6L3X
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![BU of 6l3x by Molmil](/molmil-images/mine/6l3x) | Discovery of novel peptidomimetic boronate ClpP inhibitors with noncanonical enzyme mechanism as potent virulence blockers in vitro and in vivo | 分子名称: | ATP-dependent Clp protease proteolytic subunit, [(1~{R})-1-[[(2~{S})-2-[[2,5-bis(chloranyl)phenyl]carbonylamino]-3-(1~{H}-indol-3-yl)propanoyl]amino]-3-methyl-butyl]boronic acid | 著者 | Luo, Y.F, Bao, R, Ju, Y, He, L.H. | 登録日 | 2019-10-15 | 公開日 | 2020-08-26 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.3054 Å) | 主引用文献 | Discovery of Novel Peptidomimetic Boronate ClpP Inhibitors with Noncanonical Enzyme Mechanism as Potent Virulence Blockersin Vitroandin Vivo. J.Med.Chem., 63, 2020
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7DEK
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3IBH
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![BU of 3ibh by Molmil](/molmil-images/mine/3ibh) | Crystal structure of Saccharomyces cerevisiae Gtt2 in complex with glutathione | 分子名称: | GLUTATHIONE, Saccharomyces cerevisiae Gtt2 | 著者 | Ma, X.X, Jiang, Y.L, He, Y.X, Bao, R, Chen, Y.X, Zhou, C.Z. | 登録日 | 2009-07-15 | 公開日 | 2009-10-13 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structures of yeast glutathione-S-transferase Gtt2 reveal a new catalytic type of GST family. Embo Rep., 10, 2009
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3PUB
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![BU of 3pub by Molmil](/molmil-images/mine/3pub) | Crystal structure of the Bombyx mori low molecular weight lipoprotein 7 (Bmlp7) | 分子名称: | 30kDa protein | 著者 | Yang, J.-P, Ma, X.-X, He, Y.-X, Li, W.-F, Kang, Y, Bao, R, Chen, Y, Zhou, C.-Z. | 登録日 | 2010-12-03 | 公開日 | 2011-06-01 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.91 Å) | 主引用文献 | Crystal structure of the 30 K protein from the silkworm Bombyx mori reveals a new member of the beta-trefoil superfamily J.Struct.Biol., 175, 2011
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3B54
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8GXF
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![BU of 8gxf by Molmil](/molmil-images/mine/8gxf) | Pseudomonas flexibilis GCN5 family acetyltransferase | 分子名称: | COENZYME A, GCN5 family acetyltransferase | 著者 | Song, Y.J, Bao, R. | 登録日 | 2022-09-20 | 公開日 | 2022-10-19 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (3.04 Å) | 主引用文献 | The novel type II toxin-antitoxin PacTA modulates Pseudomonas aeruginosa iron homeostasis by obstructing the DNA-binding activity of Fur. Nucleic Acids Res., 50, 2022
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8GXJ
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8GXK
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![BU of 8gxk by Molmil](/molmil-images/mine/8gxk) | Pseudomonas jinjuensis N-acetyltransferase | 分子名称: | COENZYME A, Protein N-acetyltransferase, RimJ/RimL family | 著者 | Song, Y.J, Bao, R. | 登録日 | 2022-09-20 | 公開日 | 2022-10-12 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.78 Å) | 主引用文献 | The novel type II toxin-antitoxin PacTA modulates Pseudomonas aeruginosa iron homeostasis by obstructing the DNA-binding activity of Fur. Nucleic Acids Res., 50, 2022
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8JU7
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8KHL
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![BU of 8khl by Molmil](/molmil-images/mine/8khl) | (S)-citramalyl-CoA lyase | 分子名称: | COENZYME A, Probable acyl-CoA lyase beta chain | 著者 | Huang, Q, Bao, R. | 登録日 | 2023-08-22 | 公開日 | 2024-05-15 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Structural and functional characterization of itaconyl-CoA hydratase and citramalyl-CoA lyase involved in itaconate metabolism of Pseudomonas aeruginosa. Structure, 2024
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8KHG
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![BU of 8khg by Molmil](/molmil-images/mine/8khg) | Itaconyl-CoA hydratase PaIch | 分子名称: | CITRIC ACID, Itaconyl-CoA hydratase | 著者 | Huang, Q, Bao, R. | 登録日 | 2023-08-21 | 公開日 | 2024-05-15 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Structural and functional characterization of itaconyl-CoA hydratase and citramalyl-CoA lyase involved in itaconate metabolism of Pseudomonas aeruginosa. Structure, 2024
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8YLB
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![BU of 8ylb by Molmil](/molmil-images/mine/8ylb) | Cocrystal structures of agonists compound 1 with HsClpP | 分子名称: | 5-[(2-methylphenyl)methyl]-11-(phenylmethyl)-2,5,7,11-tetrazatricyclo[7.4.0.0^{2,6}]trideca-1(9),6-dien-8-one, ATP-dependent Clp protease proteolytic subunit, mitochondrial | 著者 | Zhao, N, Zhu, Y, Bao, R. | 登録日 | 2024-03-06 | 公開日 | 2024-05-15 | 実験手法 | X-RAY DIFFRACTION (2.15 Å) | 主引用文献 | Rational Design of a Novel Class of Human ClpP Agonists through a Ring-Opening Strategy with Enhanced Antileukemia Activity. J.Med.Chem., 67, 2024
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8Z6G
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8WCO
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![BU of 8wco by Molmil](/molmil-images/mine/8wco) | (S)-citramalyl-CoA lyase | 分子名称: | ACETYL COENZYME *A, Probable acyl-CoA lyase beta chain | 著者 | Huang, Q, Bao, R. | 登録日 | 2023-09-13 | 公開日 | 2024-05-15 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Structural and functional characterization of itaconyl-CoA hydratase and citramalyl-CoA lyase involved in itaconate metabolism of Pseudomonas aeruginosa. Structure, 2024
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5WYB
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![BU of 5wyb by Molmil](/molmil-images/mine/5wyb) | Structure of Pseudomonas aeruginosa DspI | 分子名称: | (4R)-2-METHYLPENTANE-2,4-DIOL, ACETATE ION, Probable enoyl-CoA hydratase/isomerase | 著者 | Liu, L, Peng, C, Li, T, Li, C, He, L, Song, Y, Zhu, Y, Shen, Y, Bao, R. | 登録日 | 2017-01-12 | 公開日 | 2018-01-17 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Structural and functional studies on Pseudomonas aeruginosa DspI: implications for its role in DSF biosynthesis. Sci Rep, 8, 2018
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6L40
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![BU of 6l40 by Molmil](/molmil-images/mine/6l40) | Discovery of novel peptidomimetic boronate ClpP inhibitors with noncanonical enzyme mechanism as potent virulence blockers in vitro and in vivo | 分子名称: | ATP-dependent Clp protease proteolytic subunit, [(1S)-3-methyl-1-[[(2S)-3-phenyl-2-(pyrazin-2-ylcarbonylamino)propanoyl]amino]butyl]boronic acid | 著者 | Luo, Y.F, Bao, R, Ju, Y, He, L.H. | 登録日 | 2019-10-15 | 公開日 | 2020-07-08 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.209 Å) | 主引用文献 | Discovery of Novel Peptidomimetic Boronate ClpP Inhibitors with Noncanonical Enzyme Mechanism as Potent Virulence Blockersin Vitroandin Vivo. J.Med.Chem., 63, 2020
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5YKJ
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![BU of 5ykj by Molmil](/molmil-images/mine/5ykj) | Structural basis of the thiol resolving mechanism in yeast mitochondrial 1-Cys peroxiredoxin via glutathione/thioredoxin systems | 分子名称: | GLYCEROL, Peroxiredoxin PRX1, mitochondrial, ... | 著者 | Li, C.C, Yang, J, Yang, M.J, Liu, L, Peng, C.T, Li, T, He, L.H, Song, Y.J, Zhu, Y.B, Zhao, N.L, Zhao, C, Bao, R. | 登録日 | 2017-10-14 | 公開日 | 2018-10-24 | 最終更新日 | 2019-11-06 | 実験手法 | X-RAY DIFFRACTION (1.53 Å) | 主引用文献 | Structural basis of the thiol resolving mechanism in yeast mitochondrial 1-Cys peroxiredoxin via glutathione/thioredoxin systems To be published
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5YEI
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![BU of 5yei by Molmil](/molmil-images/mine/5yei) | Mechanistic insight into the regulation of Pseudomonas aeruginosa aspartate kinase | 分子名称: | Aspartokinase, GLYCEROL, LYSINE, ... | 著者 | Li, C, Yang, M, Liu, L, Peng, C, Li, T, He, L, Song, Y, Zhu, Y, Bao, R. | 登録日 | 2017-09-17 | 公開日 | 2018-08-29 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.301 Å) | 主引用文献 | Mechanistic insights into the allosteric regulation of Pseudomonas aeruginosa aspartate kinase. Biochem.J., 475, 2018
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5YKW
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![BU of 5ykw by Molmil](/molmil-images/mine/5ykw) | Structural basis of the thiol resolving mechanism in yeast mitochondrial 1-Cys peroxiredoxin via glutathione/thioredoxin systems | 分子名称: | Thioredoxin-3, mitochondrial, peptide THR-PRO-VAL-CYS-THR-THR-GLU-VAL | 著者 | Li, C.C, Yang, J, Yang, M.J, Liu, L, Peng, C.T, Li, T, He, L.H, Song, Y.J, Zhu, Y.B, Zhao, N.L, Zhao, C, Bao, R. | 登録日 | 2017-10-16 | 公開日 | 2018-10-24 | 最終更新日 | 2019-11-06 | 実験手法 | X-RAY DIFFRACTION (2.08 Å) | 主引用文献 | Structural basis of the thiol resolving mechanism in yeast mitochondrial 1-Cys peroxiredoxin via glutathione/thioredoxin systems to be published
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5YLO
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![BU of 5ylo by Molmil](/molmil-images/mine/5ylo) | Structural of Pseudomonas aeruginosa PA4980 | 分子名称: | GLYCEROL, Probable enoyl-CoA hydratase/isomerase | 著者 | Liu, L, Li, T, Peng, C.T, Li, C.C, Xiao, Q.J, He, L.H, Wang, N.Y, Bao, R. | 登録日 | 2017-10-18 | 公開日 | 2018-08-22 | 最終更新日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (2.39 Å) | 主引用文献 | Structural characterization of a Delta3, Delta2-enoyl-CoA isomerase from Pseudomonas aeruginosa: implications for its involvement in unsaturated fatty acid metabolism. J.Biomol.Struct.Dyn., 37, 2019
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5WYD
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![BU of 5wyd by Molmil](/molmil-images/mine/5wyd) | Structural of Pseudomonas aeruginosa DspI | 分子名称: | (4R)-2-METHYLPENTANE-2,4-DIOL, (4S)-2-METHYL-2,4-PENTANEDIOL, ISOPROPYL ALCOHOL, ... | 著者 | Liu, L, Peng, C, Li, T, Li, C, He, L, Song, Y, Zhu, Y, Shen, Y, Bao, R. | 登録日 | 2017-01-12 | 公開日 | 2018-01-31 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.101 Å) | 主引用文献 | Structural and functional studies on Pseudomonas aeruginosa DspI: implications for its role in DSF biosynthesis. Sci Rep, 8, 2018
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6JAU
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![BU of 6jau by Molmil](/molmil-images/mine/6jau) | The complex structure of Pseudomonas aeruginosa MucA/MucB. | 分子名称: | CALCIUM ION, GLYCEROL, HEXAETHYLENE GLYCOL, ... | 著者 | Li, T, He, L.H, Li, C.C, Liu, L, Peng, C.T, Shen, Y.L, Qin, X.F, Xiao, Q.J, Zhu, Y.B, Song, Y.J, Zhao, N.l, Zhao, C, Yang, J, Mu, X.Y, Huang, Q, Bao, R. | 登録日 | 2019-01-25 | 公開日 | 2020-01-29 | 最終更新日 | 2020-08-19 | 実験手法 | X-RAY DIFFRACTION (1.905 Å) | 主引用文献 | Molecular basis of the lipid-induced MucA-MucB dissociation in Pseudomonas aeruginosa. Commun Biol, 3, 2020
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3EVI
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![BU of 3evi by Molmil](/molmil-images/mine/3evi) | Crystal structure of the thioredoxin-fold domain of human phosducin-like protein 2 | 分子名称: | DI(HYDROXYETHYL)ETHER, Phosducin-like protein 2, SODIUM ION | 著者 | Lou, X, Bao, R, Zhou, C, Chen, Y. | 登録日 | 2008-10-13 | 公開日 | 2009-03-03 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Structure of the thioredoxin-fold domain of human phosducin-like protein 2 Acta Crystallogr.,Sect.F, 65, 2009
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3F3R
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![BU of 3f3r by Molmil](/molmil-images/mine/3f3r) | Crystal structure of yeast Thioredoxin1-glutathione mixed disulfide complex | 分子名称: | GLUTATHIONE, SULFATE ION, Thioredoxin-1 | 著者 | Zhang, Y.R, Bao, R, Zhou, C.Z, Chen, Y.X. | 登録日 | 2008-10-31 | 公開日 | 2009-10-20 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Structural and kinetic analysis of Saccharomyces cerevisiae thioredoxin Trx1: implications for the catalytic mechanism of GSSG reduced by the thioredoxin system Biochim.Biophys.Acta, 1794, 2009
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3F3H
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![BU of 3f3h by Molmil](/molmil-images/mine/3f3h) | Crystal structure and anti-tumor activity of LZ-8 from the fungus Ganoderma lucidium | 分子名称: | Immunomodulatory protein Ling Zhi-8 | 著者 | Zhou, C.Z, Huang, L, He, Y.X, Bao, R, Sun, F, Liang, C, Liu, L. | 登録日 | 2008-10-30 | 公開日 | 2009-09-15 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Crystal structure of LZ-8 from the medicinal fungus Ganoderma lucidium Proteins, 75, 2009
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