4WQN
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![BU of 4wqn by Molmil](/molmil-images/mine/4wqn) | Crystal structure of N6-methyladenosine RNA reader YTHDF2 | 分子名称: | 1,2-ETHANEDIOL, GLYCEROL, YTH domain-containing family protein 2 | 著者 | Zhu, T, Roundtree, I.A, Wang, P, Wang, X, Wang, L, Sun, C, Tian, Y, Li, J, He, C, Xu, Y. | 登録日 | 2014-10-22 | 公開日 | 2014-11-19 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.121 Å) | 主引用文献 | Crystal structure of the YTH domain of YTHDF2 reveals mechanism for recognition of N6-methyladenosine. Cell Res., 24, 2014
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1I3O
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![BU of 1i3o by Molmil](/molmil-images/mine/1i3o) | CRYSTAL STRUCTURE OF THE COMPLEX OF XIAP-BIR2 AND CASPASE 3 | 分子名称: | BACULOVIRAL IAP REPEAT-CONTAINING PROTEIN 4, CASPASE 3, ZINC ION | 著者 | Riedl, S.J, Renatus, M, Schwarzenbacher, R, Zhou, Q, Sun, C, Fesik, S.W, Liddington, R.C, Salvesen, G.S. | 登録日 | 2001-02-15 | 公開日 | 2001-03-21 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Structural basis for the inhibition of caspase-3 by XIAP. Cell(Cambridge,Mass.), 104, 2001
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1G3F
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![BU of 1g3f by Molmil](/molmil-images/mine/1g3f) | NMR STRUCTURE OF A 9 RESIDUE PEPTIDE FROM SMAC/DIABLO COMPLEXED TO THE BIR3 DOMAIN OF XIAP | 分子名称: | INHIBITOR OF APOPTOSIS PROTEIN 3, SMAC, ZINC ION | 著者 | Liu, Z, Sun, C, Olejniczak, E.T, Meadows, R.P, Betz, S.F, Oost, T, Herrmann, J, Wu, J.C, Fesik, S.W. | 登録日 | 2000-10-24 | 公開日 | 2001-01-10 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Structural basis for binding of Smac/DIABLO to the XIAP BIR3 domain. Nature, 408, 2000
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4MGJ
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![BU of 4mgj by Molmil](/molmil-images/mine/4mgj) | Crystal structure of cytochrome P450 2B4 F429H in complex with 4-CPI | 分子名称: | 4-(4-CHLOROPHENYL)IMIDAZOLE, Cytochrome P450 2B4, PROTOPORPHYRIN IX CONTAINING FE | 著者 | Yang, Y, Zhang, H, Usharani, D, Bu, W, Im, S, Tarasev, M, Rwere, F, Meagher, J, Sun, C, Stuckey, J, Shaik, S, Waskell, L. | 登録日 | 2013-08-28 | 公開日 | 2014-08-13 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.41 Å) | 主引用文献 | Structural and Functional Characterization of a Cytochrome P450 2B4 F429H Mutant with an Axial Thiolate-Histidine Hydrogen Bond. Biochemistry, 53, 2014
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5V33
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![BU of 5v33 by Molmil](/molmil-images/mine/5v33) | R. sphaeroides photosythetic reaction center mutant - Residue L223, Ser to Trp - Room Temperature Structure Solved on X-ray Transparent Microfluidic Chip | 分子名称: | BACTERIOCHLOROPHYLL A, BACTERIOPHEOPHYTIN A, FE (III) ION, ... | 著者 | Schieferstein, J.M, Pawate, A.S, Sun, C, Wan, F, Broecker, J, Ernst, O.P, Gennis, R.B, Kenis, P.J.A. | 登録日 | 2017-03-06 | 公開日 | 2017-04-12 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (3.487 Å) | 主引用文献 | X-ray transparent microfluidic chips for high-throughput screening and optimization of in meso membrane protein crystallization. Biomicrofluidics, 11, 2017
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3NEW
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![BU of 3new by Molmil](/molmil-images/mine/3new) | p38-alpha complexed with Compound 10 | 分子名称: | 4-(trifluoromethyl)-3-[3-(trifluoromethyl)phenyl]-1,7-dihydro-6H-pyrazolo[3,4-b]pyridin-6-one, Mitogen-activated protein kinase 14 | 著者 | Goedken, E.R, Comess, K.M, Sun, C, Argiriadi, M, Jia, Y, Quinn, C.M, Banach, D.L, Marcotte, D, Borhani, D. | 登録日 | 2010-06-09 | 公開日 | 2010-12-01 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.51 Å) | 主引用文献 | Discovery and Characterization of Non-ATP Site Inhibitors of the Mitogen Activated Protein (MAP) Kinases. Acs Chem.Biol., 6, 2011
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8J2G
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6MX4
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![BU of 6mx4 by Molmil](/molmil-images/mine/6mx4) | CryoEM structure of chimeric Eastern Equine Encephalitis Virus | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Capsid, ... | 著者 | Hasan, S.S, Sun, C, Kim, A.S, Watanabe, Y, Chen, C.L, Klose, T, Buda, G, Crispin, M, Diamond, M.S, Klimstra, W.B, Rossmann, M.G. | 登録日 | 2018-10-30 | 公開日 | 2018-12-19 | 最終更新日 | 2020-07-29 | 実験手法 | ELECTRON MICROSCOPY (4.4 Å) | 主引用文献 | Cryo-EM Structures of Eastern Equine Encephalitis Virus Reveal Mechanisms of Virus Disassembly and Antibody Neutralization. Cell Rep, 25, 2018
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6MWC
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![BU of 6mwc by Molmil](/molmil-images/mine/6mwc) | CryoEM structure of chimeric Eastern Equine Encephalitis Virus with Fab of EEEV-5 antibody | 分子名称: | E1, E2, EEEV-5 antibody heavy chain, ... | 著者 | Hasan, S.S, Sun, C, Kim, A.S, Watanabe, Y, Chen, C.L, Klose, T, Buda, G, Crispin, M, Diamond, M.S, Klimstra, W.B, Rossmann, M.G. | 登録日 | 2018-10-29 | 公開日 | 2018-12-19 | 最終更新日 | 2019-12-18 | 実験手法 | ELECTRON MICROSCOPY (7.5 Å) | 主引用文献 | Cryo-EM Structures of Eastern Equine Encephalitis Virus Reveal Mechanisms of Virus Disassembly and Antibody Neutralization. Cell Rep, 25, 2018
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5CPR
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![BU of 5cpr by Molmil](/molmil-images/mine/5cpr) | The novel SUV4-20 inhibitor A-196 verifies a role for epigenetics in genomic integrity | 分子名称: | 6,7-dichloro-N-cyclopentyl-4-(pyridin-4-yl)phthalazin-1-amine, Histone-lysine N-methyltransferase SUV420H1, S-ADENOSYLMETHIONINE, ... | 著者 | Jakob, C.G, Upadhyay, A.K, Sun, C. | 登録日 | 2015-07-21 | 公開日 | 2017-01-25 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.22 Å) | 主引用文献 | The SUV4-20 inhibitor A-196 verifies a role for epigenetics in genomic integrity. Nat. Chem. Biol., 13, 2017
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5C56
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![BU of 5c56 by Molmil](/molmil-images/mine/5c56) | Crystal structure of USP7/HAUSP in complex with ICP0 | 分子名称: | Ubiquitin E3 ligase ICP0, Ubiquitin carboxyl-terminal hydrolase 7 | 著者 | Cheng, J, Li, Z, Gong, R, Fang, J, Yang, Y, Sun, C, Yang, H, Xu, Y. | 登録日 | 2015-06-19 | 公開日 | 2015-07-08 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.685 Å) | 主引用文献 | Molecular mechanism for the substrate recognition of USP7. Protein Cell, 6, 2015
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2A9H
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![BU of 2a9h by Molmil](/molmil-images/mine/2a9h) | NMR structural studies of a potassium channel / charybdotoxin complex | 分子名称: | Voltage-gated potassium channel, charybdotoxin | 著者 | Yu, L, Sun, C, Song, D, Shen, J, Xu, N, Gunasekera, A, Hajduk, P.J, Olejniczak, E.T. | 登録日 | 2005-07-11 | 公開日 | 2006-01-10 | 最終更新日 | 2021-10-20 | 実験手法 | SOLUTION NMR | 主引用文献 | Nuclear magnetic resonance structural studies of a potassium channel-charybdotoxin complex. Biochemistry, 44, 2005
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4OQ5
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![BU of 4oq5 by Molmil](/molmil-images/mine/4oq5) | Crystal Structure of Human MCL-1 Bound to Inhibitor 4-(4-methylnaphthalen-1-yl)-2-{[(4-phenoxyphenyl)sulfonyl]amino}benzoic acid | 分子名称: | 4-(4-methylnaphthalen-1-yl)-2-{[(4-phenoxyphenyl)sulfonyl]amino}benzoic acid, Induced myeloid leukemia cell differentiation protein Mcl-1 | 著者 | Petros, A.M, Swann, S.L, Song, D, Swinger, K, Park, C, Zhang, H, Wendt, M.D, Kunzer, A.R, Souers, A.J, Sun, C. | 登録日 | 2014-02-07 | 公開日 | 2014-03-12 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.86 Å) | 主引用文献 | Fragment-based discovery of potent inhibitors of the anti-apoptotic MCL-1 protein. Bioorg.Med.Chem.Lett., 24, 2014
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4OQ6
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![BU of 4oq6 by Molmil](/molmil-images/mine/4oq6) | Crystal Structure of Human MCL-1 Bound to Inhibitor 4-hydroxy-4'-propylbiphenyl-3-carboxylic acid | 分子名称: | 4-hydroxy-4'-propylbiphenyl-3-carboxylic acid, Induced myeloid leukemia cell differentiation protein Mcl-1 | 著者 | Petros, A.M, Swann, S.L, Song, D, Swinger, K, Park, C, Zhang, H, Wendt, M.D, Kunzer, A.R, Souers, A.J, Sun, C. | 登録日 | 2014-02-07 | 公開日 | 2014-03-12 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.81 Å) | 主引用文献 | Fragment-based discovery of potent inhibitors of the anti-apoptotic MCL-1 protein. Bioorg.Med.Chem.Lett., 24, 2014
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2NW4
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![BU of 2nw4 by Molmil](/molmil-images/mine/2nw4) | Crystal Structure of the Rat Androgen Receptor Ligand Binding Domain Complex with BMS-564929 | 分子名称: | 2-CHLORO-4-[(7R,7AS)-7-HYDROXY-1,3-DIOXOTETRAHYDRO-1H-PYRROLO[1,2-C]IMIDAZOL-2(3H)-YL]-3-METHYLBENZONITRILE, Androgen receptor | 著者 | Ostrowski, J, Kuhns, J.E, Lupisella, J.A, Manfredi, M.C, Beehler, B.C, Krystek, S.R, Bi, Y, Sun, C, Seethala, R, Golla, R, Sleph, P.G, Fura, A, An, Y, Kish, K.F, Sack, J.S, Mookhtiar, K.A, Grover, G.J, Hamann, L.G. | 登録日 | 2006-11-14 | 公開日 | 2006-12-12 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Pharmacological and x-ray structural characterization of a novel selective androgen receptor modulator: potent hyperanabolic stimulation of skeletal muscle with hypostimulation of prostate in rats. Endocrinology, 148, 2007
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7K5W
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![BU of 7k5w by Molmil](/molmil-images/mine/7k5w) | Cryo-EM structure of heterologous protein complex loaded Thermotoga maritima encapsulin capsid | 分子名称: | Maritimacin | 著者 | Xiong, X, Sun, C, Vago, F.S, Klose, T, Zhu, J, Jiang, W. | 登録日 | 2020-09-17 | 公開日 | 2020-10-07 | 最終更新日 | 2024-03-06 | 実験手法 | ELECTRON MICROSCOPY (2.87 Å) | 主引用文献 | Cryo-EM Structure of Heterologous Protein Complex Loaded Thermotoga Maritima Encapsulin Capsid. Biomolecules, 10, 2020
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2E6W
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![BU of 2e6w by Molmil](/molmil-images/mine/2e6w) | Solution structure and calcium binding properties of EF-hands 3 and 4 of calsenilin | 分子名称: | CALCIUM ION, Calsenilin | 著者 | Yu, L, Sun, C, Mendoza, R, Hebert, E, Pereda-Lopez, A, Hajduk, P.J, Olejniczak, E.T. | 登録日 | 2007-01-05 | 公開日 | 2007-11-27 | 最終更新日 | 2024-05-29 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure and calcium-binding properties of EF-hands 3 and 4 of calsenilin. Protein Sci., 16, 2007
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4QG6
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![BU of 4qg6 by Molmil](/molmil-images/mine/4qg6) | crystal structure of PKM2-Y105E mutant | 分子名称: | PROLINE, Pyruvate kinase PKM | 著者 | Wang, P, Sun, C, Zhu, T, Xu, Y. | 登録日 | 2014-05-22 | 公開日 | 2015-02-25 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (3.207 Å) | 主引用文献 | Structural insight into mechanisms for dynamic regulation of PKM2. Protein Cell, 6, 2015
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4QG8
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![BU of 4qg8 by Molmil](/molmil-images/mine/4qg8) | crystal structure of PKM2-K305Q mutant | 分子名称: | GLYCEROL, MAGNESIUM ION, MALONATE ION, ... | 著者 | Wang, P, Sun, C, Zhu, T, Xu, Y. | 登録日 | 2014-05-22 | 公開日 | 2015-02-25 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structural insight into mechanisms for dynamic regulation of PKM2. Protein Cell, 6, 2015
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4QGC
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![BU of 4qgc by Molmil](/molmil-images/mine/4qgc) | crystal structure of PKM2-K422R mutant | 分子名称: | GLYCEROL, POTASSIUM ION, Pyruvate kinase PKM, ... | 著者 | Wang, P, Sun, C, Zhu, T, Xu, Y. | 登録日 | 2014-05-22 | 公開日 | 2015-02-25 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (2.296 Å) | 主引用文献 | Structural insight into mechanisms for dynamic regulation of PKM2. Protein Cell, 6, 2015
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4QG9
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![BU of 4qg9 by Molmil](/molmil-images/mine/4qg9) | crystal structure of PKM2-R399E mutant | 分子名称: | ACETATE ION, MAGNESIUM ION, Pyruvate kinase PKM | 著者 | Wang, P, Sun, C, Zhu, T, Xu, Y. | 登録日 | 2014-05-22 | 公開日 | 2015-02-25 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (2.381 Å) | 主引用文献 | Structural insight into mechanisms for dynamic regulation of PKM2. Protein Cell, 6, 2015
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6MW9
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![BU of 6mw9 by Molmil](/molmil-images/mine/6mw9) | CryoEM structure of chimeric Eastern Equine Encephalitis Virus with Fab of EEEV-3 antibody | 分子名称: | E1, E2, EEEV-3 antibody heavy chain, ... | 著者 | Hasan, S.S, Sun, C, Kim, A.S, Watanabe, Y, Chen, C.L, Klose, T, Buda, G, Crispin, M, Diamond, M.S, Klimstra, W.B, Rossmann, M.G. | 登録日 | 2018-10-29 | 公開日 | 2018-12-19 | 最終更新日 | 2019-12-18 | 実験手法 | ELECTRON MICROSCOPY (7.3 Å) | 主引用文献 | Cryo-EM Structures of Eastern Equine Encephalitis Virus Reveal Mechanisms of Virus Disassembly and Antibody Neutralization. Cell Rep, 25, 2018
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6MWX
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![BU of 6mwx by Molmil](/molmil-images/mine/6mwx) | CryoEM structure of Chimeric Eastern Equine Encephalitis Virus with Fab of EEEV-69 Antibody | 分子名称: | E1, E2, EEEV-69 antibody heavy chain, ... | 著者 | Hasan, S.S, Sun, C, Kim, A.S, Watanabe, Y, Chen, C.L, Klose, T, Buda, G, Crispin, M, Diamond, M.S, Klimstra, W.B, Rossmann, M.G. | 登録日 | 2018-10-30 | 公開日 | 2018-12-19 | 最終更新日 | 2019-12-18 | 実験手法 | ELECTRON MICROSCOPY (8.2 Å) | 主引用文献 | Cryo-EM Structures of Eastern Equine Encephalitis Virus Reveal Mechanisms of Virus Disassembly and Antibody Neutralization. Cell Rep, 25, 2018
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6MUI
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![BU of 6mui by Molmil](/molmil-images/mine/6mui) | CryoEM structure of chimeric Eastern Equine Encephalitis Virus with Fab of EEEV-42 antibody | 分子名称: | E1, E2, EEEV-42 antibody heavy chain, ... | 著者 | Hasan, S.S, Sun, C, Kim, A.S, Watanabe, Y, Chen, C.L, Klose, T, Buda, G, Crispin, M, Diamond, M.S, Klimstra, W.B, Rossmann, M.G. | 登録日 | 2018-10-23 | 公開日 | 2018-12-19 | 最終更新日 | 2019-12-18 | 実験手法 | ELECTRON MICROSCOPY (7.7 Å) | 主引用文献 | Cryo-EM Structures of Eastern Equine Encephalitis Virus Reveal Mechanisms of Virus Disassembly and Antibody Neutralization. Cell Rep, 25, 2018
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6MX7
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![BU of 6mx7 by Molmil](/molmil-images/mine/6mx7) | CryoEM structure of chimeric Eastern Equine Encephalitis Virus: Genome-Binding Capsid N-terminal Domain | 分子名称: | Capsid | 著者 | Hasan, S.S, Sun, C, Kim, A.S, Watanabe, Y, Chen, C.L, Klose, T, Buda, G, Crispin, M, Diamond, M.S, Klimstra, W.B, Rossmann, M.G. | 登録日 | 2018-10-30 | 公開日 | 2018-12-19 | 最終更新日 | 2024-03-13 | 実験手法 | ELECTRON MICROSCOPY (4.8 Å) | 主引用文献 | Cryo-EM Structures of Eastern Equine Encephalitis Virus Reveal Mechanisms of Virus Disassembly and Antibody Neutralization. Cell Rep, 25, 2018
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