6D1N
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6AYH
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![BU of 6ayh by Molmil](/molmil-images/mine/6ayh) | Salmonella enterica GusR | 分子名称: | 4-nitrophenyl beta-D-glucopyranosiduronic acid, GLYCEROL, TetR family transcriptional regulator | 著者 | Little, M.S, Pellock, S.J. | 登録日 | 2017-09-08 | 公開日 | 2017-12-20 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | Structural basis for the regulation of beta-glucuronidase expression by human gut Enterobacteriaceae. Proc. Natl. Acad. Sci. U.S.A., 115, 2018
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6D1P
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![BU of 6d1p by Molmil](/molmil-images/mine/6d1p) | Apo structure of Bacteroides uniformis beta-glucuronidase 3 | 分子名称: | GLYCEROL, Glycosyl hydrolases family 2, sugar binding domain protein, ... | 著者 | Walton, W.G, Pellock, S.J, Redinbo, M.R. | 登録日 | 2018-04-12 | 公開日 | 2018-10-17 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.35 Å) | 主引用文献 | Three structurally and functionally distinct beta-glucuronidases from the human gut microbeBacteroides uniformis. J. Biol. Chem., 293, 2018
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6D41
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![BU of 6d41 by Molmil](/molmil-images/mine/6d41) | Bacteriodes uniformis beta-glucuronidase 1 bound to D-glucaro-1,5-lactone | 分子名称: | (2S,3S,4S,5R)-3,4,5-trihydroxy-6-oxo-oxane-2-carboxylic acid, Beta-galactosidase/beta-glucuronidase, CHLORIDE ION, ... | 著者 | Walton, W.G, Pellock, S.J, Redinbo, M.R. | 登録日 | 2018-04-17 | 公開日 | 2018-10-17 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Three structurally and functionally distinct beta-glucuronidases from the human gut microbeBacteroides uniformis. J. Biol. Chem., 293, 2018
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5DOZ
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5DOV
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6W32
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![BU of 6w32 by Molmil](/molmil-images/mine/6w32) | Crystal structure of Sfh5 | 分子名称: | PROTOPORPHYRIN IX CONTAINING FE, Phosphatidylinositol transfer protein SFH5 | 著者 | Gulten, G, Khan, D, Aggarwal, A, Krieger, I, Sacchettini, J.C, Bankaitis, V.A. | 登録日 | 2020-03-08 | 公開日 | 2020-11-25 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | A Sec14-like phosphatidylinositol transfer protein paralog defines a novel class of heme-binding proteins. Elife, 9, 2020
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6OD1
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![BU of 6od1 by Molmil](/molmil-images/mine/6od1) | IraD-bound to RssB D58P variant | 分子名称: | Anti-adapter protein IraD, Regulator of RpoS | 著者 | Deaconescu, A.M, Dorich, V. | 登録日 | 2019-03-25 | 公開日 | 2019-04-24 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structural basis for inhibition of a response regulator of sigmaSstability by a ClpXP antiadaptor. Genes Dev., 33, 2019
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5DP1
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5DP2
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7ZGB
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![BU of 7zgb by Molmil](/molmil-images/mine/7zgb) | Structure of yeast Sec14p with NPPM112 | 分子名称: | 4-fluoranyl-~{N}-[(4-pyrrolidin-1-ylphenyl)methyl]benzamide, SEC14 cytosolic factor | 著者 | Hong, Z, Johnen, P, Schaaf, G, Bono, F. | 登録日 | 2022-04-03 | 公開日 | 2023-01-25 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Mechanisms by which small molecules of diverse chemotypes arrest Sec14 lipid transfer activity. J.Biol.Chem., 299, 2023
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7ZG9
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![BU of 7zg9 by Molmil](/molmil-images/mine/7zg9) | Structure of yeast Sec14p with himbacine | 分子名称: | Himbacine, SEC14 cytosolic factor | 著者 | Hong, Z, Johnen, P, Schaaf, G, Bono, F. | 登録日 | 2022-04-03 | 公開日 | 2023-01-25 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.764 Å) | 主引用文献 | Mechanisms by which small molecules of diverse chemotypes arrest Sec14 lipid transfer activity. J.Biol.Chem., 299, 2023
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7ZGA
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![BU of 7zga by Molmil](/molmil-images/mine/7zga) | Structure of yeast Sec14p with ergoline | 分子名称: | SEC14 cytosolic factor, ~{O}9-methyl ~{O}4-[2,2,2-tris(chloranyl)ethyl] (5~{a}~{S},6~{a}~{S},9~{R},10~{a}~{S})-7-methyl-3-nitro-5,5~{a},6,6~{a},8,9,10,10~{a}-octahydroindolo[4,3-fg]quinoline-4,9-dicarboxylate | 著者 | Hong, Z, Johnen, P, Schaaf, G, Bono, F. | 登録日 | 2022-04-03 | 公開日 | 2023-01-25 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.302 Å) | 主引用文献 | Mechanisms by which small molecules of diverse chemotypes arrest Sec14 lipid transfer activity. J.Biol.Chem., 299, 2023
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7ZGC
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![BU of 7zgc by Molmil](/molmil-images/mine/7zgc) | Structure of yeast Sec14p with NPPM481 | 分子名称: | (4-chloranyl-3-nitro-phenyl)-[4-(2-fluorophenyl)piperazin-1-yl]methanone, PHOSPHATE ION, SEC14 cytosolic factor | 著者 | Hong, Z, Johnen, P, Schaaf, G, Bono, F. | 登録日 | 2022-04-03 | 公開日 | 2023-01-25 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.236 Å) | 主引用文献 | Mechanisms by which small molecules of diverse chemotypes arrest Sec14 lipid transfer activity. J.Biol.Chem., 299, 2023
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7ZGD
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![BU of 7zgd by Molmil](/molmil-images/mine/7zgd) | Structure of yeast Sec14p with NPPM244 | 分子名称: | (4-bromanyl-3-nitro-phenyl)-[4-(2-fluorophenyl)piperazin-1-yl]methanone, SEC14 cytosolic factor | 著者 | Hong, Z, Johnen, P, Schaaf, G, Bono, F. | 登録日 | 2022-04-03 | 公開日 | 2023-01-25 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.08 Å) | 主引用文献 | Mechanisms by which small molecules of diverse chemotypes arrest Sec14 lipid transfer activity. J.Biol.Chem., 299, 2023
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6F0E
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![BU of 6f0e by Molmil](/molmil-images/mine/6f0e) | Structure of yeast Sec14p with a picolinamide compound | 分子名称: | SEC14 cytosolic factor, ~{N}-(1,3-benzodioxol-5-ylmethyl)-5-bromanyl-3-fluoranyl-pyridine-2-carboxamide | 著者 | Hong, Z, Johnen, P, Schaaf, G, Bono, F. | 登録日 | 2017-11-20 | 公開日 | 2018-01-17 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Target Identification and Mechanism of Action of Picolinamide and Benzamide Chemotypes with Antifungal Properties. Cell Chem Biol, 25, 2018
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4X7U
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4X81
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![BU of 4x81 by Molmil](/molmil-images/mine/4x81) | MycF mycinamicin III 3'-O-methyltransferase (E35Q, M56A, E139A variant) in complex with Mg, SAH and mycinamicin VI (MycE substrate) | 分子名称: | DIMETHYL SULFOXIDE, MAGNESIUM ION, Mycinamicin III 3''-O-methyltransferase, ... | 著者 | Bernard, S.M, Smith, J.L. | 登録日 | 2014-12-09 | 公開日 | 2015-03-04 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.59 Å) | 主引用文献 | Structural Basis of Substrate Specificity and Regiochemistry in the MycF/TylF Family of Sugar O-Methyltransferases. Acs Chem.Biol., 10, 2015
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4X7W
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![BU of 4x7w by Molmil](/molmil-images/mine/4x7w) | MycF mycinamicin III 3'-O-methyltransferase (E35Q, E139A variant) in complex with Mg, SAH and mycinamicin VI (MycE substrate) | 分子名称: | MAGNESIUM ION, Mycinamicin III 3''-O-methyltransferase, Mycinamicin VI, ... | 著者 | Bernard, S.M, Smith, J.L. | 登録日 | 2014-12-09 | 公開日 | 2015-03-04 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Structural Basis of Substrate Specificity and Regiochemistry in the MycF/TylF Family of Sugar O-Methyltransferases. Acs Chem.Biol., 10, 2015
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4X7Z
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![BU of 4x7z by Molmil](/molmil-images/mine/4x7z) | MycF mycinamicin III 3'-O-methyltransferase (E35Q, M56A, E139A variant) in complex with Mg, SAH and mycinamicin III (substrate) | 分子名称: | DIMETHYL SULFOXIDE, MAGNESIUM ION, MYCINAMICIN III, ... | 著者 | Bernard, S.M, Smith, J.L. | 登録日 | 2014-12-09 | 公開日 | 2015-03-04 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.44 Å) | 主引用文献 | Structural Basis of Substrate Specificity and Regiochemistry in the MycF/TylF Family of Sugar O-Methyltransferases. Acs Chem.Biol., 10, 2015
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4X7X
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![BU of 4x7x by Molmil](/molmil-images/mine/4x7x) | MycF mycinamicin III 3'-O-methyltransferase (E35Q, E139A variant) in complex with Mg, SAH and macrocin | 分子名称: | 2-[(4R,5S,6S,7R,9R,11E,13E,15R,16R)-6-[(2R,3R,4R,5S,6R)-4-(dimethylamino)-5-[(2S,4R,5S,6S)-4,6-dimethyl-4,5-bis(oxidanyl)oxan-2-yl]oxy-6-methyl-3-oxidanyl-oxan-2-yl]oxy-16-ethyl-15-[[(2R,3R,4R,5S,6R)-3-methoxy-6-methyl-4,5-bis(oxidanyl)oxan-2-yl]oxymethyl]-5,9,13-trimethyl-4-oxidanyl-2,10-bis(oxidanylidene)-1-oxacyclohexadeca-11,13-dien-7-yl]ethanal, MAGNESIUM ION, Mycinamicin III 3''-O-methyltransferase, ... | 著者 | Bernard, S.M, Smith, J.L. | 登録日 | 2014-12-09 | 公開日 | 2015-03-11 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Structural Basis of Substrate Specificity and Regiochemistry in the MycF/TylF Family of Sugar O-Methyltransferases. Acs Chem.Biol., 10, 2015
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4X7Y
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4X7V
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![BU of 4x7v by Molmil](/molmil-images/mine/4x7v) | MycF mycinamicin III 3'-O-methyltransferase (E35Q, E139A variant) in complex with Mg, SAH and mycinamicin IV (product) | 分子名称: | MAGNESIUM ION, MYCINAMICIN IV, Mycinamicin III 3''-O-methyltransferase, ... | 著者 | Bernard, S.M, Smith, J.L. | 登録日 | 2014-12-09 | 公開日 | 2015-03-04 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | Structural Basis of Substrate Specificity and Regiochemistry in the MycF/TylF Family of Sugar O-Methyltransferases. Acs Chem.Biol., 10, 2015
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4XVZ
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4XVY
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