvv by Molmil
Structure of diisopropyl fluorophosphatase (DFPase) in complex with dicyclopentylphosphoroamidate (DcPPA)
分子名称: CALCIUM ION, DICYCLOPENTYL PHOSPHORAMIDATE, Phosphotriesterase
著者Chen, J.C.H, Blum, M.M.
登録日2006-05-03
公開日2006-09-19
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.73 Å)
主引用文献Binding of a designed substrate analogue to diisopropyl fluorophosphatase: implications for the phosphotriesterase mechanism.
J.Am.Chem.Soc., 128, 2006
2GVU
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BU of 2gvu by Molmil
Crystal structure of diisopropyl fluorophosphatase (DFPase), mutant D229N / N120D
分子名称: CALCIUM ION, Phosphotriesterase
著者Chen, J.C.H, Blum, M.M.
登録日2006-05-03
公開日2006-09-19
最終更新日2021-10-20
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Binding of a designed substrate analogue to diisopropyl fluorophosphatase: implications for the phosphotriesterase mechanism.
J.Am.Chem.Soc., 128, 2006
2F67
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BU of 2f67 by Molmil
Crystal structure of Nucleoside 2-deoxyribosyltransferase from Trypanosoma brucei at 1.6 A resolution with BENZO[CD]INDOL-2(1H)-ONE bound
分子名称: BENZO[CD]INDOL-2(1H)-ONE, GLYCEROL, Nucleoside 2-deoxyribosyltransferase, ...
著者Bosch, J, Robien, M.A, Hol, W.G.J, Structural Genomics of Pathogenic Protozoa Consortium (SGPP)
登録日2005-11-28
公開日2005-12-06
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Using fragment cocktail crystallography to assist inhibitor design of Trypanosoma brucei nucleoside 2-deoxyribosyltransferase.
J.Med.Chem., 49, 2006
7KSL
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BU of 7ksl by Molmil
Substrate-free human mitochondrial LONP1
分子名称: ADENOSINE-5'-DIPHOSPHATE, Lon protease homolog, mitochondrial
著者Shin, M, Watson, E.R, Song, A.S, Mindrebo, J.T, Novick, S.R, Griffin, P, Wiseman, R.L, Lander, G.C.
登録日2020-11-23
公開日2020-12-09
最終更新日2024-05-29
実験手法ELECTRON MICROSCOPY (3.5 Å)
主引用文献Structures of the human LONP1 protease reveal regulatory steps involved in protease activation.
Nat Commun, 12, 2021
2OH5
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BU of 2oh5 by Molmil
The Crystal Structure of Infectious Cypovirus Polyhedra
分子名称: ADENOSINE-5'-TRIPHOSPHATE, CHLORIDE ION, CYTIDINE-5'-TRIPHOSPHATE, ...
著者Coulibaly, F, Chiu, E, Ikeda, K, Gutmann, S, Haebel, P.W, Schulze-Briese, C, Mori, H, Metcalf, P.
登録日2007-01-09
公開日2007-03-06
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.98 Å)
主引用文献The molecular organization of cypovirus polyhedra.
Nature, 446, 2007
4M1M
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BU of 4m1m by Molmil
Corrected Structure of Mouse P-glycoprotein
分子名称: MERCURY (II) ION, Multidrug resistance protein 1A
著者Li, J, Jaimes, K.F, Aller, S.G.
登録日2013-08-03
公開日2013-11-13
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (3.8 Å)
主引用文献Refined structures of mouse P-glycoprotein.
Protein Sci., 23, 2014
7KSM
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BU of 7ksm by Molmil
Human mitochondrial LONP1 with endogenous substrate
分子名称: ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, Lon protease homolog, ...
著者Shin, M, Watson, E.R, Song, A.S, Mindrebo, J.T, Novick, S.R, Griffin, P, Wiseman, R.L, Lander, G.C.
登録日2020-11-23
公開日2020-12-02
最終更新日2024-05-29
実験手法ELECTRON MICROSCOPY (3.2 Å)
主引用文献Structures of the human LONP1 protease reveal regulatory steps involved in protease activation.
Nat Commun, 12, 2021
7KRZ
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BU of 7krz by Molmil
Human mitochondrial LONP1 in complex with Bortezomib
分子名称: ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, Endogenous co-purified substrate, ...
著者Shin, M, Watson, E.R, Song, A.S, Mindrebo, J.T, Novick, S.R, Griffin, P, Wiseman, R.L, Lander, G.C.
登録日2020-11-20
公開日2021-02-24
最終更新日2022-06-15
実験手法ELECTRON MICROSCOPY (3.2 Å)
主引用文献Structures of the human LONP1 protease reveal regulatory steps involved in protease activation.
Nat Commun, 12, 2021
2GVW
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BU of 2gvw by Molmil
Structure of diisopropyl fluorophosphatase (DFPase) holoenzyme (RT)
分子名称: CALCIUM ION, Phosphotriesterase
著者Chen, J.C.H, Blum, M.M.
登録日2006-05-03
公開日2006-09-19
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.86 Å)
主引用文献Binding of a designed substrate analogue to diisopropyl fluorophosphatase: implications for the phosphotriesterase mechanism.
J.Am.Chem.Soc., 128, 2006
3AVX
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BU of 3avx by Molmil
Structure of viral RNA polymerase complex 5
分子名称: 3'-DEOXY-GUANOSINE-5'-TRIPHOSPHATE, CALCIUM ION, Elongation factor Ts, ...
著者Takeshita, D, Tomita, K.
登録日2011-03-08
公開日2012-01-18
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.406 Å)
主引用文献Molecular basis for RNA polymerization by Q beta replicase
Nat.Struct.Mol.Biol., 19, 2012

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