1T9B
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![BU of 1t9b by Molmil](/molmil-images/mine/1t9b) | Crystal structure of yeast acetohydroxyacid synthase in complex with a sulfonylurea herbicide, chlorsulfuron | 分子名称: | 1-(2-CHLOROPHENYLSULFONYL)-3-(4-METHOXY-6-METHYL-L,3,5-TRIAZIN-2-YL)UREA, 2-{[(4-AMINO-2-METHYLPYRIMIDIN-5-YL)METHYL]AMINO}PROPANE-1-THIOL, 5-(AMINOMETHYL)-2-METHYLPYRIMIDIN-4-AMINE, ... | 著者 | McCourt, J.A, Pang, S.S, Guddat, L.W, Duggleby, R.G. | 登録日 | 2004-05-16 | 公開日 | 2004-12-21 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Elucidating the specificity of binding of sulfonylurea herbicides to acetohydroxyacid synthase. Biochemistry, 44, 2005
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1T9D
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![BU of 1t9d by Molmil](/molmil-images/mine/1t9d) | Crystal Structure Of Yeast Acetohydroxyacid Synthase In Complex With A Sulfonylurea Herbicide, Metsulfuron methyl | 分子名称: | 2,5-DIMETHYL-PYRIMIDIN-4-YLAMINE, Acetolactate synthase, mitochondrial, ... | 著者 | McCourt, J.A, Pang, S.S, Guddat, L.W, Duggleby, R.G. | 登録日 | 2004-05-16 | 公開日 | 2004-12-21 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Elucidating the specificity of binding of sulfonylurea herbicides to acetohydroxyacid synthase. Biochemistry, 44, 2005
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4R4Y
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![BU of 4r4y by Molmil](/molmil-images/mine/4r4y) | Structural basis of a point mutation that causes the genetic disease Aspartylglucosaminuria | 分子名称: | N(4)-(Beta-N-acetylglucosaminyl)-L-asparaginase, N-hydroxy-L-asparagine | 著者 | Sui, L, Damodharan, L, Pande, S, Guo, H.C. | 登録日 | 2014-08-20 | 公開日 | 2014-12-17 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structural Basis of a Point Mutation that Causes the Genetic Disease Aspartylglucosaminuria. Structure, 22, 2014
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4XX5
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![BU of 4xx5 by Molmil](/molmil-images/mine/4xx5) | Structure of PI3K gamma in complex with an inhibitor | 分子名称: | N-[5-(5-methoxypyridin-3-yl)-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl]acetamide, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform | 著者 | Collier, P.N, Messersmith, D, Le Tiran, A, Bandarage, U.K, Boucher, C, Come, J, Cottrell, K.M, Damagnez, V, Doran, J.D, Griffith, J.P, Khare-Pandit, S, Krueger, E.B, Ledeboer, M.W, Ledford, B, Liao, Y, Mahajan, S, Moody, C.S, Wang, T, Xu, J, Aronov, A.M. | 登録日 | 2015-01-29 | 公開日 | 2015-08-05 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.76 Å) | 主引用文献 | Structure of PI3K gamma in complex with an inhibitor To Be Published
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4XZ4
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![BU of 4xz4 by Molmil](/molmil-images/mine/4xz4) | Structure of PI3K gamma in complex with an inhibitor | 分子名称: | N-[5-(6-methoxypyrazin-2-yl)-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl]acetamide, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform | 著者 | Collier, P.N, Messersmith, D, Le Tiran, A, Bandarage, U.K, Boucher, C, Come, J, Cottrell, K.M, Damagnez, V, Doran, J.D, Griffith, J.P, Khare-Pandit, S, Krueger, E.B, Ledeboer, M.W, Ledford, B, Liao, Y, Mahajan, S, Moody, C.S, Wang, T, Xu, J, Aronov, A.M. | 登録日 | 2015-02-03 | 公開日 | 2016-02-03 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Structure of PI3K gamma in complex with an inhibitor To Be Published
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9EZ8
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![BU of 9ez8 by Molmil](/molmil-images/mine/9ez8) | Cryo-EM structure of the icosahedral lumazine synthase from Vicia faba. | 分子名称: | 6,7-dimethyl-8-ribityllumazine synthase | 著者 | Chee, M, Trapani, S, Hoh, F, Lai Kee Him, J, Yvon, M, Blanc, S, Bron, P. | 登録日 | 2024-04-11 | 公開日 | 2024-05-22 | 実験手法 | ELECTRON MICROSCOPY (2.7 Å) | 主引用文献 | Cryo-EM structure of the icosahedral lumazine synthase from Vicia faba. To Be Published
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6DG8
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6DG7
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6OJ3
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![BU of 6oj3 by Molmil](/molmil-images/mine/6oj3) | In situ structure of rotavirus VP1 RNA-dependent RNA polymerase (TLP) | 分子名称: | Inner capsid protein VP2, RNA-directed RNA polymerase | 著者 | Jenni, S, Salgado, E.N, Herrmann, T, Li, Z, Grant, T, Grigorieff, N, Trapani, S, Estrozi, L.F, Harrison, S.C. | 登録日 | 2019-04-10 | 公開日 | 2019-04-24 | 最終更新日 | 2024-03-20 | 実験手法 | ELECTRON MICROSCOPY (4.5 Å) | 主引用文献 | In situ Structure of Rotavirus VP1 RNA-Dependent RNA Polymerase. J.Mol.Biol., 431, 2019
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6OJ4
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![BU of 6oj4 by Molmil](/molmil-images/mine/6oj4) | In situ structure of rotavirus VP1 RNA-dependent RNA polymerase (DLP) | 分子名称: | Inner capsid protein VP2, RNA-directed RNA polymerase | 著者 | Jenni, S, Salgado, E.N, Herrmann, T, Li, Z, Grant, T, Grigorieff, N, Trapani, S, Estrozi, L.F, Harrison, S.C. | 登録日 | 2019-04-10 | 公開日 | 2019-04-24 | 最終更新日 | 2024-03-20 | 実験手法 | ELECTRON MICROSCOPY (3.3 Å) | 主引用文献 | In situ Structure of Rotavirus VP1 RNA-Dependent RNA Polymerase. J.Mol.Biol., 431, 2019
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6NP0
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![BU of 6np0 by Molmil](/molmil-images/mine/6np0) | Cryo-EM structure of 5HT3A receptor in presence of granisetron | 分子名称: | 1-methyl-N-[(1R,5S)-9-methyl-9-azabicyclo[3.3.1]nonan-3-yl]indazole-3-carboxamide, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Basak, S, Chakrapani, S. | 登録日 | 2019-01-17 | 公開日 | 2019-07-24 | 最終更新日 | 2020-07-29 | 実験手法 | ELECTRON MICROSCOPY (2.92 Å) | 主引用文献 | Molecular mechanism of setron-mediated inhibition of full-length 5-HT3Areceptor. Nat Commun, 10, 2019
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6OJ5
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![BU of 6oj5 by Molmil](/molmil-images/mine/6oj5) | In situ structure of rotavirus VP1 RNA-dependent RNA polymerase (TLP_RNA) | 分子名称: | Inner capsid protein VP2, RNA-directed RNA polymerase | 著者 | Jenni, S, Salgado, E.N, Herrmann, T, Li, Z, Grant, T, Grigorieff, N, Trapani, S, Estrozi, L.F, Harrison, S.C. | 登録日 | 2019-04-10 | 公開日 | 2019-04-24 | 最終更新日 | 2024-03-20 | 実験手法 | ELECTRON MICROSCOPY (5.2 Å) | 主引用文献 | In situ Structure of Rotavirus VP1 RNA-Dependent RNA Polymerase. J.Mol.Biol., 431, 2019
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6OJ6
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![BU of 6oj6 by Molmil](/molmil-images/mine/6oj6) | In situ structure of rotavirus VP1 RNA-dependent RNA polymerase (DLP_RNA) | 分子名称: | Inner capsid protein VP2, RNA-directed RNA polymerase, Template, ... | 著者 | Jenni, S, Salgado, E.N, Herrmann, T, Li, Z, Grant, T, Grigorieff, N, Trapani, S, Estrozi, L.F, Harrison, S.C. | 登録日 | 2019-04-10 | 公開日 | 2019-04-24 | 最終更新日 | 2024-03-20 | 実験手法 | ELECTRON MICROSCOPY (4.2 Å) | 主引用文献 | In situ Structure of Rotavirus VP1 RNA-Dependent RNA Polymerase. J.Mol.Biol., 431, 2019
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8D4Y
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![BU of 8d4y by Molmil](/molmil-images/mine/8d4y) | C-terminal SANT-SLIDE domain of human Chromodomain-helicase-DNA-binding protein 4 (CHD4) | 分子名称: | Chromodomain-helicase-DNA-binding protein 4 | 著者 | Moghaddas Sani, H, Deshpande, C.N, Panjikar, S, Patel, K, Mackay, J.P. | 登録日 | 2022-06-03 | 公開日 | 2022-12-21 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | The role of auxiliary domains in modulating CHD4 activity suggests mechanistic commonality between enzyme families. Nat Commun, 13, 2022
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7R0J
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![BU of 7r0j by Molmil](/molmil-images/mine/7r0j) | Structure of the V2 receptor Cter-arrestin2-ScFv30 complex | 分子名称: | Arrestin2, ScFv30, V2R Cter | 著者 | Bous, J, Fouillen, A, Trapani, S, Granier, S, Mouillac, B, Bron, P. | 登録日 | 2022-02-02 | 公開日 | 2022-09-14 | 実験手法 | ELECTRON MICROSCOPY (4.23 Å) | 主引用文献 | Structure of the vasopressin hormone-V2 receptor-beta-arrestin1 ternary complex. Sci Adv, 8, 2022
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7R0C
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![BU of 7r0c by Molmil](/molmil-images/mine/7r0c) | Structure of the AVP-V2R-arrestin2-ScFv30 complex | 分子名称: | AVP, Arrestin2, ScFv30, ... | 著者 | Bous, J, Fouillen, A, Trapani, S, Granier, S, Mouillac, B, Bron, P. | 登録日 | 2022-02-01 | 公開日 | 2022-09-14 | 実験手法 | ELECTRON MICROSCOPY (4.73 Å) | 主引用文献 | Structure of the vasopressin hormone-V2 receptor-beta-arrestin1 ternary complex. Sci Adv, 8, 2022
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6PCA
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4XY7
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![BU of 4xy7 by Molmil](/molmil-images/mine/4xy7) | Crystal structure of the complex of ribosome inactivating protein from Momordica balsamina with N-acetylglucosamine at 2.5 A resolution | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, GLYCEROL, Ribosome inactivating protein | 著者 | Yamini, S, Pandey, S, Kaur, P, Sharma, S, Singh, T.P. | 登録日 | 2015-02-02 | 公開日 | 2015-09-23 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Crystal structure of the complex of ribosome inactivating protein from Momordica balsamina with N- acetylglucosamine at 2.5 A resolution To Be Published
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6PCB
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6N5V
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![BU of 6n5v by Molmil](/molmil-images/mine/6n5v) | Crystal Structure of Strictosidine in complex with 1H-indole-4-ethanamine | 分子名称: | 2-(1H-indol-4-yl)ethan-1-amine, Strictosidine synthase | 著者 | Cai, Y, Shao, N, Xie, H, Futamura, Y, Panjikar, S, Liu, H, Zhu, H, Osada, H, Zou, H. | 登録日 | 2018-11-22 | 公開日 | 2019-11-27 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.549 Å) | 主引用文献 | Crystal Structure of Strictosidine in complex with 1H-indole-4-ethanamine to be published
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6UBT
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![BU of 6ubt by Molmil](/molmil-images/mine/6ubt) | |
4WVM
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![BU of 4wvm by Molmil](/molmil-images/mine/4wvm) | Stonustoxin structure | 分子名称: | Stonustoxin subunit alpha, Stonustoxin subunit beta | 著者 | Ellisdon, A.M, Panjikar, S, Whisstock, J.C, McGowan, S. | 登録日 | 2014-11-06 | 公開日 | 2015-12-02 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Stonefish toxin defines an ancient branch of the perforin-like superfamily. Proc.Natl.Acad.Sci.USA, 112, 2015
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6UD3
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![BU of 6ud3 by Molmil](/molmil-images/mine/6ud3) | Full length Glycine receptor reconstituted in lipid nanodisc in Gly/PTX-bound open/blocked conformation | 分子名称: | (1aR,2aR,3S,6R,6aS,8aS,8bR,9R)-2a-hydroxy-8b-methyl-9-(prop-1-en-2-yl)hexahydro-3,6-methano-1,5,7-trioxacyclopenta[ij]c yclopropa[a]azulene-4,8(3H)-dione, 2-acetamido-2-deoxy-beta-D-glucopyranose, GLYCINE, ... | 著者 | Kumar, A, Basak, S, Chakrapani, S. | 登録日 | 2019-09-18 | 公開日 | 2020-07-29 | 最終更新日 | 2024-03-20 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | Mechanisms of activation and desensitization of full-length glycine receptor in lipid nanodiscs. Nat Commun, 11, 2020
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6UBS
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![BU of 6ubs by Molmil](/molmil-images/mine/6ubs) | Full length Glycine receptor reconstituted in lipid nanodisc in Apo/Resting conformation | 分子名称: | 1,2-DIMYRISTOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Glycine receptor subunit alphaZ1, ... | 著者 | Kumar, A, Basak, S, Chakrapani, S. | 登録日 | 2019-09-12 | 公開日 | 2020-07-29 | 最終更新日 | 2020-08-12 | 実験手法 | ELECTRON MICROSCOPY (3.33 Å) | 主引用文献 | Mechanisms of activation and desensitization of full-length glycine receptor in lipid nanodiscs. Nat Commun, 11, 2020
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6VM0
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![BU of 6vm0 by Molmil](/molmil-images/mine/6vm0) | Full length Glycine receptor reconstituted in lipid nanodisc in Gly/IVM-conformation (State-1) | 分子名称: | (2aE,4E,5'S,6S,6'R,7S,8E,11R,13R,15S,17aR,20R,20aR,20bS)-6'-[(2S)-butan-2-yl]-20,20b-dihydroxy-5',6,8,19-tetramethyl-17 -oxo-3',4',5',6,6',10,11,14,15,17,17a,20,20a,20b-tetradecahydro-2H,7H-spiro[11,15-methanofuro[4,3,2-pq][2,6]benzodioxacy clooctadecine-13,2'-pyran]-7-yl 2,6-dideoxy-4-O-(2,6-dideoxy-3-O-methyl-alpha-L-arabino-hexopyranosyl)-3-O-methyl-alpha-L-arabino-hexopyranoside, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, GLYCINE, ... | 著者 | Kumar, A, Basak, S, Chakrapani, S. | 登録日 | 2020-01-27 | 公開日 | 2020-07-29 | 最終更新日 | 2024-03-06 | 実験手法 | ELECTRON MICROSCOPY (3.14 Å) | 主引用文献 | Mechanisms of activation and desensitization of full-length glycine receptor in lipid nanodiscs. Nat Commun, 11, 2020
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