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1DOD
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BU of 1dod by Molmil
THE MOBIL FLAVIN OF 4-OH BENZOATE HYDROXYLASE: MOTION OF A PROSTHETIC GROUP REGULATES CATALYSIS
分子名称: 2,4-DIHYDROXYBENZOIC ACID, FLAVIN-ADENINE DINUCLEOTIDE, P-HYDROXYBENZOATE HYDROXYLASE
著者Gatti, D.L, Palfey, B.A, Lah, M.S, Entsch, B, Massey, V, Ballou, D.P, Ludwig, M.L.
登録日1994-09-06
公開日1994-11-30
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献The mobile flavin of 4-OH benzoate hydroxylase.
Science, 266, 1994
1K03
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BU of 1k03 by Molmil
Crystal Structure of Old Yellow Enzyme Mutant Gln114Asn Complexed with Para-hydroxy Benzaldehyde
分子名称: FLAVIN MONONUCLEOTIDE, MAGNESIUM ION, NADPH DEHYDROGENASE 1, ...
著者Brown, B.J, Hyun, J, Duvvuri, S.D, Karplus, P.A, Massey, V.
登録日2001-09-18
公開日2001-09-26
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献The role of glutamine 114 in old yellow enzyme
J.Biol.Chem., 277, 2002
1K02
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BU of 1k02 by Molmil
Crystal Structure of Old Yellow Enzyme Mutant Gln114Asn
分子名称: FLAVIN MONONUCLEOTIDE, MAGNESIUM ION, NADPH DEHYDROGENASE 1
著者Brown, B.J, Hyun, J, Duvvuri, S.D, Karplus, P.A, Massey, V.
登録日2001-09-18
公開日2001-09-26
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献The role of glutamine 114 in old yellow enzyme
J.Biol.Chem., 277, 2002
1BWK
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BU of 1bwk by Molmil
OLD YELLOW ENZYME (OYE1) MUTANT H191N
分子名称: FLAVIN MONONUCLEOTIDE, PROTEIN (NADPH DEHYDROGENASE 1)
著者Brown, B.J, Deng, Z, Karplus, P.A, Massey, V.
登録日1998-09-24
公開日1998-09-30
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献On the active site of Old Yellow Enzyme. Role of histidine 191 and asparagine 194.
J.Biol.Chem., 273, 1998
1BWL
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BU of 1bwl by Molmil
OLD YELLOW ENZYME (OYE1) DOUBLE MUTANT H191N:N194H
分子名称: FLAVIN MONONUCLEOTIDE, PROTEIN (NADPH DEHYDROGENASE 1)
著者Brown, B.J, Deng, Z, Karplus, P.A, Massey, V.
登録日1998-09-24
公開日1998-09-30
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献On the active site of Old Yellow Enzyme. Role of histidine 191 and asparagine 194.
J.Biol.Chem., 273, 1998
1DOB
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BU of 1dob by Molmil
THE MOBIL FLAVIN OF 4-OH BENZOATE HYDROXYLASE: MOTION OF A PROSTHETIC GROUP REGULATES CATALYSIS
分子名称: FLAVIN-ADENINE DINUCLEOTIDE, P-HYDROXYBENZOATE HYDROXYLASE, P-HYDROXYBENZOIC ACID
著者Gatti, D.L, Palfey, B.A, Lah, M.S, Entsch, B, Massey, V, Ballou, D.P, Ludwig, M.L.
登録日1994-09-06
公開日1994-11-30
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献The mobile flavin of 4-OH benzoate hydroxylase.
Science, 266, 1994
1D7L
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BU of 1d7l by Molmil
STRUCTURE-FUNCTION CORRELATIONS OF THE REACTION OF REDUCED NICOTINAMIDE ANALOGS WITH P-HYDROXYBENZOATE HYDROXYLASE SUBSTITUTED WITH A SERIES OF 8-SUBSTITUTED FLAVINS
分子名称: 8-DEMETHYL-8-DIMETHYLAMINO-FLAVIN-ADENINE-DINUCLEOTIDE, P-HYDROXYBENZOATE HYDROXYLASE, P-HYDROXYBENZOIC ACID, ...
著者Ortiz-Maldonado, M, Gatti, D, Ballou, D.P, Massey, V.
登録日1999-10-18
公開日2000-01-21
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structure-function correlations of the reaction of reduced nicotinamide analogues with p-hydroxybenzoate hydroxylase substituted with a series of 8-substituted flavins.
Biochemistry, 38, 1999
8TW3
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BU of 8tw3 by Molmil
hMPV fusion protein complexed with single domain antibodies sdHMPV16 and sdHMPV12
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Fusion glycoprotein, Single domain antibody sdHMPV12, ...
著者Rush, S.A, McLellan, J.S.
登録日2023-08-19
公開日2024-01-24
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献A neutralizing single-domain antibody that targets the trimer interface of the human metapneumovirus fusion protein.
Mbio, 15, 2024
5TOJ
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BU of 5toj by Molmil
Crystal structure of the RSV F glycoprotein in complex with the neutralizing single-domain antibody F-VHH-4
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Fusion glycoprotein F0, Fibritin chimera, ...
著者Gilman, M.S.A, Kabeche, S.C, McLellan, J.S.
登録日2016-10-17
公開日2017-02-22
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献Potent single-domain antibodies that arrest respiratory syncytial virus fusion protein in its prefusion state.
Nat Commun, 8, 2017
5TP3
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BU of 5tp3 by Molmil
Crystal structure of the RSV-neutralizing single-domain antibody F-VHH-4
分子名称: F-VHH-4
著者Wrapp, D, Gilman, M.S.A, McLellan, J.S.
登録日2016-10-19
公開日2017-02-22
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.874 Å)
主引用文献Potent single-domain antibodies that arrest respiratory syncytial virus fusion protein in its prefusion state.
Nat Commun, 8, 2017
5TOK
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BU of 5tok by Molmil
Crystal structure of the RSV F glycoprotein in complex with the neutralizing single-domain antibody F-VHH-L66
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Fusion glycoprotein F0, Fibritin chimera, ...
著者Gilman, M.S.A, Kabeche, S.C, McLellan, J.S.
登録日2016-10-17
公開日2017-02-22
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (3.8 Å)
主引用文献Potent single-domain antibodies that arrest respiratory syncytial virus fusion protein in its prefusion state.
Nat Commun, 8, 2017
6VTW
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BU of 6vtw by Molmil
De novo protein design enables the precise induction of RSV-neutralizing antibodies
分子名称: 101F Fab Heavy Chain, 101F Fab Light Chain, S4_2.45
著者Jardetzky, T, Correia, B.
登録日2020-02-13
公開日2020-04-15
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献De novo protein design enables the precise induction of RSV-neutralizing antibodies.
Science, 368, 2020
8CW9
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BU of 8cw9 by Molmil
Prefusion-stabilized hMPV fusion protein bound to ADI-61026 and MPE8 Fabs
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, ADI-61026 heavy, ADI-61026 light, ...
著者Hsieh, C.-L, McLellan, J.S.
登録日2022-05-18
公開日2022-08-10
最終更新日2023-02-22
実験手法ELECTRON MICROSCOPY (3.46 Å)
主引用文献Potently neutralizing and protective anti-human metapneumovirus antibodies target diverse sites on the fusion glycoprotein.
Immunity, 55, 2022
4ZYK
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BU of 4zyk by Molmil
Crystal Structure of Quaternary-Specific RSV-Neutralizing Human Antibody AM14
分子名称: 1,2-ETHANEDIOL, ACETATE ION, AM14 Fab heavy chain, ...
著者Gilman, M.S.A, McLellan, J.S.
登録日2015-05-21
公開日2015-07-29
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Characterization of a Prefusion-Specific Antibody That Recognizes a Quaternary, Cleavage-Dependent Epitope on the RSV Fusion Glycoprotein.
Plos Pathog., 11, 2015
4ZYP
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BU of 4zyp by Molmil
Crystal Structure of Motavizumab and Quaternary-Specific RSV-Neutralizing Human Antibody AM14 in Complex with Prefusion RSV F Glycoprotein
分子名称: AM14 antibody Fab heavy chain, AM14 antibody light chain, Fusion glycoprotein F0,Fibritin, ...
著者Gilman, M.S.A, McLellan, J.S.
登録日2015-05-21
公開日2015-07-29
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (5.5 Å)
主引用文献Characterization of a Prefusion-Specific Antibody That Recognizes a Quaternary, Cleavage-Dependent Epitope on the RSV Fusion Glycoprotein.
Plos Pathog., 11, 2015
6XWI
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BU of 6xwi by Molmil
Solution NMR structure of the S0_2.126 designed protein
分子名称: S0_2.126
著者Abriata, L.A.
登録日2020-01-23
公開日2020-04-15
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献De novo protein design enables the precise induction of RSV-neutralizing antibodies.
Science, 368, 2020
6XXV
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BU of 6xxv by Molmil
Crystal Structure of a computationally designed Immunogen S2_1.2 in complex with its elicited antibody C57
分子名称: Antibody C57, Heavy Chain, Light Chain, ...
著者Yang, C, Sesterhenn, F, Correia, B.E, Pojer, F.
登録日2020-01-28
公開日2020-04-22
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.20116425 Å)
主引用文献De novo protein design enables the precise induction of RSV-neutralizing antibodies.
Science, 368, 2020
5WB0
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BU of 5wb0 by Molmil
Crystal structure of human metapneumovirus fusion glycoprotein stabilized in the prefusion state
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Fusion glycoprotein F0, ...
著者Battles, M.B, McLellan, J.S.
登録日2017-06-27
公開日2017-11-22
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.601 Å)
主引用文献Structure and immunogenicity of pre-fusion-stabilized human metapneumovirus F glycoprotein.
Nat Commun, 8, 2017
7SEM
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BU of 7sem by Molmil
Structure-based design of prefusion-stabilized human metapneumovirus fusion proteins
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Fusion glycoprotein F0, MPE8 Fab heavy chain, ...
著者Rush, S.A, Hsieh, C.-L, McLellan, J.S.
登録日2021-09-30
公開日2022-02-16
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structure-based design of prefusion-stabilized human metapneumovirus fusion proteins.
Nat Commun, 13, 2022
7SEJ
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BU of 7sej by Molmil
Structure-based design of prefusion-stabilized human metapneumovirus fusion proteins
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Fusion glycoprotein F1 subunit, Fusion glycoprotein F2 subunit
著者Hsieh, C.-L, Rush, S.A, McLellan, J.S.
登録日2021-09-30
公開日2022-02-09
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.51 Å)
主引用文献Structure-based design of prefusion-stabilized human metapneumovirus fusion proteins.
Nat Commun, 13, 2022
6S3D
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BU of 6s3d by Molmil
Structure of D25 Fab in complex with scaffold S0_2.126
分子名称: Heavy Chain, Light Chain, S0_2.126
著者Cramer, J.T, Krey, T.
登録日2019-06-25
公開日2020-04-22
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献De novo protein design enables the precise induction of RSV-neutralizing antibodies.
Science, 368, 2020
3NLL
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BU of 3nll by Molmil
CLOSTRIDIUM BEIJERINCKII FLAVODOXIN MUTANT: G57A OXIDIZED
分子名称: FLAVIN MONONUCLEOTIDE, FLAVODOXIN
著者Ludwig, M.L, Pattridge, K.A, Metzger, A.L, Dixon, M.M, Eren, M, Feng, Y, Swenson, R.
登録日1996-12-10
公開日1997-03-12
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Control of oxidation-reduction potentials in flavodoxin from Clostridium beijerinckii: the role of conformation changes.
Biochemistry, 36, 1997
6P8Z
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BU of 6p8z by Molmil
Crystal structure of human KRAS G12C covalently bound to an acryloylazetidine acetamide inhibitor
分子名称: 2-[5-chloro-2-cyclopropyl-3-(5-methoxy-3,4-dihydroisoquinoline-2(1H)-carbonyl)-7-methyl-1H-indol-1-yl]-N-(1-propanoylazetidin-3-yl)acetamide, CALCIUM ION, GTPase KRas, ...
著者Mohr, C.
登録日2019-06-08
公開日2019-08-28
最終更新日2019-10-02
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Discovery ofN-(1-Acryloylazetidin-3-yl)-2-(1H-indol-1-yl)acetamides as Covalent Inhibitors of KRASG12C.
Acs Med.Chem.Lett., 10, 2019
6PGO
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BU of 6pgo by Molmil
Crystal structure of human KRAS G12C covalently bound to a phthalazine inhibitor
分子名称: 1-{4-[7-chloro-6-(2-fluoro-6-hydroxyphenyl)-4-phenylphthalazin-1-yl]piperazin-1-yl}propan-1-one, GTPase KRas, GUANOSINE-5'-DIPHOSPHATE, ...
著者Mohr, C.
登録日2019-06-24
公開日2019-12-25
最終更新日2020-01-22
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Discovery of a Covalent Inhibitor of KRASG12C(AMG 510) for the Treatment of Solid Tumors.
J.Med.Chem., 63, 2020
6P8W
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BU of 6p8w by Molmil
Crystal structure of human KRAS G12C covalently bound to an acryloylazetidine acetamide inhibitor.
分子名称: CALCIUM ION, GTPase KRas, GUANOSINE-5'-DIPHOSPHATE, ...
著者Mohr, C.
登録日2019-06-08
公開日2019-08-28
最終更新日2019-10-02
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Discovery ofN-(1-Acryloylazetidin-3-yl)-2-(1H-indol-1-yl)acetamides as Covalent Inhibitors of KRASG12C.
Acs Med.Chem.Lett., 10, 2019

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