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1JKA
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HUMAN LYSOZYME MUTANT WITH GLU 35 REPLACED BY ASP
分子名称: LYSOZYME, NITRATE ION
著者Muraki, M, Harata, K, Goda, S, Nagahora, H.
登録日1996-11-13
公開日1997-05-15
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.66 Å)
主引用文献Importance of van der Waals contact between Glu 35 and Trp 109 to the catalytic action of human lysozyme.
Protein Sci., 6, 1997
133L
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BU of 133l by Molmil
ROLE OF ARG 115 IN THE CATALYTIC ACTION OF HUMAN LYSOZYME. X-RAY STRUCTURE OF HIS 115 AND GLU 115 MUTANTS
分子名称: HUMAN LYSOZYME
著者Harata, K, Muraki, M, Jigami, Y.
登録日1993-06-01
公開日1993-10-31
最終更新日2017-11-29
実験手法X-RAY DIFFRACTION (1.77 Å)
主引用文献Role of Arg115 in the catalytic action of human lysozyme. X-ray structure of His115 and Glu115 mutants.
J.Mol.Biol., 233, 1993
134L
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BU of 134l by Molmil
ROLE OF ARG 115 IN THE CATALYTIC ACTION OF HUMAN LYSOZYME. X-RAY STRUCTURE OF HIS 115 AND GLU 115 MUTANTS
分子名称: HUMAN LYSOZYME
著者Harata, K, Muraki, M, Jigami, Y.
登録日1993-06-01
公開日1993-10-31
最終更新日2017-11-29
実験手法X-RAY DIFFRACTION (1.77 Å)
主引用文献Role of Arg115 in the catalytic action of human lysozyme. X-ray structure of His115 and Glu115 mutants.
J.Mol.Biol., 233, 1993
1JKC
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BU of 1jkc by Molmil
HUMAN LYSOZYME MUTANT WITH TRP 109 REPLACED BY PHE
分子名称: LYSOZYME, NITRATE ION
著者Muraki, M, Harata, K, Goda, S, Nagahora, H.
登録日1996-11-13
公開日1997-05-15
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Importance of van der Waals contact between Glu 35 and Trp 109 to the catalytic action of human lysozyme.
Protein Sci., 6, 1997
1JKB
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BU of 1jkb by Molmil
HUMAN LYSOZYME MUTANT WITH GLU 35 REPLACED BY ALA
分子名称: LYSOZYME, NITRATE ION
著者Muraki, M, Harata, K, Goda, S, Nagahora, H.
登録日1996-11-13
公開日1997-05-15
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.66 Å)
主引用文献Importance of van der Waals contact between Glu 35 and Trp 109 to the catalytic action of human lysozyme.
Protein Sci., 6, 1997
8I60
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BU of 8i60 by Molmil
Crystal structure of GAS41 YEATS domain in complex with histone H3K27cr
分子名称: ALA-ARG-KCR-SER-ALA-PRO, GLYCEROL, SULFATE ION, ...
著者Konuma, T, Zhou, M.-M.
登録日2023-01-26
公開日2023-07-26
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Histone H3 lysine 27 crotonylation mediates gene transcriptional repression in chromatin.
Mol.Cell, 83, 2023
6PGM
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BU of 6pgm by Molmil
PirF geranyltransferase
分子名称: PirF Geranyltransferase
著者Nair, S.K, Hao, Y, Estrada, P.
登録日2019-06-24
公開日2019-07-03
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献A Single Amino Acid Switch Alters the Isoprene Donor Specificity in Ribosomally Synthesized and Post-Translationally Modified Peptide Prenyltransferases.
J.Am.Chem.Soc., 140, 2018
8HHV
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BU of 8hhv by Molmil
endo-alpha-D-arabinanase EndoMA1 from Microbacterium arabinogalactanolyticum
分子名称: CALCIUM ION, GLYCEROL, SODIUM ION, ...
著者Nakashima, C, Li, J, Arakawa, T, Yamada, C, Ishiwata, A, Fujita, K, Fushinobu, S.
登録日2022-11-17
公開日2023-08-16
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Identification and characterization of endo-alpha-, exo-alpha-, and exo-beta-D-arabinofuranosidases degrading lipoarabinomannan and arabinogalactan of mycobacteria.
Nat Commun, 14, 2023
7VPC
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BU of 7vpc by Molmil
Neryl diphosphate synthase from Solanum lycopersicum
分子名称: 1,2-ETHANEDIOL, D-MALATE, Neryl-diphosphate synthase 1
著者Imaizumi, R, Misawa, S, Takeshita, K, Sakai, N, Yamamoto, M, Kataoka, K, Nakayama, T, Takahashi, S, Yamashita, S.
登録日2021-10-15
公開日2022-05-18
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.94 Å)
主引用文献Structure-based engineering of a short-chain cis-prenyltransferase to biosynthesize nonnatural all-cis-polyisoprenoids: molecular mechanisms for primer substrate recognition and ultimate product chain-length determination.
Febs J., 289, 2022
6KDX
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BU of 6kdx by Molmil
Crystal structure of PDE10A in complex with a triazolopyrimidine inhibitor
分子名称: MAGNESIUM ION, N-[2-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)ethyl]quinolin-2-amine, ZINC ION, ...
著者Amano, Y, Honbou, K.
登録日2019-07-03
公開日2019-08-14
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.44 Å)
主引用文献Synthesis, SAR study, and biological evaluation of novel 2,3-dihydro-1H-imidazo[1,2-a]benzimidazole derivatives as phosphodiesterase 10A inhibitors.
Bioorg.Med.Chem., 27, 2019
6KDZ
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Crystal structure of PDE10A in complex with a triazolopyrimidine inhibitor
分子名称: 4-[2-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)ethyl]-3,7,8,10-tetrazatricyclo[7.4.0.0^{2,7}]trideca-1,3,5,8,10,12-hexaen-6-ol, MAGNESIUM ION, ZINC ION, ...
著者Amano, Y, Honbou, K.
登録日2019-07-03
公開日2019-08-14
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Synthesis, SAR study, and biological evaluation of novel 2,3-dihydro-1H-imidazo[1,2-a]benzimidazole derivatives as phosphodiesterase 10A inhibitors.
Bioorg.Med.Chem., 27, 2019
6KE0
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BU of 6ke0 by Molmil
Crystal structure of PDE10A in complex with a triazolopyrimidine inhibitor
分子名称: 2-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-1-[(2S)-2-methyl-1,2-dihydroimidazo[1,2-a]benzimidazol-3-yl]ethanone, MAGNESIUM ION, ZINC ION, ...
著者Amano, Y, Honbou, K.
登録日2019-07-03
公開日2019-08-14
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.95 Å)
主引用文献Synthesis, SAR study, and biological evaluation of novel 2,3-dihydro-1H-imidazo[1,2-a]benzimidazole derivatives as phosphodiesterase 10A inhibitors.
Bioorg.Med.Chem., 27, 2019
8E1A
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BU of 8e1a by Molmil
Structure-based study to overcome cross-reactivity of novel androgen receptor inhibitors
分子名称: 1,2-ETHANEDIOL, 4-[4-(3-fluoro-2-methoxyphenyl)-1,3-thiazol-2-yl]morpholine, Androgen receptor
著者Lallous, N, Li, H, Radaeva, M, Dalal, K, Leblanc, E, Ban, F, Ciesielski, F, Chow, B, Morin, M, Singh, K, Rennie, P.S, Cherkasov, A.
登録日2022-08-10
公開日2022-09-14
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.2 Å)
主引用文献Structure-Based Study to Overcome Cross-Reactivity of Novel Androgen Receptor Inhibitors.
Cells, 11, 2022
9FBV
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BU of 9fbv by Molmil
70S Escherichia coli ribosome with P-site initiatior tRNA.
分子名称: 16S ribosomal RNA, 23S ribosomal RNA, 30S ribosomal protein S16, ...
著者Koller, T.O, Wilson, D.N.
登録日2024-05-14
公開日2024-06-26
実験手法ELECTRON MICROSCOPY (2.4 Å)
主引用文献Paenilamicins from the honey bee pathogen Paenibacillus larvae are context-specific translocation inhibitors of protein synthesis.
Biorxiv, 2024
7OTC
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BU of 7otc by Molmil
Cryo-EM structure of an Escherichia coli 70S ribosome in complex with elongation factor G and the antibiotic Argyrin B
分子名称: 1,4-DIAMINOBUTANE, 16S ribosomal RNA, 23S ribosomal RNA, ...
著者Wieland, M, Koller, T.O, Wilson, D.N.
登録日2021-06-10
公開日2022-05-11
最終更新日2024-04-24
実験手法ELECTRON MICROSCOPY (2.9 Å)
主引用文献The cyclic octapeptide antibiotic argyrin B inhibits translation by trapping EF-G on the ribosome during translocation.
Proc.Natl.Acad.Sci.USA, 119, 2022
7EIC
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BU of 7eic by Molmil
Crystal structure of AF9 YEATS domain in complex with H4K5acK8ac peptide
分子名称: DI(HYDROXYETHYL)ETHER, GLYCEROL, Histone H4, ...
著者Kikuchi, M, Umehara, T.
登録日2021-03-30
公開日2022-04-06
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Elucidation of binding preferences of YEATS domains to site-specific acetylated nucleosome core particles.
J.Biol.Chem., 298, 2022
7EID
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BU of 7eid by Molmil
Crystal structure of AF9 YEATS domain in complex with H4K8acK12ac peptide
分子名称: GLYCEROL, Histone H4, Protein AF-9
著者Kikuchi, M, Umehara, T.
登録日2021-03-30
公開日2022-04-06
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Elucidation of binding preferences of YEATS domains to site-specific acetylated nucleosome core particles.
J.Biol.Chem., 298, 2022
7EIE
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BU of 7eie by Molmil
Crystal structure of YEATS2 YEATS domain
分子名称: GLYCEROL, YEATS domain-containing protein 2
著者Kikuchi, M, Umehara, T.
登録日2021-03-30
公開日2022-04-06
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.67 Å)
主引用文献Elucidation of binding preferences of YEATS domains to site-specific acetylated nucleosome core particles.
J.Biol.Chem., 298, 2022
7UG7
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BU of 7ug7 by Molmil
70S ribosome complex in an intermediate state of translocation bound to EF-G(GDP) stalled by Argyrin B
分子名称: 1,4-DIAMINOBUTANE, 16S rRNA, 23S rRNA, ...
著者Rundlet, E.J, Wieland, M, Holm, M, Koller, T.O, Blanchard, S.C, Wilson, D.N.
登録日2022-03-24
公開日2022-05-18
最終更新日2024-07-10
実験手法ELECTRON MICROSCOPY (2.58 Å)
主引用文献The cyclic octapeptide antibiotic argyrin B inhibits translation by trapping EF-G on the ribosome during translocation.
Proc.Natl.Acad.Sci.USA, 119, 2022
7KDT
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BU of 7kdt by Molmil
Human Tom70 in complex with SARS CoV2 Orf9b
分子名称: Mitochondrial import receptor subunit TOM70, ORF9b protein
著者QCRG Structural Biology Consortium
登録日2020-10-09
公開日2020-10-21
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (3.05 Å)
主引用文献Comparative host-coronavirus protein interaction networks reveal pan-viral disease mechanisms.
Science, 370, 2020
7EKD
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BU of 7ekd by Molmil
Crystal structure of gibberellin 3-oxidase 2 (GA3ox2) in rice
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, 2-OXOGLUTARIC ACID, Gibberellin 3-beta-dioxygenase 2, ...
著者Takehara, S, Kawai, K, Mikami, B, Ueguchi-Tanaka, M.
登録日2021-04-05
公開日2022-02-16
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.899 Å)
主引用文献Evolutionary alterations in gene expression and enzymatic activities of gibberellin 3-oxidase 1 in Oryza.
Commun Biol, 5, 2022
3GI3
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BU of 3gi3 by Molmil
Crystal structure of a N-Phenyl-N'-Naphthylurea analog in complex with p38 MAP kinase
分子名称: Mitogen-activated protein kinase 14, N-{5-tert-butyl-2-methoxy-3-[({4-[6-(morpholin-4-ylmethyl)pyridin-3-yl]naphthalen-1-yl}carbamoyl)amino]phenyl}methanesulfonamide
著者Qian, K.C.
登録日2009-03-05
公開日2009-10-20
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Discovery and characterization of the N-phenyl-N'-naphthylurea class of p38 kinase inhibitors.
Bioorg.Med.Chem.Lett., 19, 2009
3A5P
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BU of 3a5p by Molmil
Crystal structure of hemagglutinin
分子名称: Haemagglutinin I
著者Watanabe, N, Sakai, N, Nakamura, T, Nabeshima, Y, Kouno, T, Mizuguchi, M, Kawano, K.
登録日2009-08-10
公開日2010-08-11
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.82 Å)
主引用文献The Structure of Physarum polycephalum hemagglutinin I suggests a minimal carbohydrate recognition domain of legume lectin fold
J.Mol.Biol., 405, 2011
7DNF
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BU of 7dnf by Molmil
DARPin 63_B7 in complex with V3-IY (MN) crown mimetic
分子名称: DARPin 63_B7, SULFATE ION, V3-IY (MN) crown mimetic peptide
著者Wu, Y, Plueckthun, A.
登録日2020-12-09
公開日2021-12-15
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.78 Å)
主引用文献Distinct conformations of the HIV-1 V3 loop crown are targetable for broad neutralization.
Nat Commun, 12, 2021
7DNG
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BU of 7dng by Molmil
DARPin 63_B7 in complex with linear V3-crown (MN) peptide
分子名称: DARPin 63_B7, linear V3-crown (MN) peptide
著者Wu, Y, Plueckthun, A.
登録日2020-12-09
公開日2021-12-15
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.42 Å)
主引用文献Distinct conformations of the HIV-1 V3 loop crown are targetable for broad neutralization.
Nat Commun, 12, 2021

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