9PTI
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1QLQ
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![BU of 1qlq by Molmil](/molmil-images/mine/1qlq) | Bovine Pancreatic Trypsin Inhibitor (BPTI) Mutant with Altered Binding Loop Sequence | 分子名称: | PANCREATIC TRYPSIN INHIBITOR, SULFATE ION | 著者 | Czapinska, H, Krzywda, S, Sheldrick, G.M, Otlewski, J, Jaskolski, M. | 登録日 | 1999-09-10 | 公開日 | 1999-10-05 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.42 Å) | 主引用文献 | High Resolution Structure of Bovine Pancreatic Trypsin Inhibitor with Altered Binding Loop Sequence J.Mol.Biol., 295, 1999
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6PTI
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2M99
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6KZF
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![BU of 6kzf by Molmil](/molmil-images/mine/6kzf) | Racemic X-ray Structure of Calcicludine | 分子名称: | D-calcicludine, Kunitz-type serine protease inhibitor homolog calcicludine | 著者 | Qu, Q, Gao, S, Liu, L. | 登録日 | 2019-09-24 | 公開日 | 2019-11-06 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.52 Å) | 主引用文献 | Synthesis of Disulfide Surrogate Peptides Incorporating Large-Span Surrogate Bridges Through a Native-Chemical-Ligation-Assisted Diaminodiacid Strategy Angew.Chem.Int.Ed.Engl., 59, 2020
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6YHY
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![BU of 6yhy by Molmil](/molmil-images/mine/6yhy) | A lid blocking mechanism of a cone snail toxin revealed at the atomic level | 分子名称: | Conk-S1 | 著者 | Saikia, C, Altman-Gueta, H, Dym, O, Frolow, F, Gurevitz, M, Gordon, D, Reuveny, E, Karbat, I. | 登録日 | 2020-03-31 | 公開日 | 2021-04-14 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | A Molecular Lid Mechanism of K + Channel Blocker Action Revealed by a Cone Peptide. J.Mol.Biol., 433, 2021
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6A5I
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8PTI
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![BU of 8pti by Molmil](/molmil-images/mine/8pti) | CRYSTAL STRUCTURE OF A Y35G MUTANT OF BOVINE PANCREATIC TRYPSIN INHIBITOR | 分子名称: | BOVINE PANCREATIC TRYPSIN INHIBITOR | 著者 | Housset, D, Kim, K.-S, Fuchs, J, Woodward, C, Wlodawer, A. | 登録日 | 1990-12-17 | 公開日 | 1991-04-15 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Crystal structure of a Y35G mutant of bovine pancreatic trypsin inhibitor. J.Mol.Biol., 220, 1991
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6F1F
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![BU of 6f1f by Molmil](/molmil-images/mine/6f1f) | The methylene thioacetal BPTI (Bovine Pancreatic Trypsin Inhibitor) mutant structure | 分子名称: | GLYCEROL, Pancreatic trypsin inhibitor, SULFATE ION | 著者 | Lansky, S, Mousa, R, Metanis, N, Shoham, G. | 登録日 | 2017-11-21 | 公開日 | 2018-07-18 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.716 Å) | 主引用文献 | BPTI folding revisited: switching a disulfide into methylene thioacetal reveals a previously hidden path. Chem Sci, 9, 2018
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5PTI
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4PTI
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![BU of 4pti by Molmil](/molmil-images/mine/4pti) | THE GEOMETRY OF THE REACTIVE SITE AND OF THE PEPTIDE GROUPS IN TRYPSIN, TRYPSINOGEN AND ITS COMPLEXES WITH INHIBITORS | 分子名称: | TRYPSIN INHIBITOR | 著者 | Huber, R, Kukla, D, Ruehlmann, A, Epp, O, Formanek, H, Deisenhofer, J, Steigemann, W. | 登録日 | 1982-09-27 | 公開日 | 1983-01-18 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | The Geometry of the Reactive Site and of the Peptide Groups in Trypsin, Trypsinogen and its Complexes with Inhibitors Acta Crystallogr.,Sect.B, 39, 1983
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5M4V
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![BU of 5m4v by Molmil](/molmil-images/mine/5m4v) | X-ray structure of the mambaquaretin-1, a selective antagonist of the vasopressin type 2 receptor | 分子名称: | CHLORIDE ION, Mambaquaretin-1, S-1,2-PROPANEDIOL | 著者 | Stura, E.A, Vera, L, Ciolek, J, Mourier, G, Gilles, N. | 登録日 | 2016-10-19 | 公開日 | 2017-05-03 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.06 Å) | 主引用文献 | Green mamba peptide targets type-2 vasopressin receptor against polycystic kidney disease. Proc. Natl. Acad. Sci. U.S.A., 114, 2017
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2M01
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![BU of 2m01 by Molmil](/molmil-images/mine/2m01) | Solution structure of Kunitz-type neurotoxin LmKKT-1a from scorpion venom | 分子名称: | Protease inhibitor LmKTT-1a | 著者 | Luo, F, Jiang, L, Liu, M, Chen, Z, Wu, Y. | 登録日 | 2012-10-15 | 公開日 | 2013-11-13 | 最終更新日 | 2023-06-14 | 実験手法 | SOLUTION NMR | 主引用文献 | Genomic and structural characterization of Kunitz-type peptide LmKTT-1a highlights diversity and evolution of scorpion potassium channel toxins. Plos One, 8, 2013
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6NAN
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![BU of 6nan by Molmil](/molmil-images/mine/6nan) | NMR structure determination of Ixolaris and Factor X interaction reveals a noncanonical mechanism of Kunitz inhibition | 分子名称: | Ixolaris | 著者 | De Paula, V.S, Sgourakis, N.G, Francischetti, I.M.B, Almeida, F.C.L, Monteiro, R.Q, Valente, A.P. | 登録日 | 2018-12-06 | 公開日 | 2019-06-12 | 最終更新日 | 2023-06-14 | 実験手法 | SOLUTION NMR | 主引用文献 | NMR structure determination of Ixolaris and factor X(a) interaction reveals a noncanonical mechanism of Kunitz inhibition. Blood, 134, 2019
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3WNY
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5NMV
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6Q61
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![BU of 6q61 by Molmil](/molmil-images/mine/6q61) | Pore-modulating toxins exploit inherent slow inactivation to block K+ channels | 分子名称: | Kunitz-type conkunitzin-S1, SULFATE ION | 著者 | Karbat, I, Gueta, H, Fine, S, Szanto, T, Hamer-Rogotner, S, Dym, O, Frolow, F, Gordon, D, Panyi, G, Gurevitz, M, Reuveny, E. | 登録日 | 2018-12-10 | 公開日 | 2019-08-21 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | Pore-modulating toxins exploit inherent slow inactivation to block K+channels. Proc.Natl.Acad.Sci.USA, 116, 2019
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6Q6C
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![BU of 6q6c by Molmil](/molmil-images/mine/6q6c) | Pore-modulating toxins exploit inherent slow inactivation to block K+ channels | 分子名称: | 1,2-ETHANEDIOL, Kunitz-type conkunitzin-S1, NITRATE ION, ... | 著者 | Karbat, I, Gueta, H, Fine, S, Szanto, T, Hamer-Rogotner, S, Dym, O, Frolow, F, Gordon, D, Panyi, G, Gurevitz, M, Reuveny, E. | 登録日 | 2018-12-10 | 公開日 | 2019-08-21 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | Pore-modulating toxins exploit inherent slow inactivation to block K+channels. Proc.Natl.Acad.Sci.USA, 116, 2019
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4DTG
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![BU of 4dtg by Molmil](/molmil-images/mine/4dtg) | Hemostatic effect of a monoclonal antibody mAb 2021 blocking the interaction between FXa and TFPI in a rabbit hemophilia model | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, GLYCEROL, Humanized recombinant FAB fragment, ... | 著者 | Svensson, L.A, Breinholt, J, Krogh, B.O, Hilden, I. | 登録日 | 2012-02-21 | 公開日 | 2012-06-13 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Hemostatic effect of a monoclonal antibody mAb 2021 blocking the interaction between FXa and TFPI in a rabbit hemophilia model. Blood, 119, 2012
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3OFW
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![BU of 3ofw by Molmil](/molmil-images/mine/3ofw) | Crystal structure of recombinant Kunitz Type serine protease Inhibitor-1 from the Carribean sea anemone stichodactyla helianthus | 分子名称: | CHLORIDE ION, Kunitz-type proteinase inhibitor SHPI-1 | 著者 | Garcia-Fernandez, R, Redecke, L, Pons, T, Perbandt, M, Talavera, A, Gil, D, Gonzalez, Y, de los Angeles Chavez, M, Betzel, C. | 登録日 | 2010-08-16 | 公開日 | 2011-08-17 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Structure of the recombinant BPTI/Kunitz-type inhibitor rShPI-1A from the marine invertebrate Stichodactyla helianthus. Acta Crystallogr.,Sect.F, 68, 2012
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4BQD
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![BU of 4bqd by Molmil](/molmil-images/mine/4bqd) | KD1 of human TFPI in complex with a synthetic peptide | 分子名称: | GLYCEROL, PEPTIDE, TISSUE FACTOR PATHWAY INHIBITOR (LIPOPROTEIN-ASSOCIATED COAGULATION INHIBITOR) VARIANT | 著者 | Griessner, A, Brandstetter, H. | 登録日 | 2013-05-30 | 公開日 | 2013-12-04 | 最終更新日 | 2019-07-17 | 実験手法 | X-RAY DIFFRACTION (2.48 Å) | 主引用文献 | Small Peptides Blocking Inhibition of Factor Xa and Tissue Factor-Factor Viia by Tissue Factor Pathway Inhibitor (Tfpi) J.Biol.Chem., 289, 2014
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3LDI
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![BU of 3ldi by Molmil](/molmil-images/mine/3ldi) | Crystal structure of aprotinin in complex with sucrose octasulfate: unusual interactions and implication for heparin binding | 分子名称: | GLYCEROL, MERCURY (II) ION, Pancreatic trypsin inhibitor, ... | 著者 | Yang, I.S, Kim, T.G, Park, B.S, Kim, K.H. | 登録日 | 2010-01-13 | 公開日 | 2010-06-23 | 最終更新日 | 2014-02-12 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Crystal structures of aprotinin and its complex with sucrose octasulfate reveal multiple modes of interactions with implications for heparin binding Biochem.Biophys.Res.Commun., 397, 2010
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3LDJ
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![BU of 3ldj by Molmil](/molmil-images/mine/3ldj) | Crystal structure of aprotinin in complex with sucrose octasulfate: unusual interactions and implication for heparin binding | 分子名称: | 1,3,4,6-tetra-O-sulfo-beta-D-fructofuranose-(2-1)-2,3,4,6-tetra-O-sulfonato-alpha-D-glucopyranose, ACETATE ION, Pancreatic trypsin inhibitor | 著者 | Yang, I.S, Kim, T.G, Park, B.S, Kim, K.H. | 登録日 | 2010-01-13 | 公開日 | 2010-09-15 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Crystal structures of aprotinin and its complex with sucrose octasulfate reveal multiple modes of interactions with implications for heparin binding. Biochem.Biophys.Res.Commun., 2010
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3LDM
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5JB6
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