8IDE
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![BU of 8ide by Molmil](/molmil-images/mine/8ide) | Structure of an ancient TsaD-TsaC-SUA5-TcdA modular enzyme (TsaN) | 分子名称: | MANGANESE (II) ION, N(6)-L-threonylcarbamoyladenine synthase | 著者 | Zhang, Z.L, Jin, M.Q, Yu, Z.J, Chen, W, Wang, X.L, Lei, D.S, Zhang, W.H. | 登録日 | 2023-02-13 | 公開日 | 2023-07-26 | 最終更新日 | 2023-09-20 | 実験手法 | ELECTRON MICROSCOPY (3.21 Å) | 主引用文献 | Structure-function analysis of an ancient TsaD-TsaC-SUA5-TcdA modular enzyme reveals a prototype of tRNA t6A and ct6A synthetases. Nucleic Acids Res., 51, 2023
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4IAT
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4I2Z
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1JY1
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![BU of 1jy1 by Molmil](/molmil-images/mine/1jy1) | CRYSTAL STRUCTURE OF HUMAN TYROSYL-DNA PHOSPHODIESTERASE (TDP1) | 分子名称: | TYROSYL-DNA PHOSPHODIESTERASE | 著者 | Davies, D.R, Interthal, H, Champoux, J.J, Hol, W.G.J. | 登録日 | 2001-09-10 | 公開日 | 2002-02-20 | 最終更新日 | 2021-10-27 | 実験手法 | X-RAY DIFFRACTION (1.69 Å) | 主引用文献 | The crystal structure of human tyrosyl-DNA phosphodiesterase, Tdp1. Structure, 10, 2002
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4QX6
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![BU of 4qx6 by Molmil](/molmil-images/mine/4qx6) | CRYSTAL STRUCTURE OF GLYCERALDEHYDE-3-PHOSPHATE DEHYDROGENASE FROM STREPTOCOCCUS AGALACTIAE NEM316 at 2.46 ANGSTROM RESOLUTION | 分子名称: | 1,2-ETHANEDIOL, Glyceraldehyde 3-phosphate dehydrogenase, NICOTINAMIDE-ADENINE-DINUCLEOTIDE | 著者 | Ayres, C.A, Schormann, N, Banerjee, S, Chattopadhyay, D. | 登録日 | 2014-07-18 | 公開日 | 2014-10-15 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.46 Å) | 主引用文献 | Structure of Streptococcus agalactiae glyceraldehyde-3-phosphate dehydrogenase holoenzyme reveals a novel surface. Acta Crystallogr F Struct Biol Commun, 70, 2014
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3WI4
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![BU of 3wi4 by Molmil](/molmil-images/mine/3wi4) | Crystal structure of wild-type PorB from Neisseria meningitidis serogroup B | 分子名称: | Major outer membrane protein P.IB | 著者 | Kattner, C, Toussi, D, Wetzler, L.M, Ruppel, N, Massari, P, Tanabe, M. | 登録日 | 2013-09-05 | 公開日 | 2014-01-01 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (3.32 Å) | 主引用文献 | Crystallographic analysis of Neisseria meningitidis PorB extracellular loops potentially implicated in TLR2 recognition. J.Struct.Biol., 185, 2014
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1JVL
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![BU of 1jvl by Molmil](/molmil-images/mine/1jvl) | Azurin dimer, covalently crosslinked through bis-maleimidomethylether | 分子名称: | 1-[PYRROL-1-YL-2,5-DIONE-METHOXYMETHYL]-PYRROLE-2,5-DIONE, Azurin, COPPER (II) ION, ... | 著者 | van Amsterdam, I.M.C, Ubbink, M, Einsle, O, Messerschmidt, A, Merli, A, Cavazzini, D, Rossi, G.L, Canters, G.W. | 登録日 | 2001-08-30 | 公開日 | 2002-01-04 | 最終更新日 | 2021-10-27 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Dramatic modulation of electron transfer in protein complexes by crosslinking Nat.Struct.Biol., 9, 2002
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5JUE
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![BU of 5jue by Molmil](/molmil-images/mine/5jue) | Crystal Structure of UIC2 Fab | 分子名称: | GLYCEROL, heavy chain of UIC2 Fab, light chain of UIC2 Fab | 著者 | Xia, D, Esser, L. | 登録日 | 2016-05-10 | 公開日 | 2016-08-31 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | Crystal structure of the antigen-binding fragment of a monoclonal antibody specific for the multidrug-resistance-linked ABC transporter human P-glycoprotein. Acta Crystallogr.,Sect.F, 72, 2016
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6W38
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![BU of 6w38 by Molmil](/molmil-images/mine/6w38) | Crystal structure of the FAM46C/Plk4 complex | 分子名称: | Serine/threonine-protein kinase PLK4, Terminal nucleotidyltransferase 5C | 著者 | Chen, H, Lu, D.F, Shang, G.J, Zhang, X.W. | 登録日 | 2020-03-09 | 公開日 | 2020-05-06 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (4.48 Å) | 主引用文献 | Structural and Functional Analyses of the FAM46C/Plk4 Complex. Structure, 28, 2020
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1K1C
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![BU of 1k1c by Molmil](/molmil-images/mine/1k1c) | Solution Structure of Crh, the Bacillus subtilis Catabolite Repression HPr | 分子名称: | catabolite repression HPr-like protein | 著者 | Favier, A, Brutscher, B, Blackledge, M, Galinier, A, Deutscher, J, Penin, F, Marion, D. | 登録日 | 2001-09-25 | 公開日 | 2001-10-17 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure and dynamics of Crh, the Bacillus subtilis catabolite repression HPr. J.Mol.Biol., 317, 2002
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6PRX
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![BU of 6prx by Molmil](/molmil-images/mine/6prx) | oxidized Human Branched Chain Aminotransferase mutant C318A | 分子名称: | Branched-chain-amino-acid aminotransferase, mitochondrial, PYRIDOXAL-5'-PHOSPHATE | 著者 | Dong, M, Herbert, D, Gibbs, S. | 登録日 | 2019-07-11 | 公開日 | 2020-01-22 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (3.25 Å) | 主引用文献 | Crystal structure of an oxidized mutant of human mitochondrial branched-chain aminotransferase. Acta Crystallogr.,Sect.F, 76, 2020
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4IGP
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![BU of 4igp by Molmil](/molmil-images/mine/4igp) | Histone H3 Lysine 4 Demethylating Rice JMJ703 apo enzyme | 分子名称: | FE (III) ION, Os05g0196500 protein | 著者 | Chen, Q.F, Chen, X.S, Wang, Q, Zhang, F.B, Lou, Z.Y, Zhang, Q.F, Zhou, D.X. | 登録日 | 2012-12-17 | 公開日 | 2013-04-03 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (3.003 Å) | 主引用文献 | Structural basis of a histone H3 lysine 4 demethylase required for stem elongation in rice. PLoS Genet., 9, 2013
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5K2D
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![BU of 5k2d by Molmil](/molmil-images/mine/5k2d) | 1.9A angstrom A2a adenosine receptor structure with MR phasing using XFEL data | 分子名称: | (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, (2S)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, 4-{2-[(7-amino-2-furan-2-yl[1,2,4]triazolo[1,5-a][1,3,5]triazin-5-yl)amino]ethyl}phenol, ... | 著者 | Batyuk, A, Galli, L, Ishchenko, A, Han, G.W, Gati, C, Popov, P, Lee, M.-Y, Stauch, B, White, T.A, Barty, A, Aquila, A, Hunter, M.S, Liang, M, Boutet, S, Pu, M, Liu, Z.-J, Nelson, G, James, D, Li, C, Zhao, Y, Spence, J.C.H, Liu, W, Fromme, P, Katritch, V, Weierstall, U, Stevens, R.C, Cherezov, V, GPCR Network (GPCR) | 登録日 | 2016-05-18 | 公開日 | 2016-09-21 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Native phasing of x-ray free-electron laser data for a G protein-coupled receptor. Sci Adv, 2, 2016
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1JH1
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![BU of 1jh1 by Molmil](/molmil-images/mine/1jh1) | Crystal Structure of MMP-8 complexed with a 6H-1,3,4-thiadiazine derived inhibitor | 分子名称: | BUT-3-ENYL-[5-(4-CHLORO-PHENYL)-3,6-DIHYDRO-[1,3,4]THIADIAZIN-2-YLIDENE]-AMINE, CALCIUM ION, Matrix Metalloproteinase 8, ... | 著者 | Schroder, J, Henke, A, Wenzel, H, Brandstetter, H, Stammler, H.G, Stammler, A, Pfeiffer, W.D, Tschesche, H. | 登録日 | 2001-06-27 | 公開日 | 2001-12-27 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Structure-based design and synthesis of potent matrix metalloproteinase inhibitors derived from a 6H-1,3,4-thiadiazine scaffold. J.Med.Chem., 44, 2001
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2IBN
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![BU of 2ibn by Molmil](/molmil-images/mine/2ibn) | Crystal structure of Human myo-Inositol Oxygenase (MIOX) | 分子名称: | (2S,3R,4R,5S,6S)-2,3,4,5,6-PENTAHYDROXYCYCLOHEXANONE, CYSTEINE, FE (III) ION, ... | 著者 | Hallberg, B.M, Busam, R.D, Arrowsmith, C, Berglund, H, Collins, R, Edwards, A, Ehn, M, Flodin, S, Flores, A, Graslund, S, Hammarstrom, M, Hogbom, M, Holmberg-Schiavone, L, Johansson, I, Karlberg, T, Kotenyova, T, Nilsson-Ehle, P, Nordlund, P, Nyman, T, Ogg, D, Sagemark, J, Stenmark, P, Sundstrom, M, Uppenberg, J, Van Den Berg, S, Weigelt, J, Thorsell, A.G, Persson, C, Structural Genomics Consortium (SGC) | 登録日 | 2006-09-11 | 公開日 | 2006-10-17 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Structural and Biophysical Characterization of Human myo-Inositol Oxygenase J.Biol.Chem., 283, 2008
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4QR4
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![BU of 4qr4 by Molmil](/molmil-images/mine/4qr4) | Brd4 Bromodomain 1 complex with its novel inhibitors | 分子名称: | 2-chloro-N-cyclopentyl-5-(2-oxo-2,3-dihydro-1,3-thiazol-4-yl)benzenesulfonamide, Bromodomain-containing protein 4 | 著者 | Xiong, B, Cao, D.Y, Chen, T.T, Xu, Y.C. | 登録日 | 2014-06-30 | 公開日 | 2015-07-01 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.28 Å) | 主引用文献 | Fragment-based drug discovery of 2-thiazolidinones as BRD4 inhibitors: 2. Structure-based optimization J.Med.Chem., 58, 2015
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5K3S
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![BU of 5k3s by Molmil](/molmil-images/mine/5k3s) | Crystal structure of Arabidopsis thaliana acetohydroxyacid synthase in complex with a pyrimidinyl-benzoate herbicide, bispyribac-sodium | 分子名称: | (3Z)-4-{[(4-AMINO-2-METHYLPYRIMIDIN-5-YL)METHYL]AMINO}-3-MERCAPTOPENT-3-EN-1-YL TRIHYDROGEN DIPHOSPHATE, 2,6-bis[(4,6-dimethoxypyrimidin-2-yl)oxy]benzoic acid, Acetolactate synthase, ... | 著者 | Garcia, M.D, Lonhienne, T, Guddat, L.W. | 登録日 | 2016-05-19 | 公開日 | 2017-02-08 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.873 Å) | 主引用文献 | Comprehensive understanding of acetohydroxyacid synthase inhibition by different herbicide families. Proc. Natl. Acad. Sci. U.S.A., 114, 2017
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3E4A
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![BU of 3e4a by Molmil](/molmil-images/mine/3e4a) | Human IDE-inhibitor complex at 2.6 angstrom resolution | 分子名称: | 1,4-DIETHYLENE DIOXIDE, ACETIC ACID, HYDROXAMATE PEPTIDE II1, ... | 著者 | Malito, E, Leissring, M.A, Choi, S, Cuny, G.D, Tang, W.J. | 登録日 | 2008-08-11 | 公開日 | 2009-05-19 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Designed inhibitors of insulin-degrading enzyme regulate the catabolism and activity of insulin. Plos One, 5, 2010
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1JM7
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![BU of 1jm7 by Molmil](/molmil-images/mine/1jm7) | Solution structure of the BRCA1/BARD1 RING-domain heterodimer | 分子名称: | BRCA1-ASSOCIATED RING DOMAIN PROTEIN 1, BREAST CANCER TYPE 1 SUSCEPTIBILITY PROTEIN, ZINC ION | 著者 | Brzovic, P.S, Rajagopal, P, Hoyt, D.W, King, M.-C, Klevit, R.E. | 登録日 | 2001-07-17 | 公開日 | 2001-10-03 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Structure of a BRCA1-BARD1 heterodimeric RING-RING complex. Nat.Struct.Biol., 8, 2001
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4QQN
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![BU of 4qqn by Molmil](/molmil-images/mine/4qqn) | Protein arginine methyltransferase 3 in complex with compound MTV044246 | 分子名称: | 1-{2-[1-(aminomethyl)cyclohexyl]ethyl}-3-isoquinolin-6-ylurea, CHLORIDE ION, GLYCEROL, ... | 著者 | Dong, A, Dobrovetsky, E, Tempel, W, He, H, Zhao, K, Smil, D, Landon, M, Luo, X, Chen, Z, Dai, M, Yu, Z, Lin, Y, Zhang, H, Zhao, K, Schapira, M, Brown, P.J, Bountra, C, Arrowsmith, C.H, Edwards, A.M, Vedadi, M, Structural Genomics Consortium (SGC) | 登録日 | 2014-06-27 | 公開日 | 2014-09-17 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.08 Å) | 主引用文献 | Discovery of Potent and Selective Allosteric Inhibitors of Protein Arginine Methyltransferase 3 (PRMT3). J. Med. Chem., 61, 2018
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1JMM
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![BU of 1jmm by Molmil](/molmil-images/mine/1jmm) | Crystal structure of the V-region of Streptococcus mutans antigen I/II | 分子名称: | SODIUM ION, protein I/II V-region | 著者 | Troffer-Charlier, N, Ogier, J, Moras, D, Cavarelli, J. | 登録日 | 2001-07-19 | 公開日 | 2002-07-17 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Crystal Structure of the V-region of Streptococcus mutans Antigen I/II at 2.4 a Resolution Suggests a Sugar Preformed Binding Site J.Mol.Biol., 318, 2002
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2I0T
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![BU of 2i0t by Molmil](/molmil-images/mine/2i0t) | |
4QXX
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5K9S
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![BU of 5k9s by Molmil](/molmil-images/mine/5k9s) | Importin-alpha in complex with HNF1-beta peptide | 分子名称: | HNF1 beta A splice variant 2, Importin subunit alpha-1 | 著者 | Wiedmann, M.M, Aibara, S, Spring, D.R, Stewart, M, Brenton, J. | 登録日 | 2016-06-01 | 公開日 | 2016-11-23 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Importin-alpha in complex with HNF1-beta peptide To Be Published
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4ION
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![BU of 4ion by Molmil](/molmil-images/mine/4ion) | Macrolepiota procera ricin B-like lectin (MPL) | 分子名称: | GLYCEROL, Ricin B-like lectin | 著者 | Renko, M, Zurga, S, Sabotic, J, Pohleven, J, Kos, J, Turk, D. | 登録日 | 2013-01-08 | 公開日 | 2013-11-20 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Macrolepiota procera ricin B-like lectin (MPL) TO BE PUBLISHED
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