6RVA
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![BU of 6rva by Molmil](/molmil-images/mine/6rva) | STRUCTURE OF [ASP58]-IGF-I ANALOGUE | 分子名称: | Insulin-like growth factor I | 著者 | Jiracek, J, Zakova, L, Socha, O. | 登録日 | 2019-05-31 | 公開日 | 2019-10-02 | 最終更新日 | 2023-06-14 | 実験手法 | SOLUTION NMR | 主引用文献 | Mutations at hypothetical binding site 2 in insulin and insulin-like growth factors 1 and 2 result in receptor- and hormone-specific responses. J.Biol.Chem., 294, 2019
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2WS7
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![BU of 2ws7 by Molmil](/molmil-images/mine/2ws7) | Semi-synthetic analogue of human insulin ProB26-DTI | 分子名称: | CHLORIDE ION, INSULIN A CHAIN, INSULIN B CHAIN, ... | 著者 | Brzozowski, A.M, Jiracek, J, Zakova, L, Antolikova, E, Watson, C.J, Turkenburg, J.P, Dodson, G.G. | 登録日 | 2009-09-03 | 公開日 | 2010-02-09 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.59 Å) | 主引用文献 | Implications for the Active Form of Human Insulin Based on the Structural Convergence of Highly Active Hormone Analogues. Proc.Natl.Acad.Sci.USA, 107, 2010
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2WRU
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![BU of 2wru by Molmil](/molmil-images/mine/2wru) | Semi-synthetic highly active analogue of human insulin NMeAlaB26-DTI- NH2 | 分子名称: | ACETATE ION, INSULIN A CHAIN, INSULIN B CHAIN | 著者 | Brzozowski, A.M, Jiracek, J, Zakova, L, Antolikova, E, Watson, C.J, Turkenburg, J.P, Dodson, G.G. | 登録日 | 2009-09-02 | 公開日 | 2010-02-09 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.57 Å) | 主引用文献 | Implications for the Active Form of Human Insulin Based on the Structural Convergence of Highly Active Hormone Analogues. Proc.Natl.Acad.Sci.USA, 107, 2010
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2WS4
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![BU of 2ws4 by Molmil](/molmil-images/mine/2ws4) | Semi-synthetic analogue of human insulin ProB26-DTI in monomer form | 分子名称: | INSULIN A CHAIN, INSULIN B CHAIN | 著者 | Brzozowski, A.M, Jiracek, J, Zakova, L, Antolikova, E, Watson, C.J, Turkenburg, J.P, Dodson, G.G. | 登録日 | 2009-09-03 | 公開日 | 2010-02-09 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Implications for the Active Form of Human Insulin Based on the Structural Convergence of Highly Active Hormone Analogues. Proc.Natl.Acad.Sci.USA, 107, 2010
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2WS0
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![BU of 2ws0 by Molmil](/molmil-images/mine/2ws0) | Semi-synthetic analogue of human insulin NMeAlaB26-insulin at pH 7.5 | 分子名称: | INSULIN A CHAIN, INSULIN B CHAIN | 著者 | Brzozowski, A.M, Jiracek, J, Zakova, L, Antolikova, E, Watson, C.J, Turkenburg, J.P, Dodson, G.G. | 登録日 | 2009-09-03 | 公開日 | 2010-02-09 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Implications for the Active Form of Human Insulin Based on the Structural Convergence of Highly Active Hormone Analogues. Proc.Natl.Acad.Sci.USA, 107, 2010
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2WRX
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![BU of 2wrx by Molmil](/molmil-images/mine/2wrx) | Semi-synthetic analogue of human insulin NMeAlaB26-insulin at pH 3.0 | 分子名称: | INSULIN A CHAIN, INSULIN B CHAIN, SODIUM ION | 著者 | Brzozowski, A.M, Jiracek, J, Zakova, L, Antolikova, E, Watson, C.J, Turkenburg, J.P, Dodson, G.G. | 登録日 | 2009-09-02 | 公開日 | 2010-02-09 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Implications for the Active Form of Human Insulin Based on the Structural Convergence of Highly Active Hormone Analogues. Proc.Natl.Acad.Sci.USA, 107, 2010
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2WS1
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![BU of 2ws1 by Molmil](/molmil-images/mine/2ws1) | Semi-synthetic analogue of human insulin NMeTyrB26-insulin in monomer form | 分子名称: | ACETATE ION, INSULIN A CHAIN, INSULIN B CHAIN | 著者 | Brzozowski, A.M, Jiracek, J, Zakova, L, Antolikova, E, Watson, C.J, Turkenburg, J.P, Dodson, G.G. | 登録日 | 2009-09-03 | 公開日 | 2010-02-09 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Implications for the Active Form of Human Insulin Based on the Structural Convergence of Highly Active Hormone Analogues. Proc.Natl.Acad.Sci.USA, 107, 2010
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2WRV
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![BU of 2wrv by Molmil](/molmil-images/mine/2wrv) | Semi-synthetic highly active analogue of human insulin NMeHisB26-DTI- NH2 | 分子名称: | ACETATE ION, INSULIN A CHAIN, INSULIN B CHAIN | 著者 | Brzozowski, A.M, Jiracek, J, Zakova, L, Antolikova, E, Watson, C.J, Turkenburg, J.P, Dodson, G.G. | 登録日 | 2009-09-02 | 公開日 | 2010-02-09 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.15 Å) | 主引用文献 | Implications for the Active Form of Human Insulin Based on the Structural Convergence of Highly Active Hormone Analogues. Proc.Natl.Acad.Sci.USA, 107, 2010
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2WRW
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![BU of 2wrw by Molmil](/molmil-images/mine/2wrw) | Semi-synthetic highly active analogue of human insulin D-ProB26-DTI- NH2 | 分子名称: | INSULIN A CHAIN, INSULIN B CHAIN | 著者 | Brzozowski, A.M, Jiracek, J, Zakova, L, Antolikova, E, Watson, C.J, Turkenburg, J.P, Dodson, G.G. | 登録日 | 2009-09-02 | 公開日 | 2010-02-09 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.41 Å) | 主引用文献 | Implications for the Active Form of Human Insulin Based on the Structural Convergence of Highly Active Hormone Analogues. Proc.Natl.Acad.Sci.USA, 107, 2010
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2WS6
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![BU of 2ws6 by Molmil](/molmil-images/mine/2ws6) | Semi-synthetic analogue of human insulin NMeTyrB26-insulin in hexamer form | 分子名称: | CHLORIDE ION, GLYCEROL, INSULIN A CHAIN, ... | 著者 | Brzozowski, A.M, Jiracek, J, Zakova, L, Antolikova, E, Watson, C.J, Turkenburg, J.P, Dodson, G.G. | 登録日 | 2009-09-03 | 公開日 | 2010-02-09 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Implications for the Active Form of Human Insulin Based on the Structural Convergence of Highly Active Hormone Analogues. Proc.Natl.Acad.Sci.USA, 107, 2010
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4UNG
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![BU of 4ung by Molmil](/molmil-images/mine/4ung) | Human insulin B26Asn mutant crystal structure | 分子名称: | INSULIN A CHAIN, INSULIN B CHAIN, SULFATE ION | 著者 | Zakova, L, Klevtikova, E, Lepsik, M, Collinsova, M, Watson, C.J, Turkenburg, J.P, Jiracek, J, Brzozowski, A.M. | 登録日 | 2014-05-28 | 公開日 | 2014-10-15 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.81 Å) | 主引用文献 | Human Insulin Analogues Modified at the B26 Site Reveal a Hormone Conformation that is Undetected in the Receptor Complex Acta Crystallogr.,Sect.D, 70, 2014
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4UNH
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![BU of 4unh by Molmil](/molmil-images/mine/4unh) | Human insulin B26Gly mutant crystal structure | 分子名称: | INSULIN A CHAIN, INSULIN B CHAIN, SULFATE ION | 著者 | Zakova, L, Klevtikova, E, Lepsik, M, Collinsova, M, Watson, C.J, Turkenburg, J.P, Jiracek, J, Brzozowski, A.M. | 登録日 | 2014-05-28 | 公開日 | 2014-10-15 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.75 Å) | 主引用文献 | Human Insulin Analogues Modified at the B26 Site Reveal a Hormone Conformation that is Undetected in the Receptor Complex Acta Crystallogr.,Sect.D, 70, 2014
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4M3P
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![BU of 4m3p by Molmil](/molmil-images/mine/4m3p) | Betaine-Homocysteine S-Methyltransferase from Homo sapiens complexed with Homocysteine | 分子名称: | 2-AMINO-4-MERCAPTO-BUTYRIC ACID, Betaine--homocysteine S-methyltransferase 1, POTASSIUM ION, ... | 著者 | Koutmos, M, Yamada, K, Mladkova, J, Paterova, J, Diamond, C.E, Tryon, K, Jungwirth, P, Garrow, T.A, Jiracek, J. | 登録日 | 2013-08-06 | 公開日 | 2014-06-18 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.895 Å) | 主引用文献 | Specific potassium ion interactions facilitate homocysteine binding to betaine-homocysteine S-methyltransferase. Proteins, 82, 2014
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4UNE
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![BU of 4une by Molmil](/molmil-images/mine/4une) | Human insulin B26Phe mutant crystal structure | 分子名称: | INSULIN A CHAIN, INSULIN B CHAIN, SULFATE ION | 著者 | Zakova, L, Klevtikova, E, Lepsik, M, Collinsova, M, Watson, C.J, Turkenburg, J.P, Jiracek, J, Brzozowski, A.M. | 登録日 | 2014-05-28 | 公開日 | 2014-10-15 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.59 Å) | 主引用文献 | Human Insulin Analogues Modified at the B26 Site Reveal a Hormone Conformation that is Undetected in the Receptor Complex Acta Crystallogr.,Sect.D, 70, 2014
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5BOQ
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![BU of 5boq by Molmil](/molmil-images/mine/5boq) | Human insulin with intra-chain chemical crosslink between modified B24 and B29 | 分子名称: | Insulin, SULFATE ION | 著者 | Brzozowski, A.M, Turkenburg, J.P, Jiracek, J, Zakova, L. | 登録日 | 2015-05-27 | 公開日 | 2016-02-03 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Rational steering of insulin binding specificity by intra-chain chemical crosslinking. Sci Rep, 6, 2016
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5BPO
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![BU of 5bpo by Molmil](/molmil-images/mine/5bpo) | |
5BQQ
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![BU of 5bqq by Molmil](/molmil-images/mine/5bqq) | Human insulin with intra-chain chemical crosslink between modified B27 and B30 | 分子名称: | CHLORIDE ION, Insulin, PHENOL, ... | 著者 | Brzozowski, A.M, Turkenburg, J.P, Jiracek, J, Zakova, L. | 登録日 | 2015-05-29 | 公開日 | 2016-02-03 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.54 Å) | 主引用文献 | Rational steering of insulin binding specificity by intra-chain chemical crosslinking. Sci Rep, 6, 2016
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8ONP
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![BU of 8onp by Molmil](/molmil-images/mine/8onp) | |
8ONR
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![BU of 8onr by Molmil](/molmil-images/mine/8onr) | |
8OKY
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![BU of 8oky by Molmil](/molmil-images/mine/8oky) | |
1LT7
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![BU of 1lt7 by Molmil](/molmil-images/mine/1lt7) | Oxidized Homo sapiens betaine-homocysteine S-methyltransferase in complex with four Sm(III) ions | 分子名称: | BETAINE-HOMOCYSTEINE METHYLTRANSFERASE, CITRIC ACID, SAMARIUM (III) ION | 著者 | Evans, J.C, Huddler, D.P, Jiracek, J, Castro, C, Millian, N.S, Garrow, T.A, Ludwig, M.L. | 登録日 | 2002-05-20 | 公開日 | 2002-09-11 | 最終更新日 | 2021-10-27 | 実験手法 | X-RAY DIFFRACTION (2.15 Å) | 主引用文献 | Betaine-homocysteine methyltransferase: zinc in a distorted barrel. Structure, 10, 2002
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1LT8
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![BU of 1lt8 by Molmil](/molmil-images/mine/1lt8) | Reduced Homo sapiens Betaine-Homocysteine S-Methyltransferase in Complex with S-(delta-carboxybutyl)-L-Homocysteine | 分子名称: | BETAINE-HOMOCYSTEINE METHYLTRANSFERASE, CITRIC ACID, S-(D-CARBOXYBUTYL)-L-HOMOCYSTEINE, ... | 著者 | Evans, J.C, Huddler, D.P, Jiracek, J, Castro, C, Millian, N.S, Garrow, T.A, Ludwig, M.L. | 登録日 | 2002-05-20 | 公開日 | 2002-09-11 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | Betaine-homocysteine methyltransferase: zinc in a distorted barrel. Structure, 10, 2002
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4CXL
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![BU of 4cxl by Molmil](/molmil-images/mine/4cxl) | Human insulin analogue (D-ProB8)-insulin | 分子名称: | CHLORIDE ION, INSULIN A CHAIN, INSULIN B CHAIN | 著者 | Kosinova, L, Veverka, V, Novotna, P, Collinsova, M, Urbanova, M, Jiracek, J, Moody, N.R, Turkenburg, J.P, Brzozowski, A.M, Zakova, L. | 登録日 | 2014-04-07 | 公開日 | 2014-05-28 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | An Insight Into Structural and Biological Relevance of the T/R Transition of the B-Chain N-Terminus in Human Insulin. Biochemistry, 53, 2014
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4CXN
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![BU of 4cxn by Molmil](/molmil-images/mine/4cxn) | Crystal structure of human insulin analogue (NMe-AlaB8)-insulin crystal form I | 分子名称: | INSULIN A CHAIN, INSULIN B CHAIN | 著者 | Kosinova, L, Veverka, V, Novotna, P, Collinsova, M, Urbanova, M, Jiracek, J, Moody, N.R, Turkenburg, J.P, Brzozowski, A.M, Zakova, L. | 登録日 | 2014-04-07 | 公開日 | 2014-05-28 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | An Insight Into Structural and Biological Relevance of the T/R Transition of the B-Chain N-Terminus in Human Insulin. Biochemistry, 53, 2014
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4CY7
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![BU of 4cy7 by Molmil](/molmil-images/mine/4cy7) | Crystal structure of human insulin analogue (NMe-AlaB8)-insulin crystal form II | 分子名称: | ACETATE ION, INSULIN A CHAIN, INSULIN B CHAIN, ... | 著者 | Kosinova, L, Veverka, V, Novotna, P, Collinsova, M, Urbanova, M, Jiracek, J, Moody, N.R, Turkenburg, J.P, Brzozowski, A.M, Zakova, L. | 登録日 | 2014-04-10 | 公開日 | 2014-05-28 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | An Insight Into Structural and Biological Relevance of the T/R Transition of the B-Chain N-Terminus in Human Insulin. Biochemistry, 53, 2014
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