5IGH
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![BU of 5igh by Molmil](/molmil-images/mine/5igh) | Macrolide 2'-phosphotransferase type I | Descriptor: | Macrolide 2'-phosphotransferase, SULFATE ION | Authors: | Berghuis, A.M, Fong, D.H. | Deposit date: | 2016-02-28 | Release date: | 2017-04-26 | Last modified: | 2020-01-08 | Method: | X-RAY DIFFRACTION (1.55 Å) | Cite: | Structural Basis for Kinase-Mediated Macrolide Antibiotic Resistance. Structure, 25, 2017
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5IGV
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![BU of 5igv by Molmil](/molmil-images/mine/5igv) | |
5IGR
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![BU of 5igr by Molmil](/molmil-images/mine/5igr) | Macrolide 2'-phosphotransferase type I - complex with GDP and oleandomycin | Descriptor: | (3S,5R,6S,7R,8R,11R,12S,13R,14S,15S)-6-HYDROXY-5,7,8,11,13,15-HEXAMETHYL-4,10-DIOXO-14-{[3,4,6-TRIDEOXY-3-(DIMETHYLAMINO)-BETA-D-XYLO-HEXOPYRANOSYL]OXY}-1,9-DIOXASPIRO[2.13]HEXADEC-12-YL 2,6-DIDEOXY-3-O-METHYL-ALPHA-L-ARABINO-HEXOPYRANOSIDE, AMMONIUM ION, GUANOSINE-5'-DIPHOSPHATE, ... | Authors: | Berghuis, A.M, Fong, D.H. | Deposit date: | 2016-02-28 | Release date: | 2017-04-26 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.6 Å) | Cite: | Structural Basis for Kinase-Mediated Macrolide Antibiotic Resistance. Structure, 25, 2017
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5IH1
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![BU of 5ih1 by Molmil](/molmil-images/mine/5ih1) | |
1GIT
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![BU of 1git by Molmil](/molmil-images/mine/1git) | STRUCTURE OF GTP-BINDING PROTEIN | Descriptor: | G PROTEIN GI ALPHA 1, GUANOSINE-5'-DIPHOSPHATE, PHOSPHATE ION | Authors: | Berghuis, A.M, Lee, E, Sprang, S.R. | Deposit date: | 1996-10-16 | Release date: | 1997-02-12 | Last modified: | 2024-02-07 | Method: | X-RAY DIFFRACTION (2.6 Å) | Cite: | Structure of the GDP-Pi complex of Gly203-->Ala gialpha1: a mimic of the ternary product complex of galpha-catalyzed GTP hydrolysis. Structure, 4, 1996
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3Q2M
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![BU of 3q2m by Molmil](/molmil-images/mine/3q2m) | Crystal Structure of Spectinomycin Phosphotransferase, APH(9)-Ia, Protein Kinase Inhibitor CKI-7 Complex | Descriptor: | N-(2-AMINOETHYL)-5-CHLOROISOQUINOLINE-8-SULFONAMIDE, NICKEL (II) ION, Spectinomycin phosphotransferase | Authors: | Berghuis, A.M, Fong, D.H, Xiong, B, Hwang, J. | Deposit date: | 2010-12-20 | Release date: | 2011-05-18 | Last modified: | 2023-09-13 | Method: | X-RAY DIFFRACTION (2.9 Å) | Cite: | Crystal structures of two aminoglycoside kinases bound with a eukaryotic protein kinase inhibitor. Plos One, 6, 2011
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1IRV
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![BU of 1irv by Molmil](/molmil-images/mine/1irv) | |
1IRW
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![BU of 1irw by Molmil](/molmil-images/mine/1irw) | |
1GIA
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![BU of 1gia by Molmil](/molmil-images/mine/1gia) | |
2Q99
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![BU of 2q99 by Molmil](/molmil-images/mine/2q99) | |
3I1A
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![BU of 3i1a by Molmil](/molmil-images/mine/3i1a) | Crystal Structure of apo Spectinomycin Phosphotransferase, APH(9)-Ia | Descriptor: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, DIMETHYL SULFOXIDE, Spectinomycin phosphotransferase, ... | Authors: | Berghuis, A.M, Fong, D.H, Lemke, C.T, Hwang, J, Xiong, B. | Deposit date: | 2009-06-25 | Release date: | 2010-01-19 | Last modified: | 2024-02-21 | Method: | X-RAY DIFFRACTION (1.7 Å) | Cite: | Structure of the antibiotic resistance factor spectinomycin phosphotransferase from Legionella pneumophila. J.Biol.Chem., 285, 2010
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3I0Q
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![BU of 3i0q by Molmil](/molmil-images/mine/3i0q) | Crystal Structure of the AMP-bound complex of Spectinomycin Phosphotransferase, APH(9)-Ia | Descriptor: | ADENOSINE MONOPHOSPHATE, NICKEL (II) ION, Spectinomycin phosphotransferase | Authors: | Berghuis, A.M, Fong, D.H, Lemke, C.T, Hwang, J.-Y, Xiong, B. | Deposit date: | 2009-06-25 | Release date: | 2010-01-19 | Last modified: | 2023-09-06 | Method: | X-RAY DIFFRACTION (2.8 Å) | Cite: | Structure of the antibiotic resistance factor spectinomycin phosphotransferase from Legionella pneumophila. J.Biol.Chem., 285, 2010
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3TM0
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![BU of 3tm0 by Molmil](/molmil-images/mine/3tm0) | Crystal Structure of 3',5"-Aminoglycoside Phosphotransferase Type IIIa AMPPNP Butirosin A Complex | Descriptor: | (2S)-4-amino-N-[(1R,2S,3R,4R,5S)-5-amino-4-[(2,6-diamino-2,6-dideoxy-alpha-D-glucopyranosyl)oxy]-2-hydroxy-3-(beta-D-xylofuranosyloxy)cyclohexyl]-2-hydroxybutanamide, Aminoglycoside 3'-phosphotransferase, MAGNESIUM ION, ... | Authors: | Berghuis, A.M, Fong, D.H. | Deposit date: | 2011-08-30 | Release date: | 2011-10-19 | Last modified: | 2023-09-13 | Method: | X-RAY DIFFRACTION (2.1 Å) | Cite: | Structural basis of APH(3')-IIIa-mediated resistance to N1-substituted aminoglycoside antibiotics. Antimicrob.Agents Chemother., 53, 2009
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1CRI
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![BU of 1cri by Molmil](/molmil-images/mine/1cri) | |
1CRG
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![BU of 1crg by Molmil](/molmil-images/mine/1crg) | |
1CRJ
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![BU of 1crj by Molmil](/molmil-images/mine/1crj) | |
1CRH
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![BU of 1crh by Molmil](/molmil-images/mine/1crh) | |
5E96
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![BU of 5e96 by Molmil](/molmil-images/mine/5e96) | Crystal structure of aminoglycoside 6'-acetyltransferase type Ii | Descriptor: | 1,2-ETHANEDIOL, Aminoglycoside 6'-acetyltransferase, PHOSPHATE ION | Authors: | Berghuis, A.M, Burk, D.L, Baettig, O.M, Shi, K. | Deposit date: | 2015-10-14 | Release date: | 2016-07-06 | Last modified: | 2023-09-27 | Method: | X-RAY DIFFRACTION (2.1 Å) | Cite: | Comprehensive characterization of ligand-induced plasticity changes in a dimeric enzyme. Febs J., 283, 2016
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2YCC
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![BU of 2ycc by Molmil](/molmil-images/mine/2ycc) | |
1CTY
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![BU of 1cty by Molmil](/molmil-images/mine/1cty) | |
1CTZ
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![BU of 1ctz by Molmil](/molmil-images/mine/1ctz) | |
5IGJ
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![BU of 5igj by Molmil](/molmil-images/mine/5igj) | |
5IGW
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![BU of 5igw by Molmil](/molmil-images/mine/5igw) | |
5IGI
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![BU of 5igi by Molmil](/molmil-images/mine/5igi) | |
5IGT
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![BU of 5igt by Molmil](/molmil-images/mine/5igt) | |