4UTA
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![BU of 4uta by Molmil](/molmil-images/mine/4uta) | Crystal structure of dengue 2 virus envelope glycoprotein in complex with the Fab fragment of the broadly neutralizing human antibody EDE1 C8 | 分子名称: | BROADLY NEUTRALIZING HUMAN ANTIBODY EDE1 C8 HEAVY CHAIN, BROADLY NEUTRALIZING HUMAN ANTIBODY EDE1 C8 LIGHT CHAIN, ENVELOPE GLYCOPROTEIN E, ... | 著者 | Rouvinski, A, Guardado-Calvo, P, Barba-Spaeth, G, Duquerroy, S, Vaney, M.C, Rey, F.A. | 登録日 | 2014-07-18 | 公開日 | 2015-01-28 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Recognition Determinants of Broadly Neutralizing Human Antibodies Against Dengue Viruses. Nature, 520, 2015
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4V7G
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![BU of 4v7g by Molmil](/molmil-images/mine/4v7g) | Crystal Structure of Lumazine Synthase from Bacillus Anthracis | 分子名称: | 6,7-dimethyl-8-ribityllumazine synthase, PHOSPHATE ION | 著者 | Morgunova, E, Illarionov, B, Saller, S, Popov, A, Sambaiah, T, Bacher, A, Cushman, M, Fischer, M, Ladenstein, R. | 登録日 | 2009-09-16 | 公開日 | 2014-07-09 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (3.5 Å) | 主引用文献 | Structural study and thermodynamic characterization of inhibitor binding to lumazine synthase from Bacillus anthracis. Acta Crystallogr.,Sect.D, 66, 2010
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4V5M
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![BU of 4v5m by Molmil](/molmil-images/mine/4v5m) | tRNA tranlocation on the 70S ribosome: the pre-translocational translocation intermediate TI(PRE) | 分子名称: | 16S RRNA, 23S RIBOSOMAL RNA, 30S RIBOSOMAL PROTEIN S10, ... | 著者 | Ratje, A.H, Loerke, J, Mikolajka, A, Bruenner, M, Hildebrand, P.W, Starosta, A.L, Doenhoefer, A, Connell, S.R, Fucini, P, Mielke, T, Whitford, P.C, Onuchic, J.N, Yu, Y, Sanbonmatsu, K.Y, Hartmann, R.K, Penczek, P.A, Wilson, D.N, Spahn, C.M.T. | 登録日 | 2010-10-01 | 公開日 | 2014-07-09 | 最終更新日 | 2019-12-11 | 実験手法 | ELECTRON MICROSCOPY (7.8 Å) | 主引用文献 | Head Swivel on the Ribosome Facilitates Translocation by Means of Intra-Subunit tRNA Hybrid Sites. Nature, 468, 2010
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4V67
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![BU of 4v67 by Molmil](/molmil-images/mine/4v67) | Crystal structure of a translation termination complex formed with release factor RF2. | 分子名称: | 16S RRNA, 23S RRNA, 30S ribosomal protein S10, ... | 著者 | Korostelev, A, Asahara, H, Lancaster, L, Laurberg, M, Hirschi, A, Noller, H.F. | 登録日 | 2008-10-27 | 公開日 | 2014-07-09 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Crystal structure of a translation termination complex formed with release factor RF2. Proc.Natl.Acad.Sci.USA, 105, 2008
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4UXV
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![BU of 4uxv by Molmil](/molmil-images/mine/4uxv) | Cytoplasmic domain of bacterial cell division protein EzrA | 分子名称: | SEPTATION RING FORMATION REGULATOR EZRA | 著者 | Cleverley, R.M, Barrett, J.R, Basle, A, Khai-Bui, N, Hewitt, L, Solovyova, A, Xu, Z, Daniela, R.A, Dixon, N.E, Harry, E.J, Oakley, A.J, Vollmer, W, Lewis, R.J. | 登録日 | 2014-08-27 | 公開日 | 2014-10-22 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (3.961 Å) | 主引用文献 | Structure and Function of a Spectrin-Like Regulator of Bacterial Cytokinesis. Nat.Commun., 5, 2014
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4W63
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![BU of 4w63 by Molmil](/molmil-images/mine/4w63) | TORPEDO CALIFORNICA ACETYLCHOLINESTERASE IN COMPLEX WITH A TACRINE-BENZOFURAN HYBRID INHIBITOR | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Acetylcholinesterase, ... | 著者 | Pesaresi, A, Samez, S, Lamba, D. | 登録日 | 2014-08-20 | 公開日 | 2015-09-09 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Novel Tacrine-Benzofuran Hybrids as Potent Multitarget-Directed Ligands for the Treatment of Alzheimer's Disease: Design, Synthesis, Biological Evaluation, and X-ray Crystallography. J.Med.Chem., 59, 2016
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4V29
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![BU of 4v29 by Molmil](/molmil-images/mine/4v29) | |
8RRY
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![BU of 8rry by Molmil](/molmil-images/mine/8rry) | Crystal structure of copper-loaded SmAA10 | 分子名称: | CBP21, CITRIC ACID, COPPER (II) ION, ... | 著者 | Munzone, A, Pujol, M, Reglier, M, Royant, A, Simaan, A.J, Decroos, C. | 登録日 | 2024-01-24 | 公開日 | 2024-06-12 | 実験手法 | X-RAY DIFFRACTION (1.45561326 Å) | 主引用文献 | Integrated Experimental and Theoretical Investigation of Copper Active Site Properties of a Lytic Polysaccharide Monooxygenase from Serratia marcescens. Inorg.Chem., 2024
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8BTM
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![BU of 8btm by Molmil](/molmil-images/mine/8btm) | Structural and functional studies of geldanamycin amide synthase ShGdmF | 分子名称: | 1,2-ETHANEDIOL, ACETATE ION, GdmF | 著者 | Ewert, W, Zeilinger, C, Kirschning, A, Preller, M. | 登録日 | 2022-11-29 | 公開日 | 2024-06-12 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | Structural and functional studies of geldanamycin amide synthase ShGdmF To Be Published
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4V99
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![BU of 4v99 by Molmil](/molmil-images/mine/4v99) | |
8S8A
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![BU of 8s8a by Molmil](/molmil-images/mine/8s8a) | Human pyridoxal phosphatase in complex with 7,8-dihydroxyflavone without phosphate | 分子名称: | 7,8-bis(oxidanyl)-2-phenyl-chromen-4-one, CHLORIDE ION, Chronophin, ... | 著者 | Brenner, M, Gohla, A, Schindelin, H. | 登録日 | 2024-03-06 | 公開日 | 2024-06-12 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | 7,8-Dihydroxyflavone is a direct inhibitor of pyridoxal phosphatase Elife, 13:RP93094, 2024
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8P3N
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![BU of 8p3n by Molmil](/molmil-images/mine/8p3n) | |
8P3R
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![BU of 8p3r by Molmil](/molmil-images/mine/8p3r) | |
8P59
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![BU of 8p59 by Molmil](/molmil-images/mine/8p59) | |
8P8H
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![BU of 8p8h by Molmil](/molmil-images/mine/8p8h) | Crystal structure of HHD2 domain of hRTEL1 | 分子名称: | Regulator of telomere elongation helicase 1 | 著者 | Hegde, R.P, Kanade, M, Cortone, G, Graewert, M, Longo, A, Gonzalez, A, Chaves-Arquero, B, Blanco, F.J, Napolitano, L.M.R, Onesti, S. | 登録日 | 2023-06-01 | 公開日 | 2024-06-12 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Crystal structure of HHD2 domain of hRTEL1 To Be Published
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4UT5
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![BU of 4ut5 by Molmil](/molmil-images/mine/4ut5) | Crystal structure of the LecB lectin from Pseudomonas aeruginosa strain PA7 in complex with lewis a tetrasaccharide | 分子名称: | CALCIUM ION, LECB LECTIN, beta-D-galactopyranose, ... | 著者 | Boukerb, A.M, Decor, A, Tabaroni, R, Varrot, A, Debentzmann, S, Vidal, S, Imberty, A, Cournoyer, B. | 登録日 | 2014-07-18 | 公開日 | 2015-07-22 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Genomic Rearrangements and Functional Diversification of Leca and Lecb Lectin-Coding Regions Impacting the Efficacy of Glycomimetics Directed Against Pseudomonas Aeruginosa. Front.Microbiol., 7, 2016
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8QFW
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![BU of 8qfw by Molmil](/molmil-images/mine/8qfw) | Murine pyridoxal phosphatase in complex with 7,8-dihydroxyflavone | 分子名称: | 7,8-bis(oxidanyl)-2-phenyl-chromen-4-one, CITRIC ACID, Chronophin, ... | 著者 | Schindelin, H, Gohla, A. | 登録日 | 2023-09-05 | 公開日 | 2024-06-12 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | 7,8-Dihydroxyflavone is a direct inhibitor of pyridoxal phosphatase Elife, 13:RP93094, 2024
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4V4H
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![BU of 4v4h by Molmil](/molmil-images/mine/4v4h) | Crystal structure of the bacterial ribosome from Escherichia coli in complex with the antibiotic kasugamyin at 3.5A resolution. | 分子名称: | (1S,2R,3S,4R,5S,6S)-2,3,4,5,6-PENTAHYDROXYCYCLOHEXYL 2-AMINO-4-{[CARBOXY(IMINO)METHYL]AMINO}-2,3,4,6-TETRADEOXY-ALPHA-D-ARABINO-HEXOPYRANOSIDE, 16S RIBOSOMAL RNA, 23S RIBOSOMAL RNA, ... | 著者 | Schuwirth, B.S, Vila-Sanjurjo, A, Cate, J.H.D. | 登録日 | 2006-08-04 | 公開日 | 2014-07-09 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (3.46 Å) | 主引用文献 | Structural analysis of kasugamycin inhibition of translation. Nat.Struct.Mol.Biol., 13, 2006
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4V7P
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![BU of 4v7p by Molmil](/molmil-images/mine/4v7p) | Recognition of the amber stop codon by release factor RF1. | 分子名称: | 16S rRNA (1504-MER), 23S ribosomal RNA, 30S ribosomal protein S10, ... | 著者 | Korostelev, A, Zhu, J, Asahara, H, Noller, H.F. | 登録日 | 2010-04-29 | 公開日 | 2014-07-09 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (3.62 Å) | 主引用文献 | Recognition of the amber UAG stop codon by release factor RF1. Embo J., 29, 2010
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4V88
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![BU of 4v88 by Molmil](/molmil-images/mine/4v88) | The structure of the eukaryotic ribosome at 3.0 A resolution. | 分子名称: | 18S RIBOSOMAL RNA, 18S rRNA, 25S rRNA, ... | 著者 | Ben-Shem, A, Garreau de Loubresse, N, Melnikov, S, Jenner, L, Yusupova, G, Yusupov, M. | 登録日 | 2011-10-11 | 公開日 | 2014-07-09 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | The structure of the eukaryotic ribosome at 3.0 angstrom resolution. Science, 334, 2011
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4W5C
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![BU of 4w5c by Molmil](/molmil-images/mine/4w5c) | Crystal structure analysis of cruzain with three Fragments: 1 (N-(1H-benzimidazol-2-yl)-1,3-dimethyl-pyrazole-4-carboxamide), 6 (2-amino-4,6-difluorobenzothiazole) and 9 (N-(1H-benzimidazol-2-yl)-3-(4-fluorophenyl)-1H-pyrazole-4-carboxamide). | 分子名称: | 4,6-difluoro-1,3-benzothiazol-2-amine, Cruzipain, N-(1H-benzimidazol-2-yl)-1,3-dimethyl-1H-pyrazole-4-carboxamide, ... | 著者 | Tochowicz, A, McKerrow, J.H, Craik, C.S. | 登録日 | 2014-08-17 | 公開日 | 2015-04-08 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (3.27 Å) | 主引用文献 | Applying Fragments Based- Drug Design to identify multiple binding modes on cysteine protease. To Be Published
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4V0I
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![BU of 4v0i by Molmil](/molmil-images/mine/4v0i) | Water Network Determines Selectivity for a Series of Pyrimidone Indoline Amide PI3KBeta Inhibitors over PI3K-Delta | 分子名称: | 2-[2-(2-METHYL-2,3-DIHYDRO-INDOL-1-YL)-2-OXO-ETHYL]-6-MORPHOLIN-4-YL-3H-PYRIMIDIN-4-ONE, PHOSPHATIDYLINOSITOL-4,5-BISPHOSPHATE 3-KINASE CATALYTIC SUBUNIT DELTA ISOFORM | 著者 | Robinson, D, Bertrand, T, Carry, J.C, Halley, F, Karlsson, A, Mathieu, M, Minoux, H, Perrin, M.A, Robert, B, Schio, L, Sherman, W. | 登録日 | 2014-09-16 | 公開日 | 2015-09-30 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.54 Å) | 主引用文献 | Differential Water Thermodynamics Determine Pi3K-Beta/Delta Selectivity for Solvent-Exposed Ligand Modifications. J.Chem.Inf.Model., 56, 2016
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4V4J
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![BU of 4v4j by Molmil](/molmil-images/mine/4v4j) | Interactions and Dynamics of the Shine-Dalgarno Helix in the 70S Ribosome. | 分子名称: | 16S RNA, 23S LARGE SUBUNIT RIBOSOMAL RNA, 30S ribosomal protein S10, ... | 著者 | Korostelev, A, Trakhanov, S, Asahara, H, Laurberg, M, Noller, H.F. | 登録日 | 2007-07-18 | 公開日 | 2014-07-09 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (3.83 Å) | 主引用文献 | Interactions and dynamics of the Shine Dalgarno helix in the 70S ribosome. Proc.Natl.Acad.Sci.Usa, 104, 2007
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4V5D
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![BU of 4v5d by Molmil](/molmil-images/mine/4v5d) | Structure of the Thermus thermophilus 70S ribosome in complex with mRNA, paromomycin, acylated A- and P-site tRNAs, and E-site tRNA. | 分子名称: | 16S ribosomal RNA, 23S RIBOSOMAL RNA, 30S RIBOSOMAL PROTEIN S10, ... | 著者 | Voorhees, R.M, Weixlbaumer, A, Loakes, D, Kelley, A.C, Ramakrishnan, V. | 登録日 | 2009-03-24 | 公開日 | 2014-07-09 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (3.5 Å) | 主引用文献 | Insights into substrate stabilization from snapshots of the peptidyl transferase center of the intact 70S ribosome. Nat. Struct. Mol. Biol., 16, 2009
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4V5T
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![BU of 4v5t by Molmil](/molmil-images/mine/4v5t) | X-ray structure of the Grapevine Fanleaf virus | 分子名称: | COAT PROTEIN | 著者 | Schellenberger, P, Sauter, C, Lorber, B, Bron, P, Trapani, S, Bergdoll, M, Marmonier, A, Schmitt-Keichinger, C, Lemaire, O, Demangeat, G, Ritzenthaler, C. | 登録日 | 2011-02-01 | 公開日 | 2014-07-09 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Structural Insights Into Viral Determinants of Nematode Mediated Grapevine Fanleaf Virus Transmission. Plos Pathog., 7, 2011
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