Loading
PDBj
メニューPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help
PDB: 2930 件

1RZ9
DownloadVisualize
BU of 1rz9 by Molmil
Crystal Structure of AAV Rep complexed with the Rep-binding sequence
分子名称: 26-MER, Rep protein
著者Hickman, A.B, Ronning, D.R, Perez, Z.N, Kotin, R.M, Dyda, F.
登録日2003-12-24
公開日2004-02-17
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献The nuclease domain of adeno-associated virus rep coordinates replication initiation using two distinct DNA recognition interfaces.
Mol.Cell, 13, 2004
2H5F
DownloadVisualize
BU of 2h5f by Molmil
Denmotoxin: A the three-finger toxin from colubrid snake Boiga dendrophila with bird-specific activity
分子名称: PHOSPHATE ION, POTASSIUM ION, SODIUM ION, ...
著者Pawlak, J, Kini, R.M, Stura, E.A.
登録日2006-05-26
公開日2006-08-29
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Denmotoxin, a three-finger toxin from the colubrid snake Boiga dendrophila (Mangrove Catsnake) with bird-specific activity.
J.Biol.Chem., 281, 2006
4K5Y
DownloadVisualize
BU of 4k5y by Molmil
Crystal structure of human corticotropin-releasing factor receptor 1 (CRF1R) in complex with the antagonist CP-376395
分子名称: (1R)-2-{[(S)-{[(2S)-2,3-dihydroxypropyl]oxy}(hydroxy)phosphoryl]oxy}-1-[(hexadecanoyloxy)methyl]ethyl (9Z)-octadec-9-enoate, (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, 3,6-dimethyl-N-(pentan-3-yl)-2-(2,4,6-trimethylphenoxy)pyridin-4-amine, ...
著者Hollenstein, K, Kean, J, Bortolato, A, Cheng, R.K.Y, Dore, A.S, Jazayeri, A, Cooke, R.M, Weir, M, Marshall, F.H.
登録日2013-04-15
公開日2013-07-17
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.977 Å)
主引用文献Structure of class B GPCR corticotropin-releasing factor receptor 1.
Nature, 499, 2013
2F2B
DownloadVisualize
BU of 2f2b by Molmil
Crystal structure of integral membrane protein Aquaporin AqpM at 1.68A resolution
分子名称: Aquaporin aqpM, GLYCEROL
著者Lee, J.K, Kozono, D, Remis, J, Kitagawa, Y, Agre, P, Stroud, R.M, Center for Structures of Membrane Proteins (CSMP)
登録日2005-11-15
公開日2005-12-06
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.68 Å)
主引用文献Structural basis for conductance by the archaeal aquaporin AqpM at 1.68 A.
Proc.Natl.Acad.Sci.Usa, 102, 2005
3ZIR
DownloadVisualize
BU of 3zir by Molmil
minor-site specific NLS (B141)
分子名称: B141NLS, IMPORTIN SUBUNIT ALPHA-2
著者Chang, C.-W, Counago, R.M, Williams, S.J, Kobe, B.
登録日2013-01-10
公開日2013-08-21
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Distinctive Conformation of Minor Site-Specific Nuclear Localization Signals Bound to Importin-Alpha
Traffic, 14, 2013
2FLZ
DownloadVisualize
BU of 2flz by Molmil
The X-ray structure of cis-3-chloroacrylic acid dehalogenase (cis-CaaD) with a sulfate ion bound in the active site
分子名称: SULFATE ION, cis-3-chloroacrylic acid dehalogenase
著者de Jong, R.M.
登録日2006-01-06
公開日2006-11-21
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.75 Å)
主引用文献Crystal Structures of Native and Inactivated cis-3-Chloroacrylic Acid Dehalogenase: STRUCTURAL BASIS FOR SUBSTRATE SPECIFICITY AND INACTIVATION BY (R)-OXIRANE-2-CARBOXYLATE.
J.Biol.Chem., 282, 2007
2H8M
DownloadVisualize
BU of 2h8m by Molmil
N-Domain Of Grp94 In Complex With the 2-Iodo-NECA
分子名称: (2S,3S,4R,5R)-5-(6-AMINO-2-IODO-9H-PURIN-9-YL)-N-ETHYL-3,4-DIHYDROXYTETRAHYDROFURAN-2-CARBOXAMIDE, Endoplasmin, PENTAETHYLENE GLYCOL, ...
著者Immormino, R.M, Gewirth, D.T.
登録日2006-06-07
公開日2007-04-24
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献N-Domain Of Grp94 In Complex With the 2-Iodo-NECA
To be Published
5G47
DownloadVisualize
BU of 5g47 by Molmil
Structure of Gc glycoprotein from severe fever with thrombocytopenia syndrome virus in the trimeric postfusion conformation
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, CHLORIDE ION, SFTSV GC
著者Halldorsson, S, Behrens, A.J, Harlos, K, Huiskonen, J.T, Elliott, R.M, Crispin, M, Brennan, B, Bowden, T.A.
登録日2016-05-05
公開日2016-07-06
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献Structure of a Phleboviral Envelope Glycoprotein Reveals a Consolidated Model of Membrane Fusion.
Proc.Natl.Acad.Sci.USA, 113, 2016
5GWB
DownloadVisualize
BU of 5gwb by Molmil
Hen Egg White Lysozyme native crystals soaked for 2 hours in precipitant solution containing 1 M guanidine hydrochloride and 25% glycerol, before data collection
分子名称: CHLORIDE ION, GUANIDINE, Lysozyme C
著者Hosur, M.V, Kini, R.M, Yeow, C.
登録日2016-09-10
公開日2017-09-13
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.001 Å)
主引用文献Hen Egg White Lysozyme native crystals soaked for 2 hours in precipitant solution containing 1 M guanidine hydrochloride and 25% glycerol, before data collection
To Be Published
2H55
DownloadVisualize
BU of 2h55 by Molmil
Structure of human Hsp90-alpha bound to the potent water soluble inhibitor PU-DZ8
分子名称: 2-FLUORO-8-[(6-IODO-1,3-BENZODIOXOL-5-YL)METHYL]-9-[3-(ISOPROPYLAMINO)PROPYL]-9H-PURIN-6-AMINE, Heat shock protein HSP 90-alpha 4
著者Immormino, R.M, Gewirth, D.T.
登録日2006-05-25
公開日2006-10-03
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural and quantum chemical studies of 8-aryl-sulfanyl adenine class Hsp90 inhibitors.
J.Med.Chem., 49, 2006
4LYA
DownloadVisualize
BU of 4lya by Molmil
EssC (ATPases 2 and 3) from Geobacillus thermodenitrificans (SeMet)
分子名称: ADENOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, Uncharacterized protein
著者Dovala, D.L, Bendebury, A, Cox, J.S, Stroud, R.M, Rosenberg, O.S.
登録日2013-07-30
公開日2015-02-04
最終更新日2016-09-21
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献Substrates Control Multimerization and Activation of the Multi-Domain ATPase Motor of Type VII Secretion.
Cell(Cambridge,Mass.), 161, 2015
2HCH
DownloadVisualize
BU of 2hch by Molmil
N-Domain Of Grp94 In Complex With the Novel Ligand N-(2-amino)ethyl Carboxyamido Adenosine
分子名称: 5'-N-[(2-AMINO)ETHYL CARBOXAMIDO] ADENOSINE, Endoplasmin, PENTAETHYLENE GLYCOL, ...
著者Immormino, R.M, Gewirth, D.T.
登録日2006-06-16
公開日2007-05-01
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献N-Domain Of Grp94 In Complex With the Novel Ligand N-aminoethyl Carboxyamido Adenosine
To be Published
7E9F
DownloadVisualize
BU of 7e9f by Molmil
Cryo-EM structure of the 2:1 Orc1 BAH domain in complex with nucleosome
分子名称: DNA (147-mer), Histone H2A.2, Histone H2B.2, ...
著者Jiang, H, Yu, C, Liu, C.P, Han, X, Yu, Z, Xu, R.M.
登録日2021-03-04
公開日2022-09-07
実験手法ELECTRON MICROSCOPY (4 Å)
主引用文献Nucleosome binding relinquishes the association of the BAH domain of Orc1 with Sir1
To Be Published
7E9C
DownloadVisualize
BU of 7e9c by Molmil
Cryo-EM structure of the 1:1 Orc1 BAH domain in complex with nucleosome
分子名称: DNA (147-mer), Histone H2A.2, Histone H2B.2, ...
著者Jiang, H, Yu, C, Liu, C.P, Han, X, Yu, Z, Xu, R.M.
登録日2021-03-04
公開日2022-09-07
実験手法ELECTRON MICROSCOPY (3.5 Å)
主引用文献Nucleosome binding relinquishes the association of the BAH domain of Orc1 with Sir1
To Be Published
3DM9
DownloadVisualize
BU of 3dm9 by Molmil
Structures and Conformations in Solution of the Signal Recognition Particle Receptor from the archaeon Pyrococcus furiosus
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, PHOSPHATE ION, Signal recognition particle receptor
著者Egea, P.F, Tsuruta, H, Napetschnig, J, Walter, P, Stroud, R.M.
登録日2008-06-30
公開日2008-11-11
最終更新日2017-10-25
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structures of the Signal Recognition Particle Receptor from the Archaeon Pyrococcus furiosus: Implications for the Targeting Step at the Membrane.
Plos One, 3, 2008
2EVU
DownloadVisualize
BU of 2evu by Molmil
Crystal structure of aquaporin AqpM at 2.3A resolution
分子名称: Aquaporin aqpM, GLYCEROL, octyl beta-D-glucopyranoside
著者Lee, J.K, Kozono, D, Remis, J, Kitagawa, Y, Agre, P, Stroud, R.M, Center for Structures of Membrane Proteins (CSMP)
登録日2005-10-31
公開日2005-12-06
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structural basis for conductance by the archaeal aquaporin AqpM at 1.68 A.
Proc.Natl.Acad.Sci.Usa, 102, 2005
3DL0
DownloadVisualize
BU of 3dl0 by Molmil
Crystal structure of adenylate kinase variant AKlse3
分子名称: Adenylate kinase, BIS(ADENOSINE)-5'-PENTAPHOSPHATE, MAGNESIUM ION, ...
著者Bannen, R.M, Bianchetti, C.M, Bingman, C.A, McCoy, J.G.
登録日2008-06-26
公開日2009-06-09
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.58 Å)
主引用文献Effectiveness and limitations of local structural entropy optimization in the thermal stabilization of mesophilic and thermophilic adenylate kinases.
Proteins, 82, 2014
4CT1
DownloadVisualize
BU of 4ct1 by Molmil
Human PDK1-PKCzeta Kinase Chimera in Complex with Allosteric Compound PS315 Bound to the PIF-Pocket
分子名称: (2Z)-3-(biphenyl-4-yl)-5-(4-chlorophenyl)pent-2-enoic acid, 3-PHOSPHOINOSITIDE-DEPENDENT PROTEIN KINASE 1, ADENOSINE-5'-TRIPHOSPHATE, ...
著者Schulze, J.O, Zhang, H, Lopez-Garcia, L.A, Biondi, R.M.
登録日2014-03-11
公開日2014-05-28
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Molecular Mechanism of Regulation of the Atypical Protein Kinase C by N-Terminal Domains and an Allosteric Small Compound.
Chem.Biol., 21, 2014
1RML
DownloadVisualize
BU of 1rml by Molmil
NMR STUDY OF ACID FIBROBLAST GROWTH FACTOR BOUND TO 1,3,6-NAPHTHALENE TRISULPHONATE, 26 STRUCTURES
分子名称: ACIDIC FIBROBLAST GROWTH FACTOR, NAPHTHALENE TRISULFONATE
著者Lozano, R.M, Jimenez, M.A, Santoro, J, Rico, M, Gimenez-Gallego, G.
登録日1998-05-21
公開日1998-11-11
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Solution structure of acidic fibroblast growth factor bound to 1,3, 6-naphthalenetrisulfonate: a minimal model for the anti-tumoral action of suramins and suradistas.
J.Mol.Biol., 281, 1998
4LXJ
DownloadVisualize
BU of 4lxj by Molmil
Saccharomyces cerevisiae lanosterol 14-alpha demethylase with lanosterol bound
分子名称: LANOSTEROL, Lanosterol 14-alpha demethylase, OXYGEN MOLECULE, ...
著者Monk, B.C, Tomasiak, T.M, Keniya, M.V, Huschmann, F.U, Tyndall, J.D.A, O'Connell III, J.D, Cannon, R.D, McDonald, J, Rodriguez, A, Finer-Moore, J, Stroud, R.M.
登録日2013-07-29
公開日2014-01-29
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Architecture of a single membrane spanning cytochrome P450 suggests constraints that orient the catalytic domain relative to a bilayer.
Proc.Natl.Acad.Sci.USA, 111, 2014
4MAO
DownloadVisualize
BU of 4mao by Molmil
RSK2 T493M C-Terminal Kinase Domain in Complex with RMM58
分子名称: (2Z)-2-(1H-1,2,4-triazol-1-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1H-indazol-5-yl]prop-2-enenitrile, Ribosomal protein S6 kinase alpha-3, SODIUM ION
著者Miller, R.M, Taunton, J.
登録日2013-08-16
公開日2014-10-22
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Design of reversible, cysteine-targeted Michael acceptors guided by kinetic and computational analysis.
J.Am.Chem.Soc., 136, 2014
4CT2
DownloadVisualize
BU of 4ct2 by Molmil
Human PDK1-PKCzeta Kinase Chimera
分子名称: 3-PHOSPHOINOSITIDE-DEPENDENT PROTEIN KINASE 1, ADENOSINE-5'-TRIPHOSPHATE, DITHIANE DIOL, ...
著者Schulze, J.O, Zhang, H, Lopez-Garcia, L.A, Biondi, R.M.
登録日2014-03-11
公開日2014-05-28
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.25 Å)
主引用文献Molecular Mechanism of Regulation of the Atypical Protein Kinase C by N-Terminal Domains and an Allosteric Small Compound.
Chem.Biol., 21, 2014
4M55
DownloadVisualize
BU of 4m55 by Molmil
Crystal structure of Human UDP-xylose synthase R236H substitution
分子名称: NICOTINAMIDE-ADENINE-DINUCLEOTIDE, PYROPHOSPHATE 2-, SULFATE ION, ...
著者Walsh Jr, R.M, Polizzi, S.J, Wood, Z.A.
登録日2013-08-08
公開日2013-08-28
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.86 Å)
主引用文献Man o' war mutation in UDP-alpha-D-xylose synthase favors the abortive catalytic cycle and uncovers a latent potential for hexamer formation.
Biochemistry, 54, 2015
4JG6
DownloadVisualize
BU of 4jg6 by Molmil
RSK2 CTD bound to 2-cyano-3-(1H-indazol-5-yl)acrylamide
分子名称: (2S)-2-cyano-3-(1H-indazol-5-yl)propanamide, Ribosomal protein S6 kinase alpha-3, SODIUM ION
著者Miller, R.M, Paavilainen, V.O, Krishnan, S, Serafimova, I.M, Taunton, J.
登録日2013-02-28
公開日2013-04-10
最終更新日2013-04-24
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Electrophilic fragment-based design of reversible covalent kinase inhibitors.
J.Am.Chem.Soc., 135, 2013
3DZE
DownloadVisualize
BU of 3dze by Molmil
Crystal structure of bovine coupling Factor B bound with cadmium
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, ATP synthase subunit s, mitochondrial, ...
著者Lee, J.K, Stroud, R.M, Belogrudov, G.I.
登録日2008-07-29
公開日2008-08-19
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.15 Å)
主引用文献Crystal structure of bovine mitochondrial factor B at 0.96-A resolution.
Proc.Natl.Acad.Sci.Usa, 105, 2008

222926

件を2024-07-24に公開中

PDB statisticsPDBj update infoContact PDBjnumon