3DAH
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![BU of 3dah by Molmil](/molmil-images/mine/3dah) | |
3D63
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![BU of 3d63 by Molmil](/molmil-images/mine/3d63) | |
3FTP
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![BU of 3ftp by Molmil](/molmil-images/mine/3ftp) | |
3EIZ
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![BU of 3eiz by Molmil](/molmil-images/mine/3eiz) | |
6M94
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![BU of 6m94 by Molmil](/molmil-images/mine/6m94) | Monophosphorylated pSer33 b-Catenin peptide bound to b-TrCP/Skp1 Complex | 分子名称: | Catenin beta-1, DIMETHYL SULFOXIDE, F-box/WD repeat-containing protein 1A, ... | 著者 | Simonetta, K.R, Clifton, M.C, Walter, R.L, Ranieri, G.M, Carter, J.J. | 登録日 | 2018-08-22 | 公開日 | 2019-04-03 | 最終更新日 | 2019-04-10 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Prospective discovery of small molecule enhancers of an E3 ligase-substrate interaction. Nat Commun, 10, 2019
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6M91
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![BU of 6m91 by Molmil](/molmil-images/mine/6m91) | Monophosphorylated pSer33 b-Catenin peptide, b-TrCP/Skp1, NRX-103094 ternary complex | 分子名称: | 3-({4-[(2,6-dichlorophenyl)sulfanyl]-2-oxo-6-(trifluoromethyl)-1,2-dihydropyridine-3-carbonyl}amino)benzoic acid, CHLORIDE ION, Catenin beta-1, ... | 著者 | Simonetta, K.R, Clifton, M.C, Walter, R.L, Ranieri, G.M, Carter, J.J. | 登録日 | 2018-08-22 | 公開日 | 2019-04-03 | 最終更新日 | 2019-04-10 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Prospective discovery of small molecule enhancers of an E3 ligase-substrate interaction. Nat Commun, 10, 2019
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6M93
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![BU of 6m93 by Molmil](/molmil-images/mine/6m93) | Monophosphorylated pSer33 b-Catenin peptide, b-TrCP/Skp1, NRX-1933 ternary complex | 分子名称: | 2-oxo-N-[3-(1H-tetrazol-5-yl)phenyl]-6-(trifluoromethyl)-1,2-dihydropyridine-3-carboxamide, Catenin beta-1, F-box/WD repeat-containing protein 1A, ... | 著者 | Simonetta, K.R, Clifton, M.C, Walter, R.L, Ranieri, G.M, Lee, S.J. | 登録日 | 2018-08-22 | 公開日 | 2019-04-03 | 最終更新日 | 2019-04-10 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Prospective discovery of small molecule enhancers of an E3 ligase-substrate interaction. Nat Commun, 10, 2019
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6M92
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![BU of 6m92 by Molmil](/molmil-images/mine/6m92) | Monophosphorylated pSer33 b-Catenin peptide, b-TrCP/Skp1, NRX-2663 ternary complex | 分子名称: | 3-{[2-oxo-4-phenoxy-6-(trifluoromethyl)-1,2-dihydropyridine-3-carbonyl]amino}benzoic acid, Catenin beta-1, F-box/WD repeat-containing protein 1A, ... | 著者 | Simonetta, K.R, Clifton, M.C, Walter, R.L, Ranieri, G.M, Carter, J.J, Lee, S.J. | 登録日 | 2018-08-22 | 公開日 | 2019-04-03 | 最終更新日 | 2020-01-15 | 実験手法 | X-RAY DIFFRACTION (2.35 Å) | 主引用文献 | Prospective discovery of small molecule enhancers of an E3 ligase-substrate interaction. Nat Commun, 10, 2019
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6M90
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![BU of 6m90 by Molmil](/molmil-images/mine/6m90) | Monophosphorylated pSer33 b-Catenin peptide, b-TrCP/Skp1, NRX-2776 ternary complex | 分子名称: | 2-(2-fluorophenoxy)-3-{[2-oxo-6-(trifluoromethyl)-1,2-dihydropyridine-3-carbonyl]amino}benzoic acid, Catenin beta-1, F-box/WD repeat-containing protein 1A, ... | 著者 | Simonetta, K.R, Clifton, M.C, Walter, R.L, Ranieri, G.M, Carter, J.J. | 登録日 | 2018-08-22 | 公開日 | 2019-04-03 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | Prospective discovery of small molecule enhancers of an E3 ligase-substrate interaction. Nat Commun, 10, 2019
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3GVF
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![BU of 3gvf by Molmil](/molmil-images/mine/3gvf) | |
3GK3
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![BU of 3gk3 by Molmil](/molmil-images/mine/3gk3) | |
3GVG
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![BU of 3gvg by Molmil](/molmil-images/mine/3gvg) | |
3GWC
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![BU of 3gwc by Molmil](/molmil-images/mine/3gwc) | |
3H81
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![BU of 3h81 by Molmil](/molmil-images/mine/3h81) | |
3GWA
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![BU of 3gwa by Molmil](/molmil-images/mine/3gwa) | |
3HE2
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![BU of 3he2 by Molmil](/molmil-images/mine/3he2) | |
3ICO
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![BU of 3ico by Molmil](/molmil-images/mine/3ico) | |
3IML
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![BU of 3iml by Molmil](/molmil-images/mine/3iml) | |
3HZG
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![BU of 3hzg by Molmil](/molmil-images/mine/3hzg) | Crystal structure of mycobacterium tuberculosis thymidylate synthase X bound with FAD | 分子名称: | FLAVIN-ADENINE DINUCLEOTIDE, GLYCEROL, PHOSPHATE ION, ... | 著者 | Staker, B.L, Rathod, P, Hunter, J, Seattle Structural Genomics Center for Infectious Disease (SSGCID) | 登録日 | 2009-06-23 | 公開日 | 2009-07-07 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.45 Å) | 主引用文献 | Increasing the structural coverage of tuberculosis drug targets. Tuberculosis (Edinb), 95, 2015
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3HWI
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![BU of 3hwi by Molmil](/molmil-images/mine/3hwi) | |
3HWK
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![BU of 3hwk by Molmil](/molmil-images/mine/3hwk) | |
3H7F
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![BU of 3h7f by Molmil](/molmil-images/mine/3h7f) | |
3GWE
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![BU of 3gwe by Molmil](/molmil-images/mine/3gwe) | |
3GVC
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![BU of 3gvc by Molmil](/molmil-images/mine/3gvc) | |
3GK0
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![BU of 3gk0 by Molmil](/molmil-images/mine/3gk0) | |