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PDB: 47 件

7OGJ
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BU of 7ogj by Molmil
Crystal structure of human METTL1 in complex with SAH
分子名称: CHLORIDE ION, DI(HYDROXYETHYL)ETHER, GLYCEROL, ...
著者Nai, F, Bedi, R.K, Caflisch, A.
登録日2021-05-06
公開日2021-05-19
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.59 Å)
主引用文献Small-Molecule Inhibitors of the m7G-RNA Writer METTL1
Acs Bio Med Chem Au, 2023
7ZG4
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BU of 7zg4 by Molmil
Crystal structure of YTHDF2 with compound YLI_DF_042
分子名称: GLYCEROL, N-methylpyrimidine-2-carboximidamide, SULFATE ION, ...
著者Nai, F, Li, Y, Caflisch, A.
登録日2022-04-01
公開日2022-04-20
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.01 Å)
主引用文献Fragment Ligands of the m 6 A-RNA Reader YTHDF2.
Acs Med.Chem.Lett., 13, 2022
7R5F
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BU of 7r5f by Molmil
Crystal structure of YTHDF2 with compound YLI_DF_012
分子名称: 5-azanyl-6-methyl-1~{H}-pyrimidine-2,4-dione, CHLORIDE ION, SULFATE ION, ...
著者Nai, F, Li, Y, Caflisch, A.
登録日2022-02-10
公開日2022-03-02
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Fragment Ligands of the m 6 A-RNA Reader YTHDF2.
Acs Med.Chem.Lett., 13, 2022
7R5W
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BU of 7r5w by Molmil
Crystal structure of YTHDF2 with compound YLI_DF_029
分子名称: 6-cyclopropyl-1H-pyrimidine-2,4-dione, CHLORIDE ION, GLYCEROL, ...
著者Nai, F, Li, Y, Caflisch, A.
登録日2022-02-11
公開日2022-03-16
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Fragment Ligands of the m 6 A-RNA Reader YTHDF2.
Acs Med.Chem.Lett., 13, 2022
7PL1
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BU of 7pl1 by Molmil
Crystal structure of human METTL1 bound to Sinefungin
分子名称: DI(HYDROXYETHYL)ETHER, GLYCEROL, SINEFUNGIN, ...
著者Nai, F, Caflisch, A.
登録日2021-08-27
公開日2021-09-15
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Small-Molecule Inhibitors of the m7G-RNA Writer METTL1
Acs Bio Med Chem Au, 2023
7YX6
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BU of 7yx6 by Molmil
Crystal structure of YTHDF2 with compound YLI_DF_027
分子名称: 6-ethyl-1H-pyrimidine-2,4-dione, GLYCEROL, SULFATE ION, ...
著者Nai, F, Li, Y, Caflisch, A.
登録日2022-02-15
公開日2022-02-23
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Fragment Ligands of the m 6 A-RNA Reader YTHDF2.
Acs Med.Chem.Lett., 13, 2022
7YXE
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BU of 7yxe by Molmil
Crystal structure of YTHDF2 with compound ZA_143
分子名称: GLYCEROL, SODIUM ION, SULFATE ION, ...
著者Nai, F, Zalesak, F, Li, Y, Caflisch, A.
登録日2022-02-15
公開日2022-03-02
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Fragment Ligands of the m 6 A-RNA Reader YTHDF2.
Acs Med.Chem.Lett., 13, 2022
7Z26
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BU of 7z26 by Molmil
Crystal structure of YTHDF2 YTH domain in complex with m6A RNA
分子名称: GLYCEROL, RNA (5'-R(P*(6MZ)P*CP*U)-3'), SULFATE ION, ...
著者Nai, F, Nachawati, R, Li, Y, Caflisch, A.
登録日2022-02-25
公開日2022-03-16
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Fragment Ligands of the m 6 A-RNA Reader YTHDF2.
Acs Med.Chem.Lett., 13, 2022
7Z4U
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BU of 7z4u by Molmil
Crystal structure of YTHDF2 with compound YLI_DF_028
分子名称: 6-cyclopropyl-3-methyl-1H-pyrimidine-2,4-dione, CHLORIDE ION, GLYCEROL, ...
著者Nai, F, Li, Y, Caflisch, A.
登録日2022-03-04
公開日2022-03-16
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.83 Å)
主引用文献Fragment Ligands of the m 6 A-RNA Reader YTHDF2.
Acs Med.Chem.Lett., 13, 2022
7YWB
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BU of 7ywb by Molmil
Crystal structure of YTHDF2 in complex with N6-Methyladenine
分子名称: CHLORIDE ION, GLYCEROL, N-METHYL-9H-PURIN-6-AMINE, ...
著者Nai, F, Li, Y, Caflisch, A.
登録日2022-02-12
公開日2022-03-16
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.92 Å)
主引用文献Fragment Ligands of the m 6 A-RNA Reader YTHDF2.
Acs Med.Chem.Lett., 13, 2022
7Z7F
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BU of 7z7f by Molmil
Crystal structure of YTHDF2 with compound YLI_DC1_005
分子名称: CHLORIDE ION, GLYCEROL, SULFATE ION, ...
著者Nai, F, Li, Y, Dolbois, A, Caflisch, A.
登録日2022-03-15
公開日2022-03-23
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Fragment Ligands of the m 6 A-RNA Reader YTHDF2.
Acs Med.Chem.Lett., 13, 2022
7Z8P
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BU of 7z8p by Molmil
Crystal structure of YTHDF2 with compound ZA_166
分子名称: 3-bromanyl-~{N}-methyl-2~{H}-pyrazolo[4,3-d]pyrimidin-7-amine, GLYCEROL, SULFATE ION, ...
著者Nai, F, Zalesak, F, Li, Y, Caflisch, A.
登録日2022-03-18
公開日2022-03-30
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.97 Å)
主引用文献Fragment Ligands of the m 6 A-RNA Reader YTHDF2.
Acs Med.Chem.Lett., 13, 2022
7Z8W
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BU of 7z8w by Molmil
Crystal structure of YTHDF2 with compound YLI_DC1_018
分子名称: CHLORIDE ION, GLYCEROL, SULFATE ION, ...
著者Nai, F, Li, Y, Caflisch, A.
登録日2022-03-18
公開日2022-03-30
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Fragment Ligands of the m 6 A-RNA Reader YTHDF2.
Acs Med.Chem.Lett., 13, 2022
7Z93
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BU of 7z93 by Molmil
Crystal structure of YTHDF2 with compound YLI_DF_022
分子名称: 5-azanyl-6-ethyl-1H-pyrimidine-2,4-dione, CHLORIDE ION, SULFATE ION, ...
著者Nai, F, Li, Y, Caflisch, A.
登録日2022-03-19
公開日2022-03-30
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.97 Å)
主引用文献Fragment Ligands of the m 6 A-RNA Reader YTHDF2.
Acs Med.Chem.Lett., 13, 2022
7Z92
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BU of 7z92 by Molmil
Crystal structure of YTHDF2 with compound YLI_DF_024
分子名称: 5-azanyl-3,6-dimethyl-1H-pyrimidine-2,4-dione, SULFATE ION, YTH domain-containing family protein 2
著者Nai, F, Li, Y, Caflisch, A.
登録日2022-03-19
公開日2022-03-30
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.91 Å)
主引用文献Fragment Ligands of the m 6 A-RNA Reader YTHDF2.
Acs Med.Chem.Lett., 13, 2022
7Z7B
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BU of 7z7b by Molmil
Crystal structure of YTHDF2 with compound YLI_DC1_003
分子名称: CHLORIDE ION, GLYCEROL, SULFATE ION, ...
著者Nai, F, Li, Y, Dolbois, A, Caflisch, A.
登録日2022-03-15
公開日2022-06-22
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Fragment Ligands of the m 6 A-RNA Reader YTHDF2.
Acs Med.Chem.Lett., 13, 2022
7Z5M
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BU of 7z5m by Molmil
Crystal structure of YTHDF2 with compound YLI_DC1_008
分子名称: CHLORIDE ION, GLYCEROL, SULFATE ION, ...
著者Nai, F, Li, Y, Caflisch, A.
登録日2022-03-09
公開日2022-06-22
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Fragment Ligands of the m 6 A-RNA Reader YTHDF2.
Acs Med.Chem.Lett., 13, 2022
7Z54
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BU of 7z54 by Molmil
Crystal structure of YTHDF2 with compound YLI_DC1_006
分子名称: 9-cyclopropyl-~{N}-methyl-purin-6-amine, CHLORIDE ION, GLYCEROL, ...
著者Nai, F, Li, Y, Dolbois, A, Caflisch, A.
登録日2022-03-07
公開日2022-06-22
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.82 Å)
主引用文献Fragment Ligands of the m 6 A-RNA Reader YTHDF2.
Acs Med.Chem.Lett., 13, 2022
4RMK
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BU of 4rmk by Molmil
Crystal structure of the Olfactomedin domain of latrophilin 3 in P65 crystal form
分子名称: CALCIUM ION, Latrophilin-3
著者Ranaivoson, F.M, Liu, Q, Martini, F, Bergami, F, Von daake, S, Li, S, Demeler, B, Hendrickson, W.A, Comoletti, D.
登録日2014-10-21
公開日2015-08-19
最終更新日2017-11-22
実験手法X-RAY DIFFRACTION (1.606 Å)
主引用文献Structural and Mechanistic Insights into the Latrophilin3-FLRT3 Complex that Mediates Glutamatergic Synapse Development.
Structure, 23, 2015
4RML
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BU of 4rml by Molmil
Crystal structure of the Olfactomedin domain of latrophilin 3 in C2221 crystal form
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Latrophilin-3, MAGNESIUM ION
著者Ranaivoson, F.M, Liu, Q, Martini, F, Bergami, F, Von daake, S, Li, S, Demeler, B, Hendrickson, W.A, Comoletti, D.
登録日2014-10-21
公開日2015-08-19
最終更新日2015-10-07
実験手法X-RAY DIFFRACTION (1.601 Å)
主引用文献Structural and Mechanistic Insights into the Latrophilin3-FLRT3 Complex that Mediates Glutamatergic Synapse Development.
Structure, 23, 2015
8BJS
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BU of 8bjs by Molmil
Apo KIF20A[55-510] crystal structure
分子名称: Kinesin-like protein KIF20A, SULFATE ION, UNK-UNK-UNK-UNK
著者Ranaivoson, F.M, Kikuti, C, Crozet, V, Sirkia, M.E, Houdusse, A.
登録日2022-11-06
公開日2023-10-04
実験手法X-RAY DIFFRACTION (2.73 Å)
主引用文献Nucleotide-free structures of KIF20A illuminate atypical mechanochemistry in this kinesin-6.
Open Biology, 13, 2023
4YEB
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BU of 4yeb by Molmil
Structural characterization of a synaptic adhesion complex
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, Fibronectin leucine rich transmembrane protein 3, ...
著者Ranaivoson, F.M, Liu, Q, Martini, F, Bergami, F, von Daake, S, Li, S, Lee, D, Demeler, B, Hendrickson, W.A, Comoletti, D.
登録日2015-02-23
公開日2015-08-19
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (3.19 Å)
主引用文献Structural and Mechanistic Insights into the Latrophilin3-FLRT3 Complex that Mediates Glutamatergic Synapse Development.
Structure, 23, 2015
6DLF
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BU of 6dlf by Molmil
Crystal structure of NTRI homodimer
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Neurotrimin
著者Ranaivoson, F.M, Turk, L.S, Ozkan, E, Montelione, G.T, Comoletti, D.
登録日2018-06-01
公開日2019-04-10
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (3.446 Å)
主引用文献Structure of a heterodimer of neuronal cell surface proteins
Structure, 2019
6DLD
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BU of 6dld by Molmil
Crystal structure of IgLON5/NEGR1 heterodimer
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, IgLON family member 5, Neuronal growth regulator 1, ...
著者Ranaivoson, F.M, Turk, L.S, Ozkan, E, Montelione, G.T, Comoletti, D.
登録日2018-06-01
公開日2019-04-10
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献Structure of a heterodimer of neuronal cell surface proteins
Structure, 2019
6DLE
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BU of 6dle by Molmil
Crystal structure of IgLON5 homodimer
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, IgLON family member 5
著者Ranaivoson, F.M, Turk, L.S, Ozkan, E, Montelione, G.T, Comoletti, D.
登録日2018-06-01
公開日2019-04-10
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (3.994 Å)
主引用文献Structure of a heterodimer of neuronal cell surface proteins
Structure, 2019

 

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件を2024-08-28に公開中

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