7TC3
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![BU of 7tc3 by Molmil](/molmil-images/mine/7tc3) | Human APE1 in the apo form | 分子名称: | 1,2-ETHANEDIOL, DNA-(apurinic or apyrimidinic site) endonuclease, mitochondrial | 著者 | Pidugu, L.S, Pozharski, E, Drohat, A.C. | 登録日 | 2021-12-22 | 公開日 | 2022-12-21 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.252 Å) | 主引用文献 | Characterizing inhibitors of human AP endonuclease 1. Plos One, 18, 2023
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7TC2
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![BU of 7tc2 by Molmil](/molmil-images/mine/7tc2) | Human APE1 in complex with 5-nitroindole-2-carboxylic acid | 分子名称: | 1,2-ETHANEDIOL, 5-nitro-1H-indole-2-carboxylic acid, DI(HYDROXYETHYL)ETHER, ... | 著者 | Pidugu, L.S, Pozharski, E, Drohat, A.C. | 登録日 | 2021-12-22 | 公開日 | 2022-12-21 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.43 Å) | 主引用文献 | Characterizing inhibitors of human AP endonuclease 1. Plos One, 18, 2023
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5EA2
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![BU of 5ea2 by Molmil](/molmil-images/mine/5ea2) | Crystal Structure of Holo NAD(P)H dehydrogenase, quinone 1 | 分子名称: | FLAVIN-ADENINE DINUCLEOTIDE, NAD(P)H dehydrogenase [quinone] 1 | 著者 | Pidugu, L.S, Mbimba, J.E, Ahmad, M, Pozharski, E, Sausville, E.A, Emadi, A, Toth, E.A. | 登録日 | 2015-10-15 | 公開日 | 2016-02-10 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.01 Å) | 主引用文献 | A direct interaction between NQO1 and a chemotherapeutic dimeric naphthoquinone. Bmc Struct.Biol., 16, 2016
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5EAI
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![BU of 5eai by Molmil](/molmil-images/mine/5eai) | Crystal Structure of NAD(P)H dehydrogenase, quinone 1 complexed with a chemotherapeutic naphthoquinone E6a | 分子名称: | (2~{R},3~{R})-2-[(2~{S},3~{S})-3-bromanyl-1,4-bis(oxidanylidene)-2,3-dihydronaphthalen-2-yl]-3-oxidanyl-2,3-dihydronaphthalene-1,4-dione, FLAVIN-ADENINE DINUCLEOTIDE, NAD(P)H dehydrogenase [quinone] 1 | 著者 | Pidugu, L.S, Mbimba, J.E, Ahmad, M, Pozharski, E, Sausville, E.A, Emadi, A, Toth, E.A. | 登録日 | 2015-10-16 | 公開日 | 2016-02-17 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | A direct interaction between NQO1 and a chemotherapeutic dimeric naphthoquinone. Bmc Struct.Biol., 16, 2016
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6U15
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![BU of 6u15 by Molmil](/molmil-images/mine/6u15) | |
6U16
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![BU of 6u16 by Molmil](/molmil-images/mine/6u16) | Human thymine DNA glycosylase N140A mutant bound to DNA with 5-carboxyl-dC substrate | 分子名称: | 1,2-ETHANEDIOL, DNA (28-MER), G/T mismatch-specific thymine DNA glycosylase | 著者 | Pidugu, L.S, Pozharski, E, Drohat, A.C. | 登録日 | 2019-08-15 | 公開日 | 2019-11-20 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Excision of 5-Carboxylcytosine by Thymine DNA Glycosylase. J.Am.Chem.Soc., 141, 2019
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6U17
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![BU of 6u17 by Molmil](/molmil-images/mine/6u17) | Human thymine DNA glycosylase bound to DNA with 2'-F-5-carboxyl-dC substrate analog | 分子名称: | ACETATE ION, DNA (28-MER), DNA (30-MER), ... | 著者 | Pidugu, L.S, Pozharski, E, Drohat, A.C. | 登録日 | 2019-08-15 | 公開日 | 2019-11-20 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Excision of 5-Carboxylcytosine by Thymine DNA Glycosylase. J.Am.Chem.Soc., 141, 2019
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7KZ0
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![BU of 7kz0 by Molmil](/molmil-images/mine/7kz0) | Human MBD4 glycosylase domain bound to DNA containing substrate analog 2'-deoxy-pseudouridine | 分子名称: | DNA (5'-D(*CP*CP*AP*GP*CP*GP*(P2U)P*GP*CP*AP*GP*C)-3'), DNA (5'-D(*GP*CP*TP*GP*CP*GP*CP*GP*CP*TP*GP*G)-3'), GLYCEROL, ... | 著者 | Pidugu, L.S, Pozharski, E, Drohat, A.C. | 登録日 | 2020-12-09 | 公開日 | 2021-11-10 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.57 Å) | 主引用文献 | Structural Insights into the Mechanism of Base Excision by MBD4. J.Mol.Biol., 433, 2021
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7KZG
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![BU of 7kzg by Molmil](/molmil-images/mine/7kzg) | Human MBD4 glycosylase domain bound to DNA containing oxacarbenium-ion analog 1-aza-2'-deoxyribose | 分子名称: | 1,2-ETHANEDIOL, CHLORIDE ION, DI(HYDROXYETHYL)ETHER, ... | 著者 | Pidugu, L.S, Pozharski, E, Drohat, A.C. | 登録日 | 2020-12-10 | 公開日 | 2021-11-10 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.68 Å) | 主引用文献 | Structural Insights into the Mechanism of Base Excision by MBD4. J.Mol.Biol., 433, 2021
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7KZ1
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![BU of 7kz1 by Molmil](/molmil-images/mine/7kz1) | Human MBD4 glycosylase domain bound to DNA containing an abasic site | 分子名称: | 1,2-ETHANEDIOL, DNA (5'-D(*CP*CP*AP*GP*CP*GP*(ORP)P*GP*CP*AP*GP*C)-3'), DNA (5'-D(*GP*CP*TP*GP*CP*GP*CP*GP*CP*TP*GP*G)-3'), ... | 著者 | Pidugu, L.S, Bright, H, Pozharski, E, Drohat, A.C. | 登録日 | 2020-12-09 | 公開日 | 2021-11-10 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.62 Å) | 主引用文献 | Structural Insights into the Mechanism of Base Excision by MBD4. J.Mol.Biol., 433, 2021
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5T2W
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![BU of 5t2w by Molmil](/molmil-images/mine/5t2w) | |
5TKQ
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![BU of 5tkq by Molmil](/molmil-images/mine/5tkq) | |
5TK5
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![BU of 5tk5 by Molmil](/molmil-images/mine/5tk5) | |
5JXY
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![BU of 5jxy by Molmil](/molmil-images/mine/5jxy) | Enzyme-substrate complex of TDG catalytic domain bound to a G/U analog | 分子名称: | DNA (28-MER), G/T mismatch-specific thymine DNA glycosylase | 著者 | Pidugu, L.S, Pozharski, E, Malik, S.S, Drohat, A.C. | 登録日 | 2016-05-13 | 公開日 | 2016-09-28 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.71 Å) | 主引用文献 | Structural basis of damage recognition by thymine DNA glycosylase: Key roles for N-terminal residues. Nucleic Acids Res., 44, 2016
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1UH5
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![BU of 1uh5 by Molmil](/molmil-images/mine/1uh5) | Crystal Structure of Enoyl-ACP Reductase with Triclosan at 2.2angstroms | 分子名称: | NICOTINAMIDE-ADENINE-DINUCLEOTIDE, TRICLOSAN, enoyl-ACP reductase | 著者 | Swarnamukhi, P.L, Kapoor, M, Surolia, N, Surolia, A, Suguna, K. | 登録日 | 2003-06-24 | 公開日 | 2004-09-28 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Structural basis for the variation in triclosan affinity to enoyl reductases. J.Mol.Biol., 343, 2004
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1V35
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![BU of 1v35 by Molmil](/molmil-images/mine/1v35) | Crystal Structure of Eoyl-ACP Reductase with NADH | 分子名称: | 1,4-DIHYDRONICOTINAMIDE ADENINE DINUCLEOTIDE, enoyl-ACP reductase | 著者 | SwarnaMukhi, P.L, Kapoor, M, surolia, N, Surolia, A, Suguna, K. | 登録日 | 2003-10-28 | 公開日 | 2004-09-28 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Structural basis for the variation in triclosan affinity to enoyl reductases. J.Mol.Biol., 343, 2004
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5FF8
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![BU of 5ff8 by Molmil](/molmil-images/mine/5ff8) | TDG enzyme-product complex | 分子名称: | DNA, G/T mismatch-specific thymine DNA glycosylase | 著者 | Pozharski, E, Malik, S.S, Drohat, A.C. | 登録日 | 2015-12-18 | 公開日 | 2016-09-28 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Structural basis of damage recognition by thymine DNA glycosylase: Key roles for N-terminal residues. Nucleic Acids Res., 44, 2016
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5HF7
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![BU of 5hf7 by Molmil](/molmil-images/mine/5hf7) | TDG enzyme-substrate complex | 分子名称: | DNA (28-MER), G/T mismatch-specific thymine DNA glycosylase | 著者 | Pozharski, E, Malik, S.S, Drohat, A.C. | 登録日 | 2016-01-06 | 公開日 | 2016-09-28 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.54 Å) | 主引用文献 | Structural basis of damage recognition by thymine DNA glycosylase: Key roles for N-terminal residues. Nucleic Acids Res., 44, 2016
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