1UDI
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1GOW
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1QNL
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1QO0
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1UDH
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1UDG
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1LAU
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![BU of 1lau by Molmil](/molmil-images/mine/1lau) | URACIL-DNA GLYCOSYLASE | 分子名称: | DNA (5'-D(*TP*TP*T)-3'), PROTEIN (URACIL-DNA GLYCOSYLASE (E.C.3.2.2.-)) | 著者 | Pearl, L.H, Savva, R. | 登録日 | 1996-01-03 | 公開日 | 1996-06-10 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | The structural basis of specific base-excision repair by uracil-DNA glycosylase. Nature, 373, 1995
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1PEA
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1GXR
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![BU of 1gxr by Molmil](/molmil-images/mine/1gxr) | WD40 Region of Human Groucho/TLE1 | 分子名称: | CALCIUM ION, TRANSDUCIN-LIKE ENHANCER PROTEIN 1 | 著者 | Pearl, L.H, Roe, S.M, Pickles, L.M. | 登録日 | 2002-04-10 | 公開日 | 2002-06-13 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | Crystal Structure of the C-Terminal Wd40 Repeat Domain of the Human Groucho/Tle1 Transcriptional Corepressor Structure, 10, 2002
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4APE
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![BU of 4ape by Molmil](/molmil-images/mine/4ape) | THE ACTIVE SITE OF ASPARTIC PROTEINASES | 分子名称: | ENDOTHIAPEPSIN | 著者 | Pearl, L.H, Sewell, B.T, Jenkins, J.A, Cooper, J.B, Blundell, T.L. | 登録日 | 1986-06-09 | 公開日 | 1986-07-14 | 最終更新日 | 2019-10-16 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | The Active Site of Aspartic Proteinases FEBS Lett., 174, 1984
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1AM1
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1AMW
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1W4S
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6RML
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![BU of 6rml by Molmil](/molmil-images/mine/6rml) | Crystal structure of TOPBP1 BRCT0,1,2 in complex with a 53BP1 phosphopeptide | 分子名称: | 53BP1, DNA topoisomerase 2-binding protein 1 | 著者 | Day, M, Oliver, A.W, Pearl, L.H. | 登録日 | 2019-05-07 | 公開日 | 2019-06-12 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.81 Å) | 主引用文献 | Phosphorylation-mediated interactions with TOPBP1 couple 53BP1 and 9-1-1 to control the G1 DNA damage checkpoint. Elife, 8, 2019
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8OK2
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![BU of 8ok2 by Molmil](/molmil-images/mine/8ok2) | Bipartite interaction of TOPBP1 with the GINS complex | 分子名称: | DNA replication complex GINS protein PSF1, DNA replication complex GINS protein PSF2, DNA replication complex GINS protein PSF3, ... | 著者 | Day, M, Oliver, A.W, Pearl, L.H. | 登録日 | 2023-03-26 | 公開日 | 2024-03-13 | 実験手法 | ELECTRON MICROSCOPY (4.1 Å) | 主引用文献 | TopBP1 utilises a bipartite GINS binding mode to support genome replication. Nat Commun, 15, 2024
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5HY6
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6FO1
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![BU of 6fo1 by Molmil](/molmil-images/mine/6fo1) | Human R2TP subcomplex containing 1 RUVBL1-RUVBL2 hexamer bound to 1 RBD domain from RPAP3. | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, RNA polymerase II-associated protein 3, RuvB-like 1, ... | 著者 | Martino, F, Munoz-Hernandez, H, Rodriguez, C.F, Pearl, L.H, Llorca, O. | 登録日 | 2018-02-05 | 公開日 | 2018-04-04 | 最終更新日 | 2019-12-11 | 実験手法 | ELECTRON MICROSCOPY (3.57 Å) | 主引用文献 | RPAP3 provides a flexible scaffold for coupling HSP90 to the human R2TP co-chaperone complex. Nat Commun, 9, 2018
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5LOH
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![BU of 5loh by Molmil](/molmil-images/mine/5loh) | Kinase domain of human Greatwall | 分子名称: | 1,2-ETHANEDIOL, CHLORIDE ION, STAUROSPORINE, ... | 著者 | Rajasekaran, M.B, Pearl, L.H, Oliver, A.W. | 登録日 | 2016-08-09 | 公開日 | 2016-09-07 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | A first generation inhibitor of human Greatwall kinase, enabled by structural and functional characterisation of a minimal kinase domain construct. Oncotarget, 7, 2016
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7Z6H
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![BU of 7z6h by Molmil](/molmil-images/mine/7z6h) | Structure of DNA-bound human RAD17-RFC clamp loader and 9-1-1 checkpoint clamp | 分子名称: | Cell cycle checkpoint control protein RAD9A, Cell cycle checkpoint protein RAD1,Cell cycle checkpoint protein RAD17, Checkpoint protein HUS1, ... | 著者 | Day, M, Oliver, A.W, Pearl, L.H. | 登録日 | 2022-03-11 | 公開日 | 2022-05-04 | 最終更新日 | 2022-08-31 | 実験手法 | ELECTRON MICROSCOPY (3.59 Å) | 主引用文献 | Structure of the human RAD17-RFC clamp loader and 9-1-1 checkpoint clamp bound to a dsDNA-ssDNA junction. Nucleic Acids Res., 50, 2022
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1MUG
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![BU of 1mug by Molmil](/molmil-images/mine/1mug) | G:T/U MISMATCH-SPECIFIC DNA GLYCOSYLASE FROM E.COLI | 分子名称: | PROTEIN (G:T/U SPECIFIC DNA GLYCOSYLASE), SULFATE ION | 著者 | Barrett, T.E, Savva, R, Panayotou, G, Brown, T, Barlow, T, Jiricny, J, Pearl, L.H. | 登録日 | 1998-07-10 | 公開日 | 1998-07-15 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Crystal structure of a G:T/U mismatch-specific DNA glycosylase: mismatch recognition by complementary-strand interactions. Cell(Cambridge,Mass.), 92, 1998
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1MWJ
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![BU of 1mwj by Molmil](/molmil-images/mine/1mwj) | Crystal Structure of a MUG-DNA pseudo substrate complex | 分子名称: | 5'-D(*CP*GP*CP*GP*A*GP*(DU)P*TP*CP*GP*CP*G)-3', G/U mismatch-specific DNA glycosylase | 著者 | Barrett, T.E, Scharer, O, Savva, R, Brown, T, Jiricny, J, Verdine, G.L, Pearl, L.H. | 登録日 | 2002-09-30 | 公開日 | 2002-10-11 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.85 Å) | 主引用文献 | Crystal Structure of a thwarted mismatch glycosylase DNA repair complex Embo J., 18, 1999
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1MTL
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![BU of 1mtl by Molmil](/molmil-images/mine/1mtl) | Non-productive MUG-DNA complex | 分子名称: | 5'-D(*CP*GP*CP*GP*AP*GP*(AAB)P*TP*CP*GP*CP*G)-3', G/U mismatch-specific DNA glycosylase | 著者 | Barrett, T.E, Savva, R, Barlow, T, Brown, T, Jiricny, J, Pearl, L.H. | 登録日 | 2002-09-21 | 公開日 | 2002-09-27 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Structure of a DNA base-excision product resembling a cisplatin inter-strand adduct. Nat.Struct.Biol., 5, 1998
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1MWI
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![BU of 1mwi by Molmil](/molmil-images/mine/1mwi) | Crystal structure of a MUG-DNA product complex | 分子名称: | 5'-D(*CP*GP*CP*GP*AP*GP*(AAB)P*TP*CP*GP*CP*G)-3', G/U mismatch-specific DNA glycosylase | 著者 | Barrett, T.E, Savva, R, Panayotou, G, Brown, T, Barlow, T, Jiricny, J, Pearl, L.H. | 登録日 | 2002-09-30 | 公開日 | 2002-10-04 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.35 Å) | 主引用文献 | Crystal structure of a G:T/U mismatch-specific DNA glycosylase: mismatch recognition by complementary-strand interactions. Cell(Cambridge,Mass.), 92, 1998
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5ECG
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![BU of 5ecg by Molmil](/molmil-images/mine/5ecg) | Crystal structure of the BRCT domains of 53BP1 in complex with p53 and H2AX-pSer139 (gammaH2AX) | 分子名称: | Cellular tumor antigen p53, SEP-GLN-GLU-TYR, Tumor suppressor p53-binding protein 1, ... | 著者 | Day, M, Oliver, A.W, Pearl, L.H. | 登録日 | 2015-10-20 | 公開日 | 2015-12-16 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | ATM Localization and Heterochromatin Repair Depend on Direct Interaction of the 53BP1-BRCT2 Domain with gamma H2AX. Cell Rep, 13, 2015
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4UUH
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![BU of 4uuh by Molmil](/molmil-images/mine/4uuh) | X-ray crystal structure of human TNKS in complex with a small molecule inhibitor | 分子名称: | 1,2-ETHANEDIOL, 5-methyl-3-[4-(piperazin-1-ylmethyl)phenyl]isoquinolin-1(2H)-one, GLYCEROL, ... | 著者 | Oliver, A.W, Rajasekaran, M.B, Pearl, L.H. | 登録日 | 2014-07-28 | 公開日 | 2015-07-08 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.52 Å) | 主引用文献 | Design and Discovery of 3-Aryl-5-Substituted-Isoquinolin-1- Ones as Potent and Selective Tankyrase Inhibitors Medchemcommm, 6, 2015
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