5I96
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![BU of 5i96 by Molmil](/molmil-images/mine/5i96) | Crystal Structure of Human Mitochondrial Isocitrate Dehydrogenase (IDH2) R140Q Mutant Homodimer in Complex with AG-221 (Enasidenib) Inhibitor. | Descriptor: | 2-methyl-1-[(4-[6-(trifluoromethyl)pyridin-2-yl]-6-{[2-(trifluoromethyl)pyridin-4-yl]amino}-1,3,5-triazin-2-yl)amino]propan-2-ol, ACETATE ION, CALCIUM ION, ... | Authors: | Wei, W, Zhang, B, Jin, L, Jiang, F, DeLaBarre, B, Travins, J.A, Padyana, A.K. | Deposit date: | 2016-02-19 | Release date: | 2017-03-08 | Last modified: | 2023-09-27 | Method: | X-RAY DIFFRACTION (1.55 Å) | Cite: | AG-221, a First-in-Class Therapy Targeting Acute Myeloid Leukemia Harboring Oncogenic IDH2 Mutations. Cancer Discov, 7, 2017
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5I95
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![BU of 5i95 by Molmil](/molmil-images/mine/5i95) | Crystal Structure of Human Mitochondrial Isocitrate Dehydrogenase R140Q Mutant Homodimer bound to NADPH and alpha-Ketoglutaric acid | Descriptor: | 2-OXOGLUTARIC ACID, ACETATE ION, CALCIUM ION, ... | Authors: | Zhang, B, Jin, L, Wu, W, Jiang, F, DeLaBarre, B, Travins, J.A, Padyana, A.K. | Deposit date: | 2016-02-19 | Release date: | 2017-03-01 | Last modified: | 2023-09-27 | Method: | X-RAY DIFFRACTION (1.54 Å) | Cite: | AG-221, a First-in-Class Therapy Targeting Acute Myeloid Leukemia Harboring Oncogenic IDH2 Mutations. Cancer Discov, 7, 2017
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5XGA
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![BU of 5xga by Molmil](/molmil-images/mine/5xga) | Crystal structure of the EnvZ periplasmic domain with CHAPS | Descriptor: | 3-[(3-CHOLAMIDOPROPYL)DIMETHYLAMMONIO]-1-PROPANESULFONATE, ACETIC ACID, Osmolarity sensor protein EnvZ | Authors: | Hwang, E, Cheong, H.K, Jeon, Y.H, Cheong, C. | Deposit date: | 2017-04-13 | Release date: | 2017-07-19 | Last modified: | 2024-03-27 | Method: | X-RAY DIFFRACTION (1.951 Å) | Cite: | Crystal structure of the EnvZ periplasmic domain with CHAPS. FEBS Lett., 591, 2017
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1DDT
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![BU of 1ddt by Molmil](/molmil-images/mine/1ddt) | |
1VJS
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![BU of 1vjs by Molmil](/molmil-images/mine/1vjs) | |
6C6P
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![BU of 6c6p by Molmil](/molmil-images/mine/6c6p) | Human squalene epoxidase (SQLE, squalene monooxygenase) structure with FAD and NB-598 | Descriptor: | (2E)-N-({3-[([3,3'-bithiophen]-5-yl)methoxy]phenyl}methyl)-N-ethyl-6,6-dimethylhept-2-en-4-yn-1-amine, 3-[(3-CHOLAMIDOPROPYL)DIMETHYLAMMONIO]-1-PROPANESULFONATE, FLAVIN-ADENINE DINUCLEOTIDE, ... | Authors: | Padyana, A.K, Jin, L. | Deposit date: | 2018-01-19 | Release date: | 2019-01-16 | Last modified: | 2024-03-13 | Method: | X-RAY DIFFRACTION (2.5 Å) | Cite: | Structure and inhibition mechanism of the catalytic domain of human squalene epoxidase. Nat Commun, 10, 2019
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6C6N
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![BU of 6c6n by Molmil](/molmil-images/mine/6c6n) | |
6C6R
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![BU of 6c6r by Molmil](/molmil-images/mine/6c6r) | |
2G60
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![BU of 2g60 by Molmil](/molmil-images/mine/2g60) | Structure of anti-FLAG M2 Fab domain | Descriptor: | anti-FLAG M2 Fab heavy chain, anti-FLAG M2 Fab light chain | Authors: | Roosild, T.P. | Deposit date: | 2006-02-23 | Release date: | 2006-09-12 | Last modified: | 2017-10-18 | Method: | X-RAY DIFFRACTION (1.85 Å) | Cite: | Structure of anti-FLAG M2 Fab domain and its use in the stabilization of engineered membrane proteins. Acta Crystallogr.,Sect.F, 62, 2006
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2Q8R
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![BU of 2q8r by Molmil](/molmil-images/mine/2q8r) | |
2QCQ
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![BU of 2qcq by Molmil](/molmil-images/mine/2qcq) | |
2QCW
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![BU of 2qcw by Molmil](/molmil-images/mine/2qcw) | |
1SGK
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![BU of 1sgk by Molmil](/molmil-images/mine/1sgk) | NUCLEOTIDE-FREE DIPHTHERIA TOXIN | Descriptor: | DIPHTHERIA TOXIN (DIMERIC) | Authors: | Bell, C.E, Eisenberg, D. | Deposit date: | 1996-09-12 | Release date: | 1996-12-23 | Last modified: | 2023-08-09 | Method: | X-RAY DIFFRACTION (2.3 Å) | Cite: | Crystal structure of nucleotide-free diphtheria toxin. Biochemistry, 36, 1997
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1DTP
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![BU of 1dtp by Molmil](/molmil-images/mine/1dtp) | |
4MID
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![BU of 4mid by Molmil](/molmil-images/mine/4mid) | Crystal Structure of Activin A/BMP2 chimera | Descriptor: | AB204 Activin A/BMP2 chimera | Authors: | Esquivies, L. | Deposit date: | 2013-08-30 | Release date: | 2014-05-07 | Last modified: | 2019-07-17 | Method: | X-RAY DIFFRACTION (2.139 Å) | Cite: | An Activin A/BMP2 Chimera, AB204, Displays Bone-Healing Properties Superior to Those of BMP2. J.Bone Miner.Res., 29, 2014
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4N1D
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![BU of 4n1d by Molmil](/molmil-images/mine/4n1d) | Nodal/BMP2 chimera NB250 | Descriptor: | Nodal/BMP2 chimera protein | Authors: | Esquivies, L. | Deposit date: | 2013-10-04 | Release date: | 2013-12-04 | Last modified: | 2017-07-26 | Method: | X-RAY DIFFRACTION (1.912 Å) | Cite: | Designer Nodal/BMP2 Chimeras Mimic Nodal Signaling, Promote Chondrogenesis, and Reveal a BMP2-like Structure. J.Biol.Chem., 289, 2014
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2XKY
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![BU of 2xky by Molmil](/molmil-images/mine/2xky) | Single particle analysis of Kir2.1NC_4 in negative stain | Descriptor: | INWARD RECTIFIER POTASSIUM CHANNEL 2 | Authors: | Fomina, S, Howard, T.D, Sleator, O.K, Golovanova, M, O'Ryan, L, Leyland, M.L, Grossmann, J.G, Collins, R.F, Prince, S.M. | Deposit date: | 2010-07-15 | Release date: | 2011-07-20 | Last modified: | 2024-05-08 | Method: | ELECTRON MICROSCOPY (17.200001 Å), SOLUTION SCATTERING | Cite: | Self-Directed Assembly and Clustering of the Cytoplasmic Domains of Inwardly Rectifying Kir2.1 Potassium Channels on Association with Psd-95 Biochim.Biophys.Acta, 1808, 2011
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1AUR
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![BU of 1aur by Molmil](/molmil-images/mine/1aur) | |
1AUO
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![BU of 1auo by Molmil](/molmil-images/mine/1auo) | CARBOXYLESTERASE FROM PSEUDOMONAS FLUORESCENS | Descriptor: | CARBOXYLESTERASE | Authors: | Kim, K.K, Song, H.K, Suh, S.W. | Deposit date: | 1997-09-01 | Release date: | 1998-03-04 | Last modified: | 2024-02-07 | Method: | X-RAY DIFFRACTION (1.8 Å) | Cite: | Crystal structure of carboxylesterase from Pseudomonas fluorescens, an alpha/beta hydrolase with broad substrate specificity. Structure, 5, 1997
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5I05
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![BU of 5i05 by Molmil](/molmil-images/mine/5i05) | |
2HMU
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![BU of 2hmu by Molmil](/molmil-images/mine/2hmu) | |
2HMV
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![BU of 2hmv by Molmil](/molmil-images/mine/2hmv) | |
2HMS
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![BU of 2hms by Molmil](/molmil-images/mine/2hms) | |
2HMW
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![BU of 2hmw by Molmil](/molmil-images/mine/2hmw) | |
2HMT
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![BU of 2hmt by Molmil](/molmil-images/mine/2hmt) | |