6ZUJ
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![BU of 6zuj by Molmil](/molmil-images/mine/6zuj) | Human serine racemase holoenzyme from 20% DMSO soak (XChem crystallographic fragment screen). | 分子名称: | 1,2-ETHANEDIOL, CALCIUM ION, DIMETHYL SULFOXIDE, ... | 著者 | Koulouris, C.R, Bax, B.D, Roe, S.M, Atack, J.R. | 登録日 | 2020-07-23 | 公開日 | 2021-03-03 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Tyrosine 121 moves revealing a ligandable pocket that couples catalysis to ATP-binding in serine racemase. Commun Biol, 5, 2022
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6ZSP
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![BU of 6zsp by Molmil](/molmil-images/mine/6zsp) | Human serine racemase bound to ATP and malonate. | 分子名称: | 1,2-ETHANEDIOL, ADENOSINE-5'-TRIPHOSPHATE, GLYCEROL, ... | 著者 | Koulouris, C.R, Bax, B.D, Roe, S.M, Atack, J.R. | 登録日 | 2020-07-16 | 公開日 | 2021-03-03 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Tyrosine 121 moves revealing a ligandable pocket that couples catalysis to ATP-binding in serine racemase. Commun Biol, 5, 2022
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6FIE
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![BU of 6fie by Molmil](/molmil-images/mine/6fie) | Crystallographic structure of calcium loaded Calbindin-D28K. | 分子名称: | CALCIUM ION, Calbindin, THIOCYANATE ION | 著者 | Noble, J.W, Almalki, R, Roe, S.M, Wagner, A, Dumanc, R, Atack, J.R. | 登録日 | 2018-01-18 | 公開日 | 2018-10-10 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (1.51 Å) | 主引用文献 | The X-ray structure of human calbindin-D28K: an improved model. Acta Crystallogr D Struct Biol, 74, 2018
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6SLH
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![BU of 6slh by Molmil](/molmil-images/mine/6slh) | Conformational flexibility within the small domain of human serine racemase. | 分子名称: | MAGNESIUM ION, SODIUM ION, Serine racemase, ... | 著者 | Koulouris, C.R, Bax, B, Atack, J, Roe, S.M. | 登録日 | 2019-08-19 | 公開日 | 2020-02-12 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.89 Å) | 主引用文献 | Conformational flexibility within the small domain of human serine racemase. Acta Crystallogr.,Sect.F, 76, 2020
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2HHM
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![BU of 2hhm by Molmil](/molmil-images/mine/2hhm) | |
6ZK0
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![BU of 6zk0 by Molmil](/molmil-images/mine/6zk0) | 1.47A human IMPase with ebselen | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, GLYCEROL, Inositol monophosphatase 1, ... | 著者 | Bax, B.D, Fenn, G.D. | 登録日 | 2020-06-29 | 公開日 | 2020-09-23 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.47 Å) | 主引用文献 | Crystallization and structure of ebselen bound to Cys141 of human inositol monophosphatase. Acta Crystallogr.,Sect.F, 76, 2020
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5J42
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![BU of 5j42 by Molmil](/molmil-images/mine/5j42) | Crystal structure of m2hTDP2-CAT in complex with a small molecule inhibitor | 分子名称: | 1,2-ETHANEDIOL, 10-(4-hydroxyphenyl)-2,4-dioxo-2,3,4,10-tetrahydropyrimido[4,5-b]quinoline-8-carbonitrile, GLYCEROL, ... | 著者 | Hornyak, P, Pearl, L.H, Caldecott, K.W, Oliver, A.W. | 登録日 | 2016-03-31 | 公開日 | 2016-05-04 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Mode of action of DNA-competitive small molecule inhibitors of tyrosyl DNA phosphodiesterase 2. Biochem.J., 473, 2016
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5J3P
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![BU of 5j3p by Molmil](/molmil-images/mine/5j3p) | Crystal structure of the catalytic domain of human tyrosyl DNA phosphodiesterase 2 | 分子名称: | GLYCEROL, MAGNESIUM ION, Tyrosyl-DNA phosphodiesterase 2 | 著者 | Hornyak, P, Pearl, L.H, Caldecott, K.W, Oliver, A.W. | 登録日 | 2016-03-31 | 公開日 | 2016-05-04 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Mode of action of DNA-competitive small molecule inhibitors of tyrosyl DNA phosphodiesterase 2. Biochem.J., 473, 2016
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5J3Z
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![BU of 5j3z by Molmil](/molmil-images/mine/5j3z) | Crystal structure of m2hTDP2-CAT in complex with a small molecule inhibitor | 分子名称: | 1,2-ETHANEDIOL, 2,4-dioxo-10-[3-(1H-tetrazol-5-yl)phenyl]-2,3,4,10-tetrahydropyrimido[4,5-b]quinoline-8-carbonitrile, ACETATE ION, ... | 著者 | Hornyak, P, Pearl, L.H, Caldecott, K.W, Oliver, A.W. | 登録日 | 2016-03-31 | 公開日 | 2016-05-04 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Mode of action of DNA-competitive small molecule inhibitors of tyrosyl DNA phosphodiesterase 2. Biochem.J., 473, 2016
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1IMB
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![BU of 1imb by Molmil](/molmil-images/mine/1imb) | |
1IMF
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![BU of 1imf by Molmil](/molmil-images/mine/1imf) | |
1IMC
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![BU of 1imc by Molmil](/molmil-images/mine/1imc) | |
1IMA
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![BU of 1ima by Molmil](/molmil-images/mine/1ima) | |
1IME
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![BU of 1ime by Molmil](/molmil-images/mine/1ime) | |
1IMD
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![BU of 1imd by Molmil](/molmil-images/mine/1imd) | |
5J3S
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![BU of 5j3s by Molmil](/molmil-images/mine/5j3s) | Crystal structure of the catalytic domain of human tyrosyl DNA phosphodiesterase 2 in complex with a small molecule inhibitor | 分子名称: | 2,4-dioxo-10-[3-(1H-tetrazol-5-yl)phenyl]-2,3,4,10-tetrahydropyrimido[4,5-b]quinoline-8-carbonitrile, Tyrosyl-DNA phosphodiesterase 2 | 著者 | Hornyak, P, Pearl, L.H, Caldecott, K.W, Oliver, A.W. | 登録日 | 2016-03-31 | 公開日 | 2016-05-04 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (3.4 Å) | 主引用文献 | Mode of action of DNA-competitive small molecule inhibitors of tyrosyl DNA phosphodiesterase 2. Biochem.J., 473, 2016
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6GIU
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![BU of 6giu by Molmil](/molmil-images/mine/6giu) | Human IMPase with L-690330 | 分子名称: | GLYCEROL, Inositol monophosphatase 1, MANGANESE (II) ION, ... | 著者 | Kraft, L.V, Roe, S.M. | 登録日 | 2018-05-15 | 公開日 | 2018-10-17 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.39 Å) | 主引用文献 | Co-crystallization of human inositol monophosphatase with the lithium mimetic L-690,330. Acta Crystallogr D Struct Biol, 74, 2018
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6GJ0
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![BU of 6gj0 by Molmil](/molmil-images/mine/6gj0) | Human IMPase with Mn | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, GLYCEROL, Inositol monophosphatase 1, ... | 著者 | Kraft, L.V, Roe, S.M. | 登録日 | 2018-05-15 | 公開日 | 2018-10-17 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.73 Å) | 主引用文献 | Co-crystallization of human inositol monophosphatase with the lithium mimetic L-690,330. Acta Crystallogr D Struct Biol, 74, 2018
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7NBG
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![BU of 7nbg by Molmil](/molmil-images/mine/7nbg) | Crystal structure of human serine racemase in complex with DSiP fragment Z52314092, XChem fragment screen. | 分子名称: | 1,2-ETHANEDIOL, 2-(2-METHOXYETHOXY)ETHANOL, CALCIUM ION, ... | 著者 | Koulouris, C.R, Roe, S.M. | 登録日 | 2021-01-26 | 公開日 | 2021-03-03 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.53 Å) | 主引用文献 | Tyrosine 121 moves revealing a ligandable pocket that couples catalysis to ATP-binding in serine racemase. Commun Biol, 5, 2022
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7NBH
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![BU of 7nbh by Molmil](/molmil-images/mine/7nbh) | Crystal structure of human serine racemase in complex with DSiP fragment Z26781964, XChem fragment screen. | 分子名称: | 1,2-ETHANEDIOL, CALCIUM ION, CHLORIDE ION, ... | 著者 | Koulouris, C.R, Roe, S.M. | 登録日 | 2021-01-26 | 公開日 | 2021-03-03 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.77 Å) | 主引用文献 | Tyrosine 121 moves revealing a ligandable pocket that couples catalysis to ATP-binding in serine racemase. Commun Biol, 5, 2022
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7NBD
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![BU of 7nbd by Molmil](/molmil-images/mine/7nbd) | Crystal structure of human serine racemase in complex with DSiP fragment Z235449082, XChem fragment screen. | 分子名称: | 1,2-ETHANEDIOL, CALCIUM ION, GLYCEROL, ... | 著者 | Koulouris, C.R, Roe, S.M. | 登録日 | 2021-01-26 | 公開日 | 2021-03-03 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.865 Å) | 主引用文献 | Tyrosine 121 moves revealing a ligandable pocket that couples catalysis to ATP-binding in serine racemase. Commun Biol, 5, 2022
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7NBF
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![BU of 7nbf by Molmil](/molmil-images/mine/7nbf) | Crystal structure of human serine racemase in complex with DSiP fragment Z126932614, XChem fragment screen. | 分子名称: | 1,2-ETHANEDIOL, 2-[(methylsulfonyl)methyl]-1H-benzimidazole, CALCIUM ION, ... | 著者 | Koulouris, C.R, Roe, S.M. | 登録日 | 2021-01-26 | 公開日 | 2021-03-03 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Tyrosine 121 moves revealing a ligandable pocket that couples catalysis to ATP-binding in serine racemase. Commun Biol, 5, 2022
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7NBC
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![BU of 7nbc by Molmil](/molmil-images/mine/7nbc) | Crystal structure of human serine racemase in complex with DSiP fragment Z2856434779, XChem fragment screen. | 分子名称: | 1,2-ETHANEDIOL, 2-(2-METHOXYETHOXY)ETHANOL, CALCIUM ION, ... | 著者 | Koulouris, C.R, Roe, S.M. | 登録日 | 2021-01-26 | 公開日 | 2021-03-03 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.71 Å) | 主引用文献 | Tyrosine 121 moves revealing a ligandable pocket that couples catalysis to ATP-binding in serine racemase. Commun Biol, 5, 2022
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