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3EIO
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BU of 3eio by Molmil
Crystal Structure Analysis of DPPIV Inhibitor
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 4-({4-[(3R)-3-amino-4-(2,4,5-trifluorophenyl)butanoyl]-1,4-diazepan-1-yl}carbonyl)benzoic acid, ...
著者Ahn, J.H, Lee, J.-O.
登録日2008-09-17
公開日2008-11-04
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Synthesis and biological evaluation of homopiperazine derivatives with beta-aminoacyl group as dipeptidyl peptidase IV inhibitors
Bioorg.Med.Chem.Lett., 18, 2008
3Q8W
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BU of 3q8w by Molmil
A b-aminoacyl containing thiazolidine derivative and DPPIV complex
分子名称: Dipeptidyl peptidase 4, N-(4-{[({(2R)-3-[(3R)-3-amino-4-(2,4,5-trifluorophenyl)butanoyl]-1,3-thiazolidin-2-yl}carbonyl)amino]methyl}phenyl)-D-valine
著者Lee, J.O, Song, D.H.
登録日2011-01-07
公開日2011-03-16
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (3.64 Å)
主引用文献Discovery of b-aminoacyl containing thiazolidine derivatives as potent and selective dipeptidyl peptidase IV inhibitors
To be Published
1AYM
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BU of 1aym by Molmil
HUMAN RHINOVIRUS 16 COAT PROTEIN AT HIGH RESOLUTION
分子名称: HUMAN RHINOVIRUS 16 COAT PROTEIN, LAURIC ACID, MYRISTIC ACID, ...
著者Hadfield, A.T, Rossmann, M.G.
登録日1997-11-06
公開日1998-01-21
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献The refined structure of human rhinovirus 16 at 2.15 A resolution: implications for the viral life cycle.
Structure, 5, 1997
1C8M
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BU of 1c8m by Molmil
REFINED CRYSTAL STRUCTURE OF HUMAN RHINOVIRUS 16 COMPLEXED WITH VP63843 (PLECONARIL), AN ANTI-PICORNAVIRAL DRUG CURRENTLY IN CLINICAL TRIALS
分子名称: 3-{3,5-DIMETHYL-4-[3-(3-METHYL-ISOXAZOL-5-YL)-PROPOXY]-PHENYL}-5-TRIFLUOROMETHYL-[1,2,4]OXADIAZOLE, HUMAN RHINOVIRUS 16 COAT PROTEIN, ZINC ION
著者Chakravarty, S, Bator, C.M, Pevear, D.C, Diana, G.D, Rossmann, M.G.
登録日2000-05-26
公開日2000-11-22
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献THE REFINED STRUCTURE OF A PICORNAVIRUS INHIBITOR CURRENTLY IN CLINICAL TRIALS, WHEN COMPLEXED WITH HUMAN RHINOVIRUS 16
to be published
1AYN
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BU of 1ayn by Molmil
HUMAN RHINOVIRUS 16 COAT PROTEIN
分子名称: HUMAN RHINOVIRUS 16 COAT PROTEIN, LAURIC ACID, MYRISTIC ACID, ...
著者Hadfield, A.T, Oliveira, M.A, Zhao, R, Rossmann, M.G.
登録日1997-11-06
公開日1998-01-21
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献The structure of human rhinovirus 16.
Structure, 1, 1993
6CX0
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BU of 6cx0 by Molmil
Structure of AtTPC1 D376A
分子名称: (1S,3R)-1-(3-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-4-methoxyphenyl)-2,3,4,9-tetrahydro-1H-beta-carboline-3-carboxylic acid, CALCIUM ION, Two pore calcium channel protein 1
著者Kintzer, A.F, Stroud, R.M.
登録日2018-04-02
公開日2018-09-19
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (3.501 Å)
主引用文献Structural basis for activation of voltage sensor domains in an ion channel TPC1.
Proc. Natl. Acad. Sci. U.S.A., 115, 2018
8SLB
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BU of 8slb by Molmil
X-ray structure of CorA N-terminal domain in complex with conformation-specific synthetic antibody C12
分子名称: CHLORIDE ION, Cobalt/magnesium transport protein CorA, sAB C12 Heavy Chain, ...
著者Dominik, P.K, Erramilli, S.K, Reddy, B.G, Kossiakoff, A.A.
登録日2023-04-21
公開日2023-06-07
最終更新日2023-07-26
実験手法X-RAY DIFFRACTION (2.04 Å)
主引用文献Conformation-specific Synthetic Antibodies Discriminate Multiple Functional States of the Ion Channel CorA.
J.Mol.Biol., 435, 2023
5BK1
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BU of 5bk1 by Molmil
Crystal structure of maltose binding protein in complex with an endosteric synthetic antibody
分子名称: CHLORIDE ION, GLYCEROL, Maltose binding protein, ...
著者Mukherjee, S, Kossiakoff, A.A.
登録日2017-09-12
公開日2018-01-17
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Engineered synthetic antibodies as probes to quantify the energetic contributions of ligand binding to conformational changes in proteins.
J. Biol. Chem., 293, 2018
5BK2
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Crystal structure of maltose binding protein in complex with a peristeric synthetic antibody
分子名称: CHLORIDE ION, GLYCEROL, Maltose-binding periplasmic protein, ...
著者Mukherjee, S, Kossiakoff, A.A.
登録日2017-09-12
公開日2018-01-17
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Engineered synthetic antibodies as probes to quantify the energetic contributions of ligand binding to conformational changes in proteins.
J. Biol. Chem., 293, 2018
5BJZ
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BU of 5bjz by Molmil
Crystal structure of maltose binding protein in complex with an allosteric synthetic antibody
分子名称: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, CHLORIDE ION, GLYCEROL, ...
著者Mukherjee, S, Kossiakoff, A.A.
登録日2017-09-12
公開日2018-01-17
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Engineered synthetic antibodies as probes to quantify the energetic contributions of ligand binding to conformational changes in proteins.
J. Biol. Chem., 293, 2018
3D1E
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BU of 3d1e by Molmil
Crystal structure of E. coli sliding clamp (beta) bound to a polymerase II peptide
分子名称: DNA polymerase III subunit beta, decamer from polymerase II C-terminal
著者Georgescu, R.E, Yurieva, O, Seung-Sup, K, Kuriyan, J, Kong, X.-P, O'Donnell, M.
登録日2008-05-05
公開日2008-07-29
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structure of a small-molecule inhibitor of a DNA polymerase sliding clamp.
Proc.Natl.Acad.Sci.Usa, 105, 2008
3D1G
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BU of 3d1g by Molmil
Structure of a small molecule inhibitor bound to a DNA sliding clamp
分子名称: DNA polymerase III subunit beta, [(5R)-5-(2,3-dibromo-5-ethoxy-4-hydroxybenzyl)-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]acetic acid
著者Georgescu, R.E, Yurieva, O, Seung-Sup, K, Kuriyan, J, Kong, X.-P, O'Donnell, M.
登録日2008-05-05
公開日2008-07-29
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.64 Å)
主引用文献Structure of a small-molecule inhibitor of a DNA polymerase sliding clamp.
Proc.Natl.Acad.Sci.Usa, 105, 2008
1QJX
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BU of 1qjx by Molmil
HUMAN RHINOVIRUS 16 COAT PROTEIN IN COMPLEX WITH ANTIVIRAL COMPOUND WIN68934
分子名称: 2,6-DIMETHYL-1-(3-[3-METHYL-5-ISOXAZOLYL]-PROPANYL)-4-[4-METHYL-2H-TETRAZOL-2-YL]-PHENOL, MYRISTIC ACID, PROTEIN VP1, ...
著者Hadfield, A.T, Diana, G.D, Rossmann, M.G.
登録日1999-07-06
公開日1999-07-20
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Analysis of Three Structurally Related Antiviral Compounds in Complex with Human Rhinovirus 16
Proc.Natl.Acad.Sci.USA, 96, 1999
3GHE
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BU of 3ghe by Molmil
Crystal structure of anti-HIV-1 Fab 537-10D in complex with V3 peptide MN
分子名称: Envelope glycoprotein, Fab 537-10D, heavy chain, ...
著者Kong, X.P, Burke, V.J.
登録日2009-03-03
公開日2009-12-01
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structural basis of the cross-reactivity of genetically related human anti-HIV-1 mAbs: implications for design of V3-based immunogens
Structure, 17, 2009
3GHB
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BU of 3ghb by Molmil
Crystal structure of anti-HIV-1 Fab 447-52D in complex with V3 peptide W2RW020
分子名称: Envelope glycoprotein, Fab 447-52D, heavy chain, ...
著者Kong, X.P, Burke, V.J.
登録日2009-03-03
公開日2009-12-01
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Structural basis of the cross-reactivity of genetically related human anti-HIV-1 mAbs: implications for design of V3-based immunogens
Structure, 17, 2009
3MCG
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BU of 3mcg by Molmil
THREE-DIMENSIONAL STRUCTURE OF A LIGHT CHAIN DIMER CRYSTALLIZED IN WATER. CONFORMATIONAL FLEXIBILITY OF A MOLECULE IN TWO CRYSTAL FORMS
分子名称: IMMUNOGLOBULIN LAMBDA DIMER MCG (LIGHT CHAIN)
著者Ely, K.R, Herron, J.N, Edmundson, A.B.
登録日1989-05-09
公開日1990-10-15
最終更新日2019-12-25
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Three-dimensional structure of a light chain dimer crystallized in water. Conformational flexibility of a molecule in two crystal forms.
J.Mol.Biol., 210, 1989
1QJU
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BU of 1qju by Molmil
HUMAN RHINOVIRUS 16 COAT PROTEIN IN COMPLEX WITH ANTIVIRAL COMPOUND VP61209
分子名称: 2,6-DIMETHYL-1-(3-[3-METHYL-5-ISOXAZOLYL]-PROPANYL)-4-[2N-METHYL-2H-TETRAZOL-5-YL]-PHENOL, MYRISTIC ACID, PROTEIN VP1, ...
著者Hadfield, A.T, Minor, I, Diana, G.D, Rossmann, M.G.
登録日1999-07-05
公開日1999-07-20
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Analysis of Three Structurally Related Antiviral Compounds in Complex with Human Rhinovirus 16
Proc.Natl.Acad.Sci.USA, 96, 1999
1QJY
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HUMAN RHINOVIRUS 16 COAT PROTEIN IN COMPLEX WITH ANTIVIRAL COMPOUND VP65099
分子名称: 2,6-DIMETHYL-1-(3-[3-METHYL-5-ISOXAZOLYL]-PROPANYL)-4-[2-METHYL-4-ISOXAZOLYL]-PHENOL, MYRISTIC ACID, PROTEIN VP1, ...
著者Hadfield, A.T, Diana, G.D, Rossmann, M.G.
登録日1999-07-06
公開日1999-07-20
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Analysis of Three Structurally Related Antiviral Compounds in Complex with Human Rhinovirus 16
Proc.Natl.Acad.Sci.USA, 96, 1999
1RHI
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HUMAN RHINOVIRUS 3 COAT PROTEIN
分子名称: CALCIUM ION, HUMAN RHINOVIRUS 3 COAT PROTEIN
著者Zhao, R, Rossmann, M.G.
登録日1996-06-17
公開日1997-03-12
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Human rhinovirus 3 at 3.0 A resolution.
Structure, 4, 1996
2MCG
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THREE-DIMENSIONAL STRUCTURE OF A LIGHT CHAIN DIMER CRYSTALLIZED IN WATER. CONFORMATIONAL FLEXIBILITY OF A MOLECULE IN TWO CRYSTAL FORMS
分子名称: IMMUNOGLOBULIN LAMBDA DIMER MCG (LIGHT CHAIN)
著者Ely, K.R, Herron, J.N, Edmundson, A.B.
登録日1989-05-09
公開日1990-10-15
最終更新日2019-12-25
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Three-dimensional structure of a light chain dimer crystallized in water. Conformational flexibility of a molecule in two crystal forms.
J.Mol.Biol., 210, 1989
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