2ALM
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![BU of 2alm by Molmil](/molmil-images/mine/2alm) | Crystal structure analysis of a mutant beta-ketoacyl-[acyl carrier protein] synthase II from Streptococcus pneumoniae | 分子名称: | 3-oxoacyl-(acyl-carrier-protein) synthase II, MAGNESIUM ION | 著者 | Zhang, Y.M, Hurlbert, J, White, S.W, Rock, C.O. | 登録日 | 2005-08-07 | 公開日 | 2005-08-30 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Roles of the active site water, histidine 303, and phenylalanine 396 in the catalytic mechanism of the elongation condensing enzyme of Streptococcus pneumoniae. J.Biol.Chem., 281, 2006
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2A9Y
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![BU of 2a9y by Molmil](/molmil-images/mine/2a9y) | Crystal structure of T. gondii adenosine kinase complexed with N6-dimethyladenosine | 分子名称: | 6N-DIMETHYLADENOSINE, ACETATE ION, CHLORIDE ION, ... | 著者 | Zhang, Y, el Kouni, M.H, Ealick, S.E. | 登録日 | 2005-07-12 | 公開日 | 2006-07-11 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.35 Å) | 主引用文献 | Substrate analogs induce an intermediate conformational change in Toxoplasma gondii adenosine kinase Acta Crystallogr.,Sect.D, 63, 2007
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2AA0
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![BU of 2aa0 by Molmil](/molmil-images/mine/2aa0) | Crystal structure of T. gondii adenosine kinase complexed with 6-methylmercaptopurine riboside | 分子名称: | 2-HYDROXYMETHYL-5-(6-METHYLSULFANYL-PURIN-9-YL)-TETRAHYDRO-FURAN-3,4-DIOL, ACETATE ION, CHLORIDE ION, ... | 著者 | Zhang, Y, el Kouni, M.H, Ealick, S.E. | 登録日 | 2005-07-13 | 公開日 | 2006-07-25 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Substrate analogs induce an intermediate conformational change in Toxoplasma gondii adenosine kinase Acta Crystallogr.,Sect.D, 63, 2007
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2AB8
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![BU of 2ab8 by Molmil](/molmil-images/mine/2ab8) | Crystal structure of T. gondii adenosine kinase complexed with 6-methylmercaptopurine riboside and AMP-PCP | 分子名称: | 2-HYDROXYMETHYL-5-(6-METHYLSULFANYL-PURIN-9-YL)-TETRAHYDRO-FURAN-3,4-DIOL, CHLORIDE ION, PHOSPHOMETHYLPHOSPHONIC ACID ADENYLATE ESTER, ... | 著者 | Zhang, Y, el Kouni, M.H, Ealick, S.E. | 登録日 | 2005-07-14 | 公開日 | 2006-07-25 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Substrate analogs induce an intermediate conformational change in Toxoplasma gondii adenosine kinase Acta Crystallogr.,Sect.D, 63, 2007
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2ABS
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![BU of 2abs by Molmil](/molmil-images/mine/2abs) | Crystal structure of T. gondii adenosine kinase complexed with AMP-PCP | 分子名称: | CHLORIDE ION, PHOSPHOMETHYLPHOSPHONIC ACID ADENYLATE ESTER, SODIUM ION, ... | 著者 | Zhang, Y, el Kouni, M.H, Ealick, S.E. | 登録日 | 2005-07-16 | 公開日 | 2006-01-24 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.1 Å) | 主引用文献 | Structure of Toxoplasma gondii adenosine kinase in complex with an ATP analog at 1.1 angstroms resolution. Acta Crystallogr.,Sect.D, 62, 2006
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2A9Z
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![BU of 2a9z by Molmil](/molmil-images/mine/2a9z) | Crystal structure of T. gondii adenosine kinase complexed with N6-dimethyladenosine and AMP-PCP | 分子名称: | 6N-DIMETHYLADENOSINE, CHLORIDE ION, PHOSPHOMETHYLPHOSPHONIC ACID ADENYLATE ESTER, ... | 著者 | Zhang, Y, el Kouni, M.H, Ealick, S.E. | 登録日 | 2005-07-12 | 公開日 | 2006-07-11 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.35 Å) | 主引用文献 | Substrate analogs induce an intermediate conformational change in Toxoplasma gondii adenosine kinase Acta Crystallogr.,Sect.D, 63, 2007
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6XNY
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![BU of 6xny by Molmil](/molmil-images/mine/6xny) | Structure of RAG1 (R848M/E649V)-RAG2-DNA Strand Transfer Complex (Paired-Form) | 分子名称: | 12RSS integration strand (55-mer), 12RSS signal DNA top strand (34-mer), 23RSS integration strand (66-mer), ... | 著者 | Zhang, Y, Corbett, E, Wu, S, Schatz, D.G. | 登録日 | 2020-07-05 | 公開日 | 2020-08-26 | 最終更新日 | 2024-03-06 | 実験手法 | ELECTRON MICROSCOPY (2.9 Å) | 主引用文献 | Structural basis for the activation and suppression of transposition during evolution of the RAG recombinase. Embo J., 39, 2020
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4FK3
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![BU of 4fk3 by Molmil](/molmil-images/mine/4fk3) | B-Raf Kinase V600E Oncogenic Mutant in Complex with PLX3203 | 分子名称: | N-{2,4-difluoro-3-[(5-pyridin-3-yl-1H-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]phenyl}ethanesulfonamide, Serine/threonine-protein kinase B-raf | 著者 | Zhang, Y, Wang, W, Zhang, K.Y.J. | 登録日 | 2012-06-12 | 公開日 | 2012-08-08 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.65 Å) | 主引用文献 | Discovery of a selective inhibitor of oncogenic B-Raf kinase with potent antimelanoma activity. Proc.Natl.Acad.Sci.USA, 105, 2008
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6XNX
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![BU of 6xnx by Molmil](/molmil-images/mine/6xnx) | Structure of RAG1 (R848M/E649V)-RAG2-DNA Strand Transfer Complex (Dynamic-Form) | 分子名称: | 12RSS integration strand DNA (55-MER), 12RSS signal top strand DNA (34-MER), 23RSS integration strand DNA (66-MER), ... | 著者 | Zhang, Y, Corbett, E, Wu, S, Schatz, D.G. | 登録日 | 2020-07-05 | 公開日 | 2020-08-26 | 最終更新日 | 2024-03-06 | 実験手法 | ELECTRON MICROSCOPY (2.7 Å) | 主引用文献 | Structural basis for the activation and suppression of transposition during evolution of the RAG recombinase. Embo J., 39, 2020
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5JKJ
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6M0X
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![BU of 6m0x by Molmil](/molmil-images/mine/6m0x) | Crystal structure of Streptococcus thermophilus Cas9 in complex with AGGA PAM | 分子名称: | BARIUM ION, CRISPR-associated endonuclease Cas9 1, DNA (28-MER), ... | 著者 | Zhang, Y, Zhang, H, Xu, X, Wang, Y, Chen, W, Wang, Y, Wu, Z, Tang, N, Wang, Y, Zhao, S, Gan, J, Ji, Q. | 登録日 | 2020-02-23 | 公開日 | 2020-09-09 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.561 Å) | 主引用文献 | Catalytic-state structure and engineering of Streptococcus thermophilus Cas9 Nat Catal, 2020
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6M0W
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![BU of 6m0w by Molmil](/molmil-images/mine/6m0w) | Crystal structure of Streptococcus thermophilus Cas9 in complex with the AGAA PAM | 分子名称: | CRISPR-associated endonuclease Cas9 1, DNA (28-MER), DNA (5'-D(*AP*AP*AP*GP*AP*AP*GP*C)-3'), ... | 著者 | Zhang, Y, Zhang, H, Xu, X, Wang, Y, Chen, W, Wang, Y, Wu, Z, Tang, N, Wang, Y, Zhao, S, Gan, J, Ji, Q. | 登録日 | 2020-02-23 | 公開日 | 2020-09-09 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.76 Å) | 主引用文献 | Catalytic-state structure and engineering of Streptococcus thermophilus Cas9 Nat Catal, 2020
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5JKF
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![BU of 5jkf by Molmil](/molmil-images/mine/5jkf) | Crystal structure of esterase E22 | 分子名称: | Esterase E22 | 著者 | Zhang, Y, Wang, P, Yao, Q. | 登録日 | 2016-04-26 | 公開日 | 2017-04-26 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.393 Å) | 主引用文献 | Structural basis for substrate recognition and catalysis of a novel esterase E22 with a homoserine transacetylase-like fold To Be Published
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6M0V
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![BU of 6m0v by Molmil](/molmil-images/mine/6m0v) | Crsytal structure of streptococcus thermophilus Cas9 in complex with the GGAA PAM | 分子名称: | BARIUM ION, CRISPR-associated endonuclease Cas9 1, DNA (28-MER), ... | 著者 | Zhang, Y, Zhang, H, Xu, X, Wang, Y, Chen, W, Wang, Y, Wu, Z, Tang, N, Wang, Y, Zhao, S, Gan, J, Ji, Q. | 登録日 | 2020-02-22 | 公開日 | 2020-09-09 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Catalytic-state structure and engineering of Streptococcus thermophilus Cas9 Nat Catal, 2020
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6N33
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![BU of 6n33 by Molmil](/molmil-images/mine/6n33) | Crystal structure of fms kinase domain with a small molecular inhibitor, PLX5622 | 分子名称: | 6-fluoro-N-[(5-fluoro-2-methoxypyridin-3-yl)methyl]-5-[(5-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)methyl]pyridin-2-amine, Macrophage colony-stimulating factor 1 receptor | 著者 | Zhang, Y. | 登録日 | 2018-11-14 | 公開日 | 2019-09-18 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Sustained microglial depletion with CSF1R inhibitor impairs parenchymal plaque development in an Alzheimer's disease model. Nat Commun, 10, 2019
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3LC8
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3LBS
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![BU of 3lbs by Molmil](/molmil-images/mine/3lbs) | |
4Z69
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![BU of 4z69 by Molmil](/molmil-images/mine/4z69) | |
5X87
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![BU of 5x87 by Molmil](/molmil-images/mine/5x87) | |
5XZD
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3LZC
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![BU of 3lzc by Molmil](/molmil-images/mine/3lzc) | Crystal structure of Dph2 from Pyrococcus horikoshii | 分子名称: | Dph2 | 著者 | Zhang, Y, Zhu, X, Torelli, A.T, Lee, M, Dzikovski, B, Koralewski, R.M, Wang, E, Freed, J, Krebs, C, Lin, H, Ealick, S.E. | 登録日 | 2010-03-01 | 公開日 | 2010-06-23 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.261 Å) | 主引用文献 | Diphthamide biosynthesis requires an organic radical generated by an iron-sulphur enzyme. Nature, 465, 2010
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5YGB
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5YGC
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6GFM
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![BU of 6gfm by Molmil](/molmil-images/mine/6gfm) | Crystal structure of the Escherichia coli nucleosidase PpnN (pppGpp-form) | 分子名称: | Pyrimidine/purine nucleotide 5'-monophosphate nucleosidase, guanosine 5'-(tetrahydrogen triphosphate) 3'-(trihydrogen diphosphate) | 著者 | Zhang, Y, Baerentsen, R.L, Gerdes, K, Brodersen, D.E. | 登録日 | 2018-05-01 | 公開日 | 2019-04-24 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2.77 Å) | 主引用文献 | (p)ppGpp Regulates a Bacterial Nucleosidase by an Allosteric Two-Domain Switch. Mol.Cell, 74, 2019
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5LQ6
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![BU of 5lq6 by Molmil](/molmil-images/mine/5lq6) | Salmonella effector SpvD - R161 variant | 分子名称: | SODIUM ION, Virulence protein vsdE | 著者 | Zhang, Y, Grabe, G.J, Rolhion, N, Yang, Y, Holden, D.W, Hare, S.A. | 登録日 | 2016-08-16 | 公開日 | 2016-11-02 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.48 Å) | 主引用文献 | The Salmonella Effector SpvD Is a Cysteine Hydrolase with a Serovar-specific Polymorphism Influencing Catalytic Activity, Suppression of Immune Responses, and Bacterial Virulence. J. Biol. Chem., 291, 2016
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