2XIZ
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![BU of 2xiz by Molmil](/molmil-images/mine/2xiz) | Protein kinase Pim-1 in complex with fragment-3 from crystallographic fragment screen | 分子名称: | (E)-PYRIDIN-4-YL-ACRYLIC ACID, PROTO-ONCOGENE SERINE/THREONINE PROTEIN KINASE PIM-1 | 著者 | Schulz, M.N, Fanghanel, J, Schafer, M, Badock, V, Briem, H, Boemer, U, Nguyen, D, Husemann, M, Hillig, R.C. | 登録日 | 2010-07-01 | 公開日 | 2011-02-23 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (2.21 Å) | 主引用文献 | Crystallographic Fragment Screen Identifies Cinnamic Acid Derivatives as Starting Points for Potent Pim-1 Inhibitors Acta Crystallogr.,Sect.D, 67, 2011
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2XIX
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![BU of 2xix by Molmil](/molmil-images/mine/2xix) | Protein kinase Pim-1 in complex with fragment-1 from crystallographic fragment screen | 分子名称: | 3,5-DIAMINO-1H-[1,2,4]TRIAZOLE, PROTO-ONCOGENE SERINE/THREONINE-PROTEIN KINASE PIM-1 | 著者 | Schulz, M.N, Fanghanel, J, Schafer, M, Badock, V, Briem, H, Boemer, U, Nguyen, D, Husemann, M, Hillig, R.C. | 登録日 | 2010-07-01 | 公開日 | 2011-02-23 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Crystallographic Fragment Screen Identifies Cinnamic Acid Derivatives as Starting Points for Potent Pim-1 Inhibitors Acta Crystallogr.,Sect.D, 67, 2011
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6UNX
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![BU of 6unx by Molmil](/molmil-images/mine/6unx) | Structure of E. coli FtsZ(L178E)-GTP complex | 分子名称: | Cell division protein FtsZ, GUANOSINE-5'-TRIPHOSPHATE | 著者 | Schumacher, M.A. | 登録日 | 2019-10-13 | 公開日 | 2020-02-05 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | High-resolution crystal structures of Escherichia coli FtsZ bound to GDP and GTP. Acta Crystallogr.,Sect.F, 76, 2020
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5KEC
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![BU of 5kec by Molmil](/molmil-images/mine/5kec) | Structure of K. pneumonia MrkH in its apo state. | 分子名称: | Flagellar brake protein YcgR | 著者 | Schumacher, M. | 登録日 | 2016-06-09 | 公開日 | 2016-08-17 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.949 Å) | 主引用文献 | to be published:
Structures of K. pneumonia MrkH: dual utilization of the PilZ fold for c-di-GMP and DNA binding by a novel activator of biofilm genes To Be Published
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4OAY
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![BU of 4oay by Molmil](/molmil-images/mine/4oay) | BldD CTD-c-di-GMP complex | 分子名称: | 9,9'-[(2R,3R,3aS,5S,7aR,9R,10R,10aS,12S,14aR)-3,5,10,12-tetrahydroxy-5,12-dioxidooctahydro-2H,7H-difuro[3,2-d:3',2'-j][1,3,7,9,2,8]tetraoxadiphosphacyclododecine-2,9-diyl]bis(2-amino-1,9-dihydro-6H-purin-6-one), DNA-binding protein | 著者 | Schumacher, M.A, Tschowri, N, Buttner, M, Brennan, R.G. | 登録日 | 2014-01-06 | 公開日 | 2014-11-19 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Tetrameric c-di-GMP mediates effective transcription factor dimerization to control Streptomyces development. Cell(Cambridge,Mass.), 158, 2014
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5KED
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![BU of 5ked by Molmil](/molmil-images/mine/5ked) | |
4PQL
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![BU of 4pql by Molmil](/molmil-images/mine/4pql) | |
2LIQ
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![BU of 2liq by Molmil](/molmil-images/mine/2liq) | Solution structure of CCL2 in complex with glycan | 分子名称: | CCL2 lectin, alpha-L-fucopyranose-(1-3)-[2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)]methyl 2-acetamido-2-deoxy-beta-D-glucopyranoside | 著者 | Schubert, M, Bleuler-Martinez, S, Walti, M.A, Egloff, P, Aebi, M, Kuenzler, M, Allain, F.H.-T. | 登録日 | 2011-08-30 | 公開日 | 2012-06-06 | 最終更新日 | 2024-05-15 | 実験手法 | SOLUTION NMR | 主引用文献 | Plasticity of the beta-Trefoil Protein Fold in the Recognition and Control of Invertebrate Predators and Parasites by a Fungal Defence System Plos Pathog., 8, 2012
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2LIE
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![BU of 2lie by Molmil](/molmil-images/mine/2lie) | NMR structure of the lectin CCL2 | 分子名称: | CCL2 lectin | 著者 | Schubert, M, Walti, M.A, Egloff, P, Bleuler-Martinez, S, Aebi, M, Allain, F.F.-H, Kunzler, M. | 登録日 | 2011-08-29 | 公開日 | 2012-06-06 | 最終更新日 | 2024-05-15 | 実験手法 | SOLUTION NMR | 主引用文献 | Plasticity of the beta-Trefoil Protein Fold in the Recognition and Control of Invertebrate Predators and Parasites by a Fungal Defence System Plos Pathog., 8, 2012
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1UPF
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![BU of 1upf by Molmil](/molmil-images/mine/1upf) | STRUCTURE OF THE URACIL PHOSPHORIBOSYLTRANSFERASE, MUTANT C128V BOUND TO THE DRUG 5-FLUOROURACIL | 分子名称: | 5-FLUOROURACIL, SULFATE ION, URACIL PHOSPHORIBOSYLTRANSFERASE | 著者 | Schumacher, M.A, Carter, D, Scott, D, Roos, D, Ullman, B, Brennan, R.G. | 登録日 | 1998-06-17 | 公開日 | 1999-06-22 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Crystal structures of Toxoplasma gondii uracil phosphoribosyltransferase reveal the atomic basis of pyrimidine discrimination and prodrug binding. EMBO J., 17, 1998
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8T5Y
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![BU of 8t5y by Molmil](/molmil-images/mine/8t5y) | |
4PTA
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![BU of 4pta by Molmil](/molmil-images/mine/4pta) | Structure of MDR initiator | 分子名称: | Replication initiator protein | 著者 | Schumacher, M.A. | 登録日 | 2014-03-10 | 公開日 | 2014-06-25 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.6003 Å) | 主引用文献 | Mechanism of staphylococcal multiresistance plasmid replication origin assembly by the RepA protein. Proc.Natl.Acad.Sci.USA, 111, 2014
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3HZI
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![BU of 3hzi by Molmil](/molmil-images/mine/3hzi) | Structure of mdt protein | 分子名称: | 5'-D(*DAP*DCP*DTP*DAP*DTP*DCP*DCP*DCP*DCP*DTP*DTP*DAP*DAP*DGP*DGP*DGP*DGP*DAP*DTP*DAP*DG)-3', ADENOSINE-5'-TRIPHOSPHATE, HTH-type transcriptional regulator hipB, ... | 著者 | Schumacher, M.A. | 登録日 | 2009-06-23 | 公開日 | 2009-07-28 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.98 Å) | 主引用文献 | Molecular mechanisms of HipA-mediated multidrug tolerance and its neutralization by HipB. Science, 323, 2009
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3MKY
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![BU of 3mky by Molmil](/molmil-images/mine/3mky) | Structure of SopB(155-323)-18mer DNA complex, I23 form | 分子名称: | DNA (5'-D(*CP*TP*GP*GP*GP*AP*CP*CP*AP*TP*GP*GP*TP*CP*CP*CP*AP*G)-3'), Protein sopB, SULFATE ION | 著者 | Schumacher, M.A, Piro, K, Xu, W. | 登録日 | 2010-04-15 | 公開日 | 2010-05-05 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.86 Å) | 主引用文献 | Insight into F plasmid DNA segregation revealed by structures of SopB and SopB-DNA complexes. Nucleic Acids Res., 38, 2010
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4PQK
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![BU of 4pqk by Molmil](/molmil-images/mine/4pqk) | C-Terminal domain of DNA binding protein | 分子名称: | Maltose ABC transporter periplasmic protein, Truncated replication protein RepA, alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose | 著者 | Schumacher, M.A, Chinnam, N, Tonthat, N.K. | 登録日 | 2014-03-03 | 公開日 | 2014-06-18 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (3.401 Å) | 主引用文献 | Mechanism of staphylococcal multiresistance plasmid replication origin assembly by the RepA protein. Proc.Natl.Acad.Sci.USA, 111, 2014
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4PT7
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![BU of 4pt7 by Molmil](/molmil-images/mine/4pt7) | Structure of initiator | 分子名称: | Replication initiator A family protein, SULFATE ION | 著者 | Schumacher, M.A. | 登録日 | 2014-03-10 | 公開日 | 2014-06-25 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.35 Å) | 主引用文献 | Mechanism of staphylococcal multiresistance plasmid replication origin assembly by the RepA protein. Proc.Natl.Acad.Sci.USA, 111, 2014
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2NOQ
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![BU of 2noq by Molmil](/molmil-images/mine/2noq) | Structure of ribosome-bound cricket paralysis virus IRES RNA | 分子名称: | 18S ribosomal RNA, 25S ribosomal RNA, 40S ribosomal protein S5, ... | 著者 | Schuler, M, Connell, S.R, Lescoute, A, Giesebrecht, J, Dabrowski, M, Schroeer, B, Mielke, T, Penczek, P.A, Westhof, E, Spahn, C.M.T. | 登録日 | 2006-10-26 | 公開日 | 2006-11-21 | 最終更新日 | 2023-12-27 | 実験手法 | ELECTRON MICROSCOPY (7.3 Å) | 主引用文献 | Structure of the ribosome-bound cricket paralysis virus IRES RNA. Nat.Struct.Mol.Biol., 13, 2006
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4MCT
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3MKW
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![BU of 3mkw by Molmil](/molmil-images/mine/3mkw) | Structure of sopB(155-272)-18mer complex, I23 form | 分子名称: | DNA (5'-D(*CP*TP*GP*GP*GP*AP*CP*CP*AP*TP*GP*GP*TP*CP*CP*CP*AP*G)-3'), Protein sopB, SULFATE ION | 著者 | Schumacher, M.A, Piro, K, Xu, W. | 登録日 | 2010-04-15 | 公開日 | 2010-05-05 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.99 Å) | 主引用文献 | Insight into F plasmid DNA segregation revealed by structures of SopB and SopB-DNA complexes. Nucleic Acids Res., 38, 2010
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1UPU
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![BU of 1upu by Molmil](/molmil-images/mine/1upu) | STRUCTURE OF THE URACIL PHOSPHORIBOSYLTRANSFERASE, MUTANT C128V, BOUND TO PRODUCT URIDINE-1-MONOPHOSPHATE (UMP) | 分子名称: | PHOSPHATE ION, URACIL PHOSPHORIBOSYLTRANSFERASE, URIDINE-5'-MONOPHOSPHATE | 著者 | Schumacher, M.A, Carter, D, Scott, D, Roos, D, Ullman, B, Brennan, R.G. | 登録日 | 1998-04-16 | 公開日 | 1999-05-11 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Crystal structures of Toxoplasma gondii uracil phosphoribosyltransferase reveal the atomic basis of pyrimidine discrimination and prodrug binding. EMBO J., 17, 1998
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4S0R
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![BU of 4s0r by Molmil](/molmil-images/mine/4s0r) | Structure of GS-TnrA complex | 分子名称: | GLUTAMINE, Glutamine synthetase, MAGNESIUM ION, ... | 著者 | Schumacher, M.A, Chinnam, N.G, Cuthbert, B, Tonthat, N.K. | 登録日 | 2015-01-04 | 公開日 | 2015-03-04 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (3.5 Å) | 主引用文献 | Structures of regulatory machinery reveal novel molecular mechanisms controlling B. subtilis nitrogen homeostasis. Genes Dev., 29, 2015
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4E07
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![BU of 4e07 by Molmil](/molmil-images/mine/4e07) | ParF-AMPPCP-C2221 form | 分子名称: | PHOSPHOMETHYLPHOSPHONIC ACID ADENYLATE ESTER, Plasmid partitioning protein ParF | 著者 | Schumacher, M.A, Ye, Q, Barge, M.R, Barilla, D, Hayes, F. | 登録日 | 2012-03-02 | 公開日 | 2012-06-13 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Structural Mechanism of ATP-induced Polymerization of the Partition Factor ParF: IMPLICATIONS FOR DNA SEGREGATION. J.Biol.Chem., 287, 2012
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2MK1
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![BU of 2mk1 by Molmil](/molmil-images/mine/2mk1) | |
3OQO
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![BU of 3oqo by Molmil](/molmil-images/mine/3oqo) | Ccpa-hpr-ser46p-syn cre | 分子名称: | 5'-D(*CP*TP*GP*AP*AP*AP*GP*CP*GP*CP*TP*AP*AP*CP*AP*G)-3', 5'-D(*CP*TP*GP*TP*TP*AP*GP*CP*GP*CP*TP*TP*TP*CP*AP*G)-3', Catabolite control protein A, ... | 著者 | schumacher, M.A, Sprehe, M, Bartholomae, M, Hillen, W, Brennan, R.G. | 登録日 | 2010-09-03 | 公開日 | 2011-10-26 | 最終更新日 | 2014-04-09 | 実験手法 | X-RAY DIFFRACTION (2.97 Å) | 主引用文献 | Structures of carbon catabolite protein A-(HPr-Ser46-P) bound to diverse catabolite response element sites reveal the basis for high-affinity binding to degenerate DNA operators. Nucleic Acids Res., 39, 2011
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4OB4
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![BU of 4ob4 by Molmil](/molmil-images/mine/4ob4) | Structure of the S. venezulae BldD DNA-binding domain | 分子名称: | Putative DNA-binding protein | 著者 | schumacher, M.A, Tschowri, N, Buttner, M, Brennan, R. | 登録日 | 2014-01-06 | 公開日 | 2014-11-19 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Tetrameric c-di-GMP mediates effective transcription factor dimerization to control Streptomyces development. Cell(Cambridge,Mass.), 158, 2014
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