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2F6N
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Crystal structure of PHD finger-linker-bromodomain fragment of human BPTF in the free form
分子名称: ZINC ION, bromodomain PHD finger transcription factor
著者Li, H, Patel, D.J.
登録日2005-11-29
公開日2006-07-11
最終更新日2024-10-09
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Molecular basis for site-specific read-out of histone H3K4me3 by the BPTF PHD finger of NURF.
Nature, 442, 2006
3U0R
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BU of 3u0r by Molmil
Helical repeat structure of apoptosis inhibitor 5 reveals protein-protein interaction modules
分子名称: Apoptosis inhibitor 5
著者Han, B.G, Kim, K.H, Jeong, K.C, Cho, J.W, Noh, K.H, Kim, T.W, Yoon, H.J, Suh, S.W, Lee, S.H, Lee, B.I.
登録日2011-09-29
公開日2012-02-22
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Helical repeat structure of apoptosis inhibitor 5 reveals protein-protein interaction modules.
J.Biol.Chem., 287, 2012
2F7X
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Protein Kinase A bound to (S)-2-(1H-Indol-3-yl)-1-[5-((E)-2-pyridin-4-yl-vinyl)-pyridin-3-yloxymethyl]-ethylamine
分子名称: (1S)-2-(1H-INDOL-3-YL)-1-[({5-[(E)-2-PYRIDIN-4-YLVINYL]PYRIDIN-3-YL}OXY)METHYL]ETHYLAMINE, PKI, inhibitory peptide, ...
著者Li, Q, Li, T, Zhu, G.D, Gong, J, Claibone, A, Dalton, C, Luo, Y, Johnson, E.F, Shi, Y, Liu, X, Klinghofer, V, Bauch, J.L, Marsh, K.C, Bouska, J.J, Arries, S, De Jong, R, Oltersdorf, T, Stoll, V.S, Jakob, C.G, Rosenberg, S.H, Giranda, V.L.
登録日2005-12-01
公開日2006-06-27
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Discovery of trans-3,4'-bispyridinylethylenes as potent and novel inhibitors of protein kinase B (PKB/Akt) for the treatment of cancer: Synthesis and biological evaluation.
Bioorg.Med.Chem.Lett., 16, 2006
4F8E
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BU of 4f8e by Molmil
Crystal structure of human PRS1 D52H mutant
分子名称: MAGNESIUM ION, Ribose-phosphate pyrophosphokinase 1, SULFATE ION
著者Chen, P, Teng, M, Li, X.
登録日2012-05-17
公開日2013-05-22
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.27 Å)
主引用文献A small disturbance, but a serious disease: the possible mechanism of D52H-mutant of human PRS1 that causes gout
Iubmb Life, 65, 2013
1BV3
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HUMAN CARBONIC ANHYDRASE II COMPLEXED WITH UREA
分子名称: 4-(HYDROXYMERCURY)BENZOIC ACID, PROTEIN (CARBONIC ANHYDRASE II), UREA, ...
著者Briganti, F, Mangani, S, Scozzafava, A, Vernaglione, G, Supuran, C.T.
登録日1998-09-22
公開日1999-09-28
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Carbonic anhydrase catalyzes cyanamide hydration to urea: is it mimicking the physiological reaction?
J.Biol.Inorg.Chem., 4, 1999
1J5N
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Solution Structure of the Non-Sequence-Specific HMGB protein NHP6A in complex with SRY DNA
分子名称: 5'-D(*CP*TP*GP*AP*AP*CP*AP*AP*TP*CP*AP*CP*CP*CP*C)-3', 5'-D(*GP*GP*GP*GP*TP*GP*AP*TP*TP*GP*TP*TP*CP*AP*G)-3', Nonhistone chromosomal protein 6A
著者Masse, J.E, Wong, B, Yen, Y.-M, Allain, F.H.-T, Johnson, R.C, Feigon, J.
登録日2002-05-15
公開日2002-10-16
最終更新日2023-12-27
実験手法SOLUTION NMR
主引用文献The S. cerevisiae architectural HMGB protein NHP6A complexed with DNA: DNA and protein conformational changes upon binding
J.Mol.Biol., 323, 2002
1S3Q
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BU of 1s3q by Molmil
Crystal structures of a novel open pore ferritin from the hyperthermophilic Archaeon Archaeoglobus fulgidus
分子名称: ZINC ION, ferritin
著者Johnson, E, Cascio, D, Sawaya, M, Schroeder, I.
登録日2004-01-13
公開日2005-04-12
最終更新日2024-11-13
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Crystal structures of a tetrahedral open pore ferritin from the hyperthermophilic archaeon Archaeoglobus fulgidus.
Structure, 13, 2005
2FD3
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Crystal Structure of Thioredoxin Mutant P34H
分子名称: Thioredoxin 1
著者Gavira, J.A, Perez-Jimenez, R, Ibarra-Molero, B, Sanchez-Ruiz, J.M.
登録日2005-12-13
公開日2005-12-27
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献Crystal Structure of Thioredoxin Mutant P34H
To be Published
3U5O
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Crystal structure of the complex of TRIM33 PHD-Bromo and H3(1-22)K9me3K14acK18ac histone peptide
分子名称: E3 ubiquitin-protein ligase TRIM33, Histone H3.1, ZINC ION
著者Wang, Z, Patel, D.J.
登録日2011-10-11
公開日2012-01-18
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献A poised chromatin platform for TGF-beta access to master regulators
Cell(Cambridge,Mass.), 147, 2011
4ITP
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BU of 4itp by Molmil
Structure of human carbonic anhydrase II bound to a benzene sulfonamide
分子名称: 2-phenyl-N-(4-sulfamoylbenzyl)acetamide, Carbonic anhydrase 2, DIMETHYL SULFOXIDE, ...
著者Biswas, S, McKenna, R.
登録日2013-01-18
公開日2014-01-01
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.697 Å)
主引用文献Structural study of the location of the phenyl tail of benzene sulfonamides and the effect on human carbonic anhydrase inhibition.
Bioorg.Med.Chem., 21, 2013
2EV6
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BU of 2ev6 by Molmil
Bacillus subtilis manganese transport regulator (MNTR) bound to zinc
分子名称: CITRATE ANION, GLYCEROL, Transcriptional regulator mntR, ...
著者Kliegman, J.I, Griner, S.L, Helmann, J.D, Brennan, R.G, Glasfeld, A.
登録日2005-10-31
公開日2006-03-07
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structural Basis for the Metal-Selective Activation of the Manganese Transport Regulator of Bacillus subtilis.
Biochemistry, 45, 2006
3H52
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Crystal structure of the antagonist form of human glucocorticoid receptor
分子名称: 11-(4-DIMETHYLAMINO-PHENYL)-17-HYDROXY-13-METHYL-17-PROP-1-YNYL-1,2,6,7,8,11,12,13,14,15,16,17-DODEC AHYDRO-CYCLOPENTA[A]PHENANTHREN-3-ONE, GLYCEROL, Glucocorticoid receptor, ...
著者Schoch, G.A, Benz, J, D'Arcy, B, Stihle, M, Burger, D, Thoma, R, Ruf, A.
登録日2009-04-21
公開日2009-12-01
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Molecular switch in the glucocorticoid receptor: active and passive antagonist conformations
J.Mol.Biol., 395, 2010
3MYQ
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Crystal structure of human carbonic anhydrase isozyme II with 2-chloro-5-[(1H-imidazo[4,5-c]quinolin-2-ylsulfanyl)acetyl]benzenesulfonamide
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 2-chloro-5-[(1H-imidazo[4,5-c]quinolin-2-ylsulfanyl)acetyl]benzenesulfonamide, Carbonic anhydrase 2, ...
著者Grazulis, S, Manakova, E, Golovenko, D.
登録日2010-05-11
公開日2011-02-02
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.35 Å)
主引用文献Indapamide-like benzenesulfonamides as inhibitors of carbonic anhydrases I, II, VII, and XIII.
Bioorg.Med.Chem., 18, 2010
5COC
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BU of 5coc by Molmil
Fusion protein of human calmodulin and B4 domain of protein A from staphylococcal aureus
分子名称: CALCIUM ION, Immunoglobulin G-binding protein A,Calmodulin
著者Jeong, W.H, Lee, H, Song, D.H, Lee, J.O.
登録日2015-07-20
公開日2016-03-30
最終更新日2024-11-06
実験手法X-RAY DIFFRACTION (2.6691 Å)
主引用文献Connecting two proteins using a fusion alpha helix stabilized by a chemical cross linker.
Nat Commun, 7, 2016
3U45
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Human Carbonic Anhydrase II V143A
分子名称: Carbonic anhydrase 2, GLYCEROL, ZINC ION
著者West, D, Mckenna, R.
登録日2011-10-07
公開日2012-10-10
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.699 Å)
主引用文献Structural Modification of the hydrophobic pocket in Human Carbonic Anhydrase II
To be Published
2EWM
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BU of 2ewm by Molmil
Crystal Structure of the (S)-Specific 1-Phenylethanol Dehydrogenase of the Denitrifying Bacterium Strain EbN1
分子名称: (S)-1-Phenylethanol dehydrogenase, NICOTINAMIDE-ADENINE-DINUCLEOTIDE, SULFATE ION
著者Hoeffken, H.W.
登録日2005-11-04
公開日2006-03-14
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Crystal Structure and Enzyme kinetics of the (S)-Specific 1-Phenylethanol Dehydrogenase of the denitrifying bacterium Strain EbN1
Biochemistry, 45, 2006
1C3T
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ROTAMER STRAIN AS A DETERMINANT OF PROTEIN STRUCTURAL SPECIFICITY
分子名称: PROTEIN (1D8 UBIQUITIN)
著者Lazar, G.A, Johnson, E.C, Desjarlais, J.R, Handel, T.M.
登録日1999-07-28
公開日1999-08-20
最終更新日2024-04-10
実験手法SOLUTION NMR
主引用文献Rotamer strain as a determinant of protein structural specificity.
Protein Sci., 8, 1999
2EZ7
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BU of 2ez7 by Molmil
Carbonic anhydrase activators. Activation of isozymes I, II, IV, VA, VII and XIV with L- and D-histidine and crystallographic analysis of their adducts with isoform II: engineering proton transfer processes within the active site of an enzyme
分子名称: Carbonic anhydrase 2, D-HISTIDINE, MERCURY (II) ION, ...
著者Temperini, C, Scozzafava, A, Vullo, D, Supuran, C.T.
登録日2005-11-10
公開日2006-07-18
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Carbonic Anhydrase Activators. Activation of Isozymes I, II, IV, VA, VII, and XIV with L- and D-Histidine and Crystallographic Analysis of Their Adducts with Isoform II: Engineering Proton-Transfer Processes within the Active Site of an Enzyme.
Chemistry, 12, 2006
4C74
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Phenylacetone monooxygenase: Reduced enzyme in complex with APADP
分子名称: 3-ACETYLPYRIDINE ADENINE DINUCLEOTIDE, FLAVIN-ADENINE DINUCLEOTIDE, HEXAETHYLENE GLYCOL, ...
著者Martinoli, C, Fraaije, M.W, Mattevi, A.
登録日2013-09-19
公開日2014-02-05
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.97 Å)
主引用文献Beyond the Protein Matrix: Probing Cofactor Variants in a Baeyer-Villiger Oxygenation Reaction.
Acs Catal., 3, 2013
3RAV
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BU of 3rav by Molmil
Horse spleen apo-ferritin with bound Pentobarbital
分子名称: 5-ethyl-5-[(2S)-pentan-2-yl]pyrimidine-2,4,6(1H,3H,5H)-trione, CADMIUM ION, Ferritin light chain, ...
著者Oakley, S.H, Vedula, L.S, Xi, J, Liu, R, Eckenhoff, R.G, Loll, P.J.
登録日2011-03-28
公開日2011-05-11
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献High resolution view of barbiturate recognition by a protein binding site
to be published
3RD0
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BU of 3rd0 by Molmil
Horse spleen apo-ferritin with bound thiopental
分子名称: 5-ethyl-5-[(2R)-pentan-2-yl]-2-thioxodihydropyrimidine-4,6(1H,5H)-dione, CADMIUM ION, Ferritin light chain, ...
著者Oakley, S.H, Vedula, L.S, Xi, J, Liu, R, Eckenhoff, R.G, Loll, P.J.
登録日2011-03-31
公開日2011-05-11
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献High resolution view of barbiturate recognition by a protein binding site
to be published
1TLL
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BU of 1tll by Molmil
CRYSTAL STRUCTURE OF RAT NEURONAL NITRIC-OXIDE SYNTHASE REDUCTASE MODULE AT 2.3 A RESOLUTION.
分子名称: FLAVIN MONONUCLEOTIDE, FLAVIN-ADENINE DINUCLEOTIDE, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ...
著者Garcin, E.D, Bruns, C.M, Lloyd, S.J, Hosfield, D.J, Tiso, M, Gachhui, R, Stuehr, D.J, Tainer, J.A, Getzoff, E.D.
登録日2004-06-09
公開日2004-08-31
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structural basis for isozyme-specific regulation of electron transfer in nitric-oxide synthase
J.Biol.Chem., 279, 2004
5BS5
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EPSP synthase from Acinetobacter baumannii
分子名称: 3-phosphoshikimate 1-carboxyvinyltransferase
著者Sutton, K.A, Schultz, L.W, Russo, T.A, Breen, J, Umland, T.C.
登録日2015-06-01
公開日2016-02-24
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (2.49 Å)
主引用文献EPSP synthase from Acinetobacter baumannii
Acta Crystallogr.,Sect.F, 2016
1J7J
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Crystal Structure of the HPRT from Salmonella typhimurium
分子名称: MAGNESIUM ION, hypoxanthine phosphoribosyltransferase
著者Lee, C.C, Focia, P.J, Spraggon, G, Eakin, A.E.
登録日2001-05-16
公開日2003-07-29
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal Structure of the HPRT from Salmonella Typhimurium at 2.3 A Resolution
To be Published
1J7O
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Solution structure of Calcium-calmodulin N-terminal domain
分子名称: CALCIUM ION, Calmodulin
著者Chou, J.J, Klee, C.B, Bax, A.
登録日2001-05-17
公開日2001-11-07
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Solution structure of Ca(2+)-calmodulin reveals flexible hand-like properties of its domains.
Nat.Struct.Biol., 8, 2001

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