3V4O
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3V6L
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![BU of 3v6l by Molmil](/molmil-images/mine/3v6l) | Crystal Structure of caspase-6 inactivation mutation | 分子名称: | Caspase-6 | 著者 | Cao, Q, Wang, X.J, Liu, D.F, Li, L.F, Su, X.D. | 登録日 | 2011-12-20 | 公開日 | 2012-03-28 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Inhibitory mechanism of caspase-6 phosphorylation revealed by crystal structures, molecular dynamics simulations, and biochemical assays J.Biol.Chem., 287, 2012
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3V6M
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![BU of 3v6m by Molmil](/molmil-images/mine/3v6m) | Inhibition of caspase-6 activity by single mutation outside the active site | 分子名称: | Caspase-6 | 著者 | Cao, Q, Wang, X.J, Liu, D.F, Li, L.F, Su, X.D. | 登録日 | 2011-12-20 | 公開日 | 2012-03-28 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.692 Å) | 主引用文献 | Inhibitory mechanism of caspase-6 phosphorylation revealed by crystal structures, molecular dynamics simulations, and biochemical assays J.Biol.Chem., 287, 2012
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6BFJ
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![BU of 6bfj by Molmil](/molmil-images/mine/6bfj) | Caspase-3 Mutant - T245D,S249D | 分子名称: | AZIDE ION, Ac-Asp-Glu-Val-Asp-CMK, Caspase-3 | 著者 | Thomas, M.E, Grinshpon, R, Swartz, P.D, Clark, A.C. | 登録日 | 2017-10-26 | 公開日 | 2018-02-21 | 最終更新日 | 2018-04-25 | 実験手法 | X-RAY DIFFRACTION (1.543 Å) | 主引用文献 | Modifications to a common phosphorylation network provide individualized control in caspases. J. Biol. Chem., 293, 2018
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6BG0
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![BU of 6bg0 by Molmil](/molmil-images/mine/6bg0) | Caspase-3 Mutant - D9A,D28A,S150D | 分子名称: | AC-ASP-GLU-VAL-ASP-CMK, AZIDE ION, Caspase-3, ... | 著者 | Thomas, M.E, Grinshpon, R, Swartz, P.D, Clark, A.C. | 登録日 | 2017-10-27 | 公開日 | 2018-02-21 | 最終更新日 | 2018-04-25 | 実験手法 | X-RAY DIFFRACTION (2.125 Å) | 主引用文献 | Modifications to a common phosphorylation network provide individualized control in caspases. J. Biol. Chem., 293, 2018
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6BFL
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![BU of 6bfl by Molmil](/molmil-images/mine/6bfl) | Caspase-3 Mutant- D9A,D28A,T245D | 分子名称: | AC-ASP-GLU-VAL-ASP-CMK, AZIDE ION, Caspase-3 | 著者 | Thomas, M.E, Grinshpon, R, Swartz, P.D, Clark, A.C. | 登録日 | 2017-10-26 | 公開日 | 2018-02-21 | 最終更新日 | 2018-04-25 | 実験手法 | X-RAY DIFFRACTION (1.87 Å) | 主引用文献 | Modifications to a common phosphorylation network provide individualized control in caspases. J. Biol. Chem., 293, 2018
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6BFO
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![BU of 6bfo by Molmil](/molmil-images/mine/6bfo) | Caspase-3 Mutant- T245D | 分子名称: | AC-ASP-GLU-VAL-ASP-CMK, AZIDE ION, Caspase-3, ... | 著者 | Thomas, M.E, Grinshpon, R, Swartz, P.D, Clark, A.C. | 登録日 | 2017-10-26 | 公開日 | 2018-02-21 | 最終更新日 | 2018-04-25 | 実験手法 | X-RAY DIFFRACTION (1.54 Å) | 主引用文献 | Modifications to a common phosphorylation network provide individualized control in caspases. J. Biol. Chem., 293, 2018
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6BG4
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![BU of 6bg4 by Molmil](/molmil-images/mine/6bg4) | Caspase-3 Mutant- T152D | 分子名称: | AC-ASP-GLU-VAL-ASP-CMK, AZIDE ION, CHLORIDE ION, ... | 著者 | Thomas, M.E, Grinshpon, R, Swartz, P.D, Clark, A.C. | 登録日 | 2017-10-27 | 公開日 | 2018-02-21 | 最終更新日 | 2018-04-25 | 実験手法 | X-RAY DIFFRACTION (1.87 Å) | 主引用文献 | Modifications to a common phosphorylation network provide individualized control in caspases. J. Biol. Chem., 293, 2018
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6BFK
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![BU of 6bfk by Molmil](/molmil-images/mine/6bfk) | Caspase-3 Mutant- T245A | 分子名称: | AC-ASP-GLU-VAL-ASP-CMK, Caspase-3, SODIUM ION | 著者 | Thomas, M.E, Grinshpon, R, Swartz, P.D, Clark, A.C. | 登録日 | 2017-10-26 | 公開日 | 2018-02-21 | 最終更新日 | 2018-04-25 | 実験手法 | X-RAY DIFFRACTION (1.753 Å) | 主引用文献 | Modifications to a common phosphorylation network provide individualized control in caspases. J. Biol. Chem., 293, 2018
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6BDV
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![BU of 6bdv by Molmil](/molmil-images/mine/6bdv) | Crystal structure of Caspase 3 S150A | 分子名称: | AZIDE ION, Acetyl-Asp-Glu-Val-Asp-CMK, CHLORIDE ION, ... | 著者 | Thomas, M.E, Grinshpon, R, Swartz, P.D, Clark, A.C. | 登録日 | 2017-10-24 | 公開日 | 2018-02-14 | 最終更新日 | 2018-04-25 | 実験手法 | X-RAY DIFFRACTION (1.938 Å) | 主引用文献 | Modifications to a common phosphorylation network provide individualized control in caspases. J. Biol. Chem., 293, 2018
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6BG1
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![BU of 6bg1 by Molmil](/molmil-images/mine/6bg1) | Caspase-3 Mutant - D9A,D28A,S150E | 分子名称: | AC-ASP-GLU-VAL-ASP-CMK, Caspase-3, SODIUM ION | 著者 | Thomas, M.E, Grinshpon, R, Swartz, P.D, Clark, A.C. | 登録日 | 2017-10-27 | 公開日 | 2018-02-21 | 最終更新日 | 2018-04-25 | 実験手法 | X-RAY DIFFRACTION (1.88 Å) | 主引用文献 | Modifications to a common phosphorylation network provide individualized control in caspases. J. Biol. Chem., 293, 2018
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6BGR
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![BU of 6bgr by Molmil](/molmil-images/mine/6bgr) | Caspase-3 Mutant - S150E | 分子名称: | AZIDE ION, Ac-Asp-Glu-Val-Asp-CMK, Caspase-3 | 著者 | Thomas, M.E, Grinshpon, R, Swartz, P.D, Clark, A.C. | 登録日 | 2017-10-29 | 公開日 | 2018-02-21 | 最終更新日 | 2018-04-25 | 実験手法 | X-RAY DIFFRACTION (2.16 Å) | 主引用文献 | Modifications to a common phosphorylation network provide individualized control in caspases. J. Biol. Chem., 293, 2018
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6CL0
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6CL1
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6BH9
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![BU of 6bh9 by Molmil](/molmil-images/mine/6bh9) | Caspase-3 Mutant - T152A | 分子名称: | Ac-Asp-Glu-Val-Asp-CMK, CHLORIDE ION, Caspase-3, ... | 著者 | Thomas, M.E, Grinshpon, R, Swartz, P.D, Clark, A.C. | 登録日 | 2017-10-30 | 公開日 | 2018-02-21 | 最終更新日 | 2018-04-25 | 実験手法 | X-RAY DIFFRACTION (1.94 Å) | 主引用文献 | Modifications to a common phosphorylation network provide individualized control in caspases. J. Biol. Chem., 293, 2018
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6BGS
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![BU of 6bgs by Molmil](/molmil-images/mine/6bgs) | Caspase-3 Mutant - S150Y | 分子名称: | Ac-Asp-Glu-Val-Asp-CMK, Caspase-3 | 著者 | Thomas, M.E, Grinshpon, R, Swartz, P.D, Clark, A.C. | 登録日 | 2017-10-29 | 公開日 | 2018-02-21 | 最終更新日 | 2018-04-25 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Modifications to a common phosphorylation network provide individualized control in caspases. J. Biol. Chem., 293, 2018
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6CL2
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6CKZ
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6BGQ
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![BU of 6bgq by Molmil](/molmil-images/mine/6bgq) | Caspase-3 Mutant - S150D | 分子名称: | AZIDE ION, Ac-Asp-Glu-Val-Asp-CMK, CHLORIDE ION, ... | 著者 | Thomas, M.E, Grinshpon, R, Swartz, P.D, Clark, A.C. | 登録日 | 2017-10-29 | 公開日 | 2018-02-21 | 最終更新日 | 2018-04-25 | 実験手法 | X-RAY DIFFRACTION (1.97 Å) | 主引用文献 | Modifications to a common phosphorylation network provide individualized control in caspases. J. Biol. Chem., 293, 2018
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6BHA
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![BU of 6bha by Molmil](/molmil-images/mine/6bha) | Caspase-3 Mutant - T152V | 分子名称: | Ac-Asp-Glu-Val-Asp-CMK, Caspase-3 | 著者 | Thomas, M.E, Grinshpon, R, Swartz, P.D, Clark, A.C. | 登録日 | 2017-10-30 | 公開日 | 2018-02-21 | 最終更新日 | 2018-04-25 | 実験手法 | X-RAY DIFFRACTION (1.603 Å) | 主引用文献 | Modifications to a common phosphorylation network provide individualized control in caspases. J. Biol. Chem., 293, 2018
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6BGK
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![BU of 6bgk by Molmil](/molmil-images/mine/6bgk) | Caspase-3 Mutant- D9A,D28A,T152D | 分子名称: | ACE-ASP-GLU-VAL-ASP-0QE, AZIDE ION, CHLORIDE ION, ... | 著者 | Thomas, M.E, Grinshpon, R, Swartz, P.D, Clark, A.C. | 登録日 | 2017-10-28 | 公開日 | 2018-02-21 | 最終更新日 | 2018-04-25 | 実験手法 | X-RAY DIFFRACTION (1.87 Å) | 主引用文献 | Modifications to a common phosphorylation network provide individualized control in caspases. J. Biol. Chem., 293, 2018
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6BZ9
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![BU of 6bz9 by Molmil](/molmil-images/mine/6bz9) | Crystal structure of human caspase-1 in complex with Ac-FLTD-CMK | 分子名称: | Ac-FLTD-CMK, Caspase-1, DI(HYDROXYETHYL)ETHER | 著者 | Xiao, T.S, Yang, J, Liu, Z, Wang, C, Yang, R. | 登録日 | 2017-12-22 | 公開日 | 2018-06-13 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.796 Å) | 主引用文献 | Mechanism of gasdermin D recognition by inflammatory caspases and their inhibition by a gasdermin D-derived peptide inhibitor. Proc. Natl. Acad. Sci. U.S.A., 115, 2018
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6DEU
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![BU of 6deu by Molmil](/molmil-images/mine/6deu) | Human caspase-6 A109T | 分子名称: | Caspase-6 | 著者 | Tubeleviciute-Aydin, A, Beautrait, A, Lynham, J, Sharma, G, Gorelik, A, Deny, L.J, Soya, N, Lukacs, G.L, Nagar, B, Marinier, A, LeBlanc, A.C. | 登録日 | 2018-05-13 | 公開日 | 2019-03-27 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.796 Å) | 主引用文献 | Identification of Allosteric Inhibitors against Active Caspase-6. Sci Rep, 9, 2019
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6DEV
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![BU of 6dev by Molmil](/molmil-images/mine/6dev) | Human caspase-6 E35K | 分子名称: | Caspase-6 | 著者 | Tubeleviciute-Aydin, A, Beautrait, A, Lynham, J, Sharma, G, Gorelik, A, Deny, L.J, Soya, N, Lukacs, G.L, Nagar, B, Marinier, A, LeBlanc, A.C. | 登録日 | 2018-05-13 | 公開日 | 2019-03-27 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.348 Å) | 主引用文献 | Identification of Allosteric Inhibitors against Active Caspase-6. Sci Rep, 9, 2019
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7PAW
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![BU of 7paw by Molmil](/molmil-images/mine/7paw) | MALT1 in complex with compound 1 | 分子名称: | Mucosa-associated lymphoid tissue lymphoma translocation protein 1, ~{N}1-(3-chloranyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)-~{N}4-[2-(trifluoromethyl)pyrimidin-4-yl]cyclohexane-1,4-diamine | 著者 | Kack, H, Oster, L. | 登録日 | 2021-07-30 | 公開日 | 2021-11-17 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.19 Å) | 主引用文献 | Discovery and optimization of cyclohexane-1,4-diamines as allosteric MALT1 inhibitors. Eur.J.Med.Chem., 227, 2021
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