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1IUW
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P-HYDROXYBENZOATE HYDROXYLASE COMPLEXED WITH 4-4-HYDROXYBENZOATE AT PH 7.4
分子名称: FLAVIN-ADENINE DINUCLEOTIDE, P-HYDROXYBENZOATE HYDROXYLASE, P-HYDROXYBENZOIC ACID
著者Gatti, D.L, Entsch, B, Ballou, D.P, Ludwig, M.L.
登録日1995-11-22
公開日1996-07-11
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献pH-dependent structural changes in the active site of p-hydroxybenzoate hydroxylase point to the importance of proton and water movements during catalysis.
Biochemistry, 35, 1996
1IVY
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PHYSIOLOGICAL DIMER HPP PRECURSOR
分子名称: 2-acetamido-2-deoxy-alpha-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Rudenko, G, Bonten, E, D'Azzo, A, Hol, W.G.J.
登録日1996-06-12
公開日1997-04-21
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Three-dimensional structure of the human 'protective protein': structure of the precursor form suggests a complex activation mechanism.
Structure, 3, 1995
1INP
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CRYSTAL STRUCTURE OF INOSITOL POLYPHOSPHATE 1-PHOSPHATASE AT 2.3 ANGSTROMS RESOLUTION
分子名称: INOSITOL POLYPHOSPHATE 1-PHOSPHATASE, MAGNESIUM ION
著者York, J.D, Ponder, J.W, Chen, Z, Mathews, F.S, Majerus, P.W.
登録日1994-10-04
公開日1995-01-26
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal structure of inositol polyphosphate 1-phosphatase at 2.3-A resolution.
Biochemistry, 33, 1994
1IZ2
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Interactions causing the kinetic trap in serpin protein folding
分子名称: alpha-D-glucopyranose-(1-2)-(5R)-5-[(2R)-2-hydroxynonyl]-beta-D-xylulofuranose, alpha1-antitrypsin
著者Im, H, Woo, M.-S, Hwang, K.Y, Yu, M.-H.
登録日2002-09-19
公開日2003-02-11
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Interactions causing the kinetic trap in serpin protein folding
J.BIOL.CHEM., 277, 2002
5SVA
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Mediator-RNA Polymerase II Pre-Initiation Complex
分子名称: 108bp HIS4 Promoter Non-template Strand (-92/+16), 108bp HIS4 Promoter Template Strand (+16/-92), DNA repair helicase RAD25, ...
著者Robinson, P.J, Bushnell, D.A, Kornberg, R.D.
登録日2016-08-05
公開日2016-09-28
最終更新日2019-11-27
実験手法ELECTRON MICROSCOPY (15.3 Å)
主引用文献Structure of a Complete Mediator-RNA Polymerase II Pre-Initiation Complex.
Cell, 166, 2016
1JYH
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Crystal Structure of the Escherichia coli SbmC protein (AKA Gyrase Inhibitory Protein GyrI, AKA YeeB)
分子名称: DNA Gyrase inhibitory protein
著者Romanowski, M.J, Gibney, S.A, Burley, S.K, New York SGX Research Center for Structural Genomics (NYSGXRC)
登録日2001-09-12
公開日2002-04-10
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Crystal structure of the Escherichia coli SbmC protein that protects cells from the DNA replication inhibitor microcin B17.
Proteins, 47, 2002
1K0G
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THE CRYSTAL STRUCTURE OF AMINODEOXYCHORISMATE SYNTHASE FROM PHOSPHATE GROWN CRYSTALS
分子名称: PHOSPHATE ION, TRYPTOPHAN, p-aminobenzoate synthase component I
著者Parsons, J.F, Jensen, P.Y, Pachikara, A.S, Howard, A.J, Eisenstein, E, Ladner, J.E.
登録日2001-09-19
公開日2002-02-27
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Structure of Escherichia coli aminodeoxychorismate synthase: architectural conservation and diversity in chorismate-utilizing enzymes.
Biochemistry, 41, 2002
1JON
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GROEL (HSP60 CLASS) FRAGMENT COMPRISING RESIDUES 191-345
分子名称: GROEL, HSP60 CLASS
著者Buckle, A.M, Fersht, A.R.
登録日1996-05-30
公開日1997-03-12
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Chaperone activity and structure of monomeric polypeptide binding domains of GroEL.
Proc.Natl.Acad.Sci.USA, 93, 1996
1JP3
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Structure of E.coli undecaprenyl pyrophosphate synthase
分子名称: 2-(2-{2-[2-(2-{2-[2-(2-{2-[4-(1,1,3,3-TETRAMETHYL-BUTYL)-PHENOXY]-ETHOXY}-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHANOL, undecaprenyl pyrophosphate synthase
著者Ko, T.P, Chen, Y.K, Robinson, H, Tsai, P.C, Gao, Y.G, Chen, A.P.C, Wang, A.H.J, Liang, P.H.
登録日2001-07-31
公開日2001-08-15
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Mechanism of product chain length determination and the role of a flexible loop in Escherichia coli undecaprenyl-pyrophosphate synthase catalysis.
J.Biol.Chem., 276, 2001
1K25
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PBP2x from a Highly Penicillin-resistant Streptococcus pneumoniae Clinical Isolate
分子名称: low-affinity PENICILLIN-BINDING PROTEIN 2X
著者Dessen, A, Mouz, N, Hopkins, J, Dideberg, O.
登録日2001-09-26
公開日2001-10-31
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Crystal structure of PBP2x from a highly penicillin-resistant Streptococcus pneumoniae clinical isolate: a mosaic framework containing 83 mutations.
J.Biol.Chem., 276, 2001
1K1J
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BOVINE TRYPSIN-INHIBITOR COMPLEX
分子名称: CALCIUM ION, N-ALPHA-(2-NAPHTHYLSULFONYL)-N(3-AMIDINO-L-PHENYLALANINYL)ISOPIPECOLINIC ACID METHYL ESTER, SULFATE ION, ...
著者Stubbs, M.T.
登録日2001-09-25
公開日2001-11-28
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Factorising ligand affinity: a combined thermodynamic and crystallographic study of trypsin and thrombin inhibition.
J.Mol.Biol., 313, 2001
1K1M
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BOVINE TRYPSIN-INHIBITOR COMPLEX
分子名称: CALCIUM ION, N-ALPHA-(2-NAPHTHYLSULFONYL)-N(3-AMIDINO-L-PHENYLALANINYL)-4-ACETYL-PIPERAZINE, SULFATE ION, ...
著者Stubbs, M.T.
登録日2001-09-25
公開日2001-11-28
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Factorising ligand affinity: a combined thermodynamic and crystallographic study of trypsin and thrombin inhibition.
J.Mol.Biol., 313, 2001
5T5N
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Calcium-activated chloride channel bestrophin-1 (BEST1), triple mutant: I76A, F80A, F84A; in complex with an Fab antibody fragment, chloride, and calcium
分子名称: CALCIUM ION, CHLORIDE ION, Fab antibody fragment, ...
著者Long, S.B, Vaisey, G.
登録日2016-08-31
公開日2016-11-30
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Distinct regions that control ion selectivity and calcium-dependent activation in the bestrophin ion channel.
Proc. Natl. Acad. Sci. U.S.A., 113, 2016
5T96
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Crystal structure of the infectious salmon anemia virus (ISAV) HE viral receptor complex
分子名称: 4-O-acetyl-5-acetamido-3,5-dideoxy-L-glycero-alpha-D-galacto-non-2-ulopyranosonic acid, FORMIC ACID, GLYCEROL, ...
著者Cook, J.D, Sultana, A, Lee, J.E.
登録日2016-09-09
公開日2017-03-22
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structure of the infectious salmon anemia virus receptor complex illustrates a unique binding strategy for attachment.
Proc. Natl. Acad. Sci. U.S.A., 114, 2017
5T6R
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Nmd3 is a structural mimic of eIF5A, and activates the cpGTPase Lsg1 during 60S ribosome biogenesis: 60S-Nmd3 Complex
分子名称: 25S Ribosomal RNA, 5.8S Ribosomal RNA, 5S Ribosomal RNA, ...
著者Malyutin, A.G, Musalgaonkar, S, Patchett, S, Frank, J, Johnson, A.W.
登録日2016-09-01
公開日2017-02-08
最終更新日2024-03-13
実験手法ELECTRON MICROSCOPY (4.2 Å)
主引用文献Nmd3 is a structural mimic of eIF5A, and activates the cpGTPase Lsg1 during 60S ribosome biogenesis.
EMBO J., 36, 2017
1JYQ
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Xray Structure of Grb2 SH2 Domain Complexed with a Highly Affine Phospho Peptide
分子名称: GROWTH FACTOR RECEPTOR-BOUND PROTEIN 2, mAZ-pY-(alpha Me)pY-N-NH2 peptide inhibitor
著者Nioche, P, Liu, W.-Q, Broutin, I, Charbonnier, F, Latreille, M.-T, Vidal, M, Roques, B, Garbay, C, Ducruix, A.
登録日2001-09-13
公開日2002-03-13
最終更新日2024-07-10
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal structures of the SH2 domain of Grb2: highlight on the binding of a new high-affinity inhibitor.
J.Mol.Biol., 315, 2002
1K1P
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BOVINE TRYPSIN-INHIBITOR COMPLEX
分子名称: CALCIUM ION, TRYPSIN, [((1R)-2-{(2S)-2-[({4-[AMINO(IMINO)METHYL]BENZYL}AMINO)CARBONYL]AZETIDINYL}-1-CYCLOHEXYL-2-OXOETHYL)AMINO]ACETIC ACID
著者Stubbs, M.T.
登録日2001-09-25
公開日2001-11-28
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Factorising ligand affinity: a combined thermodynamic and crystallographic study of trypsin and thrombin inhibition.
J.Mol.Biol., 313, 2001
1K1Y
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Crystal structure of thermococcus litoralis 4-alpha-glucanotransferase complexed with acarbose
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 4,6-dideoxy-4-{[(1S,4R,5S,6S)-4,5,6-trihydroxy-3-(hydroxymethyl)cyclohex-2-en-1-yl]amino}-alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose, 4-ALPHA-GLUCANOTRANSFERASE, ...
著者Imamura, H, Fushinobu, S, Kumasaka, T, Yamamoto, M, Jeon, B.S, Wakagi, T, Matsuzawa, H.
登録日2001-09-26
公開日2003-06-17
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Crystal structures of 4-alpha-glucanotransferase from Thermococcus litoralis and its complex with an inhibitor
J.BIOL.CHEM., 278, 2003
1JKK
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2.4A X-RAY STRUCTURE OF TERNARY COMPLEX OF A CATALYTIC DOMAIN OF DEATH-ASSOCIATED PROTEIN KINASE WITH ATP ANALOGUE AND MG.
分子名称: DEATH-ASSOCIATED PROTEIN KINASE, MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER
著者Tereshko, V, Teplova, M, Brunzelle, J, Watterson, D.M, Egli, M.
登録日2001-07-12
公開日2002-04-01
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Crystal structures of the catalytic domain of human protein kinase associated with apoptosis and tumor suppression.
Nat.Struct.Biol., 8, 2001
1JLD
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Potent hiv protease inhibitors containing a novel (hydroxyethyl)amide isostere
分子名称: (2S)-2-tert-butyl-N~4~-(1-ethylpropyl)-N~1~-[(2R,3S)-2-hydroxy-4-phenyl-3-{[N-(quinolin-2-ylcarbonyl)-L-threonyl]amino}butyl]butanediamide, Pol polyprotein
著者Tong, L.
登録日1997-05-31
公開日1997-12-03
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Potent HIV protease inhibitors containing a novel (hydroxyethyl)amide isostere.
J.Med.Chem., 40, 1997
1JQ3
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Crystal Structure of Spermidine Synthase in Complex with Transition State Analogue AdoDATO
分子名称: S-ADENOSYL-1,8-DIAMINO-3-THIOOCTANE, Spermidine synthase
著者Korolev, S, Ikeguchi, Y, Skarina, T, Beasley, S, Edwards, A, Joachimiak, A, Pegg, A.E, Savchenko, A, Midwest Center for Structural Genomics (MCSG)
登録日2001-08-03
公開日2001-11-21
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献The crystal structure of spermidine synthase with a multisubstrate adduct inhibitor.
Nat.Struct.Biol., 9, 2002
1JS6
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Crystal Structure of DOPA decarboxylase
分子名称: DOPA decarboxylase, PYRIDOXAL-5'-PHOSPHATE
著者Burkhard, P, Dominici, P, Borri-Voltattorni, C, Jansonius, J.N, Malashkevich, V.N.
登録日2001-08-16
公開日2001-10-26
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Structural insight into Parkinson's disease treatment from drug-inhibited DOPA decarboxylase.
Nat.Struct.Biol., 8, 2001
1JXO
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Crystal Structure of the SH3-HOOK-GK Fragment of PSD-95
分子名称: postsynaptic density protein
著者Tavares, G.A, Panepucci, E.H, Brunger, A.T.
登録日2001-09-07
公開日2002-01-16
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structural characterization of the intramolecular interaction between the SH3 and guanylate kinase domains of PSD-95.
Mol.Cell, 8, 2001
1JMF
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CONTRIBUTIONS OF ORIENTATION AND HYDROGEN BONDING TO CATALYSIS IN ASN-229 MUTANTS OF THYMIDYLATE SYNTHASE
分子名称: 2'-DEOXYURIDINE 5'-MONOPHOSPHATE, THYMIDYLATE SYNTHASE
著者Finer-Moore, J, Stroud, R.M.
登録日1997-09-13
公開日1998-01-28
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Contributions of orientation and hydrogen bonding to catalysis in Asn229 mutants of thymidylate synthase.
J.Mol.Biol., 276, 1998
1JAH
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H-RAS P21 PROTEIN MUTANT G12P, COMPLEXED WITH GUANOSINE-5'-[BETA,GAMMA-METHYLENE] TRIPHOSPHATE AND MAGNESIUM
分子名称: C-HA-RAS, MAGNESIUM ION, PHOSPHOMETHYLPHOSPHONIC ACID GUANYLATE ESTER
著者Schweins, T, Scheffzek, K, Assheuer, R, Wittinghofer, A.
登録日1996-12-15
公開日1997-07-23
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献The role of the metal ion in the p21ras catalysed GTP-hydrolysis: Mn2+ versus Mg2+.
J.Mol.Biol., 266, 1997

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