4GWQ
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![BU of 4gwq by Molmil](/molmil-images/mine/4gwq) | Structure of the Mediator Head Module from S. cerevisiae in complex with the carboxy-terminal domain (CTD) of RNA Polymerase II Rpb1 subunit | 分子名称: | DNA-directed RNA polymerase II subunit RPB1, Mediator of RNA polymerase II transcription subunit 11, Mediator of RNA polymerase II transcription subunit 17, ... | 著者 | Robinson, P.J.J, Bushnell, D.A, Trnka, M.J, Burlingame, A.L, Kornberg, R.D. | 登録日 | 2012-09-03 | 公開日 | 2012-10-31 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (4.5 Å) | 主引用文献 | Structure of the Mediator Head module bound to the carboxy-terminal domain of RNA polymerase II. Proc.Natl.Acad.Sci.USA, 109, 2012
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4GWP
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![BU of 4gwp by Molmil](/molmil-images/mine/4gwp) | Structure of the Mediator Head Module from S. cerevisiae | 分子名称: | Mediator of RNA polymerase II transcription subunit 11, Mediator of RNA polymerase II transcription subunit 17, Mediator of RNA polymerase II transcription subunit 18, ... | 著者 | Robinson, P.J.J, Bushnell, D.A, Trnka, M.J, Burlingame, A.L, Kornberg, R.D. | 登録日 | 2012-09-03 | 公開日 | 2012-10-31 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (4.2 Å) | 主引用文献 | Structure of the Mediator Head module bound to the carboxy-terminal domain of RNA polymerase II. Proc.Natl.Acad.Sci.USA, 109, 2012
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2X5W
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![BU of 2x5w by Molmil](/molmil-images/mine/2x5w) | X-ray structure of Mycobacterium tuberculosis cytochrome P450 CYP125 in complex with substrate cholest-4-en-3-one | 分子名称: | (8ALPHA,9BETA)-CHOLEST-4-EN-3-ONE, 1,2-ETHANEDIOL, PROTOPORPHYRIN IX CONTAINING FE, ... | 著者 | Ouellet, H, Guan, S, Johnston, J.B, Chow, E.D, Kells, P.M, Burlingame, A.L, Cox, J.S, Podust, L.M, Ortiz de Montellano, P.R. | 登録日 | 2010-02-10 | 公開日 | 2010-06-16 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.58 Å) | 主引用文献 | Mycobacterium Tuberculosis Cyp125A1, a Steroid C27 Monooxygenase that Detoxifies Intracellularly Generated Cholest-4-En-3-One. Mol.Microbiol., 77, 2010
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8JHU
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![BU of 8jhu by Molmil](/molmil-images/mine/8jhu) | Legionella effector protein SidI | 分子名称: | Legionella pneumophila effector protein SidI | 著者 | Wang, L, Subramanian, A, Mukherjee, S, Walter, P. | 登録日 | 2023-05-25 | 公開日 | 2023-08-30 | 最終更新日 | 2024-05-08 | 実験手法 | ELECTRON MICROSCOPY (3.1 Å) | 主引用文献 | A Legionella toxin exhibits tRNA mimicry and glycosyl transferase activity to target the translation machinery and trigger a ribotoxic stress response. Nat.Cell Biol., 25, 2023
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7FIC
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![BU of 7fic by Molmil](/molmil-images/mine/7fic) | |
1WMA
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![BU of 1wma by Molmil](/molmil-images/mine/1wma) | Crystal structure of human CBR1 in complex with Hydroxy-PP | 分子名称: | 3,6,9,12,15,18,21,24-OCTAOXAHEXACOSAN-1-OL, 3,6,9,12,15,18-HEXAOXAICOSANE-1,20-DIOL, 3-(4-AMINO-1-TERT-BUTYL-1H-PYRAZOLO[3,4-D]PYRIMIDIN-3-YL)PHENOL, ... | 著者 | Rauh, D, Bateman, R, Shokat, K.M. | 登録日 | 2004-07-06 | 公開日 | 2005-04-26 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (1.24 Å) | 主引用文献 | An unbiased cell morphology-based screen for new, biologically active small molecules Plos Biol., 3, 2005
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6C3R
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![BU of 6c3r by Molmil](/molmil-images/mine/6c3r) | |
5SVA
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![BU of 5sva by Molmil](/molmil-images/mine/5sva) | Mediator-RNA Polymerase II Pre-Initiation Complex | 分子名称: | 108bp HIS4 Promoter Non-template Strand (-92/+16), 108bp HIS4 Promoter Template Strand (+16/-92), DNA repair helicase RAD25, ... | 著者 | Robinson, P.J, Bushnell, D.A, Kornberg, R.D. | 登録日 | 2016-08-05 | 公開日 | 2016-09-28 | 最終更新日 | 2019-11-27 | 実験手法 | ELECTRON MICROSCOPY (15.3 Å) | 主引用文献 | Structure of a Complete Mediator-RNA Polymerase II Pre-Initiation Complex. Cell, 166, 2016
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5U8L
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5IX2
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![BU of 5ix2 by Molmil](/molmil-images/mine/5ix2) | Crystal structure of mouse Morc3 ATPase-CW cassette in complex with AMPPNP and unmodified H3 peptide | 分子名称: | MAGNESIUM ION, MORC family CW-type zinc finger protein 3, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, ... | 著者 | Li, S, Du, J, Patel, D.J. | 登録日 | 2016-03-23 | 公開日 | 2016-08-17 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Mouse MORC3 is a GHKL ATPase that localizes to H3K4me3 marked chromatin Proc.Natl.Acad.Sci.USA, 113, 2016
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5IX1
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![BU of 5ix1 by Molmil](/molmil-images/mine/5ix1) | Crystal structure of mouse Morc3 ATPase-CW cassette in complex with AMPPNP and H3K4me3 peptide | 分子名称: | MAGNESIUM ION, MORC family CW-type zinc finger protein 3, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, ... | 著者 | Li, S, Du, J, Patel, D.J. | 登録日 | 2016-03-23 | 公開日 | 2016-08-17 | 最終更新日 | 2016-09-14 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Mouse MORC3 is a GHKL ATPase that localizes to H3K4me3 marked chromatin Proc.Natl.Acad.Sci.USA, 113, 2016
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5K9I
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![BU of 5k9i by Molmil](/molmil-images/mine/5k9i) | Crystal structure of c-SRC in complex with a covalent lysine probe | 分子名称: | 4-[(4-{4-[(3-cyclopropyl-1H-pyrazol-5-yl)amino]-6-[(prop-2-yn-1-yl)carbamoyl]pyrimidin-2-yl}piperazin-1-yl)methyl]benzene-1-sulfonyl fluoride, Proto-oncogene tyrosine-protein kinase Src | 著者 | Wan, X, Ouyang, S, Zhao, Q, Taunton, J. | 登録日 | 2016-05-31 | 公開日 | 2017-02-01 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Broad-Spectrum Kinase Profiling in Live Cells with Lysine-Targeted Sulfonyl Fluoride Probes. J. Am. Chem. Soc., 139, 2017
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6U98
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![BU of 6u98 by Molmil](/molmil-images/mine/6u98) | Hsp90a NTD K58R bound reversibly to sulfonyl fluoride 6 | 分子名称: | 3-{[(3R)-3-({6-amino-8-[(6-iodo-2H-1,3-benzodioxol-5-yl)sulfanyl]-9H-purin-9-yl}methyl)piperidin-1-yl]methyl}benzene-1-sulfonyl fluoride, Heat shock protein HSP 90-alpha, POTASSIUM ION, ... | 著者 | Cuesta, A, Wan, X, Taunton, J. | 登録日 | 2019-09-06 | 公開日 | 2020-02-19 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Ligand Conformational Bias Drives Enantioselective Modification of a Surface-Exposed Lysine on Hsp90. J.Am.Chem.Soc., 142, 2020
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6U9B
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![BU of 6u9b by Molmil](/molmil-images/mine/6u9b) | Hsp90a NTD covalently bound to sulfonyl fluoride 5 at K58 | 分子名称: | 3-{[(3S)-3-({6-amino-8-[(6-iodo-2H-1,3-benzodioxol-5-yl)sulfanyl]-9H-purin-9-yl}methyl)piperidin-1-yl]methyl}benzene-1-sulfonyl fluoride, Heat shock protein HSP 90-alpha | 著者 | Cuesta, A, Wan, X, Taunton, J. | 登録日 | 2019-09-07 | 公開日 | 2020-02-19 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Ligand Conformational Bias Drives Enantioselective Modification of a Surface-Exposed Lysine on Hsp90. J.Am.Chem.Soc., 142, 2020
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6U99
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![BU of 6u99 by Molmil](/molmil-images/mine/6u99) | Hsp90a NTD covalently bound to sulfonyl fluoride probe 1 at K58 | 分子名称: | 3-{[(3-{6-amino-8-[(6-iodo-2H-1,3-benzodioxol-5-yl)sulfanyl]-9H-purin-9-yl}propyl)amino]methyl}benzene-1-sulfinic acid, Heat shock protein HSP 90-alpha | 著者 | Cuesta, A, Wan, X, Taunton, J. | 登録日 | 2019-09-06 | 公開日 | 2020-02-19 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Ligand Conformational Bias Drives Enantioselective Modification of a Surface-Exposed Lysine on Hsp90. J.Am.Chem.Soc., 142, 2020
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6U9A
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![BU of 6u9a by Molmil](/molmil-images/mine/6u9a) | Hsp90a NTD K58R bound reversibly to sulfonyl fluoride 5 | 分子名称: | 3-{[(3S)-3-({6-amino-8-[(6-iodo-2H-1,3-benzodioxol-5-yl)sulfanyl]-9H-purin-9-yl}methyl)piperidin-1-yl]methyl}benzene-1-sulfonyl fluoride, Heat shock protein HSP 90-alpha | 著者 | Cuesta, A, Wan, X, Taunton, J. | 登録日 | 2019-09-07 | 公開日 | 2020-02-19 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | Ligand Conformational Bias Drives Enantioselective Modification of a Surface-Exposed Lysine on Hsp90. J.Am.Chem.Soc., 142, 2020
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6W6L
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1PEN
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![BU of 1pen by Molmil](/molmil-images/mine/1pen) | ALPHA-CONOTOXIN PNI1 | 分子名称: | ALPHA-CONOTOXIN PNIA | 著者 | Hu, S.-H, Gehrmann, J, Guddat, L.W, Alewood, P.F, Craik, D.J, Martin, J.L. | 登録日 | 1996-01-29 | 公開日 | 1997-04-21 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.1 Å) | 主引用文献 | The 1.1 A crystal structure of the neuronal acetylcholine receptor antagonist, alpha-conotoxin PnIA from Conus pennaceus. Structure, 4, 1996
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2Y4I
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![BU of 2y4i by Molmil](/molmil-images/mine/2y4i) | KSR2-MEK1 heterodimer | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, CHLORIDE ION, DUAL SPECIFICITY MITOGEN-ACTIVATED PROTEIN KINASE KINASE 1, ... | 著者 | Brennan, D.F, Barford, D. | 登録日 | 2011-01-06 | 公開日 | 2011-01-19 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (3.46 Å) | 主引用文献 | A Raf-Induced Allosteric Transition of Ksr Stimulates Ksr and Raf Phosphorylation of Mek Nature, 472, 2011
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