5WI1
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5X5Y
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![BU of 5x5y by Molmil](/molmil-images/mine/5x5y) | A membrane protein complex | 分子名称: | Probable ATP-binding component of ABC transporter, Uncharacterized protein | 著者 | Luo, Q, Yang, X, Huang, Y. | 登録日 | 2017-02-18 | 公開日 | 2017-04-05 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (3.465 Å) | 主引用文献 | Structural basis for lipopolysaccharide extraction by ABC transporter LptB2FG Nat. Struct. Mol. Biol., 24, 2017
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2FIE
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2FIX
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2H96
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![BU of 2h96 by Molmil](/molmil-images/mine/2h96) | Discovery of Potent, Highly Selective, and Orally Bioavailable Pyridine Carboxamide C-jun NH2-terminal Kinase Inhibitors | 分子名称: | 5-CYANO-N-(2,5-DIMETHOXYBENZYL)-6-ETHOXYPYRIDINE-2-CARBOXAMIDE, C-jun-amino-terminal kinase-interacting protein 1, GLYCEROL, ... | 著者 | Abad-Zapatero, C. | 登録日 | 2006-06-09 | 公開日 | 2006-07-25 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Discovery of potent, highly selective, and orally bioavailable pyridine carboxamide c-Jun NH2-terminal kinase inhibitors. J.Med.Chem., 49, 2006
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3P9U
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![BU of 3p9u by Molmil](/molmil-images/mine/3p9u) | Crystal structure of TetX2 from Bacteroides thetaiotaomicron with substrate analogue | 分子名称: | FLAVIN-ADENINE DINUCLEOTIDE, SULFATE ION, TetX2 protein | 著者 | Walkiewicz, K, Davlieva, M, Sun, C, Lau, K, Shamoo, Y. | 登録日 | 2010-10-18 | 公開日 | 2011-04-27 | 最終更新日 | 2017-11-08 | 実験手法 | X-RAY DIFFRACTION (2.81 Å) | 主引用文献 | Crystal structure of Bacteroides thetaiotaomicron TetX2: a tetracycline degrading monooxygenase at 2.8 A resolution. Proteins, 79, 2011
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7EJV
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![BU of 7ejv by Molmil](/molmil-images/mine/7ejv) | The co-crystal structure of DYRK2 with YK-2-69 | 分子名称: | Dual specificity tyrosine-phosphorylation-regulated kinase 2, [6-[[4-[2-(dimethylamino)-1,3-benzothiazol-6-yl]-5-fluoranyl-pyrimidin-2-yl]amino]pyridin-3-yl]-(4-ethylpiperazin-1-yl)methanone | 著者 | Li, Z, Xiao, Y, Yuan, K, Kuang, W, Xiuquan, Y, Yang, P. | 登録日 | 2021-04-02 | 公開日 | 2022-04-06 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Targeting dual-specificity tyrosine phosphorylation-regulated kinase 2 with a highly selective inhibitor for the treatment of prostate cancer. Nat Commun, 13, 2022
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2JHB
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3WXT
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3WXU
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4W4Q
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![BU of 4w4q by Molmil](/molmil-images/mine/4w4q) | Glucose isomerase structure determined by serial femtosecond crystallography at SACLA | 分子名称: | CALCIUM ION, Xylose isomerase | 著者 | Nango, E, Tanaka, T, Sugahara, M, Suzuki, M, Iwata, S. | 登録日 | 2014-08-15 | 公開日 | 2014-11-05 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Grease matrix as a versatile carrier of proteins for serial crystallography Nat.Methods, 12, 2015
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4KTD
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![BU of 4ktd by Molmil](/molmil-images/mine/4ktd) | Fab fragment of HIV vaccine-elicited CD4bs-directed antibody, GE136, from non-human primate | 分子名称: | GE136 Heavy Chain Fab, GE136 Light Chain Fab, GLYCEROL, ... | 著者 | Poulsen, C, Tran, K, Standfield, R, Wyatt, R.T. | 登録日 | 2013-05-20 | 公開日 | 2014-02-05 | 最終更新日 | 2017-11-15 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Vaccine-elicited primate antibodies use a distinct approach to the HIV-1 primary receptor binding site informing vaccine redesign. Proc.Natl.Acad.Sci.USA, 111, 2014
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4KTE
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![BU of 4kte by Molmil](/molmil-images/mine/4kte) | Fab fragment of HIV vaccine-elicited CD4bs-directed antibody, GE148, from non-human primate | 分子名称: | GE148 Heavy Chain Fab, GE148 Light Chain Fab, GLYCEROL, ... | 著者 | Poulsen, C, Tran, K, Stanfield, R, Wyatt, R.T. | 登録日 | 2013-05-20 | 公開日 | 2014-02-05 | 最終更新日 | 2019-12-25 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Vaccine-elicited primate antibodies use a distinct approach to the HIV-1 primary receptor binding site informing vaccine redesign. Proc.Natl.Acad.Sci.USA, 111, 2014
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6U9U
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![BU of 6u9u by Molmil](/molmil-images/mine/6u9u) | Structure of GM9_TH8seq732127 FAB | 分子名称: | 1,2-ETHANEDIOL, FORMIC ACID, GM9_TH8seq732127 FAB heavy chain, ... | 著者 | Singh, S, Liban, T.J, Pancera, M. | 登録日 | 2019-09-09 | 公開日 | 2019-11-06 | 最終更新日 | 2019-12-25 | 実験手法 | X-RAY DIFFRACTION (2.26 Å) | 主引用文献 | Extensive dissemination and intraclonal maturation of HIV Env vaccine-induced B cell responses. J.Exp.Med., 217, 2020
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6U3Z
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![BU of 6u3z by Molmil](/molmil-images/mine/6u3z) | Structure of VD20_5A4 Fab | 分子名称: | ACETATE ION, CHLORIDE ION, GLYCEROL, ... | 著者 | Dionne, G, Shapiro, L. | 登録日 | 2019-08-22 | 公開日 | 2019-11-20 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.99002314 Å) | 主引用文献 | Extensive dissemination and intraclonal maturation of HIV Env vaccine-induced B cell responses. J.Exp.Med., 217, 2020
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8GNG
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![BU of 8gng by Molmil](/molmil-images/mine/8gng) | Crystal structure of human adenosine A2A receptor in complex with istradefylline. | 分子名称: | (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, 8-[(~{E})-2-(3,4-dimethoxyphenyl)ethenyl]-1,3-diethyl-7-methyl-purine-2,6-dione, Adenosine receptor A2a, ... | 著者 | Suzuki, M, Saito, J, Miyagi, H, Yasunaga, M. | 登録日 | 2022-08-23 | 公開日 | 2023-03-22 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | In Vitro Pharmacological Profile of KW-6356, a Novel Adenosine A 2A Receptor Antagonist/Inverse Agonist. Mol.Pharmacol., 103, 2023
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8GNE
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![BU of 8gne by Molmil](/molmil-images/mine/8gne) | Crystal structure of human adenosine A2A receptor in complex with an insurmountable inverse agonist, KW-6356. | 分子名称: | (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, 2-{2-[2-(2-{2-[2-(2-ETHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHOXY]-ETHOXY}-ETHANOL, Adenosine receptor A2a,Soluble cytochrome b562, ... | 著者 | Suzuki, M, Saito, J, Miyagi, H, Yasunaga, M. | 登録日 | 2022-08-23 | 公開日 | 2023-03-22 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | In Vitro Pharmacological Profile of KW-6356, a Novel Adenosine A 2A Receptor Antagonist/Inverse Agonist. Mol.Pharmacol., 103, 2023
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4YZF
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![BU of 4yzf by Molmil](/molmil-images/mine/4yzf) | Crystal structure of the anion exchanger domain of human erythrocyte Band 3 | 分子名称: | 2,2'-ethane-1,2-diylbis{5-[(sulfanylmethyl)amino]benzenesulfonic acid}, Band 3 anion transport protein, FAB fragment of Immunoglobulin (IgG) molecule | 著者 | Alguel, Y, Arakawa, T, Yugiri, T.K, Iwanari, H, Hatae, H, Iwata, M, Abe, Y, Hino, T, Suno, C.I, Kuma, H, Kang, D, Murata, T, Hamakubo, T, Cameron, A.D, Kobayashi, T, Hamasaki, N, Iwata, S. | 登録日 | 2015-03-25 | 公開日 | 2015-11-04 | 最終更新日 | 2015-11-18 | 実験手法 | X-RAY DIFFRACTION (3.5 Å) | 主引用文献 | Crystal structure of the anion exchanger domain of human erythrocyte band 3. Science, 350, 2015
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3WXQ
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![BU of 3wxq by Molmil](/molmil-images/mine/3wxq) | Serial femtosecond X-ray structure of human fatty acid-binding protein type-3 (FABP3) in complex with stearic acid (C18:0) determined using X-ray free-electron laser at SACLA | 分子名称: | Fatty acid-binding protein, heart, STEARIC ACID | 著者 | Mizohata, E, Suzuki, M, Kakinouchi, K, Sugiyama, S, Murata, M, Sugahara, M, Nango, E, Tanaka, T, Tanaka, R, Tono, K, Song, C, Hatsui, T, Joti, Y, Yabashi, M, Iwata, S. | 登録日 | 2014-08-04 | 公開日 | 2014-11-05 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Grease matrix as a versatile carrier of proteins for serial crystallography Nat. Methods, 12, 2015
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3WUM
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3WUL
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3WXS
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![BU of 3wxs by Molmil](/molmil-images/mine/3wxs) | Thaumatin structure determined by SPring-8 Angstrom Compact free electron Laser (SACLA) | 分子名称: | L(+)-TARTARIC ACID, thaumatin I | 著者 | Masuda, T, Nango, E, Sugahara, M, Mizohata, E, Tanaka, T, Tanaka, R, Suzuki, M, Mikami, B, Iwata, S. | 登録日 | 2014-08-07 | 公開日 | 2014-11-05 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Grease matrix as a versatile carrier of proteins for serial crystallography Nat. Methods, 12, 2015
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5XJM
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![BU of 5xjm by Molmil](/molmil-images/mine/5xjm) | Complex structure of angiotensin II type 2 receptor with Fab | 分子名称: | FabH, FabL, Sar1, ... | 著者 | Asada, H, Horita, S, Shimamura, T, Iwata, S. | 登録日 | 2017-05-02 | 公開日 | 2018-07-11 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | Crystal structure of the human angiotensin II type 2 receptor bound to an angiotensin II analog Nat. Struct. Mol. Biol., 25, 2018
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5XLI
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![BU of 5xli by Molmil](/molmil-images/mine/5xli) | Structure of anti-Angiotensin II type2 receptor antibody (D5711-4A03) | 分子名称: | FabH, FabL | 著者 | Asada, H, Horita, S, Iwata, S, Hirata, K. | 登録日 | 2017-05-10 | 公開日 | 2018-07-11 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.696 Å) | 主引用文献 | Crystal structure of the human angiotensin II type 2 receptor bound to an angiotensin II analog. Nat. Struct. Mol. Biol., 25, 2018
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6JOD
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![BU of 6jod by Molmil](/molmil-images/mine/6jod) | Angiotensin II type 2 receptor with ligand | 分子名称: | Angiotensin II, Heavy chain of 4A03Fab, Light chain of 4A03Fab, ... | 著者 | Asada, H, Iwata, S, Hirata, K, Shimamura, T. | 登録日 | 2019-03-20 | 公開日 | 2020-01-15 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | The Crystal Structure of Angiotensin II Type 2 Receptor with Endogenous Peptide Hormone. Structure, 28, 2020
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