6VLR
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![BU of 6vlr by Molmil](/molmil-images/mine/6vlr) | |
4ZMA
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![BU of 4zma by Molmil](/molmil-images/mine/4zma) | Crystal Structure of a FVIIa-Trypsin Chimera (ST) in Complex with Soluble Tissue Factor | 分子名称: | CACODYLATE ION, CALCIUM ION, Coagulation factor VII, ... | 著者 | Sorensen, A.B, Svensson, L.A, Gandhi, P.S. | 登録日 | 2015-05-02 | 公開日 | 2015-12-30 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Molecular Basis of Enhanced Activity in Factor VIIa-Trypsin Variants Conveys Insights into Tissue Factor-mediated Allosteric Regulation of Factor VIIa Activity. J.Biol.Chem., 291, 2016
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4Z7M
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![BU of 4z7m by Molmil](/molmil-images/mine/4z7m) | Novel Inhibitors of Bacterial Methionine Aminopeptidase with Broad-Spectrum Biochemical Activity | 分子名称: | MANGANESE (II) ION, Methionine aminopeptidase, N~2~-[(3,5-difluorophenyl)acetyl]-N-[(3S,7R)-1-methyl-2-oxo-7-phenyl-2,3,4,7-tetrahydro-1H-azepin-3-yl]-L-alaninamide | 著者 | Rose, J.A, Lahiri, S.D, McKinney, D.C, Albert, R, Morningstar, M, Shapiro, A.B, Fisher, S.F, Fleming, P.R. | 登録日 | 2015-04-07 | 公開日 | 2016-04-13 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.43 Å) | 主引用文献 | Novel Inhibitors of Bacterial Methionine Aminopeptidase with Broad-Spectrum Biochemical Activity To be Published
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4Z6A
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![BU of 4z6a by Molmil](/molmil-images/mine/4z6a) | Crystal Structure of a FVIIa-Trypsin Chimera (YT) in Complex with Soluble Tissue Factor | 分子名称: | CALCIUM ION, CITRIC ACID, Coagulation factor VII, ... | 著者 | Sorensen, A.B, Svensson, L.A, Gandhi, P.S. | 登録日 | 2015-04-04 | 公開日 | 2015-12-30 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Molecular Basis of Enhanced Activity in Factor VIIa-Trypsin Variants Conveys Insights into Tissue Factor-mediated Allosteric Regulation of Factor VIIa Activity. J.Biol.Chem., 291, 2016
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5A55
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![BU of 5a55 by Molmil](/molmil-images/mine/5a55) | The native structure of GH101 from Streptococcus pneumoniae TIGR4 | 分子名称: | 1,2-ETHANEDIOL, CALCIUM ION, ENDO-ALPHA-N-ACETYLGALACTOSAMINIDASE, ... | 著者 | Gregg, K.J, Suits, M.D.L, Deng, L, Vocadlo, D.J, Boraston, A.B. | 登録日 | 2015-06-16 | 公開日 | 2015-09-02 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Structural Analysis of a Family 101 Glycoside Hydrolase in Complex with Carbohydrates Reveals Insights Into its Mechanism. J.Biol.Chem., 290, 2015
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5AN1
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![BU of 5an1 by Molmil](/molmil-images/mine/5an1) | |
5AWN
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![BU of 5awn by Molmil](/molmil-images/mine/5awn) | |
5AMU
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![BU of 5amu by Molmil](/molmil-images/mine/5amu) | IglE I39A,Y40A,V44A | 分子名称: | IGLE | 著者 | Robb, C.S, Nano, F.E, Boraston, A.B. | 登録日 | 2015-09-01 | 公開日 | 2016-10-05 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | The Structure, Dimerisation and Impact on Intramacrophage Replication of Igle in Francisella Novicida To be Published
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5AC5
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![BU of 5ac5 by Molmil](/molmil-images/mine/5ac5) | GH20C, Beta-hexosaminidase from Streptococcus pneumoniae in complex with GlcNAc | 分子名称: | 1,2-ETHANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, GLYCEROL, ... | 著者 | Cid, M, Robb, C.S, Higgins, M.A, Boraston, A.B. | 登録日 | 2015-08-11 | 公開日 | 2015-09-23 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.84 Å) | 主引用文献 | A Second beta-Hexosaminidase Encoded in the Streptococcus pneumoniae Genome Provides an Expanded Biochemical Ability to Degrade Host Glycans. J. Biol. Chem., 290, 2015
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5ACO
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![BU of 5aco by Molmil](/molmil-images/mine/5aco) | Cryo-EM structure of PGT128 Fab in complex with BG505 SOSIP.664 Env trimer | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, HIV-1 ENVELOPE GLYCOPROTEIN, ... | 著者 | Lee, J.H, Ward, A.B. | 登録日 | 2015-08-17 | 公開日 | 2015-09-30 | 最終更新日 | 2020-07-29 | 実験手法 | ELECTRON MICROSCOPY (4.36 Å) | 主引用文献 | Model Building and Refinement of a Natively Glycosylated HIV-1 Env Protein by High-Resolution Cryoelectron Microscopy. Structure, 23, 2015
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5A6B
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![BU of 5a6b by Molmil](/molmil-images/mine/5a6b) | GH20C, Beta-hexosaminidase from Streptococcus pneumoniae in complex with PUGNAc | 分子名称: | MAGNESIUM ION, N-ACETYL-BETA-D-GLUCOSAMINIDASE, O-(2-ACETAMIDO-2-DEOXY D-GLUCOPYRANOSYLIDENE) AMINO-N-PHENYLCARBAMATE | 著者 | Cid, M, Robb, C.S, Higgins, M.A, Boraston, A.B. | 登録日 | 2015-06-24 | 公開日 | 2015-09-23 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.77 Å) | 主引用文献 | A Second beta-Hexosaminidase Encoded in the Streptococcus pneumoniae Genome Provides an Expanded Biochemical Ability to Degrade Host Glycans. J. Biol. Chem., 290, 2015
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5AC4
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![BU of 5ac4 by Molmil](/molmil-images/mine/5ac4) | GH20C, Beta-hexosaminidase from Streptococcus pneumoniae in complex with GalNAc | 分子名称: | 2-acetamido-2-deoxy-beta-D-galactopyranose, N-ACETYL-BETA-D-GLUCOSAMINIDASE | 著者 | Cid, M, Robb, C.S, Higgins, M.A, Boraston, A.B. | 登録日 | 2015-08-11 | 公開日 | 2015-09-23 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.08 Å) | 主引用文献 | A Second beta-Hexosaminidase Encoded in the Streptococcus pneumoniae Genome Provides an Expanded Biochemical Ability to Degrade Host Glycans. J. Biol. Chem., 290, 2015
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5A58
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![BU of 5a58 by Molmil](/molmil-images/mine/5a58) | The structure of GH101 D764N mutant from Streptococcus pneumoniae TIGR4 in complex with serinyl T-antigen | 分子名称: | 1,2-ETHANEDIOL, CALCIUM ION, CITRIC ACID, ... | 著者 | Gregg, K.J, Suits, M.D.L, Deng, L, Vocadlo, D.J, Boraston, A.B. | 登録日 | 2015-06-16 | 公開日 | 2015-09-02 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Structural Analysis of a Family 101 Glycoside Hydrolase in Complex with Carbohydrates Reveals Insights Into its Mechanism. J.Biol.Chem., 290, 2015
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5A69
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![BU of 5a69 by Molmil](/molmil-images/mine/5a69) | GH20C, Beta-hexosaminidase from Streptococcus pneumoniae in complex with Gal-PUGNAc | 分子名称: | N-ACETYL-BETA-D-GLUCOSAMINIDASE, [(Z)-[(3R,4R,5R,6R)-3-acetamido-6-(hydroxymethyl)-4,5-bis(oxidanyl)oxan-2-ylidene]amino] N-phenylcarbamate | 著者 | Cid, M, Robb, C.S, Higgins, M.A, Boraston, A.B. | 登録日 | 2015-06-24 | 公開日 | 2015-09-23 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | A Second beta-Hexosaminidase Encoded in the Streptococcus pneumoniae Genome Provides an Expanded Biochemical Ability to Degrade Host Glycans. J. Biol. Chem., 290, 2015
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5A6A
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![BU of 5a6a by Molmil](/molmil-images/mine/5a6a) | GH20C, Beta-hexosaminidase from Streptococcus pneumoniae in complex with NGT | 分子名称: | 1,2-ETHANEDIOL, 3AR,5R,6S,7R,7AR-5-HYDROXYMETHYL-2-METHYL-5,6,7,7A-TETRAHYDRO-3AH-PYRANO[3,2-D]THIAZOLE-6,7-DIOL, N-ACETYL-BETA-D-GLUCOSAMINIDASE | 著者 | Cid, M, Robb, C.S, Higgins, M.A, Boraston, A.B. | 登録日 | 2015-06-24 | 公開日 | 2015-09-23 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.69 Å) | 主引用文献 | A Second beta-Hexosaminidase Encoded in the Streptococcus pneumoniae Genome Provides an Expanded Biochemical Ability to Degrade Host Glycans. J. Biol. Chem., 290, 2015
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5A57
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![BU of 5a57 by Molmil](/molmil-images/mine/5a57) | The structure of GH101 from Streptococcus pneumoniae TIGR4 in complex with PUGT | 分子名称: | (Z)-[(3R,4R,5R,6R)-3-acetamido-6-(hydroxymethyl)-4,5-bis(oxidanyl)oxan-2-ylidene]amino] N-phenylcarbamate, 1,2-ETHANEDIOL, CALCIUM ION, ... | 著者 | Gregg, K.J, Suits, M.D.L, Deng, L, Vocadlo, D.J, Boraston, A.B. | 登録日 | 2015-06-16 | 公開日 | 2015-09-02 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.46 Å) | 主引用文献 | Structural Analysis of a Family 101 Glycoside Hydrolase in Complex with Carbohydrates Reveals Insights Into its Mechanism. J.Biol.Chem., 290, 2015
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5A56
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![BU of 5a56 by Molmil](/molmil-images/mine/5a56) | The structure of GH101 from Streptococcus pneumoniae TIGR4 in complex with 1-O-methyl-T-antigen | 分子名称: | 1,2-ETHANEDIOL, CALCIUM ION, CITRIC ACID, ... | 著者 | Gregg, K.J, Suits, M.D.L, Deng, L, Vocadlo, D.J, Boraston, A.B. | 登録日 | 2015-06-16 | 公開日 | 2015-09-02 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Structural Analysis of a Family 101 Glycoside Hydrolase in Complex with Carbohydrates Reveals Insights into Its Mechanism. J.Biol.Chem., 290, 2015
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5AMT
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![BU of 5amt by Molmil](/molmil-images/mine/5amt) | Intracellular growth locus protein E | 分子名称: | 1,2-ETHANEDIOL, BROMIDE ION, IGLE | 著者 | Robb, C.S, Nano, F.E, Boraston, A.B. | 登録日 | 2015-09-01 | 公開日 | 2016-10-05 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.62 Å) | 主引用文献 | Cloning, Expression, Purification, Crystallization and Preliminary X-Ray Diffraction Analysis of Intracellular Growth Locus E (Igle) Protein from Francisella Tularensis Subsp. Novicida. Acta Crystallogr.,Sect.F, 66, 2010
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5A5A
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![BU of 5a5a by Molmil](/molmil-images/mine/5a5a) | The structure of GH101 E796Q mutant from Streptococcus pneumoniae TIGR4 in complex with PNP-T-antigen | 分子名称: | 1,2-ETHANEDIOL, CALCIUM ION, CITRIC ACID, ... | 著者 | Gregg, K.J, Suits, M.D.L, Deng, L, Vocadlo, D.J, Boraston, A.B. | 登録日 | 2015-06-16 | 公開日 | 2015-09-02 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Structural Analysis of a Family 101 Glycoside Hydrolase in Complex with Carbohydrates Reveals Insights Into its Mechanism. J.Biol.Chem., 290, 2015
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5BYK
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![BU of 5byk by Molmil](/molmil-images/mine/5byk) | Schistosoma mansoni (Blood Fluke) Sulfotransferase/S-oxamniquine Complex | 分子名称: | ADENOSINE-3'-5'-DIPHOSPHATE, SODIUM ION, Sulfotransferase, ... | 著者 | Taylor, A.B, Cao, X, Holloway, S.P, Hart, P.J. | 登録日 | 2015-06-10 | 公開日 | 2015-09-30 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.28 Å) | 主引用文献 | Structural and Functional Characterization of the Enantiomers of the Antischistosomal Drug Oxamniquine. Plos Negl Trop Dis, 9, 2015
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5AKO
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![BU of 5ako by Molmil](/molmil-images/mine/5ako) | |
5A29
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![BU of 5a29 by Molmil](/molmil-images/mine/5a29) | Family 2 Pectate Lyase from Vibrio vulnificus | 分子名称: | 1,2-ETHANEDIOL, EXOPOLYGALACTURONATE LYASE, MANGANESE (II) ION, ... | 著者 | McLean, R, Hobbs, J.K, Suits, M.D, Tuomivaara, S, Jones, D, Boraston, A.B, Abbott, D.W. | 登録日 | 2015-05-15 | 公開日 | 2015-07-01 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Functional Analyses of Resurrected and Contemporary Enzymes Illuminate an Evolutionary Path for the Emergence of Exolysis in Polysaccharide Lyase Family 2. J.Biol.Chem., 290, 2015
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5A59
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![BU of 5a59 by Molmil](/molmil-images/mine/5a59) | The structure of GH101 E796Q mutant from Streptococcus pneumoniae TIGR4 in complex with T-antigen | 分子名称: | 1,2-ETHANEDIOL, CALCIUM ION, CITRIC ACID, ... | 著者 | Gregg, K.J, Suits, M.D.L, Deng, L, Vocadlo, D.J, Boraston, A.B. | 登録日 | 2015-06-16 | 公開日 | 2015-09-02 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Structural Analysis of a Family 101 Glycoside Hydrolase in Complex with Carbohydrates Reveals Insights Into its Mechanism. J.Biol.Chem., 290, 2015
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5BYJ
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![BU of 5byj by Molmil](/molmil-images/mine/5byj) | Schistosoma mansoni (Blood Fluke) Sulfotransferase/R-oxamniquine Complex | 分子名称: | ADENOSINE-3'-5'-DIPHOSPHATE, Sulfotransferase, {(2R)-7-nitro-2-[(propan-2-ylamino)methyl]-1,2,3,4-tetrahydroquinolin-6-yl}methanol | 著者 | Taylor, A.B, Cao, X, Holloway, S.P, Hart, P.J. | 登録日 | 2015-06-10 | 公開日 | 2015-09-30 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Structural and Functional Characterization of the Enantiomers of the Antischistosomal Drug Oxamniquine. Plos Negl Trop Dis, 9, 2015
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5CCK
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![BU of 5cck by Molmil](/molmil-images/mine/5cck) | |