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8EV8
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BU of 8ev8 by Molmil
Cryo-EM structure of cGMP bound truncated human CNGA3/CNGB3 channel in lipid nanodisc, closed state
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, CYCLIC GUANOSINE MONOPHOSPHATE, Cyclic nucleotide-gated cation channel alpha-3, ...
著者Hu, Z, Yang, J.
登録日2022-10-20
公開日2023-08-09
実験手法ELECTRON MICROSCOPY (3.11 Å)
主引用文献Conformational trajectory of allosteric gating of the human cone photoreceptor cyclic nucleotide-gated channel.
Nat Commun, 14, 2023
8EVC
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BU of 8evc by Molmil
Cryo-EM structure of cGMP bound truncated human CNGA3/CNGB3 channel in lipid nanodisc, open state
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, CYCLIC GUANOSINE MONOPHOSPHATE, Cyclic nucleotide-gated cation channel alpha-3, ...
著者Hu, Z, Yang, J.
登録日2022-10-20
公開日2023-08-09
実験手法ELECTRON MICROSCOPY (3.33 Å)
主引用文献Conformational trajectory of allosteric gating of the human cone photoreceptor cyclic nucleotide-gated channel.
Nat Commun, 14, 2023
4BW9
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BU of 4bw9 by Molmil
PylRS Y306G, Y384F, I405R mutant in complex with AMP-PNP
分子名称: 1,2-ETHANEDIOL, MAGNESIUM ION, PENTAETHYLENE GLYCOL, ...
著者Schneider, S, Vrabel, M, Gattner, M.J, Fluegel, V, Lopez-Carillo, V, Carell, T.
登録日2013-07-01
公開日2013-07-31
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Structural Insights Into Incorporation of Norbornene Amino Acids for Click Modification of Proteins
Chem.Bio.Chem., 14, 2013
4BR3
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BU of 4br3 by Molmil
Determination of potential scaffolds for human choline kinase alpha 1 by chemical deconvolution studies
分子名称: 1-((4'-((6-amino-3H-purin-3-yl)methyl)biphenyl-4-yl)methyl)-4-(dimethylamino)pyridinium, 3-benzyladenine, CHOLINE KINASE ALPHA, ...
著者Sahun-Roncero, M, Rubio-Ruiz, B, Conejo-Garcia, A, Velazquez-Campoy, A, Entrena, A, Hurtado-Guerrero, R.
登録日2013-06-03
公開日2013-06-19
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Determination of Potential Scaffolds for Human Choline Kinase Alpha 1 by Chemical Deconvolution Studies
Chembiochem, 14, 2013
8ERC
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BU of 8erc by Molmil
Human Membrane-bound O-acyltransferase 7
分子名称: Lysophospholipid acyltransferase 7
著者Wang, K, Liao, M, Farese, R.V, Walther, T.C.
登録日2022-10-11
公開日2023-09-27
実験手法ELECTRON MICROSCOPY (3.7 Å)
主引用文献The structure of phosphatidylinositol remodeling MBOAT7 reveals its catalytic mechanism and enables inhibitor identification.
Nat Commun, 14, 2023
8ELI
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BU of 8eli by Molmil
Broadly neutralizing antibody VRC34-combo.1 in complex with HIV fusion peptide (residue 512-519)
分子名称: Fusion peptide, VRC34-combo.1 Fab Heavy chain, VRC34-combo.1 Fab Light chain
著者Xu, K, Kwong, P.D.
登録日2022-09-24
公開日2023-09-27
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.49 Å)
主引用文献Antibody-directed evolution reveals a mechanism for enhanced neutralization at the HIV-1 fusion peptide site.
Nat Commun, 14, 2023
8EUV
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BU of 8euv by Molmil
Cryo-EM structure of HIV-1 BG505 DS-SOSIP ENV trimer bound to VRC34.01-COMBO1 FAB
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Envelope glycoprotein gp120, ...
著者Pletnev, S, Kwong, P.
登録日2022-10-19
公開日2023-09-27
最終更新日2024-02-14
実験手法ELECTRON MICROSCOPY (2.6 Å)
主引用文献Antibody-directed evolution reveals a mechanism for enhanced neutralization at the HIV-1 fusion peptide site.
Nat Commun, 14, 2023
2MPS
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BU of 2mps by Molmil
Structure of complex of MDM2(3-109) and P73 TAD(10-25)
分子名称: E3 ubiquitin-protein ligase Mdm2, Tumor protein p73
著者Shin, J.S, Ha, J.H, Chi, S.W.
登録日2014-06-02
公開日2015-06-03
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Structural convergence of unstructured p53 family transactivation domains in MDM2 recognition
Cell Cycle, 14, 2015
8EUW
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BU of 8euw by Molmil
Cryo-EM structure of HIV-1 BG505 DS-SOSIP ENV trimer bound to VRC34.01-MM28 FAB
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Envelope glycoprotein gp120, ...
著者Pletnev, S, Kwong, P.
登録日2022-10-19
公開日2023-09-27
最終更新日2024-02-14
実験手法ELECTRON MICROSCOPY (2.7 Å)
主引用文献Antibody-directed evolution reveals a mechanism for enhanced neutralization at the HIV-1 fusion peptide site.
Nat Commun, 14, 2023
8EUU
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BU of 8euu by Molmil
Cryo-EM structure of HIV-1 BG505 DS-SOSIP ENV trimer bound to VRC34.01 FAB
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Envelope glycoprotein gp120, ...
著者Pletnev, S, Kwong, P.
登録日2022-10-19
公開日2023-09-27
最終更新日2024-02-14
実験手法ELECTRON MICROSCOPY (2.7 Å)
主引用文献Antibody-directed evolution reveals a mechanism for enhanced neutralization at the HIV-1 fusion peptide site.
Nat Commun, 14, 2023
8F5I
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BU of 8f5i by Molmil
SARS-CoV-2 S2 helix epitope scaffold bound by antibody DH1057.1
分子名称: DH1057.1 HC, DH1057.1 LC, Specialized acyl carrier protein, ...
著者Kapingidza, A.B, Wrapp, D, Winters, K, Azoitei, M.L.
登録日2022-11-14
公開日2023-10-11
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Engineered immunogens to elicit antibodies against conserved coronavirus epitopes.
Nat Commun, 14, 2023
3ZD6
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BU of 3zd6 by Molmil
Snapshot 1 of RIG-I scanning on RNA duplex
分子名称: PROBABLE ATP-DEPENDENT RNA HELICASE DDX58, RNA DUPLEX, ZINC ION
著者Luo, D, Pyle, A.M.
登録日2012-11-25
公開日2013-08-07
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Defining the Functional Determinants for RNA Surveillance by Rig-I.
Embo Rep., 14, 2013
8F5H
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BU of 8f5h by Molmil
SARS-CoV-2 S2 helix epitope scaffold
分子名称: S2hlx_EX_19
著者Kapingidza, A.B, Wrapp, D, Winters, K, Azoitei, M.L.
登録日2022-11-14
公開日2023-10-11
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Engineered immunogens to elicit antibodies against conserved coronavirus epitopes.
Nat Commun, 14, 2023
8EI9
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BU of 8ei9 by Molmil
Crystal structure of beta-catenin and the MDM2 p53-binding domain in complex with H332, a Helicon Polypeptide
分子名称: Catenin beta-1, E3 ubiquitin-protein ligase Mdm2, H332, ...
著者Li, K, Travaline, T.L, Swiecicki, J.-M, Tokareva, O.S, Thomson, T.M, Verdine, G.L, McGee, J.H.
登録日2022-09-14
公開日2023-10-25
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (3.9 Å)
主引用文献Recognition and reprogramming of E3 ubiquitin ligase surfaces by alpha-helical peptides.
Nat Commun, 14, 2023
8EI8
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BU of 8ei8 by Molmil
Crystal structure of the WWP2 HECT domain in complex with H308, a Helicon Polypeptide
分子名称: 1,2-ETHANEDIOL, H308, N,N'-(1,4-phenylene)diacetamide, ...
著者Li, K, Tokareva, O.S, Thomson, T.M, Verdine, G.L, McGee, J.H.
登録日2022-09-14
公開日2023-10-25
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Recognition and reprogramming of E3 ubiquitin ligase surfaces by alpha-helical peptides.
Nat Commun, 14, 2023
8EI1
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BU of 8ei1 by Molmil
Crystal structure of the N-terminal domain of CUL4B in complex with H316, a Helicon Polypeptide
分子名称: Cullin-4B, H316, N,N'-(1,4-phenylene)diacetamide
著者Li, K, Tokareva, O.S, Thomson, T.M, Verdine, G.L, McGee, J.H.
登録日2022-09-14
公開日2023-10-25
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.89 Å)
主引用文献Recognition and reprogramming of E3 ubiquitin ligase surfaces by alpha-helical peptides.
Nat Commun, 14, 2023
8EI7
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BU of 8ei7 by Molmil
Crystal structure of the WWP2 HECT domain in complex with H304, a Helicon Polypeptide
分子名称: 1,2-ETHANEDIOL, DI(HYDROXYETHYL)ETHER, GLYCEROL, ...
著者Li, K, Tokareva, O.S, Thomson, T.M, Verdine, G.L, McGee, J.H.
登録日2022-09-14
公開日2023-10-25
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.22 Å)
主引用文献Recognition and reprogramming of E3 ubiquitin ligase surfaces by alpha-helical peptides.
Nat Commun, 14, 2023
8ETQ
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BU of 8etq by Molmil
Designed pentafoil knot protein folded into a trefoil knot
分子名称: k-cTRP5
著者Doyle, L.A, Kibler, R.D, Bradley, P, Stoddard, B.L.
登録日2022-10-17
公開日2023-10-25
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.42 Å)
主引用文献De novo design of knotted tandem repeat proteins.
Nat Commun, 14, 2023
8EI2
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BU of 8ei2 by Molmil
Crystal structure of the N-terminal domain of CUL5 in complex with H314, a Helicon Polypeptide
分子名称: Cullin-5, H314, N,N'-(1,4-phenylene)diacetamide
著者Li, K, Tokareva, O.S, Thomson, T.M, Verdine, G.L, McGee, J.H.
登録日2022-09-14
公開日2023-10-25
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Recognition and reprogramming of E3 ubiquitin ligase surfaces by alpha-helical peptides.
Nat Commun, 14, 2023
8EIC
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BU of 8eic by Molmil
Crystal structure of beta-catenin and the MDM2 p53-binding domain in complex with H330, a Helicon Polypeptide
分子名称: Catenin beta-1, E3 ubiquitin-protein ligase Mdm2, H330, ...
著者Li, K, Travaline, T.L, Swiecicki, J.-M, Tokareva, O.S, Thomson, T.M, Verdine, G.L, McGee, J.H.
登録日2022-09-14
公開日2023-10-25
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.62 Å)
主引用文献Recognition and reprogramming of E3 ubiquitin ligase surfaces by alpha-helical peptides.
Nat Commun, 14, 2023
8EIB
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BU of 8eib by Molmil
Crystal structure of beta-catenin and the MDM2 p53-binding domain in complex with H329, a Helicon Polypeptide
分子名称: Catenin beta-1, E3 ubiquitin-protein ligase Mdm2, H329, ...
著者Li, K, Travaline, T.L, Swiecicki, J.-M, Tokareva, O.S, Thomson, T.M, Verdine, G.L, McGee, J.H.
登録日2022-09-14
公開日2023-10-25
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (3.76 Å)
主引用文献Recognition and reprogramming of E3 ubiquitin ligase surfaces by alpha-helical peptides.
Nat Commun, 14, 2023
8EHZ
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BU of 8ehz by Molmil
Crystal structure of the STUB1 TPR domain in complex with H317, a Helicon Polypeptide
分子名称: E3 ubiquitin-protein ligase CHIP, H317, N,N'-(1,4-phenylene)diacetamide
著者Li, K, Swiecicki, J.-M, Tokareva, O.S, Thomson, T.M, Verdine, G.L, McGee, J.H.
登録日2022-09-14
公開日2023-10-25
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.06 Å)
主引用文献Recognition and reprogramming of E3 ubiquitin ligase surfaces by alpha-helical peptides.
Nat Commun, 14, 2023
8EI0
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BU of 8ei0 by Molmil
Crystal structure of the STUB1 TPR domain in complex with H318, a Helicon Polypeptide
分子名称: 1,2-ETHANEDIOL, E3 ubiquitin-protein ligase CHIP, H318, ...
著者Li, K, Swiecicki, J.-M, Tokareva, O.S, Thomson, T.M, Verdine, G.L, McGee, J.H.
登録日2022-09-14
公開日2023-10-25
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.47 Å)
主引用文献Recognition and reprogramming of E3 ubiquitin ligase surfaces by alpha-helical peptides.
Nat Commun, 14, 2023
8EI3
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BU of 8ei3 by Molmil
Crystal structure of VHL in complex with H313, a Helicon Polypeptide
分子名称: Elongin-B, Elongin-C, H313, ...
著者Li, K, Tokareva, O.S, Thomson, T.M, Verdine, G.L, McGee, J.H.
登録日2022-09-14
公開日2023-10-25
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (3.49 Å)
主引用文献Recognition and reprogramming of E3 ubiquitin ligase surfaces by alpha-helical peptides.
Nat Commun, 14, 2023
8EI6
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BU of 8ei6 by Molmil
Crystal structure of the WWP2 HECT domain in complex with H305, a Helicon Polypeptide
分子名称: H305, N,N'-(1,4-phenylene)diacetamide, NEDD4-like E3 ubiquitin-protein ligase WWP2
著者Li, K, Tokareva, O.S, Thomson, T.M, Verdine, G.L, McGee, J.H.
登録日2022-09-14
公開日2023-10-25
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (3.62 Å)
主引用文献Recognition and reprogramming of E3 ubiquitin ligase surfaces by alpha-helical peptides.
Nat Commun, 14, 2023

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件を2024-09-11に公開中

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