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6SBA
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BU of 6sba by Molmil
Crystal Structure of mTEAD with a VGL4 Tertiary Structure Mimetic
Descriptor: ACETYL GROUP, GLYCEROL, Transcriptional enhancer factor TEF-3, ...
Authors:Adihou, H, Grossmann, T.N, Waldmann, H, Gasper, R.
Deposit date:2019-07-19
Release date:2020-09-30
Last modified:2024-01-24
Method:X-RAY DIFFRACTION (1.3 Å)
Cite:A protein tertiary structure mimetic modulator of the Hippo signalling pathway.
Nat Commun, 11, 2020
5VZ2
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BU of 5vz2 by Molmil
Structure of ClpP from Staphylococcus aureus in complex with Acyldepsipeptide
Descriptor: ATP-dependent Clp protease proteolytic subunit, Acyldepsipeptide
Authors:Griffith, E.C, Lee, R.E.
Deposit date:2017-05-26
Release date:2017-06-21
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (2.26 Å)
Cite:Ureadepsipeptides as ClpP Activators.
Acs Infect Dis., 2019
6DUY
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BU of 6duy by Molmil
Crystal structure of the alpha-N-catenin actin-binding domain H1 mutant
Descriptor: Catenin alpha-2
Authors:Ishiyama, N, Ikura, M.
Deposit date:2018-06-22
Release date:2018-12-19
Last modified:2023-10-11
Method:X-RAY DIFFRACTION (2.81 Å)
Cite:Force-dependent allostery of the alpha-catenin actin-binding domain controls adherens junction dynamics and functions.
Nat Commun, 9, 2018
5W18
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BU of 5w18 by Molmil
Staphylococcus aureus ClpP in complex with (S)-N-((2R,6S,8aS,14aS,20S,23aS)-2,6-dimethyl-5,8,14,19,23-pentaoxooctadecahydro-1H,5H,14H,19H-pyrido[2,1-i]dipyrrolo[2,1-c:2',1'-l][1]oxa[4,7,10,13]tetraazacyclohexadecin-20-yl)-3-phenyl-2-(3-phenylureido)propanamide
Descriptor: 9V7-PHE-SER-PRO-YCP-ALA-MP8, ATP-dependent Clp protease proteolytic subunit
Authors:Lee, R.E, Griffith, E.C.
Deposit date:2017-06-02
Release date:2017-08-09
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (2.44 Å)
Cite:Ureadepsipeptides as ClpP Activators.
Acs Infect Dis., 2019
6D1Q
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BU of 6d1q by Molmil
Crystal structure of E. coli RppH-DapF complex, monomer
Descriptor: CHLORIDE ION, Diaminopimelate epimerase, GLYCEROL, ...
Authors:Gao, A, Serganov, A.
Deposit date:2018-04-12
Release date:2018-05-23
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (2.15 Å)
Cite:Structural and kinetic insights into stimulation of RppH-dependent RNA degradation by the metabolic enzyme DapF.
Nucleic Acids Res., 46, 2018
6D13
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BU of 6d13 by Molmil
Crystal structure of E.coli RppH-DapF complex
Descriptor: CHLORIDE ION, Diaminopimelate epimerase, IODIDE ION, ...
Authors:Gao, A, Serganov, A.
Deposit date:2018-04-11
Release date:2018-05-23
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (3.06 Å)
Cite:Structural and kinetic insights into stimulation of RppH-dependent RNA degradation by the metabolic enzyme DapF.
Nucleic Acids Res., 46, 2018
6DUW
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BU of 6duw by Molmil
Crystal structure of the alpha-N-catenin actin-binding domain H1 mutant
Descriptor: Catenin alpha-2
Authors:Ishiyama, N, Ikura, M.
Deposit date:2018-06-22
Release date:2018-12-19
Last modified:2023-10-11
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Force-dependent allostery of the alpha-catenin actin-binding domain controls adherens junction dynamics and functions.
Nat Commun, 9, 2018
6DV1
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BU of 6dv1 by Molmil
Crystal structure of the alpha-E-catenin actin-binding domain
Descriptor: BROMIDE ION, Catenin alpha-1, SULFATE ION
Authors:Ishiyama, N, Ikura, M.
Deposit date:2018-06-22
Release date:2018-12-19
Last modified:2024-03-13
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Force-dependent allostery of the alpha-catenin actin-binding domain controls adherens junction dynamics and functions.
Nat Commun, 9, 2018
6E4F
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BU of 6e4f by Molmil
Crystal structure of ARQ 531 in complex with the kinase domain of BTK
Descriptor: 1,2-ETHANEDIOL, 1,5-anhydro-2-{[5-(2-chloro-4-phenoxybenzene-1-carbonyl)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino}-2,3,4-trideoxy-D-erythro-hexitol, IMIDAZOLE, ...
Authors:Eathiraj, S.
Deposit date:2018-07-17
Release date:2018-09-05
Last modified:2024-03-13
Method:X-RAY DIFFRACTION (1.15 Å)
Cite:The BTK Inhibitor ARQ 531 Targets Ibrutinib-Resistant CLL and Richter Transformation.
Cancer Discov, 8, 2018
6D1V
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BU of 6d1v by Molmil
Crystal structure of E. coli RppH-DapF complex, monomer bound to RNA
Descriptor: CHLORIDE ION, Diaminopimelate epimerase, GLYCEROL, ...
Authors:Gao, A, Serganov, A.
Deposit date:2018-04-12
Release date:2018-05-23
Last modified:2024-03-13
Method:X-RAY DIFFRACTION (1.81 Å)
Cite:Structural and kinetic insights into stimulation of RppH-dependent RNA degradation by the metabolic enzyme DapF.
Nucleic Acids Res., 46, 2018
5NZ9
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BU of 5nz9 by Molmil
NMR structure of an EphA2-Sam fragment
Descriptor: Ephrin type-A receptor 2
Authors:Mercurio, F.A, Leone, M.
Deposit date:2017-05-12
Release date:2017-12-20
Last modified:2023-06-14
Method:SOLUTION NMR
Cite:The Sam-Sam interaction between Ship2 and the EphA2 receptor: design and analysis of peptide inhibitors.
Sci Rep, 7, 2017
7SP3
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BU of 7sp3 by Molmil
E. coli RppH bound to Ap4A
Descriptor: BIS(ADENOSINE)-5'-TETRAPHOSPHATE, CHLORIDE ION, FLUORIDE ION, ...
Authors:Serganov, A.A, Vasilyev, N, Nuthanakanti, A.
Deposit date:2021-11-02
Release date:2022-03-09
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (1.6 Å)
Cite:A distinct RNA recognition mechanism governs Np 4 decapping by RppH.
Proc.Natl.Acad.Sci.USA, 119, 2022
6CFD
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BU of 6cfd by Molmil
ADEP4 bound to E. faecium ClpP
Descriptor: (4S)-2-METHYL-2,4-PENTANEDIOL, ATP-dependent Clp protease proteolytic subunit, N-[(6aS,12S,15aS,17R,21R,23aS)-17,21-dimethyl-6,11,15,20,23-pentaoxooctadecahydro-2H,6H,11H,15H-pyrido[2,1-i]dipyrrolo[2,1-c:2',1'-l][1,4,7,10,13]oxatetraazacyclohexadecin-12-yl]-3,5-difluoro-Nalpha-[(2E)-hept-2-enoyl]-L-phenylalaninamide
Authors:Lee, R.E, Griffith, E.C.
Deposit date:2018-02-14
Release date:2018-05-16
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (2.57 Å)
Cite:In VivoandIn VitroEffects of a ClpP-Activating Antibiotic against Vancomycin-Resistant Enterococci.
Antimicrob. Agents Chemother., 62, 2018
3C7X
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BU of 3c7x by Molmil
Hemopexin-like domain of matrix metalloproteinase 14
Descriptor: CHLORIDE ION, Matrix metalloproteinase-14, SODIUM ION
Authors:Tochowicz, A, Itoh, Y, Maskos, K, Bode, W, Goettig, P.
Deposit date:2008-02-08
Release date:2009-02-10
Last modified:2023-11-01
Method:X-RAY DIFFRACTION (1.7 Å)
Cite:The dimer interface of the membrane type 1 matrix metalloproteinase hemopexin domain: crystal structure and biological functions
J.Biol.Chem., 286, 2011
4OS7
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BU of 4os7 by Molmil
Crystal structure of urokinase-type plasminogen activator (uPA) complexed with bicyclic peptide UK607 (bicyclic)
Descriptor: ACETATE ION, GLYCEROL, SULFATE ION, ...
Authors:Chen, S, Pojer, F, Heinis, C.
Deposit date:2014-02-12
Release date:2014-09-24
Last modified:2021-06-02
Method:X-RAY DIFFRACTION (2 Å)
Cite:Dithiol amino acids can structurally shape and enhance the ligand-binding properties of polypeptides.
Nat Chem, 6, 2014
4OS5
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BU of 4os5 by Molmil
Crystal structure of urokinase-type plasminogen activator (uPA) complexed with bicyclic peptide UK603 (bicyclic 2)
Descriptor: SULFATE ION, Urokinase-type plasminogen activator, bicyclic peptide UK603 (bicyclic 2)
Authors:Chen, S, Pojer, F, Heinis, C.
Deposit date:2014-02-12
Release date:2014-09-24
Last modified:2021-06-02
Method:X-RAY DIFFRACTION (2.26 Å)
Cite:Dithiol amino acids can structurally shape and enhance the ligand-binding properties of polypeptides.
Nat Chem, 6, 2014
4OS1
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BU of 4os1 by Molmil
Crystal structure of urokinase-type plasminogen activator (uPA) complexed with bicyclic peptide UK601 (bicyclic 1)
Descriptor: ACETATE ION, SULFATE ION, Urokinase-type plasminogen activator, ...
Authors:Chen, S, Pojer, F, Heinis, C.
Deposit date:2014-02-12
Release date:2014-09-24
Last modified:2021-06-02
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Dithiol amino acids can structurally shape and enhance the ligand-binding properties of polypeptides.
Nat Chem, 6, 2014
4OS4
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BU of 4os4 by Molmil
Crystal structure of urokinase-type plasminogen activator (uPA) complexed with bicyclic peptide UK603 (bicyclic 1)
Descriptor: ACETATE ION, CHLORIDE ION, GLYCEROL, ...
Authors:Chen, S, Pojer, F, Heinis, C.
Deposit date:2014-02-12
Release date:2014-09-24
Last modified:2021-06-02
Method:X-RAY DIFFRACTION (2 Å)
Cite:Dithiol amino acids can structurally shape and enhance the ligand-binding properties of polypeptides.
Nat Chem, 6, 2014
4OS6
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BU of 4os6 by Molmil
Crystal structure of urokinase-type plasminogen activator (uPA) complexed with bicyclic peptide UK604 (bicyclic 2)
Descriptor: ACETATE ION, SULFATE ION, Urokinase-type plasminogen activator, ...
Authors:Chen, S, Pojer, F, Heinis, C.
Deposit date:2014-02-12
Release date:2014-09-24
Last modified:2021-06-02
Method:X-RAY DIFFRACTION (1.75 Å)
Cite:Dithiol amino acids can structurally shape and enhance the ligand-binding properties of polypeptides.
Nat Chem, 6, 2014
6O2W
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BU of 6o2w by Molmil
Crystal structure of the SARAF luminal domain Cys-lock mutant dimer
Descriptor: GLYCEROL, Store-operated calcium entry-associated regulatory factor
Authors:Kimberlin, C.R, Minor, D.L.
Deposit date:2019-02-24
Release date:2019-05-29
Last modified:2023-10-11
Method:X-RAY DIFFRACTION (2.101 Å)
Cite:SARAF Luminal Domain Structure Reveals a Novel Domain-Swapped beta-Sandwich Fold Important for SOCE Modulation.
J.Mol.Biol., 431, 2019
6O2U
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BU of 6o2u by Molmil
Crystal structure of the SARAF luminal domain
Descriptor: Store-operated calcium entry-associated regulatory factor
Authors:Kimberlin, C.R, Minor, D.L.
Deposit date:2019-02-24
Release date:2019-05-29
Last modified:2019-12-04
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:SARAF Luminal Domain Structure Reveals a Novel Domain-Swapped beta-Sandwich Fold Important for SOCE Modulation.
J.Mol.Biol., 431, 2019
6O2V
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BU of 6o2v by Molmil
Crystal structure of the SARAF luminal domain Cys-lock mutant monomer
Descriptor: FORMIC ACID, GLYCEROL, Store-operated calcium entry-associated regulatory factor
Authors:Kimberlin, C.R, Minor, D.L.
Deposit date:2019-02-24
Release date:2019-05-29
Last modified:2023-10-11
Method:X-RAY DIFFRACTION (1.58 Å)
Cite:SARAF Luminal Domain Structure Reveals a Novel Domain-Swapped beta-Sandwich Fold Important for SOCE Modulation.
J.Mol.Biol., 431, 2019
6PE6
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BU of 6pe6 by Molmil
PANK3 complex structure with compound PZ-3022
Descriptor: 6-{4-[(4-cyclopropylphenyl)acetyl]piperazin-1-yl}pyridazine-3-carbonitrile, MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, ...
Authors:White, S.W, Yun, M.
Deposit date:2019-06-20
Release date:2020-12-23
Last modified:2023-10-11
Method:X-RAY DIFFRACTION (1.6 Å)
Cite:Pantothenate kinase activation relieves coenzyme A sequestration and improves mitochondrial function in mice with propionic acidemia.
Sci Transl Med, 13, 2021
4OS2
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BU of 4os2 by Molmil
Crystal structure of urokinase-type plasminogen activator (uPA) complexed with bicyclic peptide UK602 (bicyclic 1)
Descriptor: ACETATE ION, SULFATE ION, Urokinase-type plasminogen activator, ...
Authors:Chen, S, Pojer, F, Heinis, C.
Deposit date:2014-02-12
Release date:2014-09-24
Last modified:2021-06-02
Method:X-RAY DIFFRACTION (1.79 Å)
Cite:Dithiol amino acids can structurally shape and enhance the ligand-binding properties of polypeptides.
Nat Chem, 6, 2014
3UDL
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BU of 3udl by Molmil
3-heterocyclyl quinolone bound to HCV NS5B
Descriptor: 3-(5-benzyl-1,2,4-oxadiazol-3-yl)-6-fluoro-1-[2-fluoro-4-(trifluoromethyl)benzyl]-7-(4-methylpiperazin-1-yl)quinolin-4(1H)-one, HCV NS5B polymerase
Authors:Somoza, J.R.
Deposit date:2011-10-28
Release date:2011-12-21
Method:X-RAY DIFFRACTION (2.174 Å)
Cite:Quinolones as HCV NS5B polymerase inhibitors.
Bioorg.Med.Chem.Lett., 21, 2011

221716

数据于2024-06-26公开中

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