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PDB: 12895 件

3ET1
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Structure of PPARalpha with 3-[5-Methoxy-1-(4-methoxy-benzenesulfonyl)-1H-indol-3-yl]-propionic acid
分子名称: 3-{5-methoxy-1-[(4-methoxyphenyl)sulfonyl]-1H-indol-3-yl}propanoic acid, Peroxisome proliferator-activated receptor alpha, Steroid receptor coactivator 1
著者Zhang, K.Y.J, Wang, W.
登録日2008-10-06
公開日2009-02-17
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Scaffold-based discovery of indeglitazar, a PPAR pan-active anti-diabetic agent
Proc.Natl.Acad.Sci.USA, 106, 2009
7V4Y
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TTHA1264/TTHA1265 complex
分子名称: Putative zinc protease, ZINC ION, Zinc-dependent peptidase
著者Xu, M, Xu, Q, Ran, T, Wang, W, Sun, B, Wang, Q.
登録日2021-08-16
公開日2022-06-29
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Crystal structures of TTHA1265 and TTHA1264/TTHA1265 complex reveal an intrinsic heterodimeric assembly.
Int.J.Biol.Macromol., 207, 2022
3F5V
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C2 Crystal form of mite allergen DER P 1
分子名称: CALCIUM ION, Der p 1 allergen, HEXAETHYLENE GLYCOL
著者Stura, E.A, Minor, W, Chruszcz, M, Saint Remy, J.M.
登録日2008-11-04
公開日2009-02-10
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.36 Å)
主引用文献Crystal structures of mite allergens Der f 1 and Der p 1 reveal differences in surface-exposed residues that may influence antibody binding.
J.Mol.Biol., 386, 2009
1ORW
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Crystal Structure of Porcine Dipeptidyl Peptidase IV (CD26) in Complex with a Peptidomimetic Inhibitor
分子名称: (2S)-PYRROLIDIN-2-YLMETHYLAMINE, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Engel, M, Hoffmann, T, Wagner, L, Wermann, M, Heiser, U, Kiefersauer, R, Huber, R, Bode, W, Demuth, H.U, Brandstetter, H.
登録日2003-03-16
公開日2003-05-06
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.84 Å)
主引用文献The Crystal Structure of Dipeptidyl Peptidase IV (CD26) Reveals its Functional Regulation and Enzymatic Mechanism
Proc.Natl.Acad.Sci.USA, 100, 2003
7YXA
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XFEL crystal structure of the human sphingosine 1 phosphate receptor 5 in complex with ONO-5430608
分子名称: (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, 2-acetamido-2-deoxy-beta-D-glucopyranose, 4-[6-(2-naphthalen-1-ylethoxy)-2,3,4,5-tetrahydro-1H-3-benzazepin-3-ium-3-yl]butanoic acid, ...
著者Lyapina, E, Marin, E, Gusach, A, Orekhov, P, Gerasimov, A, Luginina, A, Vakhrameev, D, Ergasheva, M, Kovaleva, M, Khusainov, G, Khorn, P, Shevtsov, M, Kovalev, K, Okhrimenko, I, Bukhdruker, S, Popov, P, Hu, H, Weierstall, U, Liu, W, Cho, Y, Gushchin, I, Rogachev, A, Bourenkov, G, Park, S, Park, G, Huyn, H.J, Park, J, Gordeliy, V, Borshchevskiy, V, Mishin, A, Cherezov, V.
登録日2022-02-15
公開日2022-08-10
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structural basis for receptor selectivity and inverse agonism in S1P 5 receptors.
Nat Commun, 13, 2022
3I4P
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Crystal structure of AsnC family transcriptional regulator from Agrobacterium tumefaciens
分子名称: ACETATE ION, CALCIUM ION, CHLORIDE ION, ...
著者Cymborowski, M, Chruszcz, M, Luo, H, Xu, X, Savchenko, A, Edwards, A, Joachimiak, A, Minor, W, Midwest Center for Structural Genomics (MCSG)
登録日2009-07-02
公開日2009-07-28
最終更新日2022-04-13
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal structure of AsnC family transcriptional regulator from Agrobacterium tumefaciens
To be Published
3VGZ
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Crystal structure of E. coli YncE
分子名称: Uncharacterized protein YncE
著者Kagawa, W, Sagawa, T, Niki, H, Kurumizaka, H.
登録日2011-08-23
公開日2011-11-16
最終更新日2011-12-14
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structural basis for the DNA-binding activity of the bacterial beta-propeller protein YncE
Acta Crystallogr.,Sect.D, 67, 2011
3EZR
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CDK-2 with indazole inhibitor 17 bound at its active site
分子名称: 3-methoxy-4-{3-[4-(4-methylpiperazin-1-yl)-1H-benzimidazol-2-yl]-1H-indazol-6-yl}aniline, Cell division protein kinase 2
著者Kiefer, J.R, Day, J.E, Caspers, N.L, Mathis, K.J, Kretzmer, K.K, Weinberg, R.A, Reitz, B.A, Stegeman, R.A, Trujillo, J.I, Huang, W, Thorarensen, A, Xing, L, Wrightstone, A, Christine, L, Compton, R, Li, X.
登録日2008-10-23
公開日2009-02-03
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献2-(6-Phenyl-1H-indazol-3-yl)-1H-benzo[d]imidazoles: Design and synthesis of a potent and isoform selective PKC-zeta inhibitor
Bioorg.Med.Chem.Lett., 19, 2009
3HS9
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Intersectin 1-peptide-AP2 beta ear complex
分子名称: AP-2 complex subunit beta-1, peptide from Intersectin-1, residues 841-851
著者Vahedi-Faridi, A, Pechstein, A, Schaefer, J.G, Saenger, W, Haucke, V.
登録日2009-06-10
公開日2010-02-23
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Regulation of synaptic vesicle recycling by complex formation between intersectin 1 and the clathrin adaptor complex AP2.
Proc.Natl.Acad.Sci.USA, 107, 2010
1OPX
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Crystal structure of the traffic ATPase (HP0525) of the Helicobacter pylori type IV secretion system bound by sulfate
分子名称: NONAETHYLENE GLYCOL, SULFATE ION, virB11 homolog
著者Savvides, S.N, Yeo, H.J, Beck, M.R, Blaesing, F, Lurz, R, Lanka, E, Buhrdorf, R, Fischer, W, Haas, R, Waksman, G.
登録日2003-03-06
公開日2003-05-06
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献VirB11 ATPases are dynamic hexameric assemblies: New insights into bacterial type IV secretion
Embo J., 22, 2003
3VLK
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Crystal Structure Analysis of the Ser305Ala variant of KatG from Haloarcula marismortui
分子名称: Catalase-peroxidase 2, PROTOPORPHYRIN IX CONTAINING FE
著者Sato, T, Higuchi, W, Yoshimatsu, K, Fujiwara, T.
登録日2011-12-01
公開日2012-12-05
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal Structure and Kinetics Studies on Ser305Ala variant of KatG from HALOARCULA MARISMORTUI and its Complexes with Inhibitor SHA
To be Published
3F2R
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Crystal structure of human choline kinase alpha in complex with hemicholinium-3
分子名称: (2S,2'S)-2,2'-biphenyl-4,4'-diylbis(2-hydroxy-4,4-dimethylmorpholin-4-ium), Choline kinase alpha, UNKNOWN ATOM OR ION
著者Hong, B, Tempel, W, Rabeh, W.M, MacKenzie, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Weigelt, J, Bochkarev, A, Park, H, Structural Genomics Consortium (SGC)
登録日2008-10-30
公開日2008-11-11
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Crystal structure of human choline kinase alpha in complex with hemicholinium-3
To be Published
1OT3
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BU of 1ot3 by Molmil
Crystal structure of Drosophila deoxyribonucleotide kinase complexed with the substrate deoxythymidine
分子名称: Deoxyribonucleoside Kinase, SULFATE ION, THYMIDINE
著者Mikkelsen, N.E, Johansson, K, Karlsson, A, Knecht, W, Andersen, G, Piskur, J, Munch-Petersen, B, Eklund, H.
登録日2003-03-21
公開日2003-05-27
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural Basis for Feedback Inhibition of the Deoxyribonucleoside Salvage Pathway: Studies of the Drosophila Deoxyribonucleoside Kinase.
Biochemistry, 42, 2003
3VPV
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Crystal Structure of Pseudomonas aeruginosa Tsi2
分子名称: Tse2 specific immunity protein 2
著者Wang, W, Ding, J, Wang, D.C.
登録日2012-03-13
公開日2012-03-28
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Crystal Structure of Pseudomonas aeruginosa Tsi2
To be Published
3HXB
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BU of 3hxb by Molmil
Engineered RabGGTase in complex with a peptidomimetic inhibitor (compound 6)
分子名称: Geranylgeranyl transferase type-2 subunit alpha, Geranylgeranyl transferase type-2 subunit beta, N-[(benzyloxy)carbonyl]-D-tyrosyl-L-phenylalanyl-L-tyrosine, ...
著者Guo, Z, Alexandrov, K, Waldmann, H, Goody, R.S, Blankenfeldt, W.
登録日2009-06-20
公開日2009-09-08
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Design, synthesis, and characterization of Peptide-based rab geranylgeranyl transferase inhibitors
J.Med.Chem., 52, 2009
2JUV
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AbaA3-DKP-insulin
分子名称: Insulin A chain, Insulin B chain
著者Huang, K, Chan, S, Hua, Q, Chu, Y, Wang, R, Klaproth, B, Jia, W, Whittaker, J, De Meyts, P, Nakagawa, S.H, Steiner, D.F, Katsoyannis, P.G, Weiss, M.A.
登録日2007-09-05
公開日2007-10-16
最終更新日2021-10-20
実験手法SOLUTION NMR
主引用文献The A-chain of Insulin Contacts the Insert Domain of the Insulin Receptor: PHOTO-CROSS-LINKING AND MUTAGENESIS OF A DIABETES-RELATED CREVICE.
J.Biol.Chem., 282, 2007
3F7T
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Structure of active IspH shows a novel fold with a [3Fe-4S] cluster in the catalytic centre
分子名称: 4-hydroxy-3-methylbut-2-enyl diphosphate reductase, FE3-S4 CLUSTER, PHOSPHATE ION, ...
著者Graewert, T, Eppinger, J, Rohdich, F, Bacher, A, Eisenreich, W, Groll, M.
登録日2008-11-10
公開日2009-07-07
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structure of active IspH enzyme from Escherichia coli provides mechanistic insights into substrate reduction.
Angew.Chem.Int.Ed.Engl., 48, 2009
3F1J
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Crystal structure of the Borna disease virus matrix protein (BDV-M) reveals RNA binding properties
分子名称: CYTIDINE-5'-MONOPHOSPHATE, Matrix protein, SULFATE ION
著者Neumann, P, Lieber, D, Meyer, S, Dautel, P, Kerth, A, Kraus, I, Garten, W, Stubbs, M.T.
登録日2008-10-28
公開日2009-02-03
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.65 Å)
主引用文献Crystal structure of the Borna disease virus matrix protein (BDV-M) reveals ssRNA binding properties
Proc.Natl.Acad.Sci.USA, 106, 2009
2JPC
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SSRB DNA Binding Protein
分子名称: SsrB
著者Liao, X, Kenney, L, Sheng, W, Integrated Center for Structure and Function Innovation (ISFI)
登録日2007-05-03
公開日2007-07-03
最終更新日2023-12-20
実験手法SOLUTION NMR
主引用文献SSRB DNA Binding Protein
To be Published
3FK2
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Crystal structure of the RhoGAP domain of human glucocorticoid receptor DNA-binding factor 1
分子名称: Glucocorticoid receptor DNA-binding factor 1, UNKNOWN ATOM OR ION
著者Nedyalkova, L, Tong, Y, Tempel, W, Loppnau, P, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Weigelt, J, Bochkarev, A, Park, H, Structural Genomics Consortium (SGC)
登録日2008-12-15
公開日2008-12-23
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Crystal structure of the RhoGAP domain of human glucocorticoid receptor DNA-binding factor 1
To be Published
3HTQ
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the hemagglutinin structure of an avian H1N1 influenza A virus in complex with LSTc
分子名称: 2-acetamido-2-deoxy-alpha-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose, Hemagglutinin, ...
著者Wang, G, Li, A, Zhang, Q, Wu, C, Zhang, R, Cai, Q, Song, W, Yuen, K.-Y.
登録日2009-06-12
公開日2009-08-11
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.955 Å)
主引用文献The hemagglutinin structure of an avian H1N1 influenza A virus
Virology, 392, 2009
7YOA
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High-resolution crystal structure of the mouse alpha-defensin cryptdin 14
分子名称: Alpha-defensin 14, SULFATE ION
著者Yang, Y, Lu, W.
登録日2022-08-01
公開日2022-11-30
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.67 Å)
主引用文献Mouse alpha-Defensins: Structural and Functional Analysis of the 17 Cryptdin Isoforms Identified from a Single Jejunal Crypt.
Infect.Immun., 91, 2023
3F5K
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Semi-active E176Q mutant of rice BGlu1, a plant exoglucanase/beta-glucosidase
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, Beta-glucosidase, GLYCEROL, ...
著者Chuenchor, W, Ketudat Cairns, J.R, Pengthaisong, S, Robinson, R.C, Yuvaniyama, J, Chen, C.-J.
登録日2008-11-03
公開日2009-11-03
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献The structural basis of oligosaccharide binding by rice BGlu1 beta-glucosidase
J.Struct.Biol., 173, 2011
3HXI
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Crystal structure of Schistosome eIF4E complexed with m7GpppG and 4E-BP
分子名称: 7-METHYL-GUANOSINE-5'-TRIPHOSPHATE-5'-GUANOSINE, Eukaryotic Translation Initiation 4E, Eukaryotic translation initiation factor 4E-binding protein 1
著者Liu, W, Zhao, R, Jones, D.N.M, Davis, R.E.
登録日2009-06-20
公開日2009-08-25
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structural insights into parasite EIF4E binding specificity for m7G and m2,2,7G mRNA cap.
J.Biol.Chem., 284, 2009
2K20
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Solution structure of Par-3 PDZ3 in complex with PTEN peptide
分子名称: Partitioning-defective 3 homolog, Protein tyrosine phosphatase and tensin homolog
著者Feng, W, Wu, H, Chan, L, Zhang, M.
登録日2008-03-18
公開日2008-06-10
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of Par-3 PDZ3 in complex with PTEN peptide
To be Published

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