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3VPT
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BU of 3vpt by Molmil
Crystal structure of Bombyx mori sigma-class glutathione transferase in apo form
分子名称: DI(HYDROXYETHYL)ETHER, Glutathione S-transferase sigma, S-1,2-PROPANEDIOL, ...
著者Yamamoto, K, Higashiura, A, Suzuki, M, Nakagawa, A.
登録日2012-03-13
公開日2013-03-06
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystal structure of a Bombyx mori sigma-class glutathione transferase exhibiting prostaglandin E synthase activity
Biochim.Biophys.Acta, 1830, 2013
3WA3
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BU of 3wa3 by Molmil
Crystal structure of copper amine oxidase from arthrobacter globiformis in N2 condition
分子名称: 1,2-ETHANEDIOL, COPPER (II) ION, DI(HYDROXYETHYL)ETHER, ...
著者Murakawa, T, Hayashi, H, Sunami, T, Kurihara, K, Tamada, T, Kuroki, R, Suzuki, M, Tanizawa, K, Okajima, T.
登録日2013-04-22
公開日2013-09-11
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献High-resolution crystal structure of copper amine oxidase from Arthrobacter globiformis: assignment of bound diatomic molecules as O2
Acta Crystallogr.,Sect.D, 69, 2013
3WA2
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BU of 3wa2 by Molmil
High resolution crystal structure of copper amine oxidase from arthrobacter globiformis
分子名称: 1,2-ETHANEDIOL, COPPER (II) ION, DI(HYDROXYETHYL)ETHER, ...
著者Murakawa, T, Hayashi, H, Sunami, T, Kurihara, K, Tamada, T, Kuroki, R, Suzuki, M, Tanizawa, K, Okajima, T.
登録日2013-04-22
公開日2013-09-11
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.08 Å)
主引用文献High-resolution crystal structure of copper amine oxidase from Arthrobacter globiformis: assignment of bound diatomic molecules as O2
Acta Crystallogr.,Sect.D, 69, 2013
3WD6
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BU of 3wd6 by Molmil
Crystal structure of Bombyx mori omega-class glutathione transferase in complex with GSH
分子名称: 1,2-ETHANEDIOL, DI(HYDROXYETHYL)ETHER, GLUTATHIONE, ...
著者Yamamoto, K, Suzuki, M, Higashiura, A, Nakagawa, A.
登録日2013-06-07
公開日2014-07-16
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Three-dimensional structure of a Bombyx mori Omega-class glutathione transferase.
Biochem.Biophys.Res.Commun., 438, 2013
2ZPM
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BU of 2zpm by Molmil
Crystal structure analysis of PDZ domain B
分子名称: Regulator of sigma E protease
著者Inaba, K, Suzuki, M.
登録日2008-07-17
公開日2008-10-21
最終更新日2017-10-11
実験手法X-RAY DIFFRACTION (0.98 Å)
主引用文献Crystal Structure analysis of PDZ-domain B
To be Published
3AHR
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BU of 3ahr by Molmil
Inactive human Ero1
分子名称: ERO1-like protein alpha, FLAVIN-ADENINE DINUCLEOTIDE
著者Inaba, K, Sitia, R, Suzuki, M.
登録日2010-04-26
公開日2010-12-22
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (3.07 Å)
主引用文献Crystal structures of human Ero1-alpha reveal the mechanisms of regulated and targeted oxidation of PDI
Embo J., 29, 2010
3WHO
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BU of 3who by Molmil
X-ray-Crystallographic Structure of an RNase Po1 Exhibiting Anti-tumor Activity
分子名称: Guanyl-specific ribonuclease Po1
著者Kobayashi, H, Katsurtani, T, Hara, Y, Motoyoshi, N, Itagaki, T, Akita, F, Higashiura, A, Yamada, Y, Suzuki, M, Inokuchi, N.
登録日2013-08-30
公開日2014-07-02
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献X-ray crystallographic structure of RNase Po1 that exhibits anti-tumor activity.
Biol.Pharm.Bull., 37, 2014
3ALP
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BU of 3alp by Molmil
Cell adhesion protein
分子名称: CITRIC ACID, HEXANE-1,6-DIOL, Poliovirus receptor-related protein 1
著者Narita, H, Nakagawa, A, Suzuki, M.
登録日2010-08-05
公開日2011-02-16
最終更新日2017-10-11
実験手法X-RAY DIFFRACTION (2.804 Å)
主引用文献Crystal Structure of the cis-Dimer of Nectin-1: implications for the architecture of cell-cell junctions
J.Biol.Chem., 286, 2011
2ZPL
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BU of 2zpl by Molmil
Crystal structure analysis of PDZ domain A
分子名称: GLYCEROL, NICKEL (II) ION, Regulator of sigma E protease
著者Inaba, K, Suzuki, M.
登録日2008-07-17
公開日2008-10-21
最終更新日2021-11-10
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Crystal structure analysis of PDZ-domain A
To be Published
3AHQ
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BU of 3ahq by Molmil
hyperactive human Ero1
分子名称: ERO1-like protein alpha, FLAVIN-ADENINE DINUCLEOTIDE
著者Inaba, K, Sitia, R, Suzuki, M.
登録日2010-04-26
公開日2010-12-22
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Crystal structures of human Ero1-alpha reveal the mechanisms of regulated and targeted oxidation of PDI
Embo J., 29, 2010
8H7X
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BU of 8h7x by Molmil
Crystal structure of EGFR T790M/C797S mutant in complex with brigatinib
分子名称: 5-chloro-N~4~-[2-(dimethylphosphoryl)phenyl]-N~2~-{2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl}pyrimidine-2,4-diamine, Epidermal growth factor receptor
著者Kukimoto-Niino, M, Shirouzu, M.
登録日2022-10-21
公開日2023-10-25
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (3.404 Å)
主引用文献A macrocyclic kinase inhibitor overcomes triple resistant mutations in EGFR-positive lung cancer.
NPJ Precis Oncol, 8, 2024
2EI6
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BU of 2ei6 by Molmil
FACTOR XA IN COMPLEX WITH THE INHIBITOR (-)-cis-N1-[(5-Chloroindol-2-yl)carbonyl]-N2-[(5-methyl-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridin-2-yl)carbonyl]-1,2-cyclohexanediamine
分子名称: CALCIUM ION, Coagulation factor X, heavy chain, ...
著者Suzuki, M.
登録日2007-03-12
公開日2008-03-18
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Cycloalkanediamine derivatives as novel blood coagulation factor Xa inhibitors.
Bioorg.Med.Chem.Lett., 17, 2007
2EI7
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BU of 2ei7 by Molmil
FACTOR XA IN COMPLEX WITH THE INHIBITOR trans-N1-[(5-Chloroindol-2-yl)carbonyl]-N2-[(5-methyl-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridin-2-yl)carbonyl]-1,2-cyclohexanediamine
分子名称: CALCIUM ION, Coagulation factor X, heavy chain, ...
著者Suzuki, M.
登録日2007-03-12
公開日2008-03-18
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Cycloalkanediamine derivatives as novel blood coagulation factor Xa inhibitors
To be Published
6LKM
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BU of 6lkm by Molmil
Crystal structure of Ribonucleotide reductase R1 subunit, RRM1 in complex with 5-chloro-N-((1S,2R)-2-(6-fluoro-2,3-dimethylphenyl)-1-(5-oxo-4,5-dihydro-1,3,4-oxadiazol-2-yl)propyl)-4-methyl-3,4-dihydro-2H-benzo[b][1,4]oxazine-8-sulfonamide
分子名称: 5-chloro-N-((1S,2R)-2-(6-fluoro-2,3-dimethylphenyl)-1-(5-oxo-4,5-dihydro-1,3,4-oxadiazol-2-yl)propyl)-4-methyl-3,4-dihydro-2H-benzo[b][1,4]oxazine-8-sulfonamide, MAGNESIUM ION, Ribonucleoside-diphosphate reductase large subunit, ...
著者Miyahara, S, Chong, K.T, Suzuki, T.
登録日2019-12-19
公開日2020-12-23
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.55 Å)
主引用文献TAS1553, a novel small molecule ribonucleotide reductase (RNR) subunit interaction inhibitor, displays remarkable anti-tumor activity
To be published
7YNH
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BU of 7ynh by Molmil
Catalytic intermediate of copper amine oxidase determined by serial femtosecond X-ray crystallography using a single-flow liquid jet system
分子名称: COPPER (II) ION, PHENYLACETALDEHYDE, Phenylethylamine oxidase, ...
著者Murakawa, T, Okajima, T.
登録日2022-07-31
公開日2022-11-16
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.94 Å)
主引用文献Serial femtosecond X-ray crystallography of an anaerobically formed catalytic intermediate of copper amine oxidase.
Acta Crystallogr D Struct Biol, 78, 2022
1MR8
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BU of 1mr8 by Molmil
MIGRATION INHIBITORY FACTOR-RELATED PROTEIN 8 FROM HUMAN
分子名称: CALCIUM ION, MIGRATION INHIBITORY FACTOR-RELATED PROTEIN 8
著者Ishikawa, K, Nakagawa, A, Tanaka, I, Nishihira, J.
登録日1999-04-13
公開日2000-05-17
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献The structure of human MRP8, a member of the S100 calcium-binding protein family, by MAD phasing at 1.9 A resolution.
Acta Crystallogr.,Sect.D, 56, 2000
1DPT
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BU of 1dpt by Molmil
D-DOPACHROME TAUTOMERASE
分子名称: D-DOPACHROME TAUTOMERASE
著者Sugimoto, H, Taniguchi, M, Nakagawa, A, Tanaka, I.
登録日1998-05-11
公開日1999-03-30
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.54 Å)
主引用文献Crystal structure of human D-dopachrome tautomerase, a homologue of macrophage migration inhibitory factor, at 1.54 A resolution.
Biochemistry, 38, 1999
7YRU
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BU of 7yru by Molmil
ALK2 antibody complex
分子名称: Activin receptor type-1, antibody heavy chain, antibody light chain
著者Kawaguchi, Y, Nakamura, K, Suzuki, M, Tsuji, S, Katagiri, T.
登録日2022-08-10
公開日2023-05-17
最終更新日2023-06-07
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献A blocking monoclonal antibody reveals dimerization of intracellular domains of ALK2 associated with genetic disorders.
Nat Commun, 14, 2023
7F3O
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BU of 7f3o by Molmil
Crystal structure of the GluA2o LBD in complex with glutamate and TAK-653
分子名称: 7-(4-cyclohexyloxyphenyl)-9-methyl-4$l^{6}-thia-1$l^{4},5,8-triazabicyclo[4.4.0]deca-1(10),6,8-triene 4,4-dioxide, ACETATE ION, GLUTAMIC ACID, ...
著者Sogabe, S, Igaki, S, Hirokawa, A, Zama, Y, Lane, W, Snell, G.
登録日2021-06-16
公開日2021-07-28
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.44 Å)
主引用文献Strictly regulated agonist-dependent activation of AMPA-R is the key characteristic of TAK-653 for robust synaptic responses and cognitive improvement.
Sci Rep, 11, 2021
6L4A
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BU of 6l4a by Molmil
H3-H3-H3 tri-nucleosome with the 22 base-pair linker DNA
分子名称: DNA (485-MER), Histone H2A type 1-B/E, Histone H2B type 1-J, ...
著者Takizawa, Y, Ho, C.-H, Tachiwana, H, Matsunami, H, Ohi, M, Wolf, M, Kurumizaka, H.
登録日2019-10-16
公開日2019-12-04
最終更新日2024-03-27
実験手法ELECTRON MICROSCOPY (12.3 Å)
主引用文献Cryo-EM Structures of Centromeric Tri-nucleosomes Containing a Central CENP-A Nucleosome.
Structure, 28, 2020
8AJZ
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BU of 8ajz by Molmil
Serial femtosecond crystallography structure of CO bound ba3- type cytochrome c oxidase at 2 milliseconds after irradiation by a 532 nm laser
分子名称: (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, CARBON MONOXIDE, COPPER (II) ION, ...
著者Safari, C, Ghosh, S, Andersson, R, Johannesson, J, Donoso, A.V, Bath, P, Bosman, R, Dahl, P, Nango, E, Tanaka, R, Zoric, D, Svensson, E, Nakane, T, Iwata, S, Neutze, R, Branden, G.
登録日2022-07-29
公開日2023-08-16
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Time-resolved serial crystallography to track the dynamics of carbon monoxide in the active site of cytochrome c oxidase.
Sci Adv, 9, 2023
4REN
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BU of 4ren by Molmil
Crystal structure of UDP-glucose: anthocyanidin 3-O-glucosyltransferase in complex with petunidin
分子名称: 2-(3,4-dihydroxy-5-methoxyphenyl)-3,5,7-trihydroxychromenium, GLYCEROL, UDP-glucose:anthocyanidin 3-O-glucosyltransferase
著者Hiromoto, T, Honjo, E, Tamada, T, Kuroki, R.
登録日2014-09-23
公開日2015-01-21
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.704 Å)
主引用文献Structural basis for acceptor-substrate recognition of UDP-glucose: anthocyanidin 3-O-glucosyltransferase from Clitoria ternatea
Protein Sci., 24, 2015
4REM
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BU of 4rem by Molmil
Crystal structure of UDP-glucose: anthocyanidin 3-O-glucosyltransferase in complex with delphinidin
分子名称: 3,5,7-trihydroxy-2-(3,4,5-trihydroxyphenyl)chromenium, GLYCEROL, UDP-glucose:anthocyanidin 3-O-glucosyltransferase
著者Hiromoto, T, Honjo, E, Tamada, T, Kuroki, R.
登録日2014-09-23
公開日2015-01-21
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.55 Å)
主引用文献Structural basis for acceptor-substrate recognition of UDP-glucose: anthocyanidin 3-O-glucosyltransferase from Clitoria ternatea
Protein Sci., 24, 2015
4REL
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BU of 4rel by Molmil
Crystal structure of UDP-glucose: anthocyanidin 3-O-glucosyltransferase in complex with kaempferol
分子名称: 3,5,7-TRIHYDROXY-2-(4-HYDROXYPHENYL)-4H-CHROMEN-4-ONE, ACETATE ION, GLYCEROL, ...
著者Hiromoto, T, Honjo, E, Tamada, T, Kuroki, R.
登録日2014-09-23
公開日2015-01-21
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.754 Å)
主引用文献Structural basis for acceptor-substrate recognition of UDP-glucose: anthocyanidin 3-O-glucosyltransferase from Clitoria ternatea
Protein Sci., 24, 2015
5JOO
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BU of 5joo by Molmil
XFEL structure of influenza A M2 wild type TM domain at low pH in the lipidic cubic phase at room temperature
分子名称: CALCIUM ION, CHLORIDE ION, Matrix protein 2
著者Thomaston, J.L, Woldeyes, R.A, Fraser, J.S, DeGrado, W.F.
登録日2016-05-02
公開日2017-08-02
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.413 Å)
主引用文献XFEL structures of the influenza M2 proton channel: Room temperature water networks and insights into proton conduction.
Proc. Natl. Acad. Sci. U.S.A., 114, 2017

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