4WUA
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![BU of 4wua by Molmil](/molmil-images/mine/4wua) | Crystal structure of human SRPK1 complexed to an inhibitor SRPIN340 | 分子名称: | CITRIC ACID, N-[2-(1-piperidinyl)-5-(trifluoromethyl)phenyl]-4-pyridinecarboxamide, SRSF protein kinase 1, ... | 著者 | Hoshina, M, Ikura, T, Hosoya, T, Hagiwara, M, Ito, N. | 登録日 | 2014-10-31 | 公開日 | 2015-09-16 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Identification of a Dual Inhibitor of SRPK1 and CK2 That Attenuates Pathological Angiogenesis of Macular Degeneration in Mice Mol.Pharmacol., 88, 2015
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2RU3
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![BU of 2ru3 by Molmil](/molmil-images/mine/2ru3) | Solution structure of c.elegans SUP-12 RRM in complex with RNA | 分子名称: | Protein SUP-12, isoform a, RNA (5'-R(*GP*UP*GP*UP*GP*C)-3') | 著者 | Takahashi, M, Kuwasako, K, Unzai, S, Tsuda, K, Yoshikawa, S, He, F, Kobayashi, N, Guntert, P, Shirouzu, M, Ito, T, Tanaka, A, Yokoyama, S, Hagiwara, M, Kuroyanagi, H, Muto, Y. | 登録日 | 2013-11-12 | 公開日 | 2014-08-13 | 最終更新日 | 2024-05-15 | 実験手法 | SOLUTION NMR | 主引用文献 | RBFOX and SUP-12 sandwich a G base to cooperatively regulate tissue-specific splicing Nat.Struct.Mol.Biol., 21, 2014
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2MGZ
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![BU of 2mgz by Molmil](/molmil-images/mine/2mgz) | Solution structure of RBFOX family ASD-1 RRM and SUP-12 RRM in ternary complex with RNA | 分子名称: | Protein ASD-1, isoform a, Protein SUP-12, ... | 著者 | Takahashi, M, Kuwasako, K, Unzai, S, Tsuda, K, Yoshikawa, S, He, F, Kobayashi, N, Guntert, P, Shirouzu, M, Ito, T, Tanaka, A, Yokoyama, S, Hagiwara, M, Kuroyanagi, H, Muto, Y. | 登録日 | 2013-11-12 | 公開日 | 2014-08-13 | 最終更新日 | 2024-05-01 | 実験手法 | SOLUTION NMR | 主引用文献 | RBFOX and SUP-12 sandwich a G base to cooperatively regulate tissue-specific splicing Nat.Struct.Mol.Biol., 21, 2014
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3ANR
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![BU of 3anr by Molmil](/molmil-images/mine/3anr) | human DYRK1A/harmine complex | 分子名称: | 7-METHOXY-1-METHYL-9H-BETA-CARBOLINE, Dual specificity tyrosine-phosphorylation-regulated kinase 1A | 著者 | Nonaka, Y, Hosoya, T, Hagiwara, M, Ito, N. | 登録日 | 2010-09-06 | 公開日 | 2010-11-10 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Development of a novel selective inhibitor of the Down syndrome-related kinase Dyrk1A Nat Commun, 1, 2010
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3ANQ
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![BU of 3anq by Molmil](/molmil-images/mine/3anq) | human DYRK1A/inhibitor complex | 分子名称: | (1Z)-1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2(3H)-ylidene)propan-2-one, Dual specificity tyrosine-phosphorylation-regulated kinase 1A | 著者 | Nonaka, Y, Hosoya, T, Hagiwara, M, Ito, N. | 登録日 | 2010-09-06 | 公開日 | 2010-11-10 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Development of a novel selective inhibitor of the Down syndrome-related kinase Dyrk1A Nat Commun, 1, 2010
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3APQ
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3APO
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![BU of 3apo by Molmil](/molmil-images/mine/3apo) | |
3APS
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![BU of 3aps by Molmil](/molmil-images/mine/3aps) | |
7C4S
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![BU of 7c4s by Molmil](/molmil-images/mine/7c4s) | Sphingosine-1-phosphate receptor 3 with a natural ligand. | 分子名称: | (2S,3R,4E)-2-amino-3-hydroxyoctadec-4-en-1-yl dihydrogen phosphate, Antibody Fab fragment heavy chain, Antibody Fab fragment light chain, ... | 著者 | Iwata, S, Maeda, S, Luo, F, Nango, E, hirata, K, Asada, H. | 登録日 | 2020-05-18 | 公開日 | 2021-06-09 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | Endogenous agonist-bound S1PR3 structure reveals determinants of G protein-subtype bias. Sci Adv, 7, 2021
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3VWU
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![BU of 3vwu by Molmil](/molmil-images/mine/3vwu) | |
3VWV
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![BU of 3vwv by Molmil](/molmil-images/mine/3vwv) | |
3VWW
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![BU of 3vww by Molmil](/molmil-images/mine/3vww) | |
3W8J
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![BU of 3w8j by Molmil](/molmil-images/mine/3w8j) | Crystal structure of P5 a0 in a complex with Prx4 c-term | 分子名称: | C-terminal peptide from Peroxiredoxin-4, GLYCEROL, POTASSIUM ION, ... | 著者 | Inaba, K, Suzuki, M, Kojima, R. | 登録日 | 2013-03-13 | 公開日 | 2013-09-04 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Synergistic cooperation of PDI family members in peroxiredoxin 4-driven oxidative protein folding Sci Rep, 3, 2013
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1YDT
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![BU of 1ydt by Molmil](/molmil-images/mine/1ydt) | STRUCTURE OF CAMP-DEPENDENT PROTEIN KINASE, ALPHA-CATALYTIC SUBUNIT IN COMPLEX WITH H89 PROTEIN KINASE INHIBITOR N-[2-(4-BROMOCINNAMYLAMINO)ETHYL]-5-ISOQUINOLINE | 分子名称: | C-AMP-DEPENDENT PROTEIN KINASE, N-[2-(4-BROMOCINNAMYLAMINO)ETHYL]-5-ISOQUINOLINE SULFONAMIDE, PROTEIN KINASE INHIBITOR PEPTIDE | 著者 | Engh, R.A, Girod, A, Kinzel, V, Huber, R, Bossemeyer, D. | 登録日 | 1996-07-24 | 公開日 | 1997-04-01 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Crystal structures of catalytic subunit of cAMP-dependent protein kinase in complex with isoquinolinesulfonyl protein kinase inhibitors H7, H8, and H89. Structural implications for selectivity. J.Biol.Chem., 271, 1996
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