7Q72
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![BU of 7q72 by Molmil](/molmil-images/mine/7q72) | Structure of Pla1 in complex with Red1 | 分子名称: | NURS complex subunit red1, Poly(A) polymerase pla1 | 著者 | Soni, K, Wild, K, Sinning, I. | 登録日 | 2021-11-09 | 公開日 | 2022-12-07 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Mechanistic insights into RNA surveillance by the canonical poly(A) polymerase Pla1 of the MTREC complex. Nat Commun, 14, 2023
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7Q73
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![BU of 7q73 by Molmil](/molmil-images/mine/7q73) | Structure of Pla1 apo | 分子名称: | GLYCEROL, Poly(A) polymerase pla1 | 著者 | Soni, K, Wild, K, Sinning, I. | 登録日 | 2021-11-09 | 公開日 | 2022-12-07 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Mechanistic insights into RNA surveillance by the canonical poly(A) polymerase Pla1 of the MTREC complex. Nat Commun, 14, 2023
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7Q74
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![BU of 7q74 by Molmil](/molmil-images/mine/7q74) | |
7EA6
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![BU of 7ea6 by Molmil](/molmil-images/mine/7ea6) | Crystal structure of TCR-017 ectodomain | 分子名称: | T cell receptor 017 alpha chain, T cell receptor 017 beta chain | 著者 | Nagae, M, Yamasaki, S. | 登録日 | 2021-03-06 | 公開日 | 2021-10-13 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.18000245 Å) | 主引用文献 | Identification of conserved SARS-CoV-2 spike epitopes that expand public cTfh clonotypes in mild COVID-19 patients. J.Exp.Med., 218, 2021
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6UNQ
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![BU of 6unq by Molmil](/molmil-images/mine/6unq) | Kinase domain of ALK2-K493A with AMPPNP | 分子名称: | Activin receptor type-1, MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER | 著者 | Agnew, C, Jura, N. | 登録日 | 2019-10-13 | 公開日 | 2021-07-07 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Structural basis for ALK2/BMPR2 receptor complex signaling through kinase domain oligomerization. Nat Commun, 12, 2021
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6UNR
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![BU of 6unr by Molmil](/molmil-images/mine/6unr) | Kinase domain of ALK2-K492A/K493A with AMPPNP | 分子名称: | Activin receptor type-1, MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER | 著者 | Agnew, C, Jura, N. | 登録日 | 2019-10-13 | 公開日 | 2021-07-07 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Structural basis for ALK2/BMPR2 receptor complex signaling through kinase domain oligomerization. Nat Commun, 12, 2021
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6UNP
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![BU of 6unp by Molmil](/molmil-images/mine/6unp) | Crystal structure of the kinase domain of BMPR2-D485G | 分子名称: | 1,2-ETHANEDIOL, ADENOSINE-5'-DIPHOSPHATE, Bone morphogenetic protein receptor type-2, ... | 著者 | Agnew, C, Jura, N. | 登録日 | 2019-10-13 | 公開日 | 2021-07-07 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structural basis for ALK2/BMPR2 receptor complex signaling through kinase domain oligomerization. Nat Commun, 12, 2021
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6UNS
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![BU of 6uns by Molmil](/molmil-images/mine/6uns) | Kinase domain of ALK2-K492A/K493A with LDN-193189 | 分子名称: | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline, Activin receptor type-1 | 著者 | Agnew, C, Jura, N. | 登録日 | 2019-10-13 | 公開日 | 2021-07-07 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structural basis for ALK2/BMPR2 receptor complex signaling through kinase domain oligomerization. Nat Commun, 12, 2021
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7YOW
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7DEQ
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![BU of 7deq by Molmil](/molmil-images/mine/7deq) | Lysozyme-sugar complex in D2O | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CHLORIDE ION, Lysozyme C, ... | 著者 | Tanaka, I, Chatake, T. | 登録日 | 2020-11-04 | 公開日 | 2021-03-10 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.03 Å) | 主引用文献 | Recent structural insights into the mechanism of lysozyme hydrolysis. Acta Crystallogr D Struct Biol, 77, 2021
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7DER
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![BU of 7der by Molmil](/molmil-images/mine/7der) | Lysozyme alone in H2O | 分子名称: | CHLORIDE ION, Lysozyme C, SODIUM ION | 著者 | Tanaka, I, Chatake, T. | 登録日 | 2020-11-04 | 公開日 | 2021-03-10 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.03 Å) | 主引用文献 | Recent structural insights into the mechanism of lysozyme hydrolysis. Acta Crystallogr D Struct Biol, 77, 2021
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7BR5
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![BU of 7br5 by Molmil](/molmil-images/mine/7br5) | Lysozyme-sugar complex in H2O | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CHLORIDE ION, Lysozyme C, ... | 著者 | Tanaka, I, Chatake, T. | 登録日 | 2020-03-26 | 公開日 | 2021-03-10 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1 Å) | 主引用文献 | Recent structural insights into the mechanism of lysozyme hydrolysis. Acta Crystallogr D Struct Biol, 77, 2021
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4Q9K
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![BU of 4q9k by Molmil](/molmil-images/mine/4q9k) | P-glycoprotein cocrystallised with QZ-Leu | 分子名称: | (30F)L(30F)L(30F)L Peptide, Multidrug resistance protein 1A | 著者 | McGrath, A.P, Szewczyk, P, Chang, G. | 登録日 | 2014-05-01 | 公開日 | 2015-03-04 | 最終更新日 | 2024-07-10 | 実験手法 | X-RAY DIFFRACTION (3.8 Å) | 主引用文献 | Snapshots of ligand entry, malleable binding and induced helical movement in P-glycoprotein. Acta Crystallogr.,Sect.D, 71, 2015
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4Q9I
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![BU of 4q9i by Molmil](/molmil-images/mine/4q9i) | P-glycoprotein cocrystallised with QZ-Ala | 分子名称: | (30F)A(30F)A(30F)A Peptide, Multidrug resistance protein 1A | 著者 | McGrath, A.P, Szewczyk, P, Chang, G. | 登録日 | 2014-05-01 | 公開日 | 2015-03-04 | 最終更新日 | 2024-07-10 | 実験手法 | X-RAY DIFFRACTION (3.781 Å) | 主引用文献 | Snapshots of ligand entry, malleable binding and induced helical movement in P-glycoprotein. Acta Crystallogr.,Sect.D, 71, 2015
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4Q9J
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![BU of 4q9j by Molmil](/molmil-images/mine/4q9j) | P-glycoprotein cocrystallised with QZ-Val | 分子名称: | Multidrug resistance protein 1A, N-{[5-AMINO-1-(5-O-PHOSPHONO-BETA-D-ARABINOFURANOSYL)-1H-IMIDAZOL-4-YL]CARBONYL}-L-ASPARTIC ACID | 著者 | McGrath, A.P, Szewczyk, P, Chang, G. | 登録日 | 2014-05-01 | 公開日 | 2015-03-04 | 最終更新日 | 2024-07-10 | 実験手法 | X-RAY DIFFRACTION (3.6 Å) | 主引用文献 | Snapshots of ligand entry, malleable binding and induced helical movement in P-glycoprotein. Acta Crystallogr.,Sect.D, 71, 2015
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4Q9H
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![BU of 4q9h by Molmil](/molmil-images/mine/4q9h) | |
4DIR
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![BU of 4dir by Molmil](/molmil-images/mine/4dir) | |
4Q9L
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![BU of 4q9l by Molmil](/molmil-images/mine/4q9l) | P-glycoprotein cocrystallised with QZ-Phe | 分子名称: | (30F)F(30F)F(30F)F Peptide, Multidrug resistance protein 1A | 著者 | McGrath, A.P, Szewczyk, P, Chang, G. | 登録日 | 2014-05-01 | 公開日 | 2015-03-04 | 最終更新日 | 2024-07-10 | 実験手法 | X-RAY DIFFRACTION (3.8 Å) | 主引用文献 | Snapshots of ligand entry, malleable binding and induced helical movement in P-glycoprotein. Acta Crystallogr.,Sect.D, 71, 2015
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3BRK
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8H78
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![BU of 8h78 by Molmil](/molmil-images/mine/8h78) | Crystal structure of human MMP-2 catalytic domain in complex with inhibitor | 分子名称: | (2~{R})-2-[[4-[(4-aminocarbonylphenyl)carbonylamino]phenyl]sulfonylamino]-5-[(2~{S},4~{S})-4-azanyl-2-[[(2~{S})-1-[[(2~{S})-1-[(5-azanyl-5-oxidanylidene-pentyl)amino]-5-oxidanyl-1,5-bis(oxidanylidene)pentan-2-yl]-methyl-amino]-4-methyl-1-oxidanylidene-pentan-2-yl]carbamoyl]pyrrolidin-1-yl]-5-oxidanylidene-pentanoic acid, CALCIUM ION, DIHYDROGENPHOSPHATE ION, ... | 著者 | Kamitani, M, Takeuchi, T, Mima, M. | 登録日 | 2022-10-19 | 公開日 | 2023-01-18 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Discovery of TP0597850: A Selective, Chemically Stable, and Slow Tight-Binding Matrix Metalloproteinase-2 Inhibitor with a Phenylbenzamide-Pentapeptide Hybrid Scaffold. J.Med.Chem., 66, 2023
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6L0V
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![BU of 6l0v by Molmil](/molmil-images/mine/6l0v) | Structure of RLD2 BRX domain bound to LZY3 CCL motif | 分子名称: | 1,2-ETHANEDIOL, DI(HYDROXYETHYL)ETHER, NGR2, ... | 著者 | Hirano, Y, Futrutani, M, Nishimura, T, Taniguchi, M, Morita, M.T, Hakoshima, T. | 登録日 | 2019-09-27 | 公開日 | 2020-02-05 | 最終更新日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (1.347 Å) | 主引用文献 | Polar recruitment of RLD by LAZY1-like protein during gravity signaling in root branch angle control. Nat Commun, 11, 2020
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6L0W
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![BU of 6l0w by Molmil](/molmil-images/mine/6l0w) | Structure of RLD2 BRX domain bound to LZY3 CCL motif | 分子名称: | 1,2-ETHANEDIOL, CITRATE ANION, NGR2, ... | 著者 | Hirano, Y, Futrutani, M, Nishimura, T, Taniguchi, M, Morita, M.T, Hakoshima, T. | 登録日 | 2019-09-27 | 公開日 | 2020-02-05 | 実験手法 | X-RAY DIFFRACTION (1.591 Å) | 主引用文献 | Polar recruitment of RLD by LAZY1-like protein during gravity signaling in root branch angle control. Nat Commun, 11, 2020
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6KB0
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![BU of 6kb0 by Molmil](/molmil-images/mine/6kb0) | X-ray structure of human PPARalpha ligand binding domain-5,8,11,14-eicosatetraynoic acid (ETYA) co-crystals obtained by soaking | 分子名称: | GLYCEROL, Peroxisome proliferator-activated receptor alpha, icosa-5,8,11,14-tetraynoic acid | 著者 | Kamata, S, Suda, K, Saito, K, Oyama, T, Ishii, I. | 登録日 | 2019-06-24 | 公開日 | 2020-11-11 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.35 Å) | 主引用文献 | PPAR alpha Ligand-Binding Domain Structures with Endogenous Fatty Acids and Fibrates. Iscience, 23, 2020
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6KB1
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![BU of 6kb1 by Molmil](/molmil-images/mine/6kb1) | X-ray structure of human PPARalpha ligand binding domain-tetradecylthioacetic acid (TTA) co-crystals obtained by soaking | 分子名称: | 2-tetradecylsulfanylethanoic acid, GLYCEROL, Peroxisome proliferator-activated receptor alpha | 著者 | Kamata, S, Suda, K, Saito, K, Oyama, T, Ishii, I. | 登録日 | 2019-06-24 | 公開日 | 2020-11-11 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.25 Å) | 主引用文献 | PPAR alpha Ligand-Binding Domain Structures with Endogenous Fatty Acids and Fibrates. Iscience, 23, 2020
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6KAZ
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![BU of 6kaz by Molmil](/molmil-images/mine/6kaz) | X-ray structure of human PPARalpha ligand binding domain-pemafibrate co-crystals obtained by soaking | 分子名称: | (2~{R})-2-[3-[[1,3-benzoxazol-2-yl-[3-(4-methoxyphenoxy)propyl]amino]methyl]phenoxy]butanoic acid, GLYCEROL, Peroxisome proliferator-activated receptor alpha | 著者 | Kamata, S, Suda, K, Saito, K, Oyama, T, Ishii, I. | 登録日 | 2019-06-24 | 公開日 | 2020-11-11 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.48 Å) | 主引用文献 | PPAR alpha Ligand-Binding Domain Structures with Endogenous Fatty Acids and Fibrates. Iscience, 23, 2020
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