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2JB7
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PAE2307 with AMP
分子名称: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, ACETATE ION, ADENOSINE MONOPHOSPHATE, ...
著者Rajasekaran, K, Lott, J.S, Johnston, J.M.
登録日2006-12-04
公開日2008-08-05
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Pae2307 a Phosphotransferase
To be Published
2JB8
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Deacetoxycephalosporin C synthase complexed with 5-hydroxy-4-keto valeric acid
分子名称: 4,5-DIOXOPENTANOIC ACID, DEACETOXYCEPHALOSPORIN C SYNTHETASE, FE (III) ION
著者Cicero, G, Carbonera, C, Valegard, K, Hajdu, J, Andersson, I, Ranghino, G.
登録日2006-12-05
公開日2008-02-05
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.53 Å)
主引用文献Study of the Oxidative Half-Reaction Catalysed by a Non-Heme Ferrous Catalytic Centre by Means of Structural and Computational Methodologies
Int.J.Quantum Chem., 107, 2007
2JB9
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PhoB response regulator receiver domain constitutively-active double mutant D10A and D53E.
分子名称: PHOSPHATE REGULON TRANSCRIPTIONAL REGULATORY PROTEIN PHOB
著者Ferrer-Orta, C, Arribas-Bosacoma, R, Kim, S.-K, Blanco, A.G, Pereira, P.J.B, Gomis-Ruth, F.X, Wanner, B.L, Coll, M, Sola, M.
登録日2006-12-05
公開日2007-01-04
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献The X-Ray Crystal Structures of Two Constitutively Active Mutants of the E. Coli Phob Receiver Domain Give Insights Into Activation
J.Mol.Biol., 366, 2007
2JBA
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PhoB response regulator receiver domain constitutively-active double mutant D53A and Y102C.
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, PHOSPHATE REGULON TRANSCRIPTIONAL REGULATORY PROTEIN PHOB, SODIUM ION
著者Arribas-Bosacoma, R, Ferrer-Orta, C, Kim, S.-K, Blanco, A.G, Pereira, P.J.B, Gomis-Ruth, F.X, Wanner, B.L, Coll, M, Sola, M.
登録日2006-12-05
公開日2007-01-04
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献The X-Ray Crystal Structures of Two Constitutively Active Mutants of the Escherichia Coli Phob Receiver Domain Give Insights Into Activation.
J.Mol.Biol., 366, 2007
2JBF
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Structure of PBP-A, L158E mutant. Acyl-enzyme complex with penicillin- G.
分子名称: GLYCEROL, OPEN FORM - PENICILLIN G, TLL2115 PROTEIN
著者Evrard, C, Declercq, J.-P.
登録日2006-12-06
公開日2008-02-05
最終更新日2019-07-24
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structure of Pbp-A from Thermosynechococcus Elongatus, a Penicillin-Binding Protein Closely Related to Class a Beta-Lactamases.
J.Mol.Biol., 386, 2009
2JBG
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crystal structure of the mutant N560A of the nuclease domain of ColE7 in complex with Im7
分子名称: COLICIN E7, COLICIN-E7 IMMUNITY PROTEIN, SULFATE ION, ...
著者Huang, H, Yuan, H.S.
登録日2006-12-07
公開日2007-04-03
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献The Conserved Asparagine in the Hnh Motif Serves an Important Structural Role in Metal Finger Endonucleases.
J.Mol.Biol., 368, 2007
2JBH
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Human phosphoribosyl transferase domain containing 1
分子名称: CALCIUM ION, GUANOSINE-5'-MONOPHOSPHATE, PHOSPHATE ION, ...
著者Welin, M, Stenmark, P, Arrowsmith, C, Berglund, H, Busam, R, Collins, R, Edwards, A, Eklund, H, Ericsson, U.B, Flodin, S, Flores, A, Graslund, S, Hammarstrom, M, Hallberg, B.M, Holmberg Schiavone, L, Hogbom, M, Johansson, I, Karlberg, T, Kotenyova, T, Moche, M, Nilsson, M.E, Nyman, T, Ogg, D, Persson, C, Sagemark, J, Sundstrom, M, Uppenberg, J, Thorsell, A.G, Van Den Berg, S, Weigelt, J, Nordlund, P.
登録日2006-12-07
公開日2006-12-20
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structural and Functional Studies of the Human Phosphoribosyltransferase Domain Containing Protein 1.
FEBS J., 277, 2010
2JBJ
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membrane-bound glutamate carboxypeptidase II (GCPII) in complex with 2-PMPA (2-phosphonoMethyl-pentanedioic acid)
分子名称: (2S)-2-(PHOSPHONOMETHYL)PENTANEDIOIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Mesters, J.R, Henning, K, Hilgenfeld, R.
登録日2006-12-07
公開日2006-12-18
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.19 Å)
主引用文献Human Glutamate Carboxypeptidase II Inhibition: Structures of Gcpii in Complex with Two Potent Inhibitors, Quisqualate and 2-Pmpa.
Acta Crystallogr.,Sect.D, 63, 2007
2JBK
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membrane-bound glutamate carboxypeptidase II (GCPII) in complex with quisqualic acid (quisqualate, alpha-amino-3,5-dioxo-1,2,4- oxadiazolidine-2-propanoic acid)
分子名称: (S)-2-AMINO-3-(3,5-DIOXO-[1,2,4]OXADIAZOLIDIN-2-YL)-PROPIONIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Mesters, J.R, Henning, K, Hilgenfeld, R.
登録日2006-12-07
公開日2006-12-18
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.99 Å)
主引用文献Human Glutamate Carboxypeptidase II Inhibition: Structures of Gcpii in Complex with Two Potent Inhibitors, Quisqualate and 2-Pmpa.
Acta Crystallogr.,Sect.D, 63, 2007
2JBL
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PHOTOSYNTHETIC REACTION CENTER FROM BLASTOCHLORIS VIRIDIS
分子名称: 15-cis-1,2-dihydroneurosporene, BACTERIOCHLOROPHYLL B, BACTERIOPHEOPHYTIN B, ...
著者Lancaster, C.R.D.
登録日2006-12-08
公開日2007-03-13
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献A Comparison of Stigmatellin Conformations, Free and Bound to the Photosynthetic Reaction Center and the Cytochrome Bc(1) Complex.
J.Mol.Biol., 368, 2007
2JBM
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QPRTASE STRUCTURE FROM HUMAN
分子名称: NICOTINATE-NUCLEOTIDE PYROPHOSPHORYLASE, S,R MESO-TARTARIC ACID
著者Liu, H, Naismith, J.H.
登録日2006-12-08
公開日2007-11-13
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural and Kinetic Characterization of Quinolinate Phosphoribosyltransferase (Hqprtase) from Homo Sapiens.
J.Mol.Biol., 373, 2007
2JBO
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Protein kinase MK2 in complex with an inhibitor (crystal form-1, soaking)
分子名称: 2-(2-QUINOLIN-3-YLPYRIDIN-4-YL)-1,5,6,7-TETRAHYDRO-4H-PYRROLO[3,2-C]PYRIDIN-4-ONE, MAP KINASE-ACTIVATED PROTEIN KINASE 2, PHOSPHATE ION
著者Hillig, R.C, Eberspaecher, U, Monteclaro, F, Huber, M, Nguyen, D, Mengel, A, Muller-Tiemann, B, Egner, U.
登録日2006-12-09
公開日2007-03-20
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Structural Basis for a High Affinity Inhibitor Bound to Protein Kinase Mk2.
J.Mol.Biol., 369, 2007
2JBP
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Protein kinase MK2 in complex with an inhibitor (crystal form-2, co- crystallization)
分子名称: 2-(2-QUINOLIN-3-YLPYRIDIN-4-YL)-1,5,6,7-TETRAHYDRO-4H-PYRROLO[3,2-C]PYRIDIN-4-ONE, MAP KINASE-ACTIVATED PROTEIN KINASE 2
著者Hillig, R.C, Eberspaecher, U, Monteclaro, F, Huber, M, Nguyen, D, Mengel, A, Muller-Tiemann, B, Egner, U.
登録日2006-12-09
公開日2007-03-20
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (3.31 Å)
主引用文献Structural basis for a high affinity inhibitor bound to protein kinase MK2.
J. Mol. Biol., 369, 2007
2JBR
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Structure of the monooxygenase component of p-hydroxyphenylacetate hydroxylase from Acinetobacter baumanni
分子名称: P-HYDROXYPHENYLACETATE HYDROXYLASE C2 OXYGENASE COMPONENT
著者Alfieri, A, Mattevi, A.
登録日2006-12-11
公開日2007-01-23
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structure of the Monooxygenase Component of a Two-Component Flavoprotein Monooxygenase.
Proc.Natl.Acad.Sci.USA, 104, 2007
2JBS
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Structure of the monooxygenase component of p-hydroxyphenylacetate hydroxylase from Acinetobacter baumannii
分子名称: FLAVIN MONONUCLEOTIDE, P-HYDROXYPHENYLACETATE HYDROXYLASE C2:OXYGENASE COMPONENT
著者Alfieri, A, Mattevi, A.
登録日2006-12-11
公開日2007-01-23
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structure of the Monooxygenase Component of a Two-Component Flavoprotein Monooxygenase.
Proc.Natl.Acad.Sci.USA, 104, 2007
2JBT
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Structure of the monooxygenase component of p-hydroxyphenylacetate hydroxylase from Acinetobacter baumannii
分子名称: 4-HYDROXYPHENYLACETATE, FLAVIN MONONUCLEOTIDE, P-HYDROXYPHENYLACETATE HYDROXYLASE C2:OXYGENASE COMPONENT
著者Alfieri, A, Mattevi, A.
登録日2006-12-11
公開日2007-01-23
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structure of the Monooxygenase Component of a Two-Component Flavoprotein Monooxygenase.
Proc.Natl.Acad.Sci.USA, 104, 2007
2JBU
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Crystal structure of human insulin degrading enzyme complexed with co- purified peptides.
分子名称: 1,4-DIETHYLENE DIOXIDE, CO-PURIFIED PEPTIDE, INSULIN-DEGRADING ENZYME
著者Im, H, Shen, Y, Tang, W.J.
登録日2006-12-11
公開日2007-07-03
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Structure of Substrate-Free Human Insulin Degrading Enzyme (Ide) and Biophysical Analysis of ATP-Induced Conformational Switch of Ide
J.Biol.Chem., 282, 2007
2JBV
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Crystal structure of choline oxidase reveals insights into the catalytic mechanism
分子名称: CHOLINE OXIDASE, DIMETHYL SULFOXIDE, UNKNOWN ATOM OR ION, ...
著者Lountos, G.T, Fan, F, Gadda, G, Orville, A.M.
登録日2006-12-13
公開日2007-12-25
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.86 Å)
主引用文献Role of Glu312 in Binding and Positioning of the Substrate for the Hydride Transfer Reaction in Choline Oxidase.
Biochemistry, 47, 2008
2JBW
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Crystal Structure of the 2,6-dihydroxy-pseudo-oxynicotine Hydrolase.
分子名称: 2,6-DIHYDROXY-PSEUDO-OXYNICOTINE HYDROLASE, SODIUM ION
著者Schleberger, C, Sachelaru, P, Brandsch, R, Schulz, G.E.
登録日2006-12-14
公開日2007-01-04
最終更新日2019-05-08
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Structure and Action of a Cc Bond Cleaving Alpha/Beta-Hydrolase Involved in Nicotine Degration.
J.Mol.Biol., 367, 2007
2JBX
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Crystal Structure of the myxoma virus anti-apoptotic protein M11L
分子名称: M11L PROTEIN
著者Kvansakul, M, Van Delft, M.F, Lee, E.F, Gulbis, J.M, Fairlie, W.D, Huang, D.C.S, Colman, P.M.
登録日2006-12-14
公開日2007-03-27
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (2.73 Å)
主引用文献A Structural Viral Mimic of Prosurvival Bcl-2: A Pivotal Role for Sequestering Proapoptotic Bax and Bak.
Mol.Cell, 25, 2007
2JBY
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A viral protein unexpectedly mimics the structure and function of pro- survival Bcl-2
分子名称: BCL-2 HOMOLOGOUS ANTAGONIST/KILLER 2, M11L PROTEIN, SODIUM ION
著者Kvansakul, M, Van Delft, M.F, Lee, E.F, Gulbis, J.M, Fairlie, W.D, Huang, D.C.S, Colman, P.M.
登録日2006-12-14
公開日2007-03-27
最終更新日2018-06-13
実験手法X-RAY DIFFRACTION (2.41 Å)
主引用文献A structural viral mimic of prosurvival Bcl-2: a pivotal role for sequestering proapoptotic Bax and Bak.
Mol. Cell, 25, 2007
2JBZ
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Crystal structure of the Streptomyces coelicolor holo-[Acyl-carrier-protein] Synthase (AcpS) in complex with coenzyme A at 1.6 A
分子名称: COENZYME A, HOLO-[ACYL-CARRIER-PROTEIN] SYNTHASE, MAGNESIUM ION, ...
著者Dall'Aglio, P, Arthur, C, Law, C.K.E, Crump, M.P, Crosby, J, Hadfield, A.T.
登録日2006-12-15
公開日2007-01-23
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (1.62 Å)
主引用文献Analysis of Streptomyces Coelicolor Phosphopantetheinyl Transferase, Acps, Reveals the Basis for Relaxed Substrate Specificity.
Biochemistry, 50, 2011
2JC0
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CRYSTAL STRUCTURE OF HEPATITIS C VIRUS POLYMERASE IN COMPLEX WITH INHIBITOR SB655264
分子名称: (2S,4S,5R)-2-ISOBUTYL-5-(2-THIENYL)-1-[4-(TRIFLUOROMETHYL)BENZOYL]PYRROLIDINE-2,4-DICARBOXYLIC ACID, RNA-DEPENDENT RNA-POLYMERASE
著者Wonacott, A, Skarzynski, T, Singh, O.M.
登録日2006-12-18
公開日2007-02-13
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Optimization of Novel Acyl Pyrrolidine Inhibitors of Hepatitis C Virus RNA-Dependent RNA Polymerase Leading to a Development Candidate.
J.Med.Chem., 50, 2007
2JC1
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CRYSTAL STRUCTURE OF HEPATITIS C VIRUS POLYMERASE IN COMPLEX WITH INHIBITOR SB698223
分子名称: (2S,4S,5R)-1-(4-TERT-BUTYLBENZOYL)-2-ISOBUTYL-5-(1,3-THIAZOL-2-YL)PYRROLIDINE-2,4-DICARBOXYLIC ACID, RNA-DEPENDENT RNA-POLYMERASE
著者Wonacott, A, Skarzynski, T, Singh, O.M.
登録日2006-12-18
公開日2007-02-13
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Optimization of Novel Acyl Pyrrolidine Inhibitors of Hepatitis C Virus RNA-Dependent RNA Polymerase Leading to a Development Candidate.
J.Med.Chem., 50, 2007
2JC2
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The crystal structure of the natural F112L human sorcin mutant
分子名称: SORCIN, SULFATE ION
著者Franceschini, S, Ilari, A, Colotti, G, Chiancone, E.
登録日2006-12-19
公開日2007-08-28
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Molecular Basis for the Impaired Function of the Natural F112L Sorcin Mutant: X-Ray Crystal Structure, Calcium Affinity, and Interaction with Annexin Vii and the Ryanodine Receptor.
Faseb J., 22, 2008

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